Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,440 products)
- Cytoskeletal Signaling(1,527 products)
- DNA Damage/DNA Repair(2,968 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,874 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,382 products)
- Other Inhibitors(36,042 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,444 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66686 products of "Inhibitors"
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KY-04031
CAS:KY-04031 is an inhibitor of p21-activated kinase 4.Formula:C21H20N8OColor and Shape:SolidMolecular weight:400.44TRK/ALK-IN-1
TRK/ALK-IN-1: Potent dual TRK & ALK inhibitor; IC50s: 2.2nM (TRKA), 9.3nM (ALK WT), 38nM (ALK L1196M); cancer research potential.Formula:C31H35ClF2N8O2SColor and Shape:SolidMolecular weight:657.18CB5660386
CAS:CB5660386 inhibitor of HIV-1 entry.Formula:C23H25ClN2O4SColor and Shape:SolidMolecular weight:460.97σ1 Receptor/μ Opioid receptor modulator 1
CAS:σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).Formula:C24H31FN2O2Color and Shape:SolidMolecular weight:398.51AGG-523
CAS:AGG-523, an aggrecanase inhibitor, may slow cartilage wear after joint injury by reducing ARG-aggrecan in rats.Formula:C28H29FN2O4Color and Shape:SolidMolecular weight:476.54MMT5-14
CAS:MMT5-14: potent SARS-CoV-2 inhibitor, improves antiviral activity (2-7x), boosts prodrug in plasma/lungs (200-300x), raises NTP in lungs (5x).Formula:C39H55N6O8PColor and Shape:SolidMolecular weight:766.86D 15414
CAS:D-15414, a non-marketed, nonsteroidal weak estrogen from 2-phenylindole, metabolizes from zindoxifene, binds ER, and halts ER+ MCF-7 cell growth.Formula:C17H17NO2Color and Shape:SolidMolecular weight:267.32CHMFL-PI4K-127
CAS:CHMFL-PI4K-127 (15g) selectively inhibits PfPI4K (IC50=0.9 nM), potent against Plasmodium 3D7 (EC50=25.1 nM), with oral anti-malaria activity.Formula:C18H15ClN4O3SColor and Shape:SolidMolecular weight:402.85Tridemorph
CAS:Tridemorph: fungicide inhibiting sterol biosynthesis, targets Erysiphe graminis, created by BASF (Calixin), WHO Class II hazard.Formula:C19H39NOColor and Shape:SolidMolecular weight:297.52Moexipril methyl ester
CAS:Moexipril methyl ester is a long-acting, non-sulfhydryl angiotensine-converting enzyme inhibitor.Formula:C26H32N2O7Color and Shape:SolidMolecular weight:484.55Glyoxalase I inhibitor 2
CAS:Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.Formula:C24H23N3O4SColor and Shape:SolidMolecular weight:449.52AZD-8418
CAS:AZD-8418 and AZD8529, mGlu2 receptor modulators, reduce nicotine use and cravings, with varying effects on food intake.Formula:C19H20ClN3O3Color and Shape:SolidMolecular weight:373.83JNJ-38893777
CAS:JNJ-38893777 is a potent and selective transient receptor potential vanilloid 1 (TRPV1) channel antagonist.Formula:C26H26F6N6Color and Shape:SolidMolecular weight:536.52Antitumor agent-57
CAS:Antitumor agent-57 (Compound 3o) is a potent NQO1-directed antitumor compound.Formula:C20H15NO5Color and Shape:SolidMolecular weight:349.34Marasmic acid
CAS:Marasmic acid is a bioactive antifungal.Formula:C15H18O4Color and Shape:SolidMolecular weight:262.3Inupadenant
CAS:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65SR 1903
CAS:SR 1903 modulates RORγ, LXR, PPARγ; shows anti-inflammatory and cholesterol-lowering effects in mice.Formula:C27H27F6N3OColor and Shape:SolidMolecular weight:523.51AG311
CAS:<p>AG311 inhibits complex I; destabilizes HIF-1α; triggers necrosis in cancer cells, mitochondrial depolarization, superoxide, and calcium increase.</p>Formula:C17H15N5SColor and Shape:SolidMolecular weight:321.4NP-04634
CAS:NP-04634 is a calcium antagonist and protective agent against calcium overload and mitochondrial disruption.Formula:C31H38N2O9Color and Shape:SolidMolecular weight:582.64T6603185
CAS:T6603185 is a novel inhibitor of peroxiredoxin (Prx) and thioredoxin (Trx) systems.Formula:C21H30N6O2Color and Shape:SolidMolecular weight:398.5ST638
CAS:ST638 is a potent inhibitor of tyrosine kinase with an IC 50 of 370 nM [1].Formula:C19H18N2O3SColor and Shape:SolidMolecular weight:354.42Lexanopadol
CAS:Lexanopadol (GRT6006): Potent ORL-1 agonist for moderate/severe chronic and neuropathic pain.Formula:C23H25FN2OColor and Shape:SolidMolecular weight:364.46LEQ-506
CAS:LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.Formula:C27H29N5OColor and Shape:SolidMolecular weight:439.55NSC-4231
CAS:NSC-4231 is a novel Rho-Kinase-II Inhibitor with Vasodilatory Activity.Formula:C21H17NO3Color and Shape:SolidMolecular weight:331.36Nafagrel
