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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • 3'-Chloromethotrexate

    CAS:
    <p>'3'-Chloromethotrexate: cancer/autoimmune treatment, pregnancy termination, chemo, immunosuppressant.</p>
    Formula:C20H21ClN8O5
    Color and Shape:Solid
    Molecular weight:488.88
  • EGFR-IN-88

    CAS:
    <p>EGFR-IN-88 (Compound 4i), an EGFR inhibitor with an IC50 of 87 nM, exhibits cytotoxic effects on A549 cells at an IC50 of 3.902 μM and can induce cell apoptosis</p>
    Formula:C22H18Cl2N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.37
  • CAY10773

    CAS:
    <p>CAY10773, a sorafenib derivative, inhibits cancer cells over non-cancerous ones and induces apoptosis or ferroptosis in T24 cells.</p>
    Formula:C22H17Cl2N5O
    Color and Shape:Solid
    Molecular weight:438.31
  • ALR2-IN-3


    <p>ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.</p>
    Formula:C17H12N2O3S2
    Color and Shape:Solid
    Molecular weight:356.42
  • DHMEQ racemate

    CAS:
    <p>DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ.</p>
    Formula:C13H11NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:261.23
  • CGP 7930

    CAS:
    <p>Positive allosteric modulator of GABAB receptors</p>
    Formula:C19H32O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.46
  • Nucleoside-Analog-1

    CAS:
    Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.
    Formula:C9H9N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.2
  • CAY10762

    CAS:
    <p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>
    Formula:C15H13NOS
    Color and Shape:Solid
    Molecular weight:255.33
  • Homidium Cl

    CAS:
    <p>Homidium Chloride, a trypanosomicide and DNA intercalator, is toxic and blocks nicotinic acetylcholine receptors.</p>
    Formula:C21H20ClN3
    Color and Shape:Solid
    Molecular weight:349.862
  • HS79

    CAS:
    <p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>
    Formula:C19H22N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.47
  • EP2 receptor antagonist-1

    CAS:
    <p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>
    Formula:C24H22N4O5
    Color and Shape:Solid
    Molecular weight:446.46
  • Olanexidine Hydrochloride semihydrate

    CAS:
    <p>Olanexidine is a monobiguanide compound with the activity of bactericidal.</p>
    Formula:C17H31Cl4N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.27
  • NB-598 hydrochloride

    CAS:
    <p>NB-598 hydrochloride is a competitive squalene epoxidase (SE) inhibitor.</p>
    Formula:C27H32ClNOS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.13
  • Laidlomycin butyrate

    CAS:
    <p>Laidlomycin butyrate is a ionophore with enhanced intraruminal activity.</p>
    Formula:C41H68O13
    Color and Shape:Solid
    Molecular weight:768.97
  • SMM-189

    CAS:
    <p>SMM-189 is a potent and selective CB2 inverse agonist.</p>
    Formula:C19H12Cl2O3
    Color and Shape:Solid
    Molecular weight:359.2
  • simufilamum

    CAS:
    <p>Simufilam (PTI-125): Low-toxicity, oral drug activating FLNA, correcting its structure, aiding Alzheimer's research.</p>
    Formula:C15H21N3O
    Color and Shape:Solid
    Molecular weight:259.35
  • Sermetacin

    CAS:
    <p>Sermetacin is an anti-inflammatory agent.</p>
    Formula:C22H21ClN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.86
  • SKLB0565

    CAS:
    <p>SKLB0565 inhibits tubulin and colorectal cancer growth (IC50: 0.012-0.081 μM), causes G2/M arrest, triggers apoptosis, and prevents HUVEC migration.</p>
    Formula:C20H25ClN6O
    Color and Shape:Solid
    Molecular weight:400.91
  • DMP 696

    CAS:
    <p>DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.</p>
    Formula:C18H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.3
  • Pelanserin Free Base

    CAS:
    <p>Pelanserin Free Base is an antagonist of the 5-HT2 and α1-adrenergic receptors.</p>
    Formula:C21H24N4O2
    Color and Shape:Solid
    Molecular weight:364.44
  • VRX 03011 Potassium salt

    CAS:
    <p>VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.</p>
    Formula:C19H27KN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.6
  • CJ-17493 (free base)

    CAS:
    <p>CJ-17493 (free base) is a Neurokinin-1 Receptor Antagonist.</p>
    Formula:C24H29F3N2O2
    Color and Shape:Solid
    Molecular weight:434.49
  • Etamiphylline Camsylate

    CAS:
    <p>Etamiphylline Camsylate is used for the treatment of chronic obstructive pulmonary disease (COPD).</p>
    Formula:C23H37N5O6S
    Color and Shape:Solid
    Molecular weight:511.64
  • Aspirin Aluminum

    CAS:
    <p>Aspirin Aluminum is an intermolecular compound that can inhibit gastrointestinal mucosal disorders induced by NSAIDs.</p>
    Formula:C18H15AlO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.29
  • Deramciclane

    CAS:
    Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.
    Formula:C20H31NO
    Color and Shape:Solid
    Molecular weight:301.47
  • COX-2-IN-20

    CAS:
    <p>COX-2-IN-20 (Compound 5d) is a selective and orally active inhibitor of COX-2 (IC 50 = 17.9 nM) with anti-inflammatory activity [1].</p>
    Formula:C11H9ClFN3O2
    Color and Shape:Solid
    Molecular weight:269.66
  • IM-54

    CAS:
    <p>IM-54 is a cell-permeable, effective, and selective necrosis inhibitor.</p>
    Formula:C19H23N3O2
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:325.4
  • Temechine hydrobromide

    CAS:
    <p>Temechine hydrobromide is used for the identification of new diterpenoidal alkaloid leads as tyrosinase inhibitors.</p>
    Formula:C11H22BrN
    Color and Shape:Solid
    Molecular weight:248.21
  • (S)-GFB-12811

