Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65630 products of "Quinazoline and Quinoline Derivatives"
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Minoxidil Sulfate
CAS:Controlled ProductFormula:C9H15N5O4SColor and Shape:NeatMolecular weight:289.31Dasatinib Carboxylic Acid Ethyl Ester
CAS:Controlled Product<p>Applications Protected Dasatinib Carboxylic Acid (D193605). An oxidative metabolite of Dasatinib (M6 metabolite); used in the treatment of cancers and immune diseases. It is a COVID19-related research product.<br>References Jaworski, T., et al.: Xenobiotica, 21, 1451 (1991), Shah, N., et al.: Science, 305, 399 (2004), O'Hare, T., et al.: Cancer Res., 65, 4500 (2005), Das, J., et al.: J. Med. Chem., 49, 6819 (2006), Christopher, L., et al.: Drug Metab. Dispos., 36, 1341 (2008),<br></p>Formula:C24H28ClN7O3SColor and Shape:NeatMolecular weight:530.04Iso Loratadine
CAS:Controlled Product<p>Impurity Loratadine EP Impurity E<br>Applications Iso Loratadine (Loratadine EP Impurity E) is a Loratadine (L469575) impurity. An isomer of Loratadine used for preparation of tricyclic amides and ureas useful for inhibition of G-protein function and for treatment of proliferative diseases.<br>References Billah., et al.: Lipids, 26, 1172 (1991), Piwinski., et al.: J. Med. Chem., 34, 457 (1991),<br></p>Formula:C22H23ClN2O2Color and Shape:NeatMolecular weight:382.88N-Desmethyl Diphenhydramine Hydrochloride
CAS:<p>Applications N-Desmethyl Diphenhydramine is an impurity of Diphenhydramine (D486900) with antihistaminic activity.<br>References Nauta, W. T. et al.: Med. Chem., Spec. Contrib. Int. Symp., 3rd, 125 (1973);<br></p>Formula:C16H19NO·ClHColor and Shape:White To Light BeigeMolecular weight:277.79Hydroxy Dimetridazole-d3
CAS:Controlled Product<p>Applications A labelled metabolite of Dimetridazole (D479660).<br>References Voogd, C., et al.: Mutat. Res., 86, 243 (1981), Polzer, J., et al.: Anal. Chim. Acta., 529, 299 (2005), Mohamed, R., et al.: J. Agric .Food Chem., 56, 3500 (2008),<br></p>Formula:C52H3H4N3O3Color and Shape:BeigeMolecular weight:160.15(R)-(-)-Chlorpheniramine Maleate
CAS:Formula:C16H19ClN2•C4H4O4Color and Shape:NeatMolecular weight:274.7911607rac-Ruxolitinib-d9 (major)
CAS:Controlled Product<p>Applications Labelled racemic analogue of Ruxolitinib (R702000). Ruxolitinib is a selective Janus tyrosine kinase (JAK1 and JAK2) inhibitor used in the treatment of myeloproliferative neoplasms and psoriasis.<br>References Shilling, A.D. et al.: Drug Metab. Disp., 38, 2023 (2010); Mesa, R.A.: IDrugs, 13, 394 (2010); Campas-Moya, C.: Drugs Fut., 35, 457 (2010);<br></p>Formula:C17H9D9N6Color and Shape:White To Light YellowMolecular weight:315.42Teneligliptin Hydrobromide (2:5)
CAS:Controlled Product<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formula:C22H32·5Br2·5N6OSColor and Shape:NeatMolecular weight:628.86Celecoxib Carboxylic Acid Acyl-β-D-glucuronide
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Celecoxib Carboxylic Acid Acyl-β-D-glucuronide is a glucuronide metabolite of Celecoxib (C251000), a Cox-2 inhibitor.<br>References Penning, T., et al.: J. Med. Chem., 40, 1347 (1997), Barta, T., et al.: Bioorg. Med. Chem. Lett., 8, 3443 (1998), Paulson, S., et al.: Drug Metab. Dispos., 28, 514 (2000),<br></p>Formula:C23H20F3N3O10SPurity:>80%Color and Shape:NeatMolecular weight:587.48Risperidone Z-Oxime Impurity
CAS:Controlled Product<p>Impurity Risperidone EP Impurity B<br>Applications Risperidone Z-Oxime (Risperidone EP Impurity B) is an impurity of Risperidone (R525000). Risperidone impurity per USP.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Jannssen, P.A.J., et al.: J. Pharmacol. Exp. Ther., 244, 685 (1988), Gelders, Y.G., et al.: Pharmacopsychiatry, 23, 206 (1990), Green, B.: Curr. Med. Res. Opin., 16, 57 (2000)<br></p>Formula:C23H28F2N4O2Color and Shape:NeatMolecular weight:430.494’-O-Benzyloxy Ezetimibe
