Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,825 products)
- Apoptosis(6,305 products)
- Cell Cycle/Checkpoint(4,863 products)
- Chromatin/Epigenetics(2,608 products)
- Cytoskeletal Signaling(1,555 products)
- DNA Damage/DNA Repair(2,875 products)
- Endocrinology/Hormones(3,752 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,999 products)
- Immunology and Inflammation(3,863 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,253 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,145 products)
- Microbiology/Virology(7,618 products)
- Neuroscience(10,356 products)
- Other Inhibitors(35,866 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,426 products)
- Proteases/Proteasome(1,688 products)
- Stem Cell and Derivatives(737 products)
- Tyrosine Kinase/Adaptors(1,976 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66548 products of "Inhibitors"
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Cap-dependent endonuclease-IN-25
CAS:Cap-dependent endonuclease-IN-25 is a potent inhibitor of CEN, useful in studying Orthomyxoviridae viruses. (See WO2020075080A1, compound 4.)Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48S1PR1 agonist 2
CAS:S1PR1 agonist 2 is potent for autoimmune research (from WO2021175225A1).Formula:C25H25N5O4Color and Shape:SolidMolecular weight:459.50Gallinamide A
CAS:Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.Formula:C31H52N4O7Color and Shape:SolidMolecular weight:592.77U 75875
CAS:U 75875 is a protease inhibitor.Formula:C45H61N7O7Color and Shape:SolidMolecular weight:812.01Aristoforin
CAS:Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.Formula:C37H54O6Color and Shape:SolidMolecular weight:594.82ZD6021
CAS:ZD6021 is an antagonist of neurokinin 1 receptor.Formula:C35H35Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:632.64TLR7/8 antagonist 2
TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.Formula:C22H26FN5Color and Shape:SolidMolecular weight:379.47SphK1-IN-1
SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.Formula:C22H22N6O2Color and Shape:SolidMolecular weight:402.45MI-1481
CAS:MI-1481: potent MML1 inhibitor, IC50 3.6 nM; disrupts menin-MLL1, active in MLL leukemia.Formula:C29H30F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:597.65Musettamycin
CAS:Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.Formula:C36H45NO14Color and Shape:SolidMolecular weight:715.74Antibacterial agent 88
Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus.Formula:C31H44N2O6SColor and Shape:SolidMolecular weight:572.76Desacetylravidomycin
CAS:Desacetylravidomycin is a new inhibitor of IL-4 signal transduction, produced by Streptomyces sp. WK-6326.Formula:C29H31NO8Color and Shape:SolidMolecular weight:521.56AKR1C3-IN-7
AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.Formula:C24H20N2O4Color and Shape:SolidMolecular weight:400.43Hypoglycemic agent 1
CAS:Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.Formula:C25H24FN5O4Purity:98%Color and Shape:SolidMolecular weight:477.49GPX4-IN-3
CAS:GPX4-IN-3 (26a) is a potent GPX4 inhibitor, inducing selective ferroptosis with 71.7% inhibition at 1 μM.Formula:C29H24ClN3O3SColor and Shape:SolidMolecular weight:530.04AA 497 (Free Base)
CAS:AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.Formula:C14H21NO3Purity:98%Color and Shape:SolidMolecular weight:251.32TT15
CAS:TT15 is an agonist of the GLP-1R.Formula:C51H44Cl2N4O6Color and Shape:SolidMolecular weight:879.82UK 356618
CAS:UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).Formula:C34H43N3O4Purity:98%Color and Shape:SolidMolecular weight:557.72Glutaminyl cyclases-IN-1
Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.Formula:C25H30N6O2SColor and Shape:SolidMolecular weight:478.61LY210073
CAS:LY210073 is an antagonist of the Leukotriene B4 (LTB4) receptor (IC50: 6.2 nM).Formula:C30H28O8Purity:98%Color and Shape:SolidMolecular weight:516.54hCAII-IN-5
CAS:hCAII-IN-5 (compound 12h) is a potent, selective inhibitor of human carbonic anhydrase II (hCA II) with an inhibition constant (IC50) of 4.55 µM [1].Formula:C29H18N2O7Color and Shape:SolidMolecular weight:506.46PD-1-IN-17
CAS:PD-1-IN-17 is an inhibitor of programmed cell death-1 (PD-1). PD-1-IN-17 inhibits 92% splenocyte proliferation at 100 nM.Formula:C13H22N6O7Purity:99.6%Color and Shape:SolidMolecular weight:374.35NTPDase-IN-3
