Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:98%Color and Shape:SolidMolecular weight:250.12Rivanicline
CAS:Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.Formula:C10H14N2Purity:98%Color and Shape:SolidMolecular weight:162.23Peliglitazar racemate
CAS:Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesityFormula:C30H30N2O7Purity:97.75%Color and Shape:SolidMolecular weight:530.57Ethacrynate Sodium
CAS:Ethacrynate Sodium, a sodium salt, blocks chloride, potassium, and sodium transport mainly in Henle's loop.Formula:C13H12Cl2NaO4Purity:98%Color and Shape:SolidMolecular weight:326.12EL-102
CAS:EL-102 is a HIF1α inhibitor with anticancer activity that inhibits microtubule protein polymerization and can be used to study prostate cancer.Formula:C19H16N2O3S2Purity:99.34%Color and Shape:SolidMolecular weight:384.47SARS-CoV-2-IN-41
CAS:SARS-CoV-2-IN-41 (compound 2) is a potent inhibitor of SARS-CoV-2 3CL protease, exhibiting an IC50 of 0.022 µM and demonstrating antiviral efficacy [1].Formula:C22H30F3N5O4S2Purity:98%Color and Shape:SolidMolecular weight:549.63Octaaminocryptand 1
CAS:Octaaminocryptand 1 is an aminocryptand ligand.Formula:C36H54N8Purity:98%Color and Shape:SolidMolecular weight:598.87TWIK-1/TREK-1-IN-1
CAS:Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers andFormula:C21H24F3NO3Purity:98%Color and Shape:SolidMolecular weight:395.42IMM-02
CAS:IMM-02 is a DID-DAD binding inhibitor.Formula:C13H17F2N3OSPurity:98%Color and Shape:SolidMolecular weight:301.36c-Fms-IN-1
CAS:c-Fms-IN-1 is an inhibitor of c-FMS kinase (IC50 = 0.8 nM).Formula:C22H27N5O2Purity:99.94%Color and Shape:SolidMolecular weight:393.4820(S)-Hydroxycholesterol
CAS:20(S)-Hydroxycholesterol (20α-Hydroxycholesterol) is an allosteric activator of the oncoprotein smoothened (Smo).Formula:C27H46O2Purity:99.25% - 99.79%Color and Shape:SolidMolecular weight:402.652,6-Dichlorodiphenylamine
CAS:2,6-Dichlorodiphenylamine shows activity against Candida albicans infections. 2,6-Dichlorodiphenylamine elevated the MIC by 4-fold of diclofenac sodium (DFNa).Formula:C12H9Cl2NPurity:99.81%Color and Shape:Off White To Cream Coloured Crystalline SolidMolecular weight:238.113HOI-BA-01
CAS:3HOI-BA-01 is a mammalian targeting effective rapamycin activation inhibitor.Formula:C19H15NO5Purity:98%Color and Shape:SolidMolecular weight:337.33L748337
CAS:L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formula:C26H31N3O5SPurity:99.67% - >99.99%Color and Shape:SolidMolecular weight:497.61BPN-15606
CAS:BPN-15606, an oral γ-secretase modulator, reduces Aβ42/Aβ40 with IC50 of 7/17 nM; promising PK/PD, lowers Aβ in rodent CNS.Formula:C23H23FN6OColor and Shape:SolidMolecular weight:418.47BDM14471
CAS:BDM14471 is a selective inhibitor of hydroxamate PfAM1.Formula:C17H15FN2O3Purity:98%Color and Shape:SolidMolecular weight:314.31Ro 24-6392
CAS:Ro 24-6392, an ester co-drug of ciprofloxacin and desacetylcefotaxime, combats various aerobic bacteria.Formula:C31H31FN8O8S2Purity:98%Color and Shape:SolidMolecular weight:726.76Liothyronine HCl
CAS:Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.Formula:C15H13ClI3NO4Purity:98%Color and Shape:SolidMolecular weight:687.43Ketocaine
CAS:Ketocaine（Rec 7-0518） is a local anesthetic commonly used in animal experiments with potential antitumor activity for pain relief.Formula:C18H29NO2Purity:98.59%Color and Shape:SolidMolecular weight:291.43GNF-2-PEG-acid
GNF-2-PEG-acid is usually used as a fluorescent probe.Formula:C26H27F3N4O7Purity:98%Color and Shape:SolidMolecular weight:564.51BLM-IN-1
CAS:BLM-IN-1: BLM inhibitor, KD 1.81 μM, IC50 0.95 μM; causes DNA damage, apoptosis, stops cancer cell growth.Formula:C28H35FN4OColor and Shape:SolidMolecular weight:462.6L-Acosamine nucleoside
CAS:L-Acosamine nucleoside has antiviral activity against HIV and HSV-1.Formula:C21H21N3O7Purity:98%Color and Shape:SolidMolecular weight:427.41CB-7921220
CAS:<p>CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.</p>Formula:C14H12N2O2Purity:99.59%Color and Shape:SolidMolecular weight:240.26Valategrast hydrochloride
CAS:Valategrast hydrochloride (R411), a dual antagonist of integrin α4β1 (VLA-4), is used for the potential treatment of asthma.Formula:C30H33Cl4N3O4Purity:98%Color and Shape:SolidMolecular weight:641.41JNJ28871063 hydrochloride