CAS:Controlled Product<p>Impurity Ezetimibe Benzyl Ether Impurity<br>Applications Protected Ezetimibe, used for the synthesis of related derivatives.<br>References Raman, B., et al.: J. Pharm. Biomed. Anal., 52, 73 (2010),<br></p>Formula:C31H27F2NO3Color and Shape:NeatMolecular weight:499.55(R)-Etiracetam Acid
CAS:Controlled Product<p>Applications Levetiracetam Acid can be used as reactant/reagent in synthesis, Aβ42/tau aggregation, acetylcholinesterase/butyrylcholinesterase inhibitory activities, acute toxicity, and docking studies of levetiracetam-huprine/tacrine hybrids as anti-Alzheimer's agents.<br>References Sola, I., et al.: J Med Chem, 58, 6018 (2015)<br></p>Formula:C8H13NO3Color and Shape:Off-WhiteMolecular weight:171.19Pyraclostrobin
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Pyraclostrobin is a fungicide for use in seed grass and food crops. Useful in cannabis testing kits as a component of pesticide mixes (P698240).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Gyldenkaerne, S., et al.: Pestic Sci., 55, 1210 (1999), Pennington, D., et al.: Environ. Sci. Technol., 39, 1119 (2005), Wang, S., et al.: Food Control., 18, 731 (2007),<br></p>Formula:C19H18ClN3O4Color and Shape:YellowMolecular weight:387.823-[(5S)-(4-Fluorophenyl)-5-hydroxypentanoyl]-(4S)-phenyl-1,3-oxazolidin-2-one
CAS:Controlled Product<p>Applications 3-[(5S)-(4-Fluorophenyl)-5-hydroxypentanoyl]-(4S)-phenyl-1,3-oxazolidin-2-one is an intermediate of Ezetimibe (E975000, E975002), an antihyperlipoproteinemic. A cholesterol absorption inhibitor.<br>References Singh, A., et. al.: J. Molecular Catal. B., 85, 99 (2013); van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997); van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Formula:C20H20FNO4Color and Shape:NeatMolecular weight:357.38Nifuratel
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Nifuratel is a drug used as an antibacterial, antifungal, antiprotozoal (Trichomonas). Nifuratel appears to have a broad antibacterial spectrum of action and is effective against Chlamydia trachomatis and Mycoplasma spp. as well as fungal infections from Candida spp.<br>References Nam, H., et al.: J. Microbiol., 45, 515 (2007), Costerton, W., et al.: J. Clin. Invest., 112, 1466 (2003), Ferris, M., et al.: J. Clin. Microbiol., 42, 5892 (2004),<br></p>Formula:C10H11N3O5SColor and Shape:Yellow To Dark YellowMolecular weight:285.284’-(Trifluoromethyl)valerophenone-(E)-O-2-(2-aminoethyl) Oxime Maleate
Controlled Product<p>Applications 4’-(Trifluoromethyl)valerophenone(E)-O-2-(2-aminoethyl) Oxime Maleate is an impurity in the synthesis of Fluvoxamine (F603500), a selective serotonin reuptake inhibitor (SSRI) used as an anti-depressant. Antiobsessional.<br>References Claassen, V., et al.: Br. J. Pharmacol., 60, 505 (1977), Koran, L.M., et al.: J. Clin. Psychopharmacol., 16, 121 (1996), Ware, M.R., et al.: J. Clin. Psychiatry, 58, Suppl. 5, 15 (1997), Inazu, M., et al.: Neurochem. Int., 39, 39 (2001)<br></p>Formula:C20H28F3N3O5Color and Shape:NeatMolecular weight:447.452-(chloromethyl)-5-(5-methylthiophen-2-yl)-1H,4H-thieno[2,3-d]pyrimidin-4-one
CAS:Purity:95%Molecular weight:296.7900085449219Clozapine-d8
CAS:Controlled Product<p>Applications An antipsychotic.A representative lot was 92% d8, 8% d7.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Stille, et al: Farnaco, Ed. Prat., 26, 603 (1971), Hane, J.M., et al.: Psychopharmacol. Bull., 24, 62 (1988), Meltzer, H.Y.: J. Clin. Psychiatry, 55, Suppl. B, 47 (1994)<br></p>Formula:C18H11D8ClN4Color and Shape:Light Yellow To YellowMolecular weight:334.87Dihydroxy Moxonidine
CAS:Controlled Product<p>Impurity Moxonidine Impurity 1<br>Applications Dihydroxy Moxonidine (Moxonidine Impurity 1) is an impurity of Moxonidine (M745800).<br>References Diasio, R., et al.: Antimicrob. Agents Chemother., 14, 903 (1978), Yang, L., et al.: J. Pharm. Biomed. Anal., 22, 487 (2000),<br></p>Formula:C8H11N5O2Color and Shape:NeatMolecular weight:209.21Ref: 10-F619849
