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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • ZL0516

    CAS:
    <p>ZL0516, a chromone-based oral BRD4 BD1 inhibitor, shows potent in vivo efficacy and good pharmacokinetics, suggesting use in treating inflammation.</p>
    Formula:C27H34N2O6
    Color and Shape:Solid
    Molecular weight:482.57
  • Tridihexethyl chloride

    CAS:
    <p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>
    Formula:C21H36ClNO
    Color and Shape:Solid
    Molecular weight:353.97
  • ABD56

    CAS:
    <p>ABD56 inhibits osteoclast formation and activity in vitro and in vivo.</p>
    Formula:C17H18O3
    Color and Shape:Solid
    Molecular weight:270.32
  • CAY10719

    CAS:
    <p>CAY10719 selectively inhibits ABCG2 (IC50 = 0.23 μM), reverses SN 38 resistance, and inhibits ATPase, with low ABCG1 activity.</p>
    Formula:C25H20Cl2N2O2
    Color and Shape:Solid
    Molecular weight:451.34
  • Genistein Diglucuronide

    CAS:
    <p>Genistein Diglucuronide, a Genistein metabolite, specifically inhibits tyrosine kinases and EGF receptor autophosphorylation.</p>
    Formula:C27H26O17
    Color and Shape:Solid
    Molecular weight:622.49
  • VEC6

    CAS:
    <p>VEC6 is a VEZF1–DNA interaction inhibitor that recapitulates RhoB loss in ischaemic retinopathy.</p>
    Formula:C14H20N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.34
  • PPZ2

    CAS:
    <p>PPZ2 is a novel DAG-activated TRPC3/TRPC6/TRPC7 channels activator.</p>
    Formula:C22H29N3O2
    Color and Shape:Solid
    Molecular weight:367.48
  • KFU-127


    <p>KFU-127: broad-spectrum antimicrobial; targets bacterial/fungal biofilms; toxic to eukaryotic cells.</p>
    Formula:C34H43BrN2O3
    Color and Shape:Solid
    Molecular weight:607.62
  • Zoledronate trisodium hydrate

    CAS:
    <p>Zoledronate trisodium is a Bone Resorption Inhibitor and Osteoporosis Therapy Adjunct</p>
    Formula:C25H39N10Na15O37P10
    Color and Shape:Solid
    Molecular weight:1726.2
  • Magnesium Oxaloacetate

    CAS:
    <p>Magnesium Oxaloacetate inhibits murine macrophages, aiding parasite survival in mice and C. elegans longevity under H2O2 stress.</p>
    Formula:C4H2MgO5
    Color and Shape:Solid
    Molecular weight:154.36
  • TachypleginA

    CAS:
    <p>TachypleginA is a parasite motility and invasion inhibitor.</p>
    Formula:C22H21F2NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.4
  • IRAK4-IN-21

    CAS:
    <p>IRAK4-IN-21: Oral IRAK4 inhibitor, IC50: IRAK4 5 nM, TAK1 56 nM; curbs IL-23, aids autoimmune research.</p>
    Formula:C28H28FN7O2
    Color and Shape:Solid
    Molecular weight:513.57
  • AGR-540

    CAS:
    <p>AGR-540, a prodrug of AGR-529, normalizes mouse triglycerides, possibly via adipose A1 receptors.</p>
    Formula:C23H32N6O8
    Color and Shape:Solid
    Molecular weight:520.54
  • Domipizone

    CAS:
    <p>Domipizone is a platelet aggregation inhibitor, cardiotonic and vasodilator.</p>
    Formula:C13H16N2O4
    Color and Shape:Solid
    Molecular weight:264.28
  • Hydrolapachol

    CAS:
    <p>Hydrolapachol is a novel potent and selective inhibitor of schistosoma mansoni dihydroorotate dehydrogenase (smdhodh)</p>
    Formula:C15H16O3
    Color and Shape:Solid
    Molecular weight:244.29
  • Etintidine Free Base

    CAS:
    <p>Etintidine Free Base is a Histamine H2 Antagonist.</p>
    Formula:C12H16N6S
    Color and Shape:Solid
    Molecular weight:276.36
  • AChE/MAO-IN-2


    <p>Potent AChE/MAO-B inhibitor; IC50: AChE 0.0224 μM, MAO-B 0.0412 μM, MAO-A 0.1116 μM. Antioxidant, anti-β-amyloid, for AD research.</p>
    Formula:C23H26N2O3
    Color and Shape:Solid
    Molecular weight:378.46
  • FLA-908

