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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66669 products of "Inhibitors"

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  • MI-1851

    CAS:
    <p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88
  • NK1 receptor antagonist 2

    CAS:
    NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.
    Formula:C31H35F7N4O2
    Color and Shape:Solid
    Molecular weight:628.62
  • SP inhibitor 1


    SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.
    Formula:C36H38N2O2
    Color and Shape:Solid
    Molecular weight:530.7
  • Antifungal agent 42


    Antifungal 42 blocks biofilm formation and inhibits C.albicans' CYP51.
    Formula:C22H20Cl2N4Se2
    Color and Shape:Solid
    Molecular weight:569.25
  • RORγt inverse agonist 29


    RORγt inverse agonist 29 is a potent, selective, orally active RORγt inverse agonist with an IC50 value of 21 nM.
    Formula:C25H24N2O5S
    Color and Shape:Solid
    Molecular weight:464.53
  • Topoisomerase I inhibitor 8

    CAS:
    Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.
    Formula:C24H21FN2O4
    Color and Shape:Solid
    Molecular weight:420.43
  • LSD1-IN-21


    LSD1-IN-21: potent LSD1 inhibitor, crosses blood-brain barrier, IC50 of 0.956 μM; lowers TNF-α, anti-cancer, anti-inflammatory.
    Formula:C24H25N5O2S
    Color and Shape:Solid
    Molecular weight:447.55
  • VU6005806

    CAS:
    VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.
    Formula:C17H16F3N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.41
  • Antimalarial agent 2


    Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.
    Formula:C27H25N3O5
    Color and Shape:Solid
    Molecular weight:471.5
  • LSD1/2-IN-3


    LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07
  • CDK8-IN-9


    <p>CDK8-IN-9, potent CDK8 inhibitor (IC50: 48.6 nM), curbs tumor growth, useful for colorectal cancer research.</p>
    Color and Shape:Solid
  • PPO-IN-1


    PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).
    Formula:C18H10F3N3O4S
    Color and Shape:Solid
    Molecular weight:421.35
  • KT5926

    CAS:
    KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.
    Formula:C30H27N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.55
  • MEIS-IN-1

    CAS:
    <p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>
    Formula:C24H21F3N2O4
    Color and Shape:Solid
    Molecular weight:458.43
  • Antibacterial agent 78


    <p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>
    Formula:C16H23N3S2
    Color and Shape:Solid
    Molecular weight:321.5
  • Prohibitin ligand 1


    Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.
    Formula:C20H22N2O
    Color and Shape:Solid
    Molecular weight:306.4
  • VEGFR-2-IN-12


    VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.
    Formula:C22H24N6O3S
    Color and Shape:Solid
    Molecular weight:452.53
  • (rel)-Myrislignan

    CAS:
    (rel)-Myrislignan, a lignan compound with a relative configuration, has been isolated from Myristica fragrans Houtt.
    Formula:C21H26O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.43
  • CVN636

    CAS:
    CVN636, a potent and selective allosteric agonist for the mGluR7 receptor, exhibits oral activity and CNS permeability [1], with an EC50 of 7 nM for human
    Formula:C19H20FNO4S
    Color and Shape:Solid
    Molecular weight:377.43
  • JBJ-02-112-05

    CAS:
    JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC 50 of 15 nM for EGFR L858R/T790M [1].
    Formula:C27H20N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.54