Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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Cadein1
Cadein1, an isoquinolinium derivative, induces G2/M phase delay and caspase-dependent apoptosis in cancer cells lacking functional p53.Formula:C33H48F2INO2Color and Shape:SolidMolecular weight:655.64COX-2-IN-11
CAS:<p>COX-2-IN-11 (compound 7b2) is a potent and selective COX-2 inhibitor. COX-2-IN-11 has the potential in inflammation disease research[1].</p>Formula:C12H12OS3Color and Shape:SolidMolecular weight:268.42Ici D8731
CAS:Ici D8731 is a nonpeptide angiotensin II antagonist with potential as a treatment for hypertension and heart failure.Formula:C25H21N5OColor and Shape:SolidMolecular weight:407.47SPR519
CAS:SPR519 is a potent PI3Kα/mTOR inhibitor; IC50: 30 nM (PI3Kα), 10 nM (mTOR); EC50: 0.23-0.50 μM in cancer cells A2780, PC3, SKOV3.Formula:C19H21N7O3SColor and Shape:SolidMolecular weight:427.48MNK1/2-IN-5
CAS:MNK1/2-IN-5 is a potent and selective MNK1/2 inhibitor with anticancer activity and can be used to study solid tumors and hematological malignancies.Formula:C17H16N4O2Purity:98.04%Color and Shape:SolidMolecular weight:308.33AFN941
CAS:AFN941 is a staurosporine analog, acting as a Jak3-specific inhibitor.Formula:C28H30N4O3Color and Shape:SolidMolecular weight:470.56EGFR-IN-542
CAS:EGFR-IN-542 is a novel EGFR inhibitor reducing cardiac inflammation, fibrosis, and dysfunction, promising for obesity complications.Formula:C23H18FN5Color and Shape:SolidMolecular weight:383.42Lonaprisan
CAS:Lonaprisan: an oral steroid derivative with potent, selective anti-progestogenic effects, unaffected by PKA activators, active on PR-A/B.Formula:C28H29F5O3Color and Shape:SolidMolecular weight:508.52ZLY032
CAS:ZLY032 is a FFAR1 and PPARδ agonist (EC50: 68 nM & 102 nM), selective over PPARα/γ, lowers glucose, cholesterol, and improves NASH in mice.Formula:C22H18F3NO4SColor and Shape:SolidMolecular weight:449.44Risotilide
CAS:Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.Formula:C15H27N3O4S2Purity:98%Color and Shape:SolidMolecular weight:377.52Asulacrine free base
CAS:Asulacrine (CI-921; NSC-343499; SN-21407) is a topoisomerase II inhibitor disrupting DNA replication and RNA, protein synthesis in cancer treatment.Formula:C24H24N4O4SColor and Shape:SolidMolecular weight:464.54Dalmelitinib
CAS:Dalmelitinib: oral c-Met kinase inhibitor, IC50 2.9 nM, disrupts MET, AKT, ERK in cancer cells, for NSCLC research.Formula:C22H16FN7O2SColor and Shape:SolidMolecular weight:461.47NOS-IN-3
CAS:NOS-IN-3: potent, selective iNOS inhibitor; IC50 of 4.6 µM; spares eNOS; low toxicity; potential for septic shock treatment.Formula:C10H15N3OColor and Shape:SolidMolecular weight:193.25Tylogenin
CAS:<p>Tylogenin from Tylophora sylvatica blocks IgE-induced basophil release, outperforming its glycosides and dexamethasone.</p>Formula:C28H38O10Color and Shape:SolidMolecular weight:534.6Arnebinol
CAS:Arnebinol has prostaglandin biosynthesis inhibitory activity.Formula:C16H20O2Color and Shape:SolidMolecular weight:244.33Ph CL 28A
CAS:Ph CL 28A is a 15-hydroxyprostaglandin dehydrogenase inhibitor.Formula:C18H16N2O7Color and Shape:SolidMolecular weight:372.33(R,R)-Reboxetine mesylate
CAS:(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.Formula:C20H27NO6SColor and Shape:SolidMolecular weight:409.5SKOG102
CAS:SKOG102, a potent OLIG2 inhibitor, blocks DNA binding for GBM research.Formula:C19H25Cl2N7Color and Shape:SolidMolecular weight:422.35Chaetoglobosin C
CAS:Chaetoglobosin C (Compound 4), an anthraquinone-chromone derivative of Chaetomium globosum KMITL-N0802, exhibits anti-tuberculosis activity [1].Formula:C32H36N2O5Color and Shape:SolidMolecular weight:528.64Antitubercular agent-36
CAS:<p>Antitubercular agent-36 inhibits Mycobacterium tuberculosis with MIC90 of 1.25 μg/mL, used in TB research.</p>Formula:C18H17N3O3Color and Shape:SolidMolecular weight:323.35Cenisertib benzoate
CAS:Cenisertib benzoate is an orally bioavailable, synthetic, small-molecule multi-Aurora kinase inhibitor with potential antineoplastic activity.Formula:C31H36FN7O3Color and Shape:SolidMolecular weight:573.66Cromoglicate sodium hydrate
CAS:Cromoglicic acid stabilizes mast cells, preventing histamine release, but has been superseded by leukotriene antagonists in asthma treatment.Formula:C23H24Na2O15Color and Shape:SolidMolecular weight:586.41AS-1669058 oxalate
CAS:AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist for the treatment of type 2 diabetes mellitus.Formula:C20H17BrF2N4O5Color and Shape:SolidMolecular weight:511.27Allixin