1g446.00€5gTo inquire10gTo inquire2.5g959.00€50mg95.00€100mg158.00€250mg221.00€500mg366.00€Roxatidine Acetate Hydrochloride
CAS:Controlled Product<p>Applications A histamine H2-receptor antagonist. It is used to inhibit gastric acid secretion; an antiulcer agent.<br>References Tarutani, M. et al.: Arzneim.-Forsch., 35, 703 (1985); Yagita, M. et al.: Therap. Res., 7, 96 (1987); Asai, M. et al.: Gek. Yak., 50, 922 (2008);<br></p>Formula:C19H28N2O4·ClHColor and Shape:NeatMolecular weight:384.90(R)-Ambrisentan
CAS:<p>Applications (R)-Ambrisentan is the R-isomer impurity of Ambrisentan (A575860), which is a nonpeptide endothelin ETA receptor antagonist. Antihypertensive.<br>References Riechers, H., et al.: J. Med. Chem., 39, 2123 (1996); Billman, G.E., et al.: Curr. Opin. Invest. Drugs, 3, 1483 (2002); Vatter, H., et al.: Clin. Neuropharmacol., 26, 73 (2003);<br></p>Formula:C22H22N2O4Color and Shape:White To Off-WhiteMolecular weight:378.42Perampanel
CAS:Controlled Product<p>Applications Perampanel is a novel, noncompetitive AMPA receptor antagonist for the treatment of epilepsy. Also in the treatment of primary generalized tonic-clonic seizures in idiopathic generalized epilepsy. Perampanel is a selective non-competitive α-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid receptor antagonist that reduces neuronal excitation (1,2,3,4).<br>References (1) Shih, J., et al.: Therap. Clinical Risk Management, 9, 285 (2013)(2) Rogawski, M. A., et al.: Epilepsy Curr., 11, 56 (2011)(3) Franco, V., et al.: Ther Drug Monit. 38, 744 (2016) (4) Rudzinski, L. A., et al.: J Investig Med. 64, 1087 (2016)<br></p>Formula:C23H15N3OColor and Shape:Light YellowMolecular weight:349.38Desthiazolylmethyl Ritonavir
CAS:Controlled Product<p>Impurity Ritonavir EP Impurity L<br>Applications Desthiazolylmethyl Ritonavir (Ritonavir EP Impurity L) is an analogue of the selective HIV protease inhibitor Ritonavir (R535000). It is a COVID19-related research product.<br>References Brittain, H., et al.: Pharm. Res., 8, 963 (1991), Sham, H., et al.: J. Med. Chem., 39, 392 (1996), Phadnis, N., et al.: J. Pharm. Sci.,86, 1256 (1997), Bauer, J., et al.: Pharma. Res., 18, 859 (2001),<br></p>Formula:C33H43N5O4SColor and Shape:White To Off-WhiteMolecular weight:605.79Flumequine
CAS:Controlled Product<p>Applications Fluorinated quinolone antibacterial.This compound is a contaminant of emerging concern (CECs).<br>References Stilwell, G., et al.: Antimicrob. Agents Chemother., 7, 483 (1975), Rohlfing, S.R., et al.: J. Antimicrob. Chemother., 3, 615 (1977),<br></p>Formula:C14H12FNO3Color and Shape:White Crystalline PowderMolecular weight:261.25Orbifloxacin
CAS:<p>Applications Orbifloxacin is a fluoroquinolone antibiotic used in veterinary medicine, mainly for the treatment of staphylococcal infections in dogs.<br>References Ganiere, J.P. et al.: Res. Vet. Sci., 77, 67 (2004); Scott, D.W. et al.: Can. Vet. J., 47, 999 (2006); Rubin, J. et al.: Vet. Microbiol., 131, 164 (2008);<br></p>Formula:C19H20F3N3O3Color and Shape:White To Light YellowMolecular weight:395.38Ramifenazone
CAS:<p>Applications Analgesic, antipyretic, anti-inflammatory.<br>References Tubaro, E., et al.: Arzneim.-Forsch., 20, 1024 (1970),<br></p>Formula:C14H19N3OColor and Shape:NeatMolecular weight:245.32(R)-Norfenfluramine Hydrochloride
CAS:Controlled ProductFormula:C10H12F3N·ClHColor and Shape:NeatMolecular weight:239.665N-Benzyl Hydroxymedetomidine
CAS:Controlled Product<p>Applications N-Benzyl Hydroxymedetomidine is an impurity of Medetomidine (M203250, HCl); an α2-adrenergic agonist, sedative, and analgesic.<br>References Scheinin, M., et al.: Br. J. Clin. Pharmacol., 24, 443 (1987); Stenberg, D., et al.: J. Vet. Pharmacol. Ther., 10, 319 (1987); Virtanen, R., et al.: Eur. J. Pharmacol., 150, 9 (1988); Cullen, L.K., et al.: Br. Vet. J., 152, 519 (1996)<br></p>Formula:C20H22N2OColor and Shape:NeatMolecular weight:306.4N,N'-Methylene Ambroxol Hydrochloride