CAS:ErbB receptor family inhibitorFormula:C24H28Cl2N6O3Purity:98%Color and Shape:SolidMolecular weight:519.42Deoxypheganomycin D
CAS:Deoxypheganomycin D is a specific mycobacteria inhibitor.Formula:C30H47N9O11Purity:98%Color and Shape:SolidMolecular weight:709.75GSK9027
CAS:GSK9027, a nonsteroidal GR agonist, is a partial 2×GRE reporter gene activator, less potent than dexamethasone.Formula:C27H19F4N3O2SPurity:99.31%Color and Shape:SolidMolecular weight:525.52CRT-0105446
CAS:CRT-0105446 is an effective LIMK inhibitor that acts by suppressing cofilin phosphorylation and increasing αTubulin acetylation in cells.Formula:C20H18F3N3O2SPurity:98%Color and Shape:SolidMolecular weight:421.44ALK-IN-5
CAS:ALK-IN-5 is a potent, selective, and brain-penetrant inhibitor of anaplastic lymphoma kinase (ALK, IC50: 2.9 nM).Formula:C24H25FN6O3Purity:98%Color and Shape:SolidMolecular weight:464.49BMT-145027
CAS:BMT-145027 is a positive allosteric modulator of mGluR5 without inherent agonist activity (EC50 = 47 nM).Formula:C23H14ClF3N4Purity:99.62%Color and Shape:SolidMolecular weight:438.83Tedisamil
CAS:Tedisamil blocks cardiac K+ currents, slows heart rate, is a class III antiarrhythmic, and treats angina.Formula:C19H32N2Purity:98%Color and Shape:SolidMolecular weight:288.47Lanicemine
CAS:Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).Formula:C13H14N2Purity:98%Color and Shape:SolidMolecular weight:198.26p18SMI-41
CAS:p18SMI-41 is a novel INK4C inhibitor. It also specifically blocking the bioactivity of p18 protein.Formula:C19H16N2O4Purity:98%Color and Shape:SolidMolecular weight:336.34AMG-548
CAS:AMG-548, oral p38α inhibitor (Ki=0.5 nM), >1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.Formula:C29H27N5OPurity:99.91%Color and Shape:SolidMolecular weight:461.56Utibapril
CAS:Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.Formula:C22H31N3O5SPurity:98%Color and Shape:SolidMolecular weight:449.56ML388
CAS:ML388 is an inhibitor of human NAD(+)- dependent 15- hydroxyprostaglandin dehydrogenase.Formula:C20H24N4Purity:98%Color and Shape:SolidMolecular weight:320.43ND-322 HCl
CAS:ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.Formula:C15H16ClNO3S2Purity:99.49%Color and Shape:SolidMolecular weight:357.88GV-196771A
CAS:<p>GV-196771A A novel NMDA receptor glycine site antagonist with potent antinociceptive activity.</p>Formula:C20H13Cl2N2NaO3Purity:96.43%Color and Shape:SolidMolecular weight:423.23Iferanserin
CAS:Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Formula:C23H28N2OColor and Shape:SolidMolecular weight:348.48AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purity:98%Color and Shape:SolidMolecular weight:504.53HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Formula:C22H25ClO7Purity:98%Color and Shape:SolidMolecular weight:436.88AV-1101
CAS:AV-1101, a cytokine production inhibitor, is used potentially for the treatment of HIV infection.Formula:C19H20N2O4Purity:98%Color and Shape:SolidMolecular weight:340.37M8891
CAS:M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.Formula:C20H17F2N3O3Color and Shape:SolidMolecular weight:385.36GPR40 Activator 2
CAS:GPR40 Activator 2 is a highly effective activator of the GPR40 receptor.Formula:C28H29NO6S2Purity:98%Color and Shape:SolidMolecular weight:539.66HexylHIBO
CAS:HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.Formula:C12H20N2O4Purity:99.55%Color and Shape:SolidMolecular weight:256.3(RS)-3,4-DCPG
CAS:antagonist of AMPA receptors and agonist of mGluR8Formula:C10H9NO6Purity:98%Color and Shape:SolidMolecular weight:239.18Butoprozine HCl
CAS:Butoprozine HCl is a cardiac depressant agent.Formula:C28H39ClN2O2Purity:98%Color and Shape:SolidMolecular weight:471.07IT1t
CAS:IT1t inhibits CXCL12/CXCR4 interaction with an IC50 of 2.1 nM. is a potent CXCR4 antagonist.Formula:C21H34N4S2Purity:98%Color and Shape:SolidMolecular weight:406.65CRS400393
CAS:CRS400393: Anti-tuberculosis drug, MIC - M. abs.: 0.03μg/mL, M. avium: 2μg/mL, M. intracellulare: ≤0.12 μg/mL, M. tuberculosis: ≤0.12 μg/mL.Formula:C18H20Cl2N2OSPurity:98%Color and Shape:SolidMolecular weight:383.34KF 13218
CAS:KF 13218 is a selective, potent and long lasting thromboxane B2 (TXB2) synthase inhibitor with an IC50 value of 5.3±1.3 nM.Formula:C20H20N2O3Purity:98%Color and Shape:SolidMolecular weight:336.38