CAS:NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.Formula:C22H24ClN3OS2Color and Shape:SolidMolecular weight:446.03Ph-Ph+
Ph-Ph+ is a dimerized phenanthroline derivative with antitumor, antibacterial, and antifungal effects.Formula:C24H17N4Color and Shape:SolidMolecular weight:361.42RAD51-IN-5
CAS:RAD51-IN-5 blocks RAD51; may aid mitochondrial disorder research. (WO2021164746A1, cmpd 3)Formula:C26H38N4O5S2Color and Shape:SolidMolecular weight:550.73BNTX maleate
CAS:δ1 opioid receptor antagonistFormula:C31H31NO8Purity:98%Color and Shape:SolidMolecular weight:545.58LA-810
CAS:LA-810 is a nitrous oxide donor.Formula:C15H25N5O7SColor and Shape:SolidMolecular weight:419.45Tofacitinib Prodrug-1
Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.Formula:C36H39ClN10O7Color and Shape:SolidMolecular weight:759.21CVS-1578
CAS:CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Formula:C20H30N6O5SColor and Shape:SolidMolecular weight:466.55MAP3K14-IN-173
CAS:MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.Formula:C29H31N7O2Color and Shape:SolidMolecular weight:509.60L-Afegostat
CAS:L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.Formula:C6H13NO3Color and Shape:SolidMolecular weight:147.17ONO-AE1-329
CAS:ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.Formula:C22H30O6S2Color and Shape:SolidMolecular weight:454.6MRS2179 tetrasodium hydrate
MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:576.21YM-60828 dihydrochloride
CAS:YM-60828 dihydrochloride is a Factor Xa (FXa) inhibitor and anticoagulant used in the treatment of venous thromboembolic disease.Formula:C27H33Cl2N5O5SColor and Shape:SolidMolecular weight:610.55T01-1
CAS:T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.Formula:C26H29N3O6SColor and Shape:SolidMolecular weight:511.59Ibafloxacine
CAS:Ibafloxacine (R835) is a fluoroquinolone antibiotic that is used exclusively in veterinary applications and shows zero good bacteriostatic effect againstFormula:C15H14FNO3Purity:97.67%Color and Shape:SolidMolecular weight:275.27Fonadelpar
CAS:Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.Formula:C25H23F3N2O4SPurity:98%Color and Shape:SolidMolecular weight:504.52CHK1-IN-2
CAS:CHK1-IN-2 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 6 nM).Formula:C20H22N4OSPurity:98%Color and Shape:SolidMolecular weight:366.48Leustroducsin B
CAS:Leustroducsin B is a novel colony-stimulating factor (CSF) inducer extracted from Streptomyces platensis SANK 60191.Formula:C34H56NO10PColor and Shape:SolidMolecular weight:669.78Fandosentan
CAS:Fandosentan is an endothelin receptor antagonist.Formula:C25H18F3NO6SColor and Shape:SolidMolecular weight:517.47[D-Leu-4]-OB3
CAS:[D-Leu-4]-OB3 suppresses the expression of genes associated with inflammation, proliferation, and metastasis, as well as the expression of PD-L1.Formula:C29H50N8O12SColor and Shape:SolidMolecular weight:734.82Riminkefon
CAS:Riminkefon is a kappa opioid receptor agonist .Formula:C38H57N7O6Color and Shape:SolidMolecular weight:707.9CI 922
CAS:CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.Formula:C26H30N10O6Color and Shape:SolidMolecular weight:578.58Guraxetan
Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.Formula:C20H34N4O9Color and Shape:SolidMolecular weight:474.51Antiangiogenic agent 2
Antiangiogenic agent 2 (compound 3b) is a potent inhibitor of thymidine phosphorylase (IC50: 39.71 μM) and exhibits anti-angiogenic effects.
Formula:C26H26FN3O4Color and Shape:SolidMolecular weight:463.5KR-67607
CAS:KR-67607, or NTX-101, is a novel 11β-HSD1 inhibitor that protects against eye injury by reducing cortisol and preserving eye structures.Formula:C24H29Cl2F3N4O4SColor and Shape:SolidMolecular weight:597.48LpxA-IN-1
CAS:LpxA-IN-1, a novel UDP-N-acetylglucosamine acyltransferase (LpxA) inhibitor exhibiting potent activity (IC 50 2 nM), effectively targets Pseudomonas aeruginosaFormula:C21H11D7F3N5O3Color and Shape:SolidMolecular weight:452.44PF-06305591 dihydrate
PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADMEFormula:C15H26N4O3Color and Shape:SolidMolecular weight:310.39Pateamine A
CAS:Pateamine A: marine-sourced macrolide from Mycale hentscheli; anticancer, antiviral, and translation inhibitor.Formula:C31H45N3O4SColor and Shape:SolidMolecular weight:555.77
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