Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,564 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,725 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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Falecalcitriol
CAS:Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.Formula:C27H38F6O3Purity:98%Color and Shape:SolidMolecular weight:524.58HIF-2α-IN-5
CAS:HIF-2α-IN-5 is a potent HIF-2α inhibitor with an IC 50 of < 50 nM [1].Formula:C15H12F4O3S2Color and Shape:SolidMolecular weight:380.38SLC4101431
SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.Formula:C29H28ClN7OSColor and Shape:SolidMolecular weight:558.1S100A2-p53-IN-1
CAS:S100A2-p53-IN-1 inhibits S100A2-p53 in pancreatic cancer, stunting MiaPaCa-2 cell growth at 1.2-3.4 μM.Formula:C20H20F6N2O4SColor and Shape:SolidMolecular weight:498.44Riminkefon
CAS:Riminkefon is a kappa opioid receptor agonist .Formula:C38H57N7O6Color and Shape:SolidMolecular weight:707.9Purine phosphoribosyltransferase-IN-2
Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:531.17Homopteroic Acid
CAS:Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.Formula:C15H14N6O3Color and Shape:SolidMolecular weight:326.31MLKL-IN-1
MLKL-IN-1 is a covalent inhibitor of MLKL with a Kd value of 50 μM.Formula:C19H20N2O3Color and Shape:SolidMolecular weight:324.37GLS1 Inhibitor-5
GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.Color and Shape:SolidCD73-IN-13
CD73-IN-13, a potent CD73 inhibitor, may be developed for tumor-related disease treatment.Formula:C13H11F3N4O2Color and Shape:SolidMolecular weight:312.25MK-7128
CAS:MK-7128 is a CB1 receptor inverse agonist.Formula:C29H25ClF2N4O2Color and Shape:SolidMolecular weight:534.98Antitubercular agent-13
Compound 3d: antitubercular, MIC 0.007 μg/mL vs MTB H37Rv, 1.851 μg/mL vs MDR-MTB 16833, metabolically unstable.Formula:C18H18N4O5Color and Shape:SolidMolecular weight:370.36Antifungal agent 42
Antifungal 42 blocks biofilm formation and inhibits C.albicans' CYP51.Formula:C22H20Cl2N4Se2Color and Shape:SolidMolecular weight:569.25NNTA
CAS:NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.Formula:C31H32N2O4Color and Shape:SolidMolecular weight:496.60FPDT
FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: >100 μM (astrocytes), 45-68 μM (GBM cells).Formula:C16H12FNO2SColor and Shape:SolidMolecular weight:301.34TS010
TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 μM. It holds significant promise for advancements in cancer research [1].Formula:C16H12N4O4SColor and Shape:SolidMolecular weight:356.36Canosimibe
CAS:Canosimibe is a cholesterol absorption inhibitorFormula:C44H60FN3O10Color and Shape:SolidMolecular weight:809.96Rezatapopt
CAS:Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.Formula:C28H31F4N5O2Purity:98.12%Color and Shape:SolidMolecular weight:545.57(-)-Adenophorine
CAS:(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.Formula:C8H17NO4Color and Shape:SolidMolecular weight:191.22Fosmanogepix
CAS:Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.Formula:C22H21N4O6PPurity:98%Color and Shape:SolidMolecular weight:468.40A 76889
CAS:A 76889 is an inhibitor of HIV-1 protease.Formula:C44H58N8O6Purity:98%Color and Shape:SolidMolecular weight:794.98Dyrk1A/α-synuclein-IN-1
Dyrk1A/α-synuclein-IN-1 (Compound b1) is a dual inhibitor of Dyrk1A (IC50: 177 nM) and α-synuclein aggregation (IC50: 10.5 μM).Formula:C20H21N5O3SColor and Shape:SolidMolecular weight:411.48PF-06263276
CAS:PF-06263276 selectively inhibits pan-JAK with IC50: JAK1 (2.2 nM), JAK2 (23.1 nM), JAK3 (59.9 nM), TYK2 (29.7 nM).Formula:C31H31FN8O2Purity:98%Color and Shape:SolidMolecular weight:566.63Rafutrombopag
CAS:Rafutrombopag is a thrombopoietin (TPO) agonist.Formula:C25H22N4O5Color and Shape:SolidMolecular weight:458.47KY-02327 acetate
KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.Formula:C22H31N3O6Color and Shape:SolidMolecular weight:433.5CHK1-IN-4
