Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,754 products)
- Apoptosis(6,187 products)
- Cell Cycle/Checkpoint(4,807 products)
- Chromatin/Epigenetics(2,573 products)
- Cytoskeletal Signaling(1,503 products)
- DNA Damage/DNA Repair(2,893 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,964 products)
- Immunology and Inflammation(3,697 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,246 products)
- Membrane Transporter/Ion Channel(3,137 products)
- Metabolism(10,096 products)
- Microbiology/Virology(7,552 products)
- Neuroscience(10,303 products)
- Other Inhibitors(35,769 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,402 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,921 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66573 products of "Inhibitors"
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Alkyne-probe 1
Alkyne-probe 1 is usually used as an Alkyne-labeled fluorescent or chemical probe.Formula:C14H23N5O2Purity:98%Color and Shape:SolidMolecular weight:293.36CXCR4 antagonist 3
CXCR4 antagonist 3, aka compound 12a, has 11 nM IC50, shares TIQ15 traits, and is promising in HIV research.Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52NS2B/NS3-IN-5
Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.Formula:C14H9IN2O3SColor and Shape:SolidMolecular weight:412.2Calphostin D
CAS:Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.Formula:C30H30O10Color and Shape:SolidMolecular weight:550.55AL-6556
CAS:AL-6556 is a prostaglandin DP receptor agonist.Formula:C20H33ClO5Color and Shape:SolidMolecular weight:388.93Antitumor agent-43
Antitumor agent-43 (Compound 4B) is a potent antitumor agent that induces cell cycle arrest at G2/M phase.Formula:C16H8N2O3Color and Shape:SolidMolecular weight:276.25KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Formula:C35H39F3N8O2Color and Shape:SolidMolecular weight:660.73SOS1-IN-9
SOS1-IN-9 is a potent inhibitor of SOS1 that acts on KRAS G12C-SOS1 (IC50: 116.5 nM).Formula:C22H28F3N5OColor and Shape:SolidMolecular weight:435.49P-gp modulator 2
P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.Formula:C22H20BrN3O4Color and Shape:SolidMolecular weight:470.32Carbonic anhydrase inhibitor 8
R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).Formula:C20H25N3O4SColor and Shape:SolidMolecular weight:403.5IRAK4-IN-12
IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).Formula:C24H31FN8OColor and Shape:SolidMolecular weight:466.55Epothilone E
CAS:Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumorFormula:C26H39NO7SColor and Shape:SolidMolecular weight:509.66Purine phosphoribosyltransferase-IN-2
Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:531.17(E)-10-Hydroxynortriptyline maleate
CAS:(E)-10-Hydroxy Nortriptyline maleate, a derivative of antidepressant Nortriptyline, eases depression symptoms.Formula:C23H25NO5Purity:98%Color and Shape:SolidMolecular weight:395.455BAY-364
CAS:BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+Formula:C23H19N3O4Color and Shape:SolidMolecular weight:401.41Oberadilol
CAS:Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory actionFormula:C25H30ClN5O3Color and Shape:SolidMolecular weight:483.99Anti-inflammatory agent 23
Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.Formula:C34H49NO6Color and Shape:SolidMolecular weight:567.76Metocurine chloride
CAS:Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.Formula:C40H48Cl2N2O6Color and Shape:SolidMolecular weight:723.72PKCiota-IN-1
CAS:PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).Formula:C25H22FN5OColor and Shape:SolidMolecular weight:427.47Inupadenant HCl
CAS:Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.Formula:C25H27ClF2N8O4S2Color and Shape:SolidMolecular weight:641.11FT001
CAS:FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.Formula:C25H29N3O4SPurity:99.9%Color and Shape:SolidMolecular weight:467.58Ref: TM-T27392
1mg115.00€2mg172.00€5mg255.00€10mg374.00€25mg562.00€50mg787.00€100mg1,074.00€500mg2,147.00€1mL*10mM (DMSO)299.00€COX-2-IN-7
COX-2-IN-7: potent, orally active COX-2 inhibitor with higher selectivity than Celecoxib, IC50 6.585 uM, anti-inflammatory, low ulcer risk.Formula:C15H13N3O2S2Color and Shape:SolidMolecular weight:331.41Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).Formula:C18H17N3O4S2Color and Shape:SolidMolecular weight:403.48MK-7445
CAS:MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.Formula:C21H13Cl2N7OColor and Shape:SolidMolecular weight:450.28Dopamine D3 receptor ligand-1
