Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,754 products)
- Apoptosis(6,187 products)
- Cell Cycle/Checkpoint(4,807 products)
- Chromatin/Epigenetics(2,573 products)
- Cytoskeletal Signaling(1,503 products)
- DNA Damage/DNA Repair(2,893 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,964 products)
- Immunology and Inflammation(3,697 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,246 products)
- Membrane Transporter/Ion Channel(3,137 products)
- Metabolism(10,096 products)
- Microbiology/Virology(7,552 products)
- Neuroscience(10,303 products)
- Other Inhibitors(35,769 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,402 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,921 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66573 products of "Inhibitors"
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Macbecin I
CAS:Hsp90 inhibitorFormula:C30H42N2O8Purity:98%Color and Shape:SolidMolecular weight:558.66(Z)-Lanoconazole
(Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.
Formula:C14H10ClN3S2Color and Shape:SolidMolecular weight:319.83CXCR2 antagonist 7
CXCR2 antagonist 7 is a powerful blocker with IC50s: 0.044 μM for binding, 0.66 μM for calcium mobilization.Formula:C14H14F2N6OSColor and Shape:SolidMolecular weight:352.36NNC-11-1585
CAS:NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.Formula:C18H19N3OSColor and Shape:SolidMolecular weight:325.43Tubulin inhibitor 22
Compound 4c: Strong tubulin inhibitor with anti-cancer & anti-angiogenic effects; halts MGC-803 cells in G2/M, triggers Caspase-mediated apoptosis.Formula:C20H17BrFNO4Color and Shape:SolidMolecular weight:434.26Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Formula:C80H102ClN15O14Color and Shape:SolidMolecular weight:1533.21Asimicin
CAS:Asimicin is a effective complex I inhibitor.Formula:C37H66O7Purity:98%Color and Shape:SolidMolecular weight:622.92FPDT
FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: >100 μM (astrocytes), 45-68 μM (GBM cells).Formula:C16H12FNO2SColor and Shape:SolidMolecular weight:301.34Danavorexton
CAS:Danavorexton is an orexin receptor agonist.Formula:C21H32N2O5SColor and Shape:SolidMolecular weight:424.55RhlR antagonist 1
RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.Formula:C12H10F2OColor and Shape:SolidMolecular weight:208.2EBI-1051
CAS:EBI-1051 is a highly potent and orally efficacious inhibitor of MEK (IC50: 3.9 nM).Formula:C18H15F2IN2O5Purity:98%Color and Shape:SolidMolecular weight:504.22KDOAM-25 trihydrochloride
KDOAM-25 trihydrochloride selectively inhibits KDM5 enzymes, boosts H3K4 methylation, and suppresses MM1S cell growth.Formula:C15H28Cl3N5O2Color and Shape:SolidMolecular weight:416.77Sdz 210-096
CAS:Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.Formula:C27H31NO2Color and Shape:SolidMolecular weight:401.54RGT-068A
CAS:RGT-068A is a potent, selective and oral bioavailable MALT1 inhibitor .Formula:C17H16ClN9O2Color and Shape:SolidMolecular weight:413.82Hsp90-IN-16
Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.Formula:C30H26FN3O6Color and Shape:SolidMolecular weight:543.54LXRβ agonist-2
CAS:LXRβ agonist-2 is a highly potent and β-selective liver X receptor (LXRβ) agonist with EC50 of 7 nM.Formula:C32H31F6N3O7Purity:98%Color and Shape:SolidMolecular weight:683.59Kalafungin
CAS:Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.Formula:C16H12O6Color and Shape:SolidMolecular weight:300.26AZ14145845
AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.Formula:C32H35N9OColor and Shape:SolidMolecular weight:561.68T01-1
CAS:T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.Formula:C26H29N3O6SColor and Shape:SolidMolecular weight:511.59SB 258741 hydrochloride
SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].Formula:C19H31ClN2O2SColor and Shape:SolidMolecular weight:386.98ZK-Thiazolidinone
CAS:ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.Formula:C23H26F3N5O2SColor and Shape:SolidMolecular weight:493.55SSTR5 antagonist 2 TFA
CAS:Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.Formula:C34H36F4N2O7Purity:98%Color and Shape:SolidMolecular weight:660.65KCa2 channel modulator 2
Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.Formula:C16H15ClFN5Color and Shape:SolidMolecular weight:331.78Ascofuranone
CAS:Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODHFormula:C23H29ClO5Color and Shape:SolidMolecular weight:420.93Tauro-ω-muricholic acid sodium
