Enzyme Modulators
Enzyme modulators are compounds that can enhance or inhibit the activity of enzymes, thereby regulating the rate of biochemical reactions. These modulators play a critical role in controlling metabolic pathways, cell signaling, and various physiological processes. Enzyme modulators are widely used in research and drug development to study enzyme functions and to develop therapeutic agents. At CymitQuimica, we offer a comprehensive range of high-quality enzyme modulators to support your research in enzyme regulation and drug discovery.
Subcategories of "Enzyme Modulators"
Found 693 products of "Enzyme Modulators"
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Licofelone
CAS:<p>Dual COX/5-LO inhibitor; anti-inflammatory; analgesic</p>Formula:C23H22ClNO2Purity:Min. 95%Color and Shape:PowderMolecular weight:379.88 g/molRasagiline mesylate
CAS:Controlled Product<p>Monoamine oxidase-B inhibitor; anti-parkinsonian; neuroprotective</p>Formula:C12H13N•CH4O3SPurity:Min. 95%Color and Shape:PowderMolecular weight:267.35 g/molAZD 1152
CAS:<p>AZD 1152 is an Aurora kinase inhibitor, which is a type of small-molecule therapeutic agent. It is derived from the pharmaceutical research conducted by AstraZeneca. Its primary mode of action involves the selective inhibition of Aurora B kinase, an enzyme crucial for the regulation of mitosis. By interfering with this enzyme, AZD 1152 disrupts the normal progression of cell division, leading to the inhibition of proliferation and induction of apoptosis in rapidly dividing cells.</p>Formula:C26H31FN7O6PPurity:Min. 97 Area-%Color and Shape:Slightly Yellow PowderMolecular weight:587.54 g/molCerivastatin sodium
CAS:<p>An inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase that reduces total cholesterol and low-density lipoprotein (LDL). Cerivastatin is cardioprotective and anti-atherosclerotic. Cerivastatin inhibits the expression of the atherosclerotic genes monocyte chemoattractant protein-1 (MCP-1) and C-C chemokine receptor type 2 (CCR2), whilst inducing the expression of Kruppel-like factor 2 (KLF2).</