Dopamine D 3 receptor ligand is a potent, selective, high-affinity dopamine D3 receptor ligand that is 89 times more selective for D3 (Ki: 8 nM) than D2 (Ki:Formula:C27H29N5OColor and Shape:SolidMolecular weight:439.55PD 113271
CAS:PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.Formula:C19H27O10PPurity:98%Color and Shape:SolidMolecular weight:446.39Ph-Ph+
Ph-Ph+ is a dimerized phenanthroline derivative with antitumor, antibacterial, and antifungal effects.Formula:C24H17N4Color and Shape:SolidMolecular weight:361.42Thalicarpine
CAS:Thalicarpine, a natural anticancer alkaloid, inhibits p-glycoprotein and induces DNA damage, arresting cell cycle.Formula:C41H48N2O8Color and Shape:SolidMolecular weight:696.83AZ-PFKFB3-67 quarterhydrate
AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).Formula:C26H27N5O4Color and Shape:SolidMolecular weight:460.01HDAC10-IN-2
HDAC10-IN-2, a selective HDAC10 inhibitor (IC50=20nM), modulates autophagy in FLT3-ITD+ acute myeloid leukemia.Formula:C19H22N2O2Color and Shape:SolidMolecular weight:310.39IRAK4-IN-9
CAS:IRAK4-IN-9 is a potent IRAK4 inhibitor with an IC50 of 1.5 nM, promising for inflammatory, autoimmune diseases, and cancer research.Formula:C22H25N7Color and Shape:SolidMolecular weight:387.48Cathepsin C-IN-3
Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).Formula:C28H21F3N6OSColor and Shape:SolidMolecular weight:546.57AM Toxin II
CAS:AM Toxin II is a Cyclic tetradepsipeptide isolated from Alternaria mali.Formula:C22H29N3O5Color and Shape:SolidMolecular weight:415.49BRD5631
CAS:BRD5631 is an autophagy enhancer, enhances autophagy through an mTOR-independent pathway.Formula:C30H35N3O4Purity:98%Color and Shape:SolidMolecular weight:501.62Antibacterial agent 112
Compound 112: Powerful antibacterial, MIC 1250 μM against B. subtilis, E. coli, E. faecalis, S. typhimurium, S. aureus; also an HIV-1 antibody.Formula:C35H23N5O5Color and Shape:SolidMolecular weight:593.59Antileishmanial agent-5
Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.Formula:C17H17ClN4O4Color and Shape:SolidMolecular weight:376.79Onalespib lactate
CAS:Onalespib lactate is a second-generation, potent and selective HSP90 Inhibitor with antitumor activity.Formula:C27H37N3O6Color and Shape:SolidMolecular weight:499.6HCV-IN-40
CAS:HCV-IN-39 is a potent oral drug inhibiting HCV, effective on GT1a (EC50: 0.259μM), GT1b (EC50: 0.434μM), GT1b CES1 (EC50: 0.069μM) replicons.Formula:C21H26BrFN3O9PColor and Shape:SolidMolecular weight:594.32G-4120
CAS:G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.Formula:C26H36N8O11SColor and Shape:SolidMolecular weight:668.68Top/HDAC-IN-1
Top/HDAC-IN-1: Dual Top/HDAC inhibitor, potent against HDAC1-3,6,8 and HCT116 cells; blocks G2 phase, induces apoptosis.Formula:C29H27N5O4Color and Shape:SolidMolecular weight:509.56Zalunfiban dihydrochloride
Zalunfiban (RUC-4) is a potent αIIbβ3 platelet antagonist, IC50 45 nM, used in myocardial infarction research.Formula:C16H20Cl2N8O2SColor and Shape:SolidMolecular weight:459.35ORIC-101
CAS:ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.Formula:C34H47NO2Purity:98%Color and Shape:SolidMolecular weight:501.74Rafutrombopag
CAS:Rafutrombopag is a thrombopoietin (TPO) agonist.Formula:C25H22N4O5Color and Shape:SolidMolecular weight:458.47CD73-IN-12
CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.Formula:C17H14F2N4O2Color and Shape:SolidMolecular weight:344.329(S),10(S),13(S)-TriHOME
CAS:9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.Formula:C18H34O5Color and Shape:SolidMolecular weight:330.46AChE/BChE-IN-1
AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.Formula:C32H35ClN6O3Color and Shape:SolidMolecular weight:587.11Cap-dependent endonuclease-IN-14
CAS:Cap-dependent endonuclease-IN-14 hinders CEN and could treat influenza virus infections. (Patent CN113620948A, compound 1-c).Formula:C30H23FN2O6SColor and Shape:SolidMolecular weight:558.58c-Met/HDAC-IN-2
CAS:Potent dual c-Met/HDAC inhibitor, IC50: HDAC1 5.4 nM, c-Met 18.49 nM; anti-cancer, induces apoptosis, G2/M arrest in HCT-116.Formula:C34H33N5O7Color and Shape:SolidMolecular weight:623.66Antitubercular agent-22
Antitubercular agent-22 combats Candida albicans (MIC: 2.34 μg/ml) and M. tuberculosis (MIC: 2 μg/ml).Formula:C24H28FN5O8Color and Shape:SolidMolecular weight:533.51AFP-07
CAS:AFP-07 is a highly selective and potent agonist. It was used for the prostacyclin receptor.Formula:C22H29F2NaO5Purity:98%Color and Shape:SolidMolecular weight:434.45