    CAS:
    <p>(S)-GFB-12811, a CDK5 inhibitor with IC50&lt;10 nM, aids research in cell cycle, neuronal growth, and cancer.</p>
    Formula:C22H23F4N5O
    Color and Shape:Solid
    Molecular weight:449.44
  • SH-053-S-CH3-2'F

    CAS:
    <p>SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.</p>
    Formula:C23H18FN3O2
    Color and Shape:Solid
    Molecular weight:387.41
  • CAY10760

    CAS:
    <p>CAY10760 inhibits RAD51-BRCA2 interaction (EC50=19 μM), reduces homologous recombination by 54%, and hinders BxPC-3/Capan-1 cancer cell proliferation.</p>
    Formula:C28H24ClN3O3
    Color and Shape:Solid
    Molecular weight:485.96
  • AC-155

    CAS:
    <p>AC-155 is a bamifylline metabolite in human plasma that may induce apoptosis selectively in cancer cells.</p>
    Formula:C16H19N5O2
    Color and Shape:Solid
    Molecular weight:313.35
  • Tunicamine

    CAS:
    Tunicamine is a reversible polyprenol-phosphate inhibitor.
    Formula:C11H21NO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:311.29
  • CAM 4750

    CAS:
    <p>CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist.</p>
    Formula:C30H31ClN4O4
    Color and Shape:Solid
    Molecular weight:547.05
  • HI5

    CAS:
    <p>HI5: potent tubulin/IDO inhibitor, IC50 70 nM (HeLa), blocks kynurenine, G2/M arrest, spurs T cell activity, &amp; triggers apoptosis.</p>
    Formula:C42H43N5O8
    Color and Shape:Solid
    Molecular weight:745.82
  • Z-VAE(OMe)-fmk

    CAS:
    <p>Z-VAE(OMe)-fmk: an irreversible, cell-permeable UCHL1 inhibitor, binds ubiquitin's C-terminal site.</p>
    Formula:C23H32FN3O7
    Color and Shape:Solid
    Molecular weight:481.51
  • EZH2-IN-11

    CAS:
    <p>EZH2-IN-11, a potent E2HZ inhibitor with potential for cancer treatment, is highlighted in patent WO2019204490A1.</p>
    Formula:C28H36ClN3O5S
    Color and Shape:Solid
    Molecular weight:562.12
  • Mabuterol, (S)-

    CAS:
    Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.
    Formula:C13H18ClF3N2O
    Color and Shape:Solid
    Molecular weight:310.74
  • BPH-1358

    CAS:
    <p>BPH-1358 (NSC-50460) inhibits FPPS and UPPS (IC50: 1.8 μM, 110 nM), active against S. aureus (MIC ~250 ng/mL).</p>
    Formula:C32H30Cl2N6O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:601.53
  • YM550

    CAS:
    <p>YM550 is an antagonist.</p>
    Formula:C21H19F6N5O
    Color and Shape:Solid
    Molecular weight:471.4
  • DRL-17822

    CAS:
    <p>DRL-17822 is a Cholesteryl Ester Transfer Protein (CETP) inhibitor.</p>
    Formula:C30H31F6N7
    Color and Shape:Solid
    Molecular weight:603.6
  • Plantainoside C

    CAS:
    <p>Plantainoside C is a useful organic compound for research related to life sciences. The catalog number is T125990 and the CAS number is 136083-86-8.</p>
    Formula:C30H38O15
    Color and Shape:Solid
    Molecular weight:638.619
  • KAI-407

    CAS:
    <p>KAI407, a non-8-aminoquinoline, kills early Plasmodium cynomolgi liver parasites with IC50 of 0.69μM for hypnozoites; similar to primaquine efficacy.</p>
    Formula:C22H14F3N5O
    Color and Shape:Solid
    Molecular weight:421.37
  • ADL-5859 HCl

    CAS:
    <p>ADL-5859 is a delta-opioid receptor agonist.</p>
    Formula:C24H28N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49
  • Antimicrobial agent-3

    CAS:
    <p>Antimicrobial agent-3 (Compound U10) is an antimicrobial agent that is used against bacterial, fungal, and tubercular infections [1].</p>
    Formula:C14H11N3OS
    Color and Shape:Solid
    Molecular weight:269.32
  • LT175

    CAS:
    <p>LT175 is a dual PPARα/γ partial agonist, insulin sensitizer, orally active, with lower adipogeny (EC50: hPPARα 0.22μm, mPPARα 0.26μm, hPPARγ 0.48μm).</p>
    Formula:C21H18O3
    Color and Shape:Solid
    Molecular weight:318.37
  • Cycloguanil nitrate

    CAS:
    <p>Cycloguanil nitrate is a dihydrofolate reductase inhibitor and is a metabolite of the antimalarial drug proguanil.</p>
    Formula:C11H15ClN6O3
    Color and Shape:Solid
    Molecular weight:314.73
  • TP-008

    CAS:
    TGFβRI-IN-2 is a selective, potent and orally active inhibitor of (Activin-Like Kinase 5) ALK 5(pIC50 and pEC50 values of 7.6 and 6.63, respectively).
    Formula:C20H15ClFN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.82
  • LP10

    CAS:
    <p>LP10 is a reverse type I inhibitor of Mycobacterium tuberculosis CYP125A1 and a Potent type II inhibitor of Trypanosoma cruzi CYP51.</p>
    Formula:C24H28N4O2
    Color and Shape:Solid
    Molecular weight:404.5
  • JNJ-56022486

    CAS:
    <p>JNJ-56022486 is a selective TARP γ‑8 AMPA receptor modulator.</p>
    Formula:C15H10ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.71