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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66669 products of "Inhibitors"

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  • THR-β agonist 4

    CAS:
    THR-β agonist 4 is a potent agonist of THR-β.
    Formula:C16H11Cl2F2N5O6S
    Color and Shape:Solid
    Molecular weight:510.26
  • CDK7-IN-17

    CAS:
    CDK7-IN-17, a pyrimidine-based CDK7 inhibitor, shows promise for various cancers, especially with abnormal transcription.
    Formula:C24H26F3N6OP
    Purity:99.60%
    Color and Shape:Solid
    Molecular weight:502.47
  • AZ14145845


    AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.
    Formula:C32H35N9O
    Color and Shape:Solid
    Molecular weight:561.68
  • Aplaviroc

    CAS:
    Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.
    Formula:C33H43N3O6
    Purity:97.98% - 98.26%
    Color and Shape:Solid
    Molecular weight:577.71
  • Nurr1 agonist 1


    Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1 which is an appealing target to treat neurodegenerative diseases.
    Formula:C16H14N2O2
    Color and Shape:Solid
    Molecular weight:266.29
  • BMS-681

    CAS:
    BMS-681 is a CCR2 antagonist blocking chemokine binding, aiding control of inflammatory and neurodegenerative diseases.
    Formula:C26H36F3N5O
    Color and Shape:Solid
    Molecular weight:491.59
  • E6201

    CAS:
    E6201, a dual kinase inhibitor, blocks MEK1/FLT3 and has anti-tumor/psoriasis effects with low IC50s: ERK2 (5.2 nM), JNK (91 nM), p38 MAPK (19 nM).
    Formula:C21H27NO6
    Color and Shape:Solid
    Molecular weight:389.44
  • Dazucorilant

    CAS:
    Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i <1 nM, useful for neurological research.
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57
  • MEIS-IN-3


    MEIS-IN-3 is a potent inhibitor of MEIS.
    Formula:C25H26N2O4
    Color and Shape:Solid
    Molecular weight:418.48
  • LSD1-IN-16


    LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.
    Formula:C20H18N2OS
    Color and Shape:Solid
    Molecular weight:334.43
  • Antitumor agent-48


    Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.
    Formula:C35H34N2O14
    Color and Shape:Solid
    Molecular weight:706.65
  • Vimirogant hydrochloride


    Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), >1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.
    Formula:C27H36ClF3N4O3S
    Color and Shape:Solid
    Molecular weight:588.21487
  • VEGFR-2/DHFR-IN-2


    VEGFR-2/DHFR-IN-2 inhibits VEGFR-2 & DHFR (IC50: 0.623 & 9.085 μM), toxic to C26, HepG2, MCF7 cells (IC50: 3.59-8.38 μM), promising for cancer study.
    Formula:C21H21NO4
    Color and Shape:Solid
    Molecular weight:351.4
  • HMG499

    CAS:
    HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.
    Formula:C33H54O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.78
  • D6808


    D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.
    Formula:C30H25F3N6O2
    Color and Shape:Solid
    Molecular weight:558.55
  • Aniline-MPB-amino-C3-PBD

    CAS:
    Aniline-MPB-amino-C3-PBD is a cytotoxic agent comprised of the non-alkylating group. It is a sequence-selective DNA minor-groove binding agent.
    Formula:C42H46N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:758.86
  • hCAII-IN-4

    CAS:
    hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.
    Formula:C31H23NO9
    Color and Shape:Solid
    Molecular weight:553.52
  • DH376

    CAS:
    DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.
    Formula:C31H28F2N4O3
    Color and Shape:Solid
    Molecular weight:542.58
  • Rubropunctatin

    CAS:
    Rubropunctatin is a monascus pigment with very potent cancer cell proliferation inhibitory effects.
    Formula:C21H23NO4
    Color and Shape:Solid
    Molecular weight:353.41
  • Pamiparib maleate

    CAS:
    Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.
    Formula:C44H42F2N8O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:944.859