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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • CFM-1

    CAS:
    <p>CFM-1 is an antagonist of the anaphase-promoting complex (APC)-2. It also is a cell cycle and apoptosis regulatory protein (CARP)-1 interaction antagonist.</p>
    Formula:C12H7BrN2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.23
  • SCH-79687

    CAS:
    <p>SCH-79687 is a histamine antagonist selective for the H3 subtype. This H3 antagonist may play a role in allergic rhinitis.</p>
    Formula:C18H16Cl2N4O
    Color and Shape:Solid
    Molecular weight:375.25
  • LY-580276

    CAS:
    <p>LY-580276 is an inhibitor of the type I transforming growth factor beta receptor (TβRI).</p>
    Formula:C18H16FN3
    Color and Shape:Solid
    Molecular weight:293.34
  • CB-64D

    CAS:
    <p>CB-64D is a sigma2R selective agonist which releases calcium in human neuroblastoma cells and produces cell death in tumor cell lines.</p>
    Formula:C22H23NO2
    Color and Shape:Solid
    Molecular weight:333.42
  • IMM-H004

    CAS:
    <p>IMM-H004 is an effective inhibitor of BV2 microglia activation.</p>
    Formula:C16H20N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.34
  • hCAXII-IN-5

    CAS:
    <p>hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI &amp; II &gt;10000, hCAIX 286.1, hCAXII 1.0 nM.</p>
    Formula:C23H22N2O4
    Color and Shape:Solid
    Molecular weight:390.43
  • NAMI-A

    CAS:
    <p>NAMI-A is a ruthenium-based compound with selective activity against tumor metastasis.NAMI-A inhibits cancer cell adhesion and migration.</p>
    Formula:C8H15Cl4N4ORuS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.18
  • JBP485

    CAS:
    <p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>
    Formula:C8H12N2O4
    Color and Shape:Solid
    Molecular weight:200.19
  • Glaucocalyxin B

    CAS:
    Glaucocalyxin B is a diterpenoid isolated from Rabdosia japonica with anticancer and antitumor activity. It decreases the growth of HL-60 cells (IC50: 5.86 μM).
    Formula:C22H30O5
    Purity:99.13% - 99.35%
    Color and Shape:Solid
    Molecular weight:374.47
  • Diazoxon

    CAS:
    <p>Diazoxon is the oxidized form of Diazinon -- an organophosphate insecticide. Diazoxon is shown to be a more potent acetylcholinesterase (AChE) inhibitor.</p>
    Formula:C12H21N2O4P
    Color and Shape:Solid
    Molecular weight:288.28
  • SMER10

    CAS:
    <p>SMER10 promotes mutant protein clearance via autophagy in Huntington's/Parkinson's cell models, without relying on rapamycin.</p>
    Formula:C16H17N3O
    Color and Shape:Solid
    Molecular weight:267.33
  • Paraprost

    CAS:
    <p>Paraprost consists of 1-glutamic acid, alanine, and glycine. It was used in prostate hypertrophy drug therapy.</p>
    Formula:C10H21N3O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:311.291
  • WAG003

    CAS:
    <p>WAG003 is a Tudor domain inhibitor.</p>
    Formula:C24H28I2NO3
    Color and Shape:Solid
    Molecular weight:632.29
  • NCG21

    CAS:
    <p>NCG21, a GPR120 agonist, boosts ERK, Ca²⁺ responses, and GLP-1 in GPR120-expressing cells; raises GLP-1 in mice.</p>
    Formula:C23H24N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.45
  • MARK-IN-4

    CAS:
    <p>MARK-IN-4 inhibits microtubule kinase (MARK) effectively (IC50: 1 nM), a target for Alzheimer's therapy.</p>
    Formula:C21H23N7OS
    Color and Shape:Solid
    Molecular weight:421.52
  • MRS1177

    CAS:
    <p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>
    Formula:C20H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.79
  • BTK-IN-23

    CAS:
    <p>BTK-IN-23: BTK inhibitor, IC50=12.8 nM; also blocks BLX (35.6 nM), BMX (5.7 nM); better selectivity than Ibrutinib.</p>
    Formula:C27H28N6O2
    Color and Shape:Solid
    Molecular weight:468.55
  • J1038

    CAS:
    <p>J1038 is a novel Histone Deacetylase 8 (HDAC8) Inhibitor .</p>
    Formula:C10H10N2O3S
    Color and Shape:Solid
    Molecular weight:238.26
  • KRAS inhibitor-16

    CAS:
    <p>KRAS inhibitor-16 blocks KRAS G12C and p-ERK in cancer cells; potential for pancreatic, colorectal, lung cancer treatment. IC50: 0.457 μM.</p>
    Formula:C20H16Cl2FN3O2S
    Color and Shape:Solid
    Molecular weight:452.33
  • AG-024104

    CAS:
    <p>AG-024104 is a broad spectrum cyclin-dependent kinase inhibitors with potential anticancer activity.</p>
    Formula:C24H28F2N6O4S2
    Color and Shape:Solid
    Molecular weight:566.64
  • Cardionogen 1

    CAS:
    Wnt signaling modulator
    Formula:C13H14N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:274.34
  • Umespirone

    CAS:
    Umespirone is a potential antipsychotic/anxiolytic drug of the azapirone class. It possesses anxiolytic and antipsychotic properties.
    Formula:C28H40N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:512.64
  • Neladenoson dalanate HCl

    CAS:
    <p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>
    Formula:C35H35Cl2N7O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:752.73
  • SB-226552

    CAS:
    <p>SB-226552 is an aryloxypropanolamine selective beta3AR agonist.</p>
    Formula:C25H36NO5P
    Color and Shape:Solid
    Molecular weight:461.53
  • CL-275838

