Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,758 products)
- Apoptosis(6,191 products)
- Cell Cycle/Checkpoint(4,808 products)
- Chromatin/Epigenetics(2,580 products)
- Cytoskeletal Signaling(1,503 products)
- DNA Damage/DNA Repair(2,887 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,965 products)
- Immunology and Inflammation(3,700 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,136 products)
- Metabolism(10,096 products)
- Microbiology/Virology(7,554 products)
- Neuroscience(10,304 products)
- Other Inhibitors(35,764 products)
- Oxidation-Reduction(39 products)
- PI3K/Akt/mTOR Signaling(1,402 products)
- Proteases/Proteasome(1,672 products)
- Stem Cell and Derivatives(741 products)
- Tyrosine Kinase/Adaptors(1,922 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66571 products of "Inhibitors"
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(Rac)-OSMI-1
(Rac)-OSMI-1, a racemate, inhibits OGT (IC50: 2.7 μM) affecting O-GlcNAcylation without changing surface glycans.Formula:C28H25N3O6S2Color and Shape:SolidMolecular weight:563.64Mf 268
CAS:Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.Formula:C28H46N4O3Color and Shape:SolidMolecular weight:486.69BET-IN-6
CAS:BET-IN-6: Potent BRD2/4 inhibitor and ligand for PROTAC BRD2/BRD4 degrader-1 synthesis.Formula:C22H20N2O6SPurity:98%Color and Shape:SolidMolecular weight:440.47Arverapamil
CAS:Arverapamil is a chiral metabolite of Verapamil.Formula:C26H36N2O4Purity:99.87%Color and Shape:SolidMolecular weight:440.58GR 122222X
CAS:GR 122222X is an inhibitor of topoisomerase II.Formula:C26H35N5O11SPurity:98%Color and Shape:SolidMolecular weight:625.65Oncopterin
CAS:Oncopterin is found in urine from patients with solid and blood cancers.Formula:C12H18N6O3Color and Shape:SolidMolecular weight:294.31Fusarisetin A
CAS:Fusarisetin A, a pentacyclic fungal metabolite, is an acinar morphogenesis inhibitor .Formula:C22H31NO5Color and Shape:SolidMolecular weight:389.49TLR8 agonist 4
TLR8 agonist 4 inhibits wild-type and lamivudine/entecavir-resistant HBV; IC50: 0.15 μM and 0.10 μM.Formula:C28H27N5O5SColor and Shape:SolidMolecular weight:545.612-Methylsorbinol
CAS:2-Methylsorbinol is a bioactive chemical.Formula:C12H11FN2O3Color and Shape:SolidMolecular weight:250.23Tofogliflozin
CAS:Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).Formula:C22H26O6Purity:98%Color and Shape:SolidMolecular weight:386.44CB1/2 agonist 1
Potent CB1/2 agonist 1; crosses blood-brain barrier; anti-inflammatory, analgesic; for multiple sclerosis research.Formula:C21H24BrFN2O2Color and Shape:SolidMolecular weight:435.33Vindeburnol
CAS:Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.Formula:C17H20N2OColor and Shape:SolidMolecular weight:268.35Sucistil
Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].Formula:C9H15NO4SColor and Shape:SolidMolecular weight:233.28BMS-986143
CAS:BMS-986143: oral BTK inhibitor, IC50=0.26 nM, potential for autoimmune research, also targets TEC, BLK, BMX, TXK, YES1, ITK.Formula:C31H24Cl2N4O4Color and Shape:SolidMolecular weight:587.45Dihydro-β-erythroidine hydrobromide
CAS:Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H22BrNO3Purity:98%Color and Shape:White SolidMolecular weight:356.26CAII-IN-2
CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.Formula:C18H19BrN4SColor and Shape:SolidMolecular weight:403.34Methyl 5-thia-6,8,11,14-eicosatetraenoate
CAS:Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.Formula:C20H32O2SColor and Shape:SolidMolecular weight:336.53P-gp inhibitor 2
CAS:Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formula:C29H26N2O6Color and Shape:SolidMolecular weight:498.53BF-168
CAS:BF-168 is a candidate probe for PET and specifically recognizes both neuritic and diffuse plaques (Ki: 6.4 nM for Aβ1-42).Formula:C18H17FN2O2Color and Shape:SolidMolecular weight:312.34MNK1/2-IN-6
MNK1/2-IN-6: Strong, selective MNK1/2 inhibitor; IC50s: MNK1 at 2.3 nM, MNK2 at 3.4 nM; triggers dose-dependent apoptosis.Formula:C27H24N6OColor and Shape:SolidMolecular weight:448.52WIN 66306
CAS:WIN 66306: Cyclic heptapeptide, blocks NK1/NK2 receptors, inhibits substance P-triggered contractions in guinea pig ileum.Formula:C41H52N8O9Color and Shape:SolidMolecular weight:800.9SS-RJW100
SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57PKG1α activator 3
PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).Formula:C27H26Cl2N2O6Color and Shape:SolidMolecular weight:545.41XIAP degrader-1
