Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,377 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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(Z)-Pitavastatin calcium
CAS:(Z)-Pitavastatin calcium is the Z-Isomer of Pitavastatin hemicacium. Pitavastatin calcium is a potent of hydroxymethylglutaryl-CoA (HMG-CoA) reductase.Formula:C50H50CaF2N2O8Purity:98%Color and Shape:SolidMolecular weight:885.031R 1485 dihydrochloride
5-HT6 antagonist,selective and high affinityFormula:C18H20FN3O3S·2HClPurity:98%Color and Shape:SolidMolecular weight:450.35Aniline, N-methyl-p-(8-phenoxyoctyloxy)-
CAS:Aniline, N-methyl-p-(8-phenoxyoctyloxy)- is a Drug / Therapeutic Agent.Formula:C21H29NO2Color and Shape:SolidMolecular weight:327.46PF-02413873
CAS:PF-02413873 is a competitive antagonist of nonsteroidal progesterone receptor with a Ki of 2.6 nM.Formula:C18H21N3O3SPurity:99.83% - 99.89%Color and Shape:SolidMolecular weight:359.44Ref: TM-T28362
1mg38.00€2mg52.00€5mg84.00€10mg119.00€25mg236.00€50mg379.00€100mg565.00€500mg1,215.00€1mL*10mM (DMSO)93.00€Prinomastat hydrochloride
CAS:Prinomastat HCl, an oral MMP (1, 3, 9) inhibitor, IC50s: 79, 6.3, 5.0 nM, shows antitumor activity.
Formula:C18H22ClN3O5S2Purity:98%Color and Shape:SolidMolecular weight:459.97LP8
CAS:LP8 is a novel inhibitor of Trypanosoma cruzi CYP51.Formula:C16H19N3O4SPurity:98%Color and Shape:SolidMolecular weight:349.4JAK3/BTK-IN-5
CAS:JAK3/BTK-IN-5 is a potent dual inhibitor targeting JAK3 and BTK with synergistic effects, valuable for related autoimmune disease research.Formula:C19H22ClN7O2Color and Shape:SolidMolecular weight:415.88WAY-151693
CAS:WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).Formula:C21H22ClN3O5SColor and Shape:SolidMolecular weight:463.93β-Lactamase-IN-1
CAS:β-Lactamase-IN-1 (4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one) is a β-Lactamase inhibitor and targets the infection of NeisseriaFormula:C11H13N3O4Purity:99.89%Color and Shape:SolidMolecular weight:251.24Ref: TM-T19206
1mg60.00€5mg146.00€10mg215.00€25mg358.00€50mg510.00€100mg692.00€1mL*10mM (DMSO)152.00€L-708906
CAS:L-708906 is the Human Immunodeficiency Virus Type 1 inhibitor.Formula:C24H20O6Purity:98%Color and Shape:SolidMolecular weight:404.41AZD0865
CAS:AZD0865 is an effective drug that inhibits gastric H(+), K(+) -ATPase activity and acid formation in vitro, with rapid onset.Formula:C21H26N4O2Color and Shape:SolidMolecular weight:366.465Anticancer agent 147
CAS:Compound 6j (Anticancer agent 147), a sophoridine derivative and ferroptosis inducer, promotes intracellular accumulation of Fe2+, reactive oxygen species (ROSFormula:C32H40BrN3O2Purity:98%Color and Shape:SolidMolecular weight:578.58AZD-3289
CAS:AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.Formula:C24H14F5N5Color and Shape:SolidMolecular weight:467.39Trelanserin
CAS:Trelanserin (SL-650472) is an antagonist of the serotonin receptor.Formula:C24H24FN5O2SColor and Shape:SolidMolecular weight:465.54GID4 Ligand 3
CAS:GID4 Ligand 3 binds GID4; Kd 110 μM, IC50 148.5 μM; useful in CRBN/VHL research.Formula:C10H12N2OSColor and Shape:SolidMolecular weight:208.28DSHS00884
CAS:DSHS00884 is a potent inhibitor of human papillomavirus E6 (IC50: 10 μM).Formula:C12H12N4O2S2Color and Shape:SolidMolecular weight:308.38NPD-001
CAS:NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).Formula:C33H40N6O4Purity:98%Color and Shape:SolidMolecular weight:584.71MRL20
CAS:MRL20 is a SPPARγM with strong anti-diabetic effects and a better therapeutic range than full PPARγ agonists in rodents.Formula:C28H24F3NO6Color and Shape:SolidMolecular weight:527.49Oxythiamine diphosphate
CAS:Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).Formula:C12H17N3O8P2SPurity:98%Color and Shape:SolidMolecular weight:425.29Erythrofuranosyladenine
CAS:ETA: Non-toxic MTAP substrate, salvage agent for T-cell leukemia therapy with L-alanosine.Formula:C9H11N5O3Color and Shape:SolidMolecular weight:237.22Foliglurax monohydrochloride
CAS:Foliglurax monohydrochloride, an antiparkinsonian, is a selective brain-penetrant mGluR4 PAM with an EC50 of 79 nM.Formula:C23H24ClN3O3SColor and Shape:SolidMolecular weight:457.97Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFormula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82CP-471474
CAS:MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.Formula:C16H17FN2O5SPurity:98%Color and Shape:SolidMolecular weight:368.38Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formula:C15H19N3O2Color and Shape:SolidMolecular weight:273.33AQ 148