CAS:Controlled Product<p>Impurity Ambroxol EP Impurity B Hydrochloride<br>Stability Hygroscopic<br>Applications Ambroxol Cyclic Impurity is a metabolite as well as an impurity of the bronchosecretolytic drug, Ambroxol (A575900).<br>References Hammer, R. et al.: Arzneim.-Forsch., 28, 899 (1978); Nieder, M. et al.: HRC & CC, 9, 561 (1986); Huq, F. et al.: J. Pharmacol. Toxicol., 3, 147 (2008);<br></p>Formula:C14H18Br2N2O·ClHColor and Shape:White To Off-WhiteMolecular weight:426.57N-Nitroso Desmethyl Olopatadine
Controlled ProductFormula:C20H20N2O4Color and Shape:NeatMolecular weight:352.3846-methoxy-N-(pyridin-3-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Purity:95.0%Molecular weight:271.3399963378906Carboxymefloquine-d3
CAS:Controlled Product<p>Applications Labelled Carboxymefloquine (C178700). Carboxymefloquine is a metabolite of Mefloquine (M207050).<br>References Crevoisier, C., et al.: Eur. J. Clin. Pharmacol., 53, 135 (1997), Ridtitid, W., et al.: J. Pharm. Pharmacol., 52, 1265 (2000),<br></p>Formula:C12H2D3F6NO2Color and Shape:NeatMolecular weight:312.182-Methylpyrazine
CAS:Controlled Product<p>Applications 2-Methyl-pyrazine is an intermediate used to synthesize 5-Methyl-2(1H)-pyrazinone (M324900) which is a derivative of 2-Hydroxypyrazine (H952710). 2-Hydroxypyrazine (H952710) is used in the synthesis of potential antioxidants.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Shi, J. et al.: J. Phys. Org. Chem., 22, 1038 (2009); Bonde, C. et al.: Ind. J. Hetero. Chem., 10, 271 (2001);<br></p>Formula:C5H6N2Color and Shape:NeatMolecular weight:94.112-(((5-((Dimethylamino)methyl)furan-2-yl)methyl)thio)ethanamine Fumarate (2:1)
CAS:Controlled Product<p>Impurity USP Ranitidine Related Compound A<br>Applications 2-(((5-((Dimethylamino)methyl)furan-2-yl)methyl)thio)ethanamine (E)-2-Butenedioate is an impurity of Ranitidine (R120000), a histamine H2-receptor antagonist which inhibits gastric acid secretion. Antiulcerative.<br>References Bradshaw, J., et al.: Brit. J. Pharmacol., 66, 464 (1979), Berstad, A., et al.: Scand. J. Gastroenterol, 15, 637 (1980), Hohnjec, M., et al.: Anal. Profiles Drug Subs., 15, 533 (1986),<br></p>Formula:C10H18N2OS·C4H4O4Color and Shape:WhiteMolecular weight:544.7276Prothioconazole
CAS:<p>Applications Prothioconazole is an antifungal metabolite used in agricultural fungicides and herbicides.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Aristimuno Ficoseco, M.E., et al.: Nat. Prod. Res (2016);<br></p>Formula:C14H15Cl2N3OSColor and Shape:NeatMolecular weight:344.264-((2R,3S,6S)-6-(4-Fluorophenyl)-3-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)phenol (Ezetimibe Impurity)
<p>Applications 4-((2R,3S,6S)-6-(4-Fluorophenyl)-3-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)phenol, is a diol impurity of Ezetimibe (E975000), a drug that lowers plasma cholesterol levels.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Formula:C18H19FO3Color and Shape:NeatMolecular weight:302.34rac N-Methyl Atomoxetine Oxalate
CAS:<p>Applications rac N-Methyl Atomoxetine Oxalate is a derivative of Atomoxetine which acts as a norepinephrine reuptake inhibitor.<br>References Farid, N.A., et al.: J. Clin. Pharmacol., 25, 296 (1985), Gehlert, D.R., et al.: J. Neurochem., 64, 2792 (1995), Hwamg. et al.: Neurosci. Lett., 265, 151 (1999), Ring, B.J., et al.: Drug Metab. Dispos., 30, 319 (2002),<br></p>Formula:C18H23NO·C2H2O4Color and Shape:Off White SolidMolecular weight:359.42N-Formyl Benzocaine