Tauro-ω-muricholic acid sodium (TωMCA sodium) is an analogue of tauro-α-muricholic acid, a bile acid of hepatic origin.Formula:C26H44NNaO7SColor and Shape:SolidMolecular weight:537.68Thielavin B
CAS:Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.Formula:C31H34O10Color and Shape:SolidMolecular weight:566.6GNE-203
CAS:GNE-203 is a Met inhibitor.Formula:C30H29Cl2F3N8O3Color and Shape:SolidMolecular weight:677.50TA-316
CAS:Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.Formula:C28H25BrN4O5S2Purity:98%Color and Shape:SolidMolecular weight:641.56EGFR-IN-18
EGFR-IN-18 strongly inhibits L858R/T790M/C797S mutant EGFR (4.9 nM) and also targets wild-type EGFR (47 nM).Formula:C33H28N6O3SColor and Shape:SolidMolecular weight:588.68Vimirogant hydrochloride
Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), >1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.Formula:C27H36ClF3N4O3SColor and Shape:SolidMolecular weight:588.21487Anti-MRSA agent 6
Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].Formula:C16H11F2N3Color and Shape:SolidMolecular weight:283.28PRMT5-IN-21
PRMT5-IN-21 (compound 1) is a potent inhibitor of cyclonucleoside PRMT5.Formula:C18H18F2N6O3Color and Shape:SolidMolecular weight:404.37PTP1B-IN-3 diammonium
PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.Formula:C12H13BrF2N3O3PColor and Shape:SolidMolecular weight:396.12Antibacterial agent 90
Antibacterial agent 90 (6n), a pleuromutilin derivative, targets Gram-positive pathogens and Mycoplasma pneumoniae.Formula:C30H42N2O6Color and Shape:SolidMolecular weight:526.66Anticancer agent 30
Anticancer agent 30 (6f-Z), a 3-arylidene-2-oxindole, selectively inhibits CDK2, showing potent anticancer potential.Formula:C22H15ClFNOColor and Shape:SolidMolecular weight:363.81AR-13324 M1 metabolite
CAS:AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.Formula:C19H19N3O2Purity:98%Color and Shape:SolidMolecular weight:321.37Acetylpepstatin
CAS:Acetylpepstatin is an inhibitor of HIV-1 protease, HIV-2 protease, aspartyl protease.Formula:C33H61N5O11Purity:98%Color and Shape:SolidMolecular weight:703.875D6808
D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.Formula:C30H25F3N6O2Color and Shape:SolidMolecular weight:558.55UTPγS trisodium salt
CAS:P2Y2 and P2Y4 receptor agonistFormula:C9H12N2Na3O14P3SPurity:98%Color and Shape:SolidMolecular weight:566.15BMS-748730
CAS:BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.Formula:C22H26ClN7O3SColor and Shape:SolidMolecular weight:504.01Tubulin inhibitor 14
Tubulin inhibitor 14 blocks NQO2 and microtubule formation, disrupts blood vessels, and may target tumors; IC50 of 1.0 μM.Formula:C15H9F2NOColor and Shape:SolidMolecular weight:257.23Haspin-IN-2
CAS:Haspin-IN-2 is a potent haspin inhibitor (IC50: 50 nM) and also inhibits CLK1 (IC50: 445 nM) and DYRK1A (IC50: 917 nM).Formula:C12H8N4O3Color and Shape:SolidMolecular weight:256.22S1P1 agonist 4
CAS:S1P1 agonist 4 exhibits enhanced potency with an EC 50 value of less than 0.05 mg/kg and a predicted human half-life (t1/2) of approximately 5 days, indicatingFormula:C24H31NO3Color and Shape:SolidMolecular weight:381.51Adecypenol
CAS:Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.Formula:C12H16N4O4Purity:98%Color and Shape:SolidMolecular weight:280.28Org-31710
CAS:Org-31710 is a progesterone receptor antagonist potentially for contraception.Formula:C30H39NO2Purity:98%Color and Shape:SolidMolecular weight:445.64Aurora/LIM kinase-IN-1
Aurora/LIM kinase-IN-1 (Compound F114) is a dual inhibitor targeting aurora and lim kinases, potentially useful in GBM cancer treatment efforts.Formula:C16H20N6OColor and Shape:SolidMolecular weight:312.37SGK1-IN-3
CAS:SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.Formula:C23H20Cl2N6O3SColor and Shape:SolidMolecular weight:531.4145-Iminodaunorubicin hydrochloride
CAS:5-Iminodaunorubicin HCl: quinone-modified anthracycline with antitumor properties, induces DNA breaks in cancer cells.Formula:C27H31ClN2O9Color and Shape:SolidMolecular weight:563.00Anticancer agent 69
Anticancer agent 69 targets PC3 cells (IC50=26 nM), raises ROS, lowers EGFR, and induces apoptosis.Formula:C19H26N8SColor and Shape:SolidMolecular weight:398.53GSK866
CAS:GSK866 is a selective glucocorticoid receptor agonist (SEGRA).Formula:C23H21Cl2F4N5O3Color and Shape:SolidMolecular weight:562.34
