Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,749 products)
- Apoptosis(6,182 products)
- Cell Cycle/Checkpoint(4,805 products)
- Chromatin/Epigenetics(2,571 products)
- Cytoskeletal Signaling(1,499 products)
- DNA Damage/DNA Repair(2,896 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,962 products)
- Immunology and Inflammation(3,694 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,246 products)
- Membrane Transporter/Ion Channel(3,135 products)
- Metabolism(10,102 products)
- Microbiology/Virology(7,552 products)
- Neuroscience(10,303 products)
- Other Inhibitors(35,763 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,922 products)
- Ubiquitination(1,715 products)
Show 16 more subcategories
Found 66575 products of "Inhibitors"
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Anti-inflammatory agent 6
Anti-inflammatory agent 6 blocks IKKα/β, IκBα, and NF-κB p65 phosphorylation, key to controlling inflammation.Formula:C22H20O12Color and Shape:SolidMolecular weight:476.39PDE4-IN-6
PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.Formula:C25H20FNO5SColor and Shape:SolidMolecular weight:465.49ATM Inhibitor-4
ATM Inhibitor -4: selective, potent (IC50: 0.32 nM), inhibits PI3K family, stable, stops mTOR at 1 μM.Formula:C26H29FN6O3Color and Shape:SolidMolecular weight:492.55Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formula:C22H32N4O4Purity:98.57%Color and Shape:SolidMolecular weight:416.51Lp-PLA2-IN-10
Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.Formula:C21H15F5N4O4Color and Shape:SolidMolecular weight:482.36SGLT inhibitor-1
CAS:SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s of 43 nM and 9 nM, respectively).Formula:C24H27FO8Purity:98%Color and Shape:SolidMolecular weight:462.46MDL-100240
CAS:MDL-100240 inhibits ACE/neprilysin, effective against hypertension-induced heart/vascular changes.Formula:C26H28N2O5SPurity:98%Color and Shape:SolidMolecular weight:480.58AChE-IN-8
AChE-IN-8 (Compound 19), potent acetylcholinesterase blocker; IC50 = 1.95 μM; potential Alzheimer's treatment.Formula:C20H22N4O2SColor and Shape:SolidMolecular weight:382.48(-)-Adenophorine
CAS:(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.Formula:C8H17NO4Color and Shape:SolidMolecular weight:191.22Atorvastatin 3-Deoxyhept-2E-Enoic Acid
CAS:Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.Formula:C33H33FN2O4Purity:98%Color and Shape:SolidMolecular weight:540.62CXCR4 modulator-1
CAS:CXCR4 modulator-1 (ZINC72372983) is potent (EC50=100nM) with uses in anti-inflammatory, anticancer, and anti-HIV research.Formula:C23H27N5O2Color and Shape:SolidMolecular weight:405.49Dihydro-β-erythroidine hydrobromide
CAS:Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H22BrNO3Purity:98%Color and Shape:White SolidMolecular weight:356.26MK-7128
CAS:MK-7128 is a CB1 receptor inverse agonist.Formula:C29H25ClF2N4O2Color and Shape:SolidMolecular weight:534.98GSK3368715 3HCl
CAS:GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81Formula:C20H41Cl3N4O2Purity:98%Color and Shape:SolidMolecular weight:475.92Eilatine
CAS:Eilatine is a novel marine alkaloid inhibits in vitro proliferation of progenitor cells in chronic myeloid leukemia patients.Formula:C24H12N4Color and Shape:SolidMolecular weight:356.38Leukotriene B4 dimethyl amide
CAS:LTB4 dimethyl amide: inhibits human neutrophil degranulation and rat lysozyme release; antagonizes LTB4 receptor on guinea pig lung membranes (Ki = 130 nM).Formula:C22H37NO3Color and Shape:SolidMolecular weight:363.53Uprosertib hydrochloride
CAS:Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).Formula:C18H17Cl3F2N4O2Purity:98%Color and Shape:SolidMolecular weight:465.71CDK2-IN-9
CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.Formula:C21H16ClN3O4SColor and Shape:SolidMolecular weight:441.89DNA Gyrase-IN-1
DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.Formula:C24H24FN7O6Color and Shape:SolidMolecular weight:525.49USP7-IN-6
CAS:USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).Formula:C41H43N7O4SPurity:98%Color and Shape:SolidMolecular weight:729.89MurB-IN-1
MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.Formula:C12H7Cl2F3N2O2Color and Shape:SolidMolecular weight:339.1MALT1-IN-5
CAS:MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.Formula:C17H17ClF2N6O3Color and Shape:SolidMolecular weight:426.80TIY-7
TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.Color and Shape:SolidMAP3K14-IN-173
CAS:MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.Formula:C29H31N7O2Color and Shape:SolidMolecular weight:509.60Burapitant
CAS:Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
Formula:C31H35Cl2F6N3O3Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:682.52PDE4B/7A-IN-1
CAS:5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.Formula:C25H35N3O3Color and Shape:SolidMolecular weight:425.56DWN-12088 HCl
CAS:DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitorFormula:C15H21Cl4N3OColor and Shape:SolidMolecular weight:401.15CVS-1578
CAS:CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Formula:C20H30N6O5SColor and Shape:SolidMolecular weight:466.55Oxythiamine diphosphate ammonium
Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).Color and Shape:SolidTRK-IN-19
TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.Formula:C22H26FN5O2Color and Shape:SolidMolecular weight:411.47Seco-Duocarmycin SA
CAS:Seco-Duocarmycin SA is a highly potent DNA alkylator used as an ADC cytotoxin.Formula:C25H24ClN3O7Purity:98%Color and Shape:SolidMolecular weight:513.93LASSBio-1632
LASSBio-1632: Novel anti-asthmatic, blocks PDE4A/D, reduces AHR & lung TNF-α, crosses BBB.Formula:C18H20N2O6SColor and Shape:SolidMolecular weight:392.43Arverapamil
CAS:Arverapamil is a chiral metabolite of Verapamil.Formula:C26H36N2O4Purity:99.87%Color and Shape:SolidMolecular weight:440.58MK-8825
CAS:MK-8825 is a CGRP receptor antagonist.Formula:C31H30F2N6O3Color and Shape:SolidMolecular weight:572.61Befiradol hydrochloride
CAS:Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.
Formula:C20H23Cl2F2N3OPurity:99.1%Color and Shape:SolidMolecular weight:430.32AS2521780
CAS:AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).Formula:C30H41N7OSPurity:98%Color and Shape:SolidMolecular weight:547.76BMS-824
CAS:BMS-824: potent HCV NS5A inhibitor, IC50 ~5 nM, therapeutic index >10,000, specific to HCV.Formula:C27H25F3N4O5Color and Shape:SolidMolecular weight:542.51Sdz 210-096
CAS:Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.Formula:C27H31NO2Color and Shape:SolidMolecular weight:401.54PAT-347
CAS:PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.Formula:C28H21ClF2N2O3SColor and Shape:SolidMolecular weight:538.99Fumarranol
CAS:Fumarranol inhibits angiogenesis and malaria growth by targeting PfMAP2.Formula:C16H24O4Color and Shape:SolidMolecular weight:280.36D4R antagonis-2
Potent D4R antagonist-2: selective, IC50=6.52 μM, good in vitro PK and brain penetration, potential for Parkinson's research.Formula:C21H23ClF2N2O2Color and Shape:SolidMolecular weight:408.87GS-9822
CAS:GS-9822 is a new LEDGIN inhibitor targeting LEDGF/p75 to alter HIV integration, showing a block-and-lock effect in cells.Formula:C36H39ClN4O4SColor and Shape:SolidMolecular weight:659.247(Z),11(Z)-Nonacosadiene
CAS:7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.Formula:C29H56Color and Shape:SolidMolecular weight:404.75KRAS G12C inhibitor 50
CAS:KRAS G12C inhibitor 50 is a KRAS G12C inhibitor (IC50: 46.7 nM).Formula:C31H34N8O2Color and Shape:SolidMolecular weight:550.65SCP1-IN-1
CAS:SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.Formula:C20H19F3N2O7S2Purity:99.53%Color and Shape:SoildMolecular weight:520.5Ref: TM-T60077
1mg49.00€5mg104.00€10mg169.00€25mg311.00€50mg472.00€100mg707.00€1mL*10mM (DMSO)119.00€Flutimide
CAS:Flutimide: Endonuclease inhibitor, IC50 = 3μM, for research on acute respiratory diseases like influenza.Formula:C12H18N2O3Color and Shape:SolidMolecular weight:238.28Macropa-NCS
CAS:Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.Formula:C27H35N5O8SPurity:98%Color and Shape:SolidMolecular weight:589.66Antitubercular agent-23
Antitubercular agent-23 combats Candida albicans (MIC: 1.1 μg/ml) and M. tuberculosis (MIC: 1 μg/ml).Formula:C20H22FN5O8SColor and Shape:SolidMolecular weight:511.48A-9758
CAS:A-9758: RORγt selective inverse agonist, IC50 5nM, inhibits IL-17A, Th17, and treats psoriasis.Formula:C25H23Cl2F3N2O3Purity:98%Color and Shape:SolidMolecular weight:527.36LSD1-IN-18
LSD1-IN-18 inhibits LSD1 (Ki: 0.156 μM, KD: 0.075 μM), blocking THP-1 and MDA-MB-231 cell growth (IC50: 0.16, 0.21 μM).Formula:C31H40N6O2Color and Shape:SolidMolecular weight:528.69