CAS:Controlled Product<p>Applications N-Formyl Benzocaine is a degradation product of Benzocaine (B202970); a compound that is used as an anesthetic (local).<br>References Kholod, Y., et al.: Environ. Sci. Technol., 43, 9208 (2009); Fliri, A., et al.: J. Med. Chem., 52, 8038 (2009); Helguera, A., et al.: J. Pharm. Sci., 98, 4557 (2009); Onoue, S., et al.: J. Pharm. Sci., 98, 3647 (2009); Koellmer, M., et al.: AAPS PharmSciTech., 14, 1333 (2013)<br></p>Formula:C10H11NO3Color and Shape:NeatMolecular weight:193.199Betrixaban
CAS:Controlled Product<p>Applications Betrixaban is a novel anticoagulant. An oral direct inhibitor of factor Xa (FXa) for use in the prevention of venous thromboembolism (VTE).<br>References Turpie, A.G.G. et al.: Thromb. Haemost., 101, 68 (2009); Gomez-Outes, A. et al.: Curr. Vasc. Pharmacol., 7, 309 (2009);<br></p>Formula:C23H22ClN5O3Color and Shape:Light YellowMolecular weight:451.91Meloxicam
CAS:<p>Applications Preferential cyclooxygenase (COX-2) inhibitor. Sudoxicam and Meloxicam are nonsteroidal anti-inflammatory drugs (NSAIDs) from the enol-carboxamide class.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hawkey, C., et al.: Br. J. Rheumatol., 35, Suppl. 1, 1 (1996), Fleischmann, R., et al.: Expert Opin. Pharmacother., 3, 1501 (2002),<br></p>Formula:C14H13N3O4S2Color and Shape:Light YellowMolecular weight:351.40rac-trans-Ambroxol-d5
CAS:Controlled Product<p>Applications A labelled metabolite of Bromohexine. Ambroxol Hydrochloride is a bronchosecretolytic drug.<br>References Jauch, R., et al.: Arzneim-Forsch., 13, 474 (1963)<br></p>Formula:C13H13D5Br2N2OColor and Shape:NeatMolecular weight:383.13Methyl 5-chloro-2-hydroxy-1-oxo-2,3-dihydro-1H-indene-2-carboxylate
CAS:Controlled Product<p>Applications Methyl 5-chloro-2-hydroxy-1-oxo-2,3-dihydro-1H-indene-2-carboxylate (cas# 144172-24-7) is a useful research chemical. It is an intermediate in the synthesis of IN-KG 433 (I627995). IN-KG 433 is an impurity of Indoxacarb (I654000), an oxadiazine pesticide that acts against lepidopteran larvae and is the active ingredient in a number of household insecticides including cockroach baits.<br>References Wang, H., et al.: Water. Sci. Technol., 61, 2733 (2010); Shono, T., et al.: Pesticide. Biochem. Physiol., 75, 1 (2003);<br></p>Formula:C11H9O4ClColor and Shape:NeatMolecular weight:240.633-Hydroxy Medetomidine
CAS:Controlled Product<p>Applications A metabolite of Medetomidine (M203250).<br>References Salonen, J.S., et al.: Xenobiotica, 20, 471 (1990),<br></p>Formula:C13H16N2OColor and Shape:NeatMolecular weight:216.284-(2,3-Epoxypropoxy)carbazole
CAS:Controlled Product<p>Impurity Carvedilol EP Impurity D; Carvedilol USP-D<br>Applications 4-(2,3-Epoxypropoxy)carbazole (Carvedilol EP Impurity D; Carvedilol USP-D) is an intermediate in the synthesis of Carvedilol (C184625).<br></p>Formula:C15H13NO2Color and Shape:Beige SolidMolecular weight:239.275-(p-Methylphenyl)-5-phenylhydantoin
CAS:<p>Applications An antibody agent.<br>References Rowell, F. J., et al.: Immunochemistry, 13, 891 (1976),<br></p>Formula:C16H14N2O2Color and Shape:NeatMolecular weight:266.29N-Ethyl-N-methyl-3-vinylphenyl Carbamate
CAS:Controlled Product<p>Impurity Rivastigmine USP Related Compound F<br>Stability Light Sensitive<br>Applications A related compound of Rivastigmine (R541000), a cholinesterase inhibitor. Rivastigmine USP Related Compound F.<br></p>Formula:C12H15NO2Color and Shape:White SolidMolecular weight:205.25Linagliptin Methyl Dimer
CAS:Controlled Product<p>Applications Linagliptin Methyldimer is an impurity of Linagliptin (L465900). Linagliptin is a novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.<br>References Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011); Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011)<br></p>Formula:C51H56N16O4Color and Shape:NeatMolecular weight:957.095N-Desmethyl 4-Hydroxy Toremifene Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A metabolite of Toremifene (T547500).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Phillips, D., et al.: Carcinogenesis, 17, 89 (1996), Davies, R., et al.: Cancer Res., 57, 1288 (1997), Moorthy, B., et al.: Biochem. Pharmacol., 53, 663 (1997),<br></p>Formula:C25H27Cl2NO2Color and Shape:NeatMolecular weight:444.392-(2-(2-morpholinothiazol-4-yl)ethyl)isoindoline-1,3-dione hydrochloride