CAS:Allixin, a garlic compound, weakly fights microbes and skin tumor growth; blocks toxin-induced mutations.Formula:C12H18O4Color and Shape:SolidMolecular weight:226.27TK4b
CAS:TK4b, a JAK inhibitor, targets leukemia/lymphoid diseases, with IC50s: 18.42 nM (JAK3) & 19.40 nM (JAK2).Formula:C21H22N2O2Color and Shape:SolidMolecular weight:334.41Avitriptan Fumarate
CAS:Amitriptan fumarate is serotonin 5HT-1B/1D receptor agonist with anti-migraine activity.Formula:C26H34N6O7SColor and Shape:SolidMolecular weight:574.65KF 17837S
CAS:KF 17837S is an adenosine A(2a) receptor antagonists.Formula:C20H26N4O4Color and Shape:SolidMolecular weight:386.44Tubulin polymerization-IN-27
CAS:Compound 5j inhibits tubulin polymerization, arrests cell cycle at G2/M phase, and induces apoptosis.Formula:C22H20N2O2Color and Shape:SolidMolecular weight:344.418-Acetyl-2-(dipropylamino)tetralin
CAS:8-Acetyl-2-(dipropylamino)tetralin is a 5-HT(1A) receptor agonist; both isomers are active, but the (S)-isomer is the most potent.Formula:C18H27NOColor and Shape:SolidMolecular weight:273.41HPK1-IN-25
CAS:HPK1-IN-25, an HPK1 inhibitor, IC50 129 nM, may aid cancer research.Formula:C23H25N5OColor and Shape:SolidMolecular weight:387.48TDP1 Inhibitor-2
CAS:TDP1 Inhibitor-2 strongly blocks TDP1 (IC50: 99 nM) & treats SCAN1 (IC50: 3.5 μM).Formula:C25H14Cl2O5Color and Shape:SolidMolecular weight:465.28Fostemsavir dihydrate
CAS:Fostemsavir dihydrate is an HIV-1 attachment inhibitor.Formula:C25H30N7O10PColor and Shape:SolidMolecular weight:619.53Pulixin
CAS:Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).Formula:C14H11NO4Color and Shape:SolidMolecular weight:257.24Posenacaftor
CAS:Posenacaftor (PTI-801) regulates CFTR protein for cystic fibrosis research.Formula:C27H27NO5Color and Shape:SolidMolecular weight:445.51Cefaparole
CAS:Cefaparole is an antibacterial compound and cell wall biosynthesis inhibitor.Formula:C19H19N5O5S3Color and Shape:SolidMolecular weight:493.58BAY-27-9955
CAS:BAY-27-9955 is a glucagon receptor antagonist.Formula:C23H31FOColor and Shape:SolidMolecular weight:342.49TC299423
CAS:TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.Formula:C11H15N3Color and Shape:SolidMolecular weight:189.26AZD-2327 sesquifumarate
CAS:AZD-2327 sesquifumarate is a delta opioid receptor agonist.Formula:C70H82F2N8O14Color and Shape:SolidMolecular weight:1297.46Ramentaceone
CAS:Ramentaceone is an antineoplastic.Formula:C11H8O3Purity:98%Color and Shape:SolidMolecular weight:188.18CD73-IN-8
CAS:CD73-IN-8 blocks CD73, hindering adenosine production that supports tumor growth, flagged as compound 57 in WO2022052886A1.Formula:C17H13ClN4O2Color and Shape:SolidMolecular weight:340.76Laccaic acid A
CAS:Laccaic acid A is a direct, DNA-competitive DNA methyltransferase 1 inhibitor.Formula:C26H19NO12Color and Shape:SolidMolecular weight:537.43VUF14480
CAS:VUF14480 is a covalent partial agonist for hH4 receptor, binding to C98(3.36) with high affinity; S98(3.36) mutation inhibits binding.Formula:C17H20N4Color and Shape:SolidMolecular weight:280.37AZD-9684
CAS:AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.Formula:C10H14N2O2SColor and Shape:SolidMolecular weight:226.3Trimetaphan camsilate
CAS:<p>Trimetaphan camsilate, short-acting IV drug, blocks cholinergic transmission at autonomic ganglia, affecting both sympathetic and parasympathetic systems.</p>Formula:C22H25N2OSColor and Shape:SolidMolecular weight:365.51Dynamin IN-1
CAS:Dynamin IN-1 is a potent dynamin inhibitor with an IC 50 value of 1.0 µM .Formula:C23H24N2OColor and Shape:SolidMolecular weight:344.45Tioclomarol
CAS:<p>Tioclomarol is a coumarin anticoagulant and a vitamin K antagonist.</p>Formula:C22H16Cl2O4SColor and Shape:SolidMolecular weight:447.33TCMDC-125457
CAS:TCMDC-125457 aids calcium redistribution and treats artemisinin-resistant parasites with artesunate, not affecting heme crystallization.Formula:C19H18ClN5O3Color and Shape:SolidMolecular weight:399.83RU 27849
CAS:<p>RU 27849 is used to study the binding of tryptamine recognition sites.</p>Formula:C11H12N2Color and Shape:SolidMolecular weight:172.23Thr101
CAS:<p>Thr101, or NOX Inhibitor VII, is a dose-dependent blocker of HDAC1-9 and NOX.</p>Formula:C14H10FNOSColor and Shape:SolidMolecular weight:259.3FR-168888 free base
CAS:FR-168888: novel Na+/H+ exchange inhibitor protecting heart from arrhythmia and cell death under ischemia.Formula:C13H14N4O2Color and Shape:SolidMolecular weight:258.28