CAS:CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.Formula:C18H18BrN7O2Purity:98%Color and Shape:SolidMolecular weight:444.29SP inhibitor 1
SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.Formula:C36H38N2O2Color and Shape:SolidMolecular weight:530.7RK-582
CAS:RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.Formula:C27H35FN6O3Color and Shape:SolidMolecular weight:510.6Dyrk1A/α-synuclein-IN-2
Dyrk1A/α-synuclein-IN-2 (Compound b20) is a dual inhibitor of Dyrk1A and α-synuclein aggregation that acts on α-synuclein (IC50: 7.8 μM).Formula:C21H16N4O4SColor and Shape:SolidMolecular weight:420.44AY-22,252
CAS:AY-22,252 is an inhibitor of beef heart & rat brain nucleoside-3',5'- monophosphate phosphodiesterase.Formula:C27H37NaO7Color and Shape:SolidMolecular weight:496.57Peridinin
CAS:Peridinin is an exceptionally potent and membrane-embedded inhibitor of bilayer lipid peroxidation.Formula:C39H50O7Color and Shape:SolidMolecular weight:630.81DAD dichloride
DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.Formula:C26H42Cl2N6OColor and Shape:SolidMolecular weight:525.56USP7-IN-6
CAS:USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).Formula:C41H43N7O4SPurity:98%Color and Shape:SolidMolecular weight:729.89SG3199
CAS:SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66Mal-PEG4-VA-PBD
CAS:Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connectedFormula:C68H79N9O17Purity:98%Color and Shape:SolidMolecular weight:1294.41LY 178210
CAS:LY 178210 is a 5-hydroxytryptamine receptor agonist.Formula:C18H25N3OColor and Shape:SolidMolecular weight:299.41PDHK-IN-3
PDHK-IN-3 (compound 7) is a potent inhibitor of pyruvate dehydrogenase kinase(PDHK) with IC50s of 0.21 and 1.54 μM for PDHK2 and PDHK4, respectively [1].Formula:C17H16N2O2Color and Shape:SolidMolecular weight:280.32Ledene
CAS:Ledene (Viridiflorene) is an essential oil produced by viridiflorene synthase.Formula:C15H24Purity:98%Color and Shape:SolidMolecular weight:204.35Lasonolide A
CAS:Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.Formula:C41H60O9Color and Shape:SolidMolecular weight:696.91CH-38083
CAS:CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.Formula:C18H24ClNO3Purity:98%Color and Shape:SolidMolecular weight:337.84GSK2578999A
CAS:GSK2578999A is a betulin derivative with antitumor activity.Formula:C46H62ClNO7Purity:98%Color and Shape:SolidMolecular weight:776.44Aeroplysinin 1
CAS:Aeroplysinin I is an antibacterial compound from the sponge. It has cytotoxic activity against colon cancer cells by promoting β-catenin degradation.Formula:C9H9Br2NO3Color and Shape:SolidMolecular weight:338.98Glycyl H-1152 hydrochloride
CAS:Glycyl-H-1152 is a potent ROCK-II inhibitor (IC50=11.8 nM) with high selectivity over CaMKII, PKG, Aurora A, PKA, and PKC. Better than Y-27632 and HA-1077.Formula:C18H26Cl2N4O3SColor and Shape:SolidMolecular weight:449.39EGFR-IN-48
EGFR-IN-48: potent EGFR inhibitor, oral, IC50: 0.193-66.7 nM, blocks EGFR mutants & BaF3/PC-9 cell proliferation.Color and Shape:SolidGlucosylceramide synthase-IN-3
Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.Formula:C21H20FN3O3Color and Shape:SolidMolecular weight:381.4Cilobamine (free base)
CAS:Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.Formula:C17H23Cl2NOColor and Shape:SolidMolecular weight:328.28GSK866
CAS:GSK866 is a selective glucocorticoid receptor agonist (SEGRA).Formula:C23H21Cl2F4N5O3Color and Shape:SolidMolecular weight:562.34Chitinase-IN-5
Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.Formula:C20H21ClFN7Color and Shape:SolidMolecular weight:413.88MEK1/2-IN-2
MEK1/2-IN-2 is a potent, ATP-competitive MEK1/2 inhibitor that exhibits equal inhibitory effects on wild-type MEK1/2 and a group of MEK1/2 mutant cells.Formula:C28H22ClFN6OColor and Shape:SolidMolecular weight:512.97Cryptopleurine
CAS:Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.Formula:C24H27NO3Purity:98%Color and Shape:SolidMolecular weight:377.48