CAS:Purity:95.0%Molecular weight:379.8599853515625Aripiprazole-d8 (Butyl-d8)
CAS:Controlled ProductFormula:C232H8H19Cl2N3O2Color and Shape:White To Off-WhiteMolecular weight:456.43(Z,Z)-5-(2-Methyl-3-phenyl-propenylidene)-4-oxo-2-thioxo-3-thiazolidineacetic Acid
CAS:Controlled Product<p>Stability Light Sensitive<br>Applications (Z,Z)-5-(2-Methyl-3-phenyl-propenylidene)-4-oxo-2-thioxo-3-thiazolidineacetic Acid is a stereoisomer of Epalrestat (E565300), an aldose reductase inhibitor. Used in the treatment of diabetic neuropathy.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Terashima, H., et al.: J. Pharmacol. Exp. Ther., 229, 226 (1983), Kikkawa, R., et al.: Diabetologia, 24, 290 (1983), Kojima, K., et al.: Jpn. J. Ophthalmol., 29, 99 (1985), Qi, M. et al.: J. Beij, Inst. Tech., 13, 445 (2004);<br></p>Formula:C15H13NO3S2Color and Shape:Yellow-Red SolidMolecular weight:319.4Desfluoro Risperidone
CAS:Controlled Product<p>Impurity Risperidone EP Impurity K<br>Applications Desfluoro Risperidone (Risperidone EP Impurity K) is a Risperidone (R525000) impurity, as antipsychotics.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Formula:C23H28N4O2Color and Shape:NeatMolecular weight:392.496-fluoro-2-methylquinoline-4-carboxylic acid
CAS:Formula:C11H8FNO2Purity:95.0%Color and Shape:Yellow powderMolecular weight:205.188Paliperidone Z-Oxime
CAS:Controlled Product<p>Applications Paliperidone Z-oxime is an impurity of Paliperidone (P141000), a known orally active antipsychotic agent.<br>References Rao, J., et al.: Pharmacia Lettre, 3, 240 (2011);<br></p>Formula:C23H28F2N4O3Color and Shape:NeatMolecular weight:446.49(S)-4-(Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl)morpholine
CAS:Purity:98.0%Molecular weight:421.27458077Bupivacaine
CAS:<p>Applications Bupivacaine is a sodium channel blocker, local anesthetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),<br></p>Formula:C18H28N2OColor and Shape:NeatMolecular weight:288.43Ref: 10-F025806
1gTo inquire2gTo inquire5gTo inquire10gTo inquire100mgTo inquire250mgTo inquire500mgTo inquireTelmisartan-d4
CAS:Controlled Product<p>Applications Telmisartan-d4 is deuterium labelled Telmisartan (T017000). Telmisartan is an angiotensin II receptor antagonist.<br>References Wienen, W. et al.: Br. J. Pharmacol., 110, 245 (1993); Neutel, J.M. et al: Adv. Therap., 15, 206 (1998)<br></p>Formula:C33D4H26N4O2Color and Shape:NeatMolecular weight:518.642,2-Diphenylglycine
CAS:Controlled Product<p>Impurity Phenytoin USP Related Compound A 2,2-Diphenylglycine<br>Stability Hygroscopic<br>Applications 2,2-Diphenylglycine (Phenytoin USP Related Compound A 2,2-Diphenylglycine) is a decomposition product of Phenytoin (D491650), which reduces incidence of grand mal seizures; appears to stabilize excitable membranes perhaps through effects on Na+, K+, and Ca2+ channels.<br>References Shah, V. et al.: J. Pharm. Sci., 75, 1113 (1986); Faucette, S., et al.: J. Pharmacol. Exp. Ther., 320, 72 (2007); Raymond, H. et al.: Teratol., 10, 237 (1974);<br></p>Formula:C14H13NO2Color and Shape:White To Off-WhiteMolecular weight:227.26Mirtazapine-d3
CAS:Controlled Product<p>Applications An α2-Adrenergic blocker; analogue of Mianserin. Antidepressant.<br>References De Boer, T., et al.: Neuropharmacology, 27, 399 (1988), Smith, W.T., et al.: Psychopharmacol. Bull., 26, 191 (1990)<br></p>Formula:C172H3H16N3Color and Shape:White To BeigeMolecular weight:268.373,7-Dihydro-3,7-dimethyl-6-[(5-oxohexyl)oxy]-2H-purin-2-one
CAS:Formula:C13H18N4O3Color and Shape:NeatMolecular weight:278.31Eltrombopag Olamine