XIAP degrader-1 is a small primary amine molecule that promotes the degradation of X-linked apoptosis inhibitory protein (XIAP).Formula:C34H45N5O4Color and Shape:SolidMolecular weight:587.75Clavicoronic acid
CAS:Clavicoronic acid, a β-lactamase inhibitor, boosts penicillin antibiotics against resistant bacteria.Formula:C15H18O4Color and Shape:SolidMolecular weight:262.3Kahweol Acetate
CAS:Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.Formula:C22H28O4Color and Shape:SolidMolecular weight:356.46CCW 28-3
CAS:CCW 28-3 is a novel potent covalent BRD4 degrader, degrading BRD4 in a proteasome- and RNF4-dependent manner without inhibiting RNF4 autoubiquitination activityFormula:C44H42Cl2N6O4SColor and Shape:SolidMolecular weight:821.81ZK168281
CAS:ZK168281 is a 1α,25(OH)2D3 analog, VDR antagonist with 0.1 nM Kd, and blocks receptor CoA interaction.Formula:C32H46O5Purity:98%Color and Shape:SolidMolecular weight:510.70MA242 free base
CAS:MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.Formula:C24H20ClN3O3SColor and Shape:SolidMolecular weight:465.95GR 83895
CAS:GR 83895 is an antagonist of prototype fibrinogen receptor.Formula:C29H39N9O8SPurity:98%Color and Shape:SolidMolecular weight:673.74hMAO-B/MB-COMT-IN-2
Dual inhibitor hMAO-B/MB-COMT-IN-2 targets hMAO-B (IC50: 4.27μM) & MB-COMT (IC50: 2.69μM), aids in neurodegenerative research.Formula:C17H18N2O3Color and Shape:SolidMolecular weight:298.34USP7-IN-10
CAS:USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.Formula:C26H29ClN4O3SColor and Shape:SolidMolecular weight:513.05PF-03715455
CAS:PF-03715455 is a potent p38 MAPK inhibitor, reducing TNFα in blood (IC50=1.7 nM) with selectivity for p38α, and may treat COPD.Formula:C35H34ClN7O3S2Purity:98%Color and Shape:SolidMolecular weight:700.27ODN 2088
CAS:ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.Color and Shape:SolidDN-F01
DN-F01 exhibits a potent calcium-dependent inhibitory effect on cardiac myofibrillar ATPase activity, with an IC50 of 11 ± 4 nmol/L.Formula:C22H16N2O2Color and Shape:SolidMolecular weight:340.37(25S)-δ7-Dafachronic acid
CAS:(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.Formula:C27H42O3Purity:98%Color and Shape:SolidMolecular weight:414.62Hcyb1
Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.Formula:C24H20N4OColor and Shape:SolidMolecular weight:380.44Barixibat
CAS:Barixibat is a bile acid transport inhibitor.Formula:C42H55N5O8Color and Shape:SolidMolecular weight:757.91EGFR-IN-24
EGFR-IN-24 is a potent inhibitor of EGFR and inhibits EGFR (del19/T790M/C797S) and EGFR (L858R/T790M/C797S).Formula:C30H35FN6O3Color and Shape:SolidMolecular weight:546.64HDAC-IN-32
HDAC-IN-32, potent inhibitor: IC50—HDAC1 (5.2 nM), HDAC2 (11 nM), HDAC6 (28 nM). Effective anti-tumor and immunity-boosting traits.Formula:C20H23N3O3Color and Shape:SolidMolecular weight:353.41Metoquizine
CAS:Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Formula:C22H27N5OPurity:98%Color and Shape:SolidMolecular weight:377.48Cap-dependent endonuclease-IN-17
CAS:CEN inhibitor IN-17 targets influenza A/H3N2; IC50: 1.29 μM. From patent CN112898346A, DSC701.Formula:C24H20F2N3O7PSColor and Shape:SolidMolecular weight:563.47Calcipotriol Impurity C
CAS:Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.Formula:C27H40O3Purity:98%Color and Shape:SolidMolecular weight:412.614MS117
MS117 is a first-in-class and cell-active irreversible covalent inhibitor of protein arginine methyltransferase 6 (PRMT6) (IC50 = 18 nM) [1].Formula:C17H22N4OColor and Shape:SolidMolecular weight:298.38MGAT2-IN-1
CAS:MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively).Formula:C27H21ClF5N7O3SColor and Shape:SolidMolecular weight:654.01STAT3-IN-8
CAS:"STAT3-IN-8 (compound H172) is a potent inhibitor of STAT3 with potential applications in cancer research [1]."Formula:C19H7F7N2O3Purity:98%Color and Shape:SolidMolecular weight:444.26UK 356618
CAS:UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).
Formula:C34H43N3O4Purity:98%Color and Shape:SolidMolecular weight:557.72Antibacterial agent 118
Antibacterial agent 118, potent against various mycobacteria, has MIC values ranging from 10.2 to 163.0 μM. Useful in TB research.Formula:C19H21N5O2SColor and Shape:SolidMolecular weight:383.47SCP1-IN-2
SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.Formula:C19H17F3N2O6S2Color and Shape:SolidMolecular weight:490.47BW-10
CAS:BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.Formula:C57H72N14O8Color and Shape:SolidMolecular weight:1081.27