CAS:Nafagrel is a thromboxane A2 synthetase inhibitor.Formula:C15H16N2O2Color and Shape:SolidMolecular weight:256.3(Rac)-MEM 1003
CAS:MEM-1003, a calcium channel blocker, is used potentially for the treatment of bipolar disorders.Formula:C22H25ClN2O5Color and Shape:SolidMolecular weight:432.9PF-05139962
CAS:PF-05139962: potent mTOR inhibitor, IC50=48nM/6nM, kinase-selective, good ADME, non-genotoxic, CYP-safe, LE=0.35, LipE=6.8.Formula:C21H27N5O4SColor and Shape:SolidMolecular weight:445.54HCV-IN-35
CAS:HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.Formula:C30H36ClN5Color and Shape:SolidMolecular weight:502.09SGC-AAK1-1N
CAS:SGC-AAK1-1N is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) with an IC 50 of 1.8 μM [1].Formula:C20H22N4O3SColor and Shape:SolidMolecular weight:398.48AM0216
CAS:AM0216 is a novel highly potent inhibitor of NF-κB inducing Kinase (NIK).Formula:C19H17N5OSColor and Shape:SolidMolecular weight:363.44ZINC36617540
CAS:ZINC36617540 is a novel Nef Protein Inhibitor with anti-HIV activity.Formula:C21H17N5OColor and Shape:SolidMolecular weight:355.39IDO1/TDO-IN-1
CAS:IDO1/TDO-IN-1 (30) inhibits IDO1 (Ki=0.23μM) & TDO (Ki=0.73μM); induces apoptosis via Bcl-2/Bax.Formula:C21H16O6Color and Shape:SolidMolecular weight:364.35Pyrethrosin
CAS:Pyrethrosin is a germacranolide.Formula:C17H22O5Color and Shape:SolidMolecular weight:306.35KRAS G12C inhibitor 48
KRAS G12C inhibitor 48: potent with IC50 639.91 nM; hampers H358, H23, A549 cell growth with IC50s of 0.796, 6.33, 16.14 µM, respectively.Formula:C36H39ClN8O2Color and Shape:SolidMolecular weight:651.2Pheniprazine
CAS:Pheniprazine, a potent and long-acting monoamine oxidase inhibitor, shows promise for depression research.Formula:C9H14N2Color and Shape:SolidMolecular weight:150.22CSV0C018875 Hydrochloride
CAS:CSV0C018875 Hydrochloride: Novel G9a inhibitor with low toxicity, effective in enzyme/cell assays, outperforms BIX-0129.Formula:C18H18Cl2N2OColor and Shape:SolidMolecular weight:349.255Fenmetozole
CAS:Fenmetozole is an antagonist of the actions of ethanol.Formula:C10H10Cl2N2OColor and Shape:SolidMolecular weight:245.11Cgp 33304
CAS:CGP 33304 blocks leukotriene receptors and inhibits PLA2, averting hypoxia from leukotriene-induced bronchoconstriction.Formula:C23H26BrN5NaO5Color and Shape:SolidMolecular weight:555.385T-5342126
CAS:T-5342126: TLR4 antagonist, lowers LPS-induced NO in cells (IC50=27.8 μM) & cytokines in blood, cuts ethanol intake & Iba1 in mice.Formula:C25H32ClN3O3Color and Shape:SolidMolecular weight:457.99MMP-9-IN-5
CAS:MMP-9-IN-5: MMP-9 and AKT inhibitor (IC50: 4.49 nM and 1.34 nM), induces apoptosis for cancer research.Formula:C27H20IN3O4Color and Shape:SolidMolecular weight:577.37Iso-Fludelone
CAS:Iso-Fludelone: a stable, soluble, potent, 3rd-gen epothilone B inhibiting cell division and inducing apoptosis, with low toxicity.Formula:C27H36F3NO6Color and Shape:SolidMolecular weight:527.57Cynodontin
CAS:Cynodontin is a strong in vitro fungicide against Sclerotinia spp. and Botrytis cinerea, less so for Verticillium dahliae.Formula:C15H10O6Color and Shape:SolidMolecular weight:286.24GLP-1R agonist 1
CAS:GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.Formula:C32H29ClFN3O5Color and Shape:SolidMolecular weight:590.04q-FTAA
CAS:q-FTAA targets Aβ1-42 fibrils (330-630 nM) and ADPBC (300-500 nM), useful in Alzheimer's disease research.Formula:C21H14O6S4Color and Shape:SolidMolecular weight:490.59myomiR-IN-1
CAS:myomiR-IN-1 inhibits myoD translation in C2C12 cells, doesn't affect myoD mRNA, and reduces differentiation markers.Formula:C33H27NO6Purity:98%Color and Shape:SolidMolecular weight:533.57EGFR-IN-557
CAS:EGFR-IN-557 is an EGFR inhibitor, attenuating Ang II-induced Kidney Fibrosis.Formula:C26H20FN5OColor and Shape:SolidMolecular weight:437.47Hexamethonium chloride dihydrate
CAS:Hexamethonium chloride dihydrate: Non-depolarizing NMJ blocker, nAChR antagonist, treats hypertension, inhibits sympathetic activity, muscle relaxant.Formula:C12H34Cl2N2O2Color and Shape:SolidMolecular weight:309.32Anticancer agent 25
CAS:Anticancer agent 25 demonstrates the highest level of cytotoxic effectiveness on PC3 cells, achieving an IC 50 value of 0.19 μM.Formula:C37H45BrN2O3Color and Shape:SolidMolecular weight:645.67Brobactam Sodium Salt
CAS:Brobactam Sodium Salt is a β-lactamase inhibitor.Formula:C8H9BrNNaO3SColor and Shape:SolidMolecular weight:302.12ANO1-IN-3
CAS:ANO1-IN-3 (Compound 3n) can induces apoptosis that is a potent and selective inhibitor of ANO1 with an IC 50 of 1.23 μM [1].Formula:C20H17NO3Color and Shape:SolidMolecular weight:319.35