CAS:<p>Stability Hygroscopic<br>Applications Eltrombopag is an agonist of the Thrombopoietin (Tpo) receptor, used as treatment for thrombocytopenia<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Bussel, J., et al.: New Eng. J. Med., 357, 2237 (2007), Marsilje, T., et al.: Bioorg. Med. Chem. Lett., 18, 5259 (2008), Alper, P., et al.: Bioorg. Med. Chem. Lett., 18, 5255 (2008)<br></p>Formula:C25H22N4O4·2C2H7NOColor and Shape:Dark RedMolecular weight:564.63Anastrozole
CAS:Controlled Product<p>Applications An aromatase inhibitor. Used as an antineoplastic.<br>References Plourde, P.V., et al.: Breast Cancer Res. Treat., 30, 103 (1994), Buzdar, A.U., et al.: Cancer, 79, 730 (1997)<br></p>Formula:C17H19N5Color and Shape:NeatMolecular weight:293.37Ref: 10-F547198
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire250mgTo inquireUvinul A Plus
CAS:<p>Applications Uvinul A Plus is a component of cosmetic emulsion with UV protection.<br>References Chang, M., et al.: J. Food Drug Anal., 9, 199 (2001), Simeoni, S., et al.: J. Pharm. Biomed. Anal., 38, 250 (2005), Vielhaber, G., et al.: Photochem. Photobiol. Sci., 5, 275 (2006), Lee, S., et al.: J. Cosmet. Sci., 59, 469 (2008),<br></p>Formula:C24H31NO4Color and Shape:White To YellowMolecular weight:397.513’-Anhydro Ezetimibe
CAS:Controlled ProductFormula:C24H19F2NO2Color and Shape:NeatMolecular weight:391.41Pamabrom
CAS:Controlled Product<p>Applications A diuretic used to reduce menstrual pains.<br>References Varga, J., et al.: Mol. Immunol., 28, 641 (1991), Marrero-Ponce, Y., et al.: Bioorg. Med. Chem., 13, 2881 (2005), Ibrahim, H., et al.: Drug Discov. Ther., 3, 168 (2009),<br></p>Formula:C7H7BrN4O2·C4H11NOColor and Shape:NeatMolecular weight:348.20Hydroxydehydro Nifedipine Carboxylate
CAS:Controlled ProductFormula:C16H14N2O7Color and Shape:NeatMolecular weight:346.29Phenylephrone-d3 Hydrochloride
CAS:Controlled Product<p>Applications Labelled impurity C of Phenylephrine.<br>References Bodor, N., et al.: J. Med. Chem., 31, 100 (1988), Goskonda, V., et al.: J. Pharm. Sci., 88, 180 (1999),<br></p>Formula:C9H9D3ClNO2Color and Shape:NeatMolecular weight:204.674-[6-(4-Methoxy-phenyl)-pyridin-3-yl]-pyrimidin-2-ylamine
Purity:95.0%Molecular weight:278.315002441406252-(4-(3-(2',8-Bis(trifluoromethyl)-10H-[3,10'-biphenothiazin]-10-yl)propyl)piperazin-1-yl)ethanol
Controlled ProductFormula:C35H32F6N4OS2Color and Shape:NeatMolecular weight:702.7842-O-tert-Butyldimethylsilyloxyethyl Rapamycin
CAS:<p>Stability Hygroscopic<br>Applications 42-O-tert-Butyldimethylsilyloxyethyl Rapamycin is a useful synthetic intermediate in the synthesis of Everolimus (E945400); an immunosuppressant macrolide and analog of the parent drug Rapamycin (R124000). Everolimus inhibits cytokine-mediated lymphocyte proliferation.<br>References Dumont, F.J., et al.: Curr. Opin. Invest. Drugs, 2, 1220 (2001); Kovarik, J. M., et al.: Clin. Pharmacol. Ther., 69, 48 (2001); Nashan, B., et al.: Ther. Drug Monit., 24, 53 (2002); Venkata, S.P., et al.: PCT Int. Appl. WO 2012066502 A1 20120524. May 24, 2012<br></p>Formula:C59H97NO14SiColor and Shape:NeatMolecular weight:1072.48Tolvaptan
CAS:Controlled Product<p>Applications Tolvaptan is a selective, competitive arginine vasopressin V2 receptor antagonist used to treat hyponatremia (low blood sodium levels) associated with congestive heart failure, cirrhosis, and the syndrome of inappropriate antidiuretic hormone (SIADH).<br>References Paterna, S., et al.: Eur. J. Heart Fail, 2, 305 (2000); Udelson, J., et al.: Circulation, 104, 2417 (2001); Goldsmith, S., et al.: J. Am. Coll Cardiol., 46, 1785 (2005); Schrier, R., et al.: N. Engl. J. Med., 355, 2099 (2006);<br></p>Formula:C26H25ClN2O3Color and Shape:White To Off-WhiteMolecular weight:448.942-Hydroxy Imipramine