CAS:AQ 148 is a potent competitive inhibitor of HIV-1 PR.Formula:C30H37N3O4Color and Shape:SolidMolecular weight:503.63Pyrazinib
CAS:Pyrazinib: novel anti-angiogenic, disrupts oesophageal cancer cell metabolism & cytokine secretion (IL-6, IL-4, IL-8, IL-13) in radioresistance.Formula:C12H10N2OColor and Shape:SolidMolecular weight:198.22CLR1501
CAS:CLR1501 is a fluorescently labeled CLR1404 analog and a cancer cell-selective fluorescence compound[1][2].Formula:C38H59BF2N3O4PPurity:98%Color and Shape:SolidMolecular weight:701.67hDHODH-IN-9
CAS:hDHODH-IN-9 is a potent hDHODH inhibitor, IC50=0.34 μM, toxic to MCF-7/A375 cells, promising for cancer research.Formula:C21H21NO4Color and Shape:SolidMolecular weight:351.4N-Retinoylphenylalanine
CAS:N-Retinoylphenylalanine is an inhibitor of alkaline phosphatase isoenzymes.Formula:C29H37NO3Purity:98%Color and Shape:SolidMolecular weight:447.61Cysteinesulfenic acid
CAS:Cysteinesulfenic acid is a protein-sulfenic acid involved in enzyme catalysis, redox regulation, and signal transduction.Formula:C3H7NO3SColor and Shape:SolidMolecular weight:137.16Nafadotride
CAS:Nafadotride is a dopamine D3 receptor antagonist.Formula:C22H27N3O2Color and Shape:SolidMolecular weight:365.47GSK2793660 HCl
CAS:GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.Formula:C22H32ClN3O3Color and Shape:SolidMolecular weight:421.96HMR1031
CAS:HMR1031 is a specific α4ß1 integrin antagonist targeting VLA-4, VCAM-1, and fibronectin.Formula:C35H41N5O6Color and Shape:SolidMolecular weight:627.73Tilarginine
CAS:Tilarginine is a nitric oxide synthetase competitive inhibitor.Formula:C7H16N4O2Purity:98%Color and Shape:SolidMolecular weight:188.23Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Color and Shape:SolidMolecular weight:403.9Fce 28260
CAS:Fce 28260 is a 5 alpha-reductase inhibitor.Formula:C28H35F3N2O2Color and Shape:SolidMolecular weight:488.58SSI-4
CAS:SSI-4 is a Stearoyl CoA desaturase 1 (SCD1) inhibitor that can be labeled with carbon-11 (11C) for use as a ligand in small animal in vivo PET/CT imagingFormula:C19H21ClN4O3Purity:98%Color and Shape:SolidMolecular weight:388.85BTP1
CAS:BTP1 blocks NFAT activation, T-cell cytokine release, and selectively inhibits SOCE over Ca2+ voltage channels.Formula:C18H10ClF6N3OColor and Shape:SolidMolecular weight:433.73c-Fms-IN-9
CAS:c-Fms-IN-9 inhibits c-FMS/uFMS and uKIT with IC50 <0.01μM and 0.1-1μM, from patent WO2014145023A1.Formula:C21H23N7O2Purity:98%Color and Shape:SolidMolecular weight:405.45KF 18259
CAS:KF 18259 is a potent and selective serotonin3 receptor antagonist with similar activity to ondansetron and granisetron in animal models.Formula:C22H29ClN2O3Color and Shape:SolidMolecular weight:404.94GPR40 Activator 1
CAS:GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes.Formula:C31H31NO3SPurity:98%Color and Shape:SolidMolecular weight:497.65Hsp90-Cdc37-IN-1
CAS:Hsp90-Cdc37-IN-1 is an Hsp90-Cdc37 interaction disruptor (IC50: 140 nM) that inhibit cell migration and reverse drug resistance.Formula:C43H57FN2O6SPurity:98%Color and Shape:SolidMolecular weight:748.99HPK1-IN-26
CAS:HPK1-IN-26, from WO2021254118A1, is a potent dual HPK1/GLK inhibitor for studying animal infections.Formula:C19H21N5OSColor and Shape:SolidMolecular weight:367.47GlyRS-IN-1
CAS:GlyRS-IN-1 is an inhibitor of glycyl-tRNA synthase (GlyRS). It can inhibit the growth of bacteria.Formula:C12H17N7O7SColor and Shape:SolidMolecular weight:403.37RSH-7
CAS:RSH-7 is a potent dual inhibitor of BTK and FLT3, with IC50s of 47 and 12 nM, respectively.RSH-7 has antiproliferative and antitumor activities, inducingFormula:C22H25FN8OPurity:99.43%Color and Shape:SolidMolecular weight:436.49NASTRp
CAS:NASTRp inhibits CREB-CBP, has anti-cancer properties, regulates cell cycle, suppresses autophagy, and induces ER stress.Formula:C18H15ClNO5PColor and Shape:SolidMolecular weight:391.74RET-IN-19
CAS:RET-IN-19, a potent RET inhibitor, anticancer: IC50 6.8 nM (RET-wt), 13.51 nM (RET V804M); for NSCLC research.Formula:C28H28N6O4SColor and Shape:SolidMolecular weight:544.62Cinuperone
CAS:Cinuperone, a D2, alpha1, sigma receptor antagonist, halts dopamine-related behaviors; antipsychotic use stopped due to orthostasis.Formula:C23H24FN3OColor and Shape:SolidMolecular weight:377.45Boc-8-aoc-oh
CAS:Boc-8-aoc-oh is a PROTAC linker with an alkane chain, terminal carboxylic acid, and Boc-protected amino, used in amide bond formation.Formula:C13H25NO4Color and Shape:SolidMolecular weight:259.34Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purity:98%Color and Shape:SolidMolecular weight:393.74