    CAS:
    <p>CL-275838 is a compound of memory-enhancing with potent antidepressant activities.</p>
    Formula:C27H25F3N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.52
  • RO27-3225 TFA

    CAS:
    <p>RO27-3225, a MC4R agonist (EC50=1nM), may treat obesity and brain damage, also acts on MC1R, and helps in hemorrhagic shock.</p>
    Formula:C41H53F3N12O8
    Color and Shape:Solid
    Molecular weight:898.9462
  • Shz 1

    CAS:
    <p>Shz 1 is a cardiogenic agent that induces phenotypic differentiation and various cardiac-specific genes including sarcomeric tropomyosin.</p>
    Formula:C13H11BrN2O3S
    Purity:99.57% - 99.91%
    Color and Shape:Solid
    Molecular weight:355.21
  • Palmoxirate sodium hydrate

    CAS:
    <p>Palmoxirate sodium hydrate is a potent inhibitor of long-chain fatty acid oxidation.</p>
    Formula:C17H35NaO5
    Color and Shape:Solid
    Molecular weight:342.45
  • CO-101244 Free Base

    CAS:
    <p>CO-101244 Free Base is an NMDA receptor NR2B subunit blocker.</p>
    Formula:C21H27NO3
    Color and Shape:Solid
    Molecular weight:341.44
  • CB1R Allosteric modulator 3

    CAS:
    <p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>
    Formula:C22H17ClN2O2
    Purity:98.18%
    Color and Shape:Solid
    Molecular weight:376.84
  • Amphenidone

    CAS:
    <p>Amphenidone is a Tranquilizer.</p>
    Formula:C11H10N2O
    Color and Shape:Solid
    Molecular weight:186.21
  • LYC-31138

    CAS:
    <p>LYC-31138 is a modulator of F1F0-ATPase that acts by significantly decreasing M2 glutamate and increasing M4 glutamate.</p>
    Formula:C22H21F4N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.43
  • ZC0101

    CAS:
    <p>ZC0101: potent oral IDO1/TrxR inhibitor. IC50: 0.084/7.98 μM. Induces apoptosis, ROS in cancer cells.</p>
    Formula:C17H15N3O2
    Color and Shape:Solid
    Molecular weight:293.32
  • NSC66098

    CAS:
    <p>NSC66098 is a novel potent inhibitor of Huntington's disease (HD) pathogenesis via targeting CAG repeats RNA and Poly Q protein.</p>
    Formula:C15H11FN2S
    Color and Shape:Solid
    Molecular weight:270.32
  • ET-JQ1-OH

    CAS:
    <p>ET-JQ1-OH is an allele-specific BET inhibitor.</p>
    Formula:C21H21ClN4O2S
    Color and Shape:Solid
    Molecular weight:428.93
  • NF-κB-IN-3

    CAS:
    <p>NF-κB-IN-3 (Compound 2) is an NF-κB inhibitor (IC50: 0.70 μM) and can be used as an anti-tumour agent.</p>
    Formula:C24H18ClF3N2O2
    Color and Shape:Solid
    Molecular weight:458.86
  • TH-162

    CAS:
    <p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>
    Formula:C19H23N5O4
    Color and Shape:Solid
    Molecular weight:385.42
  • Mocravimod

    CAS:
    <p>Mocravimod: S1P1 receptor agonist, reduces atherosclerosis in mice. KRP-203 mitigates rat heart disease, extends graft survival.</p>
    Formula:C24H26ClNO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.99
  • NNC45-0781

    CAS:
    NNC45-0781 is a tissue-selective partial-agonist of estrogen.
    Formula:C27H29NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.52
  • DC-S100

    CAS:
    <p>DC-S100 is a selective histone methyltransferase SET7 inhibitor.</p>
    Formula:C15H14N2O5
    Color and Shape:Solid
    Molecular weight:302.28
  • ADL-5859 HCl

    CAS:
    <p>ADL-5859 is a delta-opioid receptor agonist.</p>
    Formula:C24H28N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49
  • AChE-IN-12

    CAS:
    <p>AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.</p>
    Formula:C33H41NO7
    Color and Shape:Solid
    Molecular weight:563.68
  • 5-OxoETE methyl ester

    CAS:
    <p>5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.</p>
    Formula:C21H32O3
    Color and Shape:Solid
    Molecular weight:332.48
  • BPH-1358

    CAS:
    <p>BPH-1358 (NSC-50460) inhibits FPPS and UPPS (IC50: 1.8 μM, 110 nM), active against S. aureus (MIC ~250 ng/mL).</p>
    Formula:C32H30Cl2N6O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:601.53
  • photoCORM-2

    CAS:
    <p>photoCORM-2 releases CO, changes color for real-time monitoring, has good cellular uptake, and anti-tumor properties.</p>
    Formula:C17H13NO3
    Color and Shape:Solid
    Molecular weight:279.29
  • p-Valerylphenol

    CAS:
    p-Valerylphenol (NSC-49186) can be used to synthesize acylphenoxyacetic acid compounds.
    Formula:C11H14O2
    Purity:99.87%
    Color and Shape:White To Light Beige Powder
    Molecular weight:178.23
  • Scaff10-8

    CAS:
    Scaff10-8 blocks AKAP-Lbc-RhoA, aiding aquaporin-2 movement in kidney cells.
    Formula:C22H18O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.37
  • FPL-55712

    CAS:
    <p>FPL-55712 is a CysLT1 leukotriene receptor antagonist.</p>
    Formula:C27H29NaO9
    Color and Shape:Solid
    Molecular weight:520.5
  • LY 56110

    CAS:
    <p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>
    Formula:C17H12Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.2
  • UCSF648

    CAS:
    <p>UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].</p>
    Formula:C15H19ClN2O2S
    Color and Shape:Solid
    Molecular weight:326.84