CAS:Controlled Product<p>Applications A metabolite of Imipramine.<br>References De Jongh, G.D., et al.: Drug Metab. Dispos., 2, 48 (1981), Suckow, R.F., et al.: J. Pharm. Sci., 73, 1745 (1984), Fraser, A.D., et al.: J. Anal. Toxicol., 11,168 (1987),<br></p>Formula:C19H24N2OColor and Shape:Yellowish SolidMolecular weight:296.41Salbutamol Glyoxal Impurity
Controlled Product<p>Stability Hygroscopic<br>Applications Salbutamol Glyoxal Impurity that is synthesized from C369215 (3-Chloromethyl-4-hydroxyacetophenone).<br></p>Formula:C9H10O5Color and Shape:Off White SolidMolecular weight:198.17Afatinib Dimaleate
CAS:Controlled Product<p>Applications Afatinib Dimaleate is a salt of Afatinib {BIBW 2992) (B377000), an aminocrotonylamino-substituted quinazoline derivative used for treating cancer and diseases of the respiratory tract, lungs, gastrointestinal tract, bile duct, and gallbladder. An anilino-quinazoline that irreversibly inhibits EGFR and HER2 kinase activity.<br>References D, Li. et al.: Oncogene., 27, 4702 (2008); Wang, X. et al.: Cancer Res., 74, 4431 (2014);<br></p>Formula:C24H25ClFN5O3·2C4H4O4Color and Shape:NeatMolecular weight:718.08Ebastine
CAS:<p>Applications A nonsedating type histamine H1-receptor antagonist. Antihistaminic.<br>References Fliri, A., et al.: J. Med. Chem., 52, 8038 (2009), Inomata, N., et al.: J. Dermatol., 36, 224 (2009), Carvajal, A., et al.: Clin. Pharmacol. Ther., 85, 481 (2009), Yamashita, S., et al.: Mol. Pharm., 6, 48 (2009),<br></p>Formula:C32H39NO2Color and Shape:White To Off-WhiteMolecular weight:469.66Mavoglurant
CAS:Controlled Product<p>Applications Mavoglurant is a non-competitive metabotropic glutamate receptor 5 (mGlu5) receptor antagonist.<br>References Vranesic, I., et al.; Bioorg. Med. Chem., 22, 5790 (2014); Kubas, H., et al.: Bioorg. Med. Chem. Lett., 23, 6370 (2013)<br></p>Formula:C19H23NO3Color and Shape:NeatMolecular weight:313.391,4-Dibromobenzene
CAS:<p>Applications 1,4-Dibromobenzene is used in the synthesis of triarylamines as well as trans-stilbenes. Also used in the synthesis of calcium channel blockers for inhibition of TRPV6-mediated calcium transport.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Corriu, R. et al.: J. Chem. Soc. Chem. Comm., 3, 144 (1972); Lambert, C. et al.: J. Am. Chem. Soc., 121, 8434 (1999); Hofer, A. et al.: Bioorg. Med. Chem., 21, 3202 (2013);<br></p>Formula:C6H4Br2Color and Shape:Light YellowMolecular weight:235.908-Bromo-3-methyl-7-(2-butynyl)-xanthine
CAS:Controlled ProductFormula:C10H9BrN4O2Color and Shape:NeatMolecular weight:297.1086-PIPERAZIN-1-YL-4(3H)-QUINAZOLINONE-3-ACETIC ACID
CAS:Purity:97.0%Color and Shape:SolidMolecular weight:288.3070068359375PTC-124
CAS:Controlled Product<p>Applications PTC-124 is a nonaminoglycoside that has been reported to induce ribosomes to read through premature nonsense stop signals on mRNA, allowing the production of full-length functional proteins,<br>References Yu, H. et al.: Int. J. Mol. Med., 33, 729 (2014); Aditya, S. et al.: J. Biomed. Pharm. Res., 2, 21 (2013);<br></p>Formula:C15H9FN2O3Color and Shape:White To Off-WhiteMolecular weight:284.24Ranolazine Dihydrochloride
CAS:<p>Stability Hygroscopic<br>Applications Ranolazine Dihydrochloride is an anti-ischemic agent which modulates myocardial metabolism. Antianginal.<br>References Chaitman, B.R., et al.: J. Am. Coll. Cardial., 43, 1375 (2004); McCormack, J.G., et al.: Gen. Pharmacol., 30, 639 (1998); Schofield, J.A.H., et al.: Expert Opin. Invest. Drugs, 11, 117 (2002)<br></p>Formula:C24H35Cl2N3O4Color and Shape:NeatMolecular weight:500.46Ondansetron-d3
CAS:Controlled Product<p>Applications Ondansetron-d3 is a labeled specific serotonin (5-HT3) receptor antagonist. Antiemetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Kris, M.G., et al.: J. Clin. Oncol., 6, 659 (1988); Faris, P..L., et al.: Lances, 355, 792 (2000)<br></p>Formula:C18H16D3N3OColor and Shape:NeatMolecular weight:296.38
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