    CAS:
    <p>FLA-908 is a Dopamine D2 receptor antagonist and metabolite of remoxipride.</p>
    Formula:C15H21BrN2O3
    Color and Shape:Solid
    Molecular weight:357.25
  • (+)-Cembrene A

    CAS:
    <p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>
    Formula:C20H32
    Color and Shape:Solid
    Molecular weight:272.47
  • IMB-10

    CAS:
    <p>IMB-10 is an alphaMbeta2 integrin modulator, inhibiting leukocyte migration and recruitment in vitro and in vivo.</p>
    Formula:C19H15NOS2
    Color and Shape:Solid
    Molecular weight:337.46
  • NSC-668036

    CAS:
    <p>NSC-668036 is an inhibitor of Dishevelled (Dvl) protein, a key protein in wnt signaling.</p>
    Formula:C21H36N2O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.52
  • Benfluron Hydrochloride

    CAS:
    <p>Benfluron Hydrochloride is an inhibitor of HIV-1 Rev function which also acts as a cytostatic agent with substantial antiretroviral activity.</p>
    Formula:C21H20ClNO2
    Color and Shape:Solid
    Molecular weight:353.85
  • Procaine merethoxylline

    CAS:
    <p>Procaine merethoxylline is a noted sodium channel blocker with a variety of inhibitory effects.</p>
    Formula:C28H41HgN3O9
    Color and Shape:Solid
    Molecular weight:764.24
  • NK-611 free acid

    CAS:
    <p>NK-611 is a potent semisynthetic etoposide analogue that inhibits topoisomerase II and excels against various cancers in vitro.</p>
    Formula:C31H37NO12
    Color and Shape:Solid
    Molecular weight:615.62
  • Ametantrone Acetate

    CAS:
    <p>Ametantrone Acetate is a topoisomerase II inhibitor of anthrapyrazole family, which can lead to DNA covalent crosslinking.</p>
    Formula:C24H32N4O6
    Color and Shape:Solid
    Molecular weight:472.542
  • Naproxen ethyl ester

    CAS:
    <p>Naproxen ethyl ester, an NSAID similar to ibuprofen, reduces pain, fever, and inflammation. It's a non-selective COX inhibitor.</p>
    Formula:C16H18O3
    Color and Shape:Solid
    Molecular weight:258.31
  • Tinostamustine HCl

    CAS:
    <p>Tinostamustine (EDO-S101) is an alkylating HDACi fusion molecule, enhancing potency and overcoming drug resistance.</p>
    Formula:C19H29Cl3N4O2
    Color and Shape:Solid
    Molecular weight:451.82
  • HDAC6-IN-14


    <p>HDAC6-IN-14, an inhibitor of HDAC6 (HDAC), exhibits high selectivity with an IC50 value of 42 nM, demonstrating over 100-fold selectivity compared to HDAC1,</p>
    Formula:C24H30FN3O4
    Color and Shape:Solid
    Molecular weight:443.51
  • FLM-5011

    CAS:
    <p>FLM-5011 is a a lipoxygenase inhibitor with anti-inflammatory effects.</p>
    Formula:C19H31NO2
    Color and Shape:Solid
    Molecular weight:305.46
  • LY191704

    CAS:
    <p>LY 191704 is a 5α-reductase type 1 inhibitor.</p>
    Formula:C14H16ClNO
    Color and Shape:Solid
    Molecular weight:249.74
  • AVN-211

    CAS:
    <p>AVN-211 (CD-008-0173) is a novel and highly selective 5-HT6 receptor small molecule antagonist for the treatment of Alzheimer's disease.</p>
    Formula:C15H15N3O2S2
    Color and Shape:Solid
    Molecular weight:333.43
  • BAY-846

    CAS:
    <p>BAY-846: allosteric MEK inhibitor, long-lasting, highly bioavailable, low brain entry, effective in K-Ras A549 model.</p>
    Formula:C19H13F4IN4O4S
    Color and Shape:Solid
    Molecular weight:596.29
  • CGS 21595

    CAS:
    <p>CGS 21595 inhibits the formation of 5-hydroxyeicosatetraenoic acid and leukotriene B4; rapidly metabolized to CGS 19213.</p>
    Formula:C21H25NO4
    Color and Shape:Solid
    Molecular weight:355.43
  • Angiogenesis inhibitor BT2

    CAS:
    <p>BT2 inhibits angiogenesis, vascular permeability by targeting ERK, FosB, VCAM-1, and related genes, affecting MEK1 and suppressing retinal markers.</p>
    Formula:C18H18N2O4
    Color and Shape:Solid
    Molecular weight:326.35
  • Leptocarpin acetate

    CAS:
    <p>Leptocarpin acetate is used as a [35S]-methionine uptake inhibitor.</p>
    Formula:C22H28O7
    Color and Shape:Solid
    Molecular weight:404.45
  • NTZ-24

    CAS:
    <p>NTZ-24 is a novel potent STAT3 inhibitor.</p>
    Formula:C10H5Cl2N3O3S
    Color and Shape:Solid
    Molecular weight:318.14
  • BuChE-IN-4

    CAS:
    <p>BuChE-IN-4 is a potent inhibitor of BuChE (IC50: 7.7 nM) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects.</p>
    Formula:C21H21BrFN3O4S
    Color and Shape:Solid
    Molecular weight:510.38
  • Anticancer agent 34

    CAS:
    <p>Anticancer agent 34, a sulfonylurea, inhibits Mycobacterium, E. coli, C. albicans (MIC 0.039-0.156 mg/ml), and A549, PC3 cancers (IC50 8.4, 7.8 μg/ml).</p>
    Formula:C17H14BrN3O3S2
    Color and Shape:Solid
    Molecular weight:452.35
  • FWM-3

    CAS:
    <p>FWM-3 is a potent SARS-CoV-2 NSP13 helicase inhibitor [1].</p>
    Formula:C16H16N6O2S
    Color and Shape:Solid
    Molecular weight:356.4
  • MP-1

    CAS:
    <p>MP-1 inhibits FH, induces FH-dependent cytotoxicity, and targets TRMT1's Zn-finger cysteine.</p>
    Formula:C15H17NO3S
    Color and Shape:Solid
    Molecular weight:291.37
  • FTO-IN-8

    CAS:
    <p>FTO-IN-8 (FTO-43) inhibits N6-methyladenosine demethylase FTO with 5.5 μM IC50; shows anti-cancer properties.</p>
    Formula:C19H23ClN2O2
    Color and Shape:Solid
    Molecular weight:346.85
  • Aminopeptidase N Inhibitor

    CAS:
    <p>AP-N inhibitor: reversible, selective for AP-N/CD13 (IC50=25 μM), non-toxic to U937 cells at 100 μM.</p>
    Formula:C17H10N2O8
    Color and Shape:Solid
    Molecular weight:370.27
  • BRD3731

    CAS:
    <p>BRD3731 selectively inhibits GSK3β with IC50 of 15 nM; it's promising for PTSD, psychiatric issues, diabetes, and neurodegeneration.</p>
    Formula:C24H31N3O
    Color and Shape:Solid
    Molecular weight:377.52
  • α-Amylase/α-Glucosidase-IN-1

    CAS:
    <p>α-Amylase/α-Glucosidase-IN-1 (compound 33) is an effective inhibitor of α-amylase/α-glucosidase with IC 50 s of 2.01, 2.09 μM for α-amylase and α-glucosidase,</p>
    Formula:C11H9N5
    Color and Shape:Solid
    Molecular weight:211.22
  • JAK3-IN-12

    CAS:
    <p>JAK3-IN-12 (compound 15k) is a potent inhibitor of JAK3 (IC50: 9.5 nM) and can be used in the study of rheumatoid arthritis.</p>
    Formula:C19H19N5O4S
    Color and Shape:Solid
    Molecular weight:413.45
  • PDE4-IN-10

    CAS:
    <p>PDE4-IN-10 (7a), potent PDE4B inhibitor, IC50 7.01μM; selective, stable, TNF-α blocking, non-toxic in vitro.</p>
    Formula:C18H13N
    Color and Shape:Solid
    Molecular weight:243.3
  • MTR-105

    CAS:
    <p>MTR-105 is a nitric oxide synthase inhibitor.</p>
    Formula:C7H19N2O4PS
    Color and Shape:Solid
    Molecular weight:258.2728
  • AMXT1501

    CAS:
    <p>AMXT1501 is a polyamine uptake inhibitor, also inhibiting the putrescine transport in epimastigotes (the insect stage of t. cruzi)</p>
    Formula:C32H68N6O2
    Color and Shape:Solid
    Molecular weight:568.92
  • AZD-3355

    CAS:
    <p>AZD-3355, also known as Lesogaberan, is a GABA(B)-receptor agonist reflux inhibitor.</p>
    Formula:C3H7FNO2P
    Color and Shape:Solid
    Molecular weight:139.07
  • KRAS G12C inhibitor 22

    CAS:
    <p>KRAS G12C inhibitor 22 is a KRAS G12C inhibitor.</p>
    Formula:C32H41N7O2
    Color and Shape:Solid
    Molecular weight:555.71