Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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ZLM-66
ZLM-66: Doravirine analog, HIV-1 NNRTI inhibitor, IC50: 41nM, EC50: HIV-1 13nM, cIAP1 0.32nM; useful in AIDS research.Color and Shape:SolidAAA-10 formic
AAA-10 formic is an orally active inhibitor of intestinal bacterial bile salt hydrolase (BSH) against B.Formula:C26H43FO7SColor and Shape:SolidMolecular weight:518.68O-GlcNAcase-IN-1
O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.Formula:C15H22N6Color and Shape:SolidMolecular weight:286.38Aplaviroc hydrochloride
CAS:Aplaviroc, a potent CCR5 inhibitor, binds selectively, blocking HIV entry and specific monoclonal antibody attachment in vitro.Formula:C33H44ClN3O6Color and Shape:SolidMolecular weight:614.17FTI-2628
CAS:FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.Formula:C31H34N4O3SColor and Shape:SolidMolecular weight:542.69Antibacterial agent 78
Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].Formula:C16H23N3S2Color and Shape:SolidMolecular weight:321.5Camptothecin-20(S)-O-propionate
CAS:CZ-48 is a DNA topoisomerase inhibitor.Formula:C23H20N2O5Color and Shape:SolidMolecular weight:404.42Carbacyclin
CAS:Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.Formula:C21H34O4Purity:98%Color and Shape:SolidMolecular weight:350.49JAK-IN-23
"JAK-IN-23: oral dual JAK/STAT & NF-κB inhibitor; JAK1 (IC50: 8.9 nM), JAK2 (15 nM), JAK3 (46.2 nM); for IBD research."Formula:C23H22Cl2N4OColor and Shape:SolidMolecular weight:441.35BTK-IN-8
BTK-IN-8: potent, selective covalent BTK inhibitor; IC50=0.22 nM, Kd=0.91 nM; effective in blood CD69 cells (IC50=0.029 μM).Formula:C26H36N6O3Color and Shape:SolidMolecular weight:480.6Antitumor agent-37
Antitumor agent-37: strong anti-growth, anti-spread, induces DNA damage, apoptosis via Bcl-2/Bax/caspase3, boosts immune response.Formula:C16H18Cl2N2O4PtColor and Shape:SolidMolecular weight:568.32ONL-1204
CAS:ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Formula:C71H100N18O16Color and Shape:SolidMolecular weight:1461.66Antitubulin agent 1
Antitubulin agents-1 disrupts microtubules, ups α-tubulin acetylation, and has anticancer properties.Formula:C21H19N3O3Color and Shape:SolidMolecular weight:361.39S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurity:98%Color and Shape:SolidMolecular weight:340.23Resolvin E4
CAS:RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45RO5461111
CAS:RO5461111: Oral Cathepsin S inhibitor, IC50 of 0.4 nM (human) & 0.5 nM (mouse), reduces T/B cell activation, treats lung inflammation & lupus nephritis.Formula:C27H24F6N4O4SColor and Shape:SolidMolecular weight:614.56Anti-inflammatory agent 9
Benzimidazothiazole-derived Compound 28 from tilomisole targets COX-2, has potent anti-inflammatory effects & is orally bioavailable.Formula:C18H15N5O2SColor and Shape:SolidMolecular weight:365.41MK-2748
CAS:MK-2748 is an inhibitor of NS3 protease, hepatitis C virus.Formula:C42H56N6O10SColor and Shape:SolidMolecular weight:836.99ART615
ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).Formula:C21H21F3N4O2Color and Shape:SolidMolecular weight:418.41Anticancer agent 54
Anticancer agent 54 blocks cell cycle in G0/G1, induces apoptosis, and fights cancer via DNA embedding and ROS.Formula:C33H36N6Color and Shape:SolidMolecular weight:516.68SX 3202
CAS:SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.Formula:C17H11BrFN3O4Color and Shape:SolidMolecular weight:420.19NVP-CFC218
CAS:NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.Formula:C37H45ClN4O4Color and Shape:SolidMolecular weight:645.23Quinagolide Free Base
CAS:Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.Formula:C20H33N3O3SColor and Shape:SolidMolecular weight:395.56CYP1B1-IN-2
CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].Formula:C20H11F3O2Color and Shape:SolidMolecular weight:340.3BW 443C
CAS:BW 443C is a selective agonist of mu-opioid receptor.Formula:C33H46N10O10Color and Shape:SolidMolecular weight:742.791SSTR5 antagonist 2 hydrochloride
SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.Formula:C32H36ClFN2O5Color and Shape:SolidMolecular weight:583.09Norbinaltorphimine dihydrochloride
CAS:Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.Formula:C40H45Cl2N3O6Purity:98.17% - 99.88%Color and Shape:SolidMolecular weight:734.71Ref: TM-T12241
1mg35.00€5mg80.00€10mg114.00€25mg224.00€50mg388.00€100mg618.00€200mg859.00€1mL*10mM (DMSO)117.00€ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formula:C29H33ClF2N6O9Purity:98%Color and Shape:SolidMolecular weight:683.06O4
CAS:O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.Formula:C24H15NO7Purity:98%Color and Shape:SolidMolecular weight:429.38BDZ-h
CAS:BDZ-h inhibits both closed/open states of all 4 homomeric & 2 GluA2R-complex AMPA receptors.Formula:C21H21N5O3SColor and Shape:SolidMolecular weight:423.49SB 224289
CAS:SB 224289: selective 5-HT1B antagonist, pKi 8.2, 60x selectivity, effective orally.Formula:C32H32N4O3Purity:98%Color and Shape:SolidMolecular weight:520.62Pibrozelesin
CAS:Pibrozelesin, a water-soluble duocarmycin B2 derivative, binds AT-rich DNA, blocking replication and inducing cell death.Formula:C32H36BrN5O8Color and Shape:SolidMolecular weight:698.56KRAS G12C inhibitor 15
CAS:KRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor .Formula:C25H21ClF2N4O3Purity:98%Color and Shape:SolidMolecular weight:498.91Samuraciclib
CAS:Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.Formula:C22H30N6OColor and Shape:SolidMolecular weight:394.51GSK065
CAS:GSK065 is a potent inhibitor of kynurenine-3-monooxygenase (KMO).Formula:C17H15ClN2O4Color and Shape:SolidMolecular weight:346.77Indinavir monohydrate
CAS:Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.Formula:C36H49N5O5Color and Shape:SolidMolecular weight:631.82EGFR/HER2/DHFR-IN-1
Potent EGFR/HER2/DHFR inhibitor for MCF-7 breast cancer; IC50: 0.153/0.108/0.291 μM; arrests G1/S phase, triggers apoptosis.Formula:C14H11BrN4O2SColor and Shape:SolidMolecular weight:379.23GSK2578999A
CAS:GSK2578999A is a betulin derivative with antitumor activity.Formula:C46H62ClNO7Purity:98%Color and Shape:SolidMolecular weight:776.44SR 140333
CAS:SR 140333 is a NK1 receptor antagonist.Formula:C37H45Cl3N2O2Purity:98%Color and Shape:SolidMolecular weight:656.12CB 30900
CAS:CB30900 is a novel and effective thymidylate synthase inhibitor.Formula:C31H32FN5O9Color and Shape:SolidMolecular weight:637.61JAK3-IN-13
JAK3-IN-13: Oral JAK3 inhibitor, selective & potent. Acts on NK1, JNK2, JNK3, Tyk2. Anti-tumor. IC50: JNK3, 8 nM; Tyk2, 365 nM; JNK2, 2039 nM; NK1, 4728 nM.Formula:C25H33ClN6O5Color and Shape:SolidMolecular weight:533.02Luffolide
CAS:Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.Formula:C27H40O6Color and Shape:SolidMolecular weight:460.60Saussureamine C
CAS:Saussureamine C is an inhibitor of H274Y and N294S mutants.Formula:C19H26N2O5Color and Shape:SolidMolecular weight:362.42Napsagatran hydrate
CAS:Napsagatran hydrate is a novel and specific inhibitor of thrombin.Formula:C26H36N6O7SPurity:98%Color and Shape:SolidMolecular weight:576.66ML-SI1
CAS:ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).Formula:C23H26Cl2N2O3Color and Shape:SolidMolecular weight:449.37COX-2-IN-10
COX-2-IN-10 is a potent COX-2 inhibitor, reducing IL-6, TNF-α, IL-1β, PGE2 (IC50=2.54 μM), and iNOS expression.Formula:C31H32FN5O2SColor and Shape:SolidMolecular weight:557.68BMS453
CAS:BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.Formula:C27H24O2Purity:99.93%Color and Shape:SolidMolecular weight:380.48Suzetrigine
CAS:Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.Formula:C21H20F5N3O4Purity:98.08% - 99.27%Color and Shape:SolidMolecular weight:473.39Ref: TM-T69552
1mg58.00€5mg114.00€10mg170.00€25mg266.00€300g129,112.00€50mg457.00€100mg747.00€200mg1,026.00€1mL*10mM (DMSO)118.00€Dazostinag disodium
CAS:Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.Formula:C21H20F2N8Na2O10P2S2Purity:98.84% - 99.96%Color and Shape:SolidMolecular weight:754.48FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Formula:C28H27FN2O3Purity:97.45%Color and Shape:SolidMolecular weight:458.52
