Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,782 products)
- Apoptosis(6,263 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,441 products)
- Cytoskeletal Signaling(1,528 products)
- DNA Damage/DNA Repair(2,965 products)
- Endocrinology/Hormones(3,707 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,009 products)
- Immunology and Inflammation(3,875 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,209 products)
- Microbiology/Virology(7,592 products)
- Neuroscience(10,381 products)
- Other Inhibitors(36,040 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,442 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(826 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66683 products of "Inhibitors"
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AChE/BChE-IN-2
CAS:AChE/BChE-IN-2 (Compound 13b) is a potent inhibitor of AChE/BChE with IC50 values of 0.96 ± 0.14 μM and 1.23 ± 0.23 μM for AChE and BChE, respectively.Formula:C23H25N3O5Color and Shape:SolidMolecular weight:423.46HMS-I2
CAS:HMS-I2 is a chemical probe used to form heterochromatin. It works by disrupting heterochromatin mediated transcriptional gene silencing.Formula:C20H19ClFN3OSColor and Shape:SolidMolecular weight:403.9Deanol aceglumate
CAS:Deanol aceglumate, a deanol and N-acetyl-L-glutamic acid mix, aids in protecting the liver, and counters stress-related gastropathy and diabetes.Formula:C11H22N2O6Color and Shape:SolidMolecular weight:278.305Lauroylmethionine
CAS:Lauroylmethionine is a lysine salt of the product formed by the condensation of lauroyl fatty acid chloride with methionine.Formula:C17H33NO3SColor and Shape:SolidMolecular weight:331.51YM-01 Tosylate
CAS:<p>YM-01 Tosylate, a potent antitumor agent, selectively targets cancer cells and overcoming tamoxifen resistance.</p>Formula:C27H27N3O4S3Color and Shape:SolidMolecular weight:553.72V-11-0711
CAS:V-11-0711 is an inhibitor of Chk-α, which may be essential in cancer cell proliferation.Formula:C27H35NO3Purity:98%Color and Shape:SolidMolecular weight:421.57Azidothiorphan
CAS:Azidothiorphan irreversibly binds to neutral endopeptidase 24.11's active site after UV exposure; thiorphan prevents this.Formula:C12H14N4O3SColor and Shape:SolidMolecular weight:294.33hACC2-IN-1
CAS:hACC2-IN-1 is a potent inhibitor of acetyl coenzyme A carboxylase 2 (ACC2) with an IC50 value of 2.5 μM for hACC2. hACC2-IN-1 has potential for obesity studies.Formula:C23H32N2O4SColor and Shape:SolidMolecular weight:432.58Antibacterial agent 106
CAS:Compound 106 is an orally active antibacterial with biofilm-fighting properties, kills 99.7% of MRSA in macrophages.Formula:C20H24N6SColor and Shape:SolidMolecular weight:380.51Carbazomycin B
CAS:Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).Formula:C15H15NO2Color and Shape:SolidMolecular weight:241.294,5,6,7-Tetrabromobenzimidazole
CAS:4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].Formula:C7H2Br4N2Color and Shape:SolidMolecular weight:433.72CXCR4 antagonist 9
CAS:CXCR4 antagonist 9, with IC50s of 15 nM & 1.3 nM against CXCR4 & Ca²⁺ rise by CXCL12 respectively.Formula:C21H27FN6Color and Shape:SolidMolecular weight:382.48Ambenoxan hydrochloride
CAS:Ambenoxan hydrochloride is a centrally acting skeletal muscle relaxant.Formula:C14H22ClNO4Color and Shape:SolidMolecular weight:303.78M1 ligand 1
CAS:Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.Formula:C20H21NO2Color and Shape:SolidMolecular weight:307.39Metopimazine
CAS:Metopimazine is a selective and peripherally restricted dopamine D3 and D2 receptors antagonist.Formula:C22H27N3O3S2Purity:98%Color and Shape:SolidMolecular weight:445.6AS1907417
CAS:AS1907417 is a GPR119 agonist.Formula:C19H27N3O4SColor and Shape:SolidMolecular weight:393.5Dual AChE-MAO B-IN-2
CAS:Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) & MAO B (0.01 μM); promising for Alzheimer's research.Formula:C26H25NO4Color and Shape:SolidMolecular weight:415.48Antibacterial agent 48
CAS:Antibacterial agent 48 is an antimicrobial agent that reduces the MIC of the antimicrobial agent Ceftazidime.Formula:C13H18N5NaO7SColor and Shape:SolidMolecular weight:411.36S 9795
CAS:S 9795 is a methylxanthine derivative and acts as a potent inhibitor of bronchoconstriction in vivo.Formula:C29H36N6O2Color and Shape:SolidMolecular weight:500.64NITD-304
CAS:NITD-304 combats multidrug-resistant tuberculosis (MDR-TB) effectively.Formula:C17H20Cl2N2OColor and Shape:SolidMolecular weight:339.26SB 201823-A
CAS:SB 201823-A is a Ca2+ channel antagonist.Formula:C18H28Cl3NOColor and Shape:SolidMolecular weight:380.78Nivasorexant
CAS:Nivasorexant is a potent antagonist of the orexin receptor.Formula:C23H23N7O2Color and Shape:SolidMolecular weight:429.47ST7710AA1
CAS:ST7710AA1 inhibits PARP-1, effectively targets in vitro, and overcomes Pgp-associated multidrug resistance.Formula:C20H22N4OColor and Shape:SolidMolecular weight:334.41hiCE inhibitor-1
CAS:Sulfonamide-derived hiCE inhibitor-1 selectively targets human intestinal enzyme, Ki 53.3 nM, mitigates Irinotecan-induced diarrhea.Formula:C18H14Cl2N2O4S2Color and Shape:SolidMolecular weight:457.35CAI-1
CAS:CAI-1 is a vibrio cholerae quorum-sensing autoinducer.Formula:C13H26O2Color and Shape:SolidMolecular weight:214.343-Fucosyllactose
CAS:3-Fucosyllactose, a key fucosylated oligosaccharide in human milk, offers prebiotic and immune benefits.Formula:C18H32O15Color and Shape:SolidMolecular weight:488.44Rubilactone
CAS:Rubilactone is a naphthoic acid ester extracted from the roots of Rubia cordifolia L.Formula:C15H10O5Color and Shape:SolidMolecular weight:270.24Neratinib dimethylamine N-oxide
CAS:Neratinib dimethylamine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity.Formula:C30H29ClN6O4Color and Shape:SolidMolecular weight:573.04CAY10416
CAS:CAY10416: dual COX-2/5-LO inhibitor, IC50: COX-2 (50 nM), 5-LO (3 nM); >200x selectivity for COX-2; anti-inflammatory, prostate cancer agent.Formula:C29H29FN2O5SColor and Shape:SolidMolecular weight:536.61AK 275
CAS:AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.Formula:C20H31N3O4Color and Shape:SolidMolecular weight:377.48Inz-4
CAS:Inz-4 is a fungal-selective inhibitor of mitochondrial cytochrome bc1.Formula:C18H14F4N2O2Color and Shape:SolidMolecular weight:366.31Acetylaminofluorene-dG
CAS:Acetylaminofluorene-dG is a carcinogenic adduct which covalently binds DNA bases and promotes mutagenesis near the adduct site.Formula:C25H24N6O5Color and Shape:SolidMolecular weight:488.5Pifexole
CAS:Pifexole, a 1,2,4-oxadiazole derivative, shows muscle-relaxant effects in animals and is 7x more potent than chlorzoxazone in rats.Formula:C13H8ClN3OColor and Shape:SolidMolecular weight:257.68SYNTi
SYNTi, a PDZ inhibitor, disrupts syndecan/syntenin interaction with an IC50 of 400 nM, LE of 0.24, for breast cancer study.Formula:C28H24BrFN2O5Color and Shape:SolidMolecular weight:567.4TbPTR1 inhibitor 1
CAS:TbPTR1 inhibitor 1 effectively targets kinetochore PTR1 with IC50 <0.1 nM, EC50 0.66 μM against Trypanosoma brucei.Formula:C22H21N7OColor and Shape:SolidMolecular weight:399.45DC-034
CAS:DC-034, a strong MYC transcription suppressor in cancer via G4 mechanism, targets MYC more than other G4 genes.Formula:C24H25F3N2O3Color and Shape:SolidMolecular weight:446.46OX2R-IN-1
CAS:OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.Formula:C20H28ClN3O5SColor and Shape:SolidMolecular weight:457.97RDEA-806 free acid
CAS:<p>RDEA-806, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Formula:C24H18BrClN4O3SColor and Shape:SolidMolecular weight:557.85Vin-C01
CAS:Vin-C01, a potent protector of pancreatic β-cells (EC50=0.22μM), aids in type 2 diabetes research by preventing STZ-induced β-cell apoptosis.Formula:C20H24N2OColor and Shape:SolidMolecular weight:308.42MIF-IN-4 hydrochloride
CAS:MIF-IN-4 hydrochloride inhibits MIF, a cytokine; has pIC50 of 5.01-6, affecting macrophage movement.Formula:C26H29ClN6O2Color and Shape:SolidMolecular weight:493.01AJ-3941
CAS:AJ-3941: Selective calcium channel blocker, prevents lipid peroxidation, potential for treating brain vessel disorders.Formula:C35H35FN2O9Color and Shape:SolidMolecular weight:646.67Lubabegron
CAS:Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.Formula:C29H29N3O3SColor and Shape:SolidMolecular weight:499.62IMC-76
CAS:IMC-76 is a BCL2 i-motif-interactive compound that can act by destabilizing or unfolding the i-motif.Formula:C30H45NO3Color and Shape:SolidMolecular weight:467.68XR 1853
CAS:XR 1853 is a low molecular weight modulator of human plasminogen activator inhibitor-1 activity.Formula:C22H23N3O3Color and Shape:SolidMolecular weight:377.444GW0072
CAS:GW0072 is a partial agonist of PPARγ.Formula:C36H44N2O4SColor and Shape:SolidMolecular weight:600.81Plasma kallikrein-IN-3
CAS:Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.Formula:C20H23N5O2Color and Shape:SolidMolecular weight:365.43Zoleprodolol
CAS:Zoleprodolol is a antagonist of adrenoreceptor.Formula:C17H25N3O5Color and Shape:SolidMolecular weight:351.4AG-012986
CAS:AG-012986: a selective CDK inhibitor with in vitro and in vivo antitumor effects; low IC50 in 14/18 cancer cell types; CAS# 486414-35-1.Formula:C22H23F2N5O2SColor and Shape:SolidMolecular weight:459.51MEISi-1
CAS:MEISi-1: Novel inhibitor of MEIS, blocks MEIS-luciferase, boosts murine & human HSC self-renewal ex vivo.Formula:C24H24N2O3Color and Shape:SolidMolecular weight:388.46AChE-IN-6
CAS:AChE-IN-6: inhibits EeAChE (IC50=0.20μM), HuAChE (IC50=37.02nM), and modulates Aβ1-42 aggregation (IC50=~1.86μM). Potential Alzheimer's research.Formula:C29H41N5O2Color and Shape:SolidMolecular weight:491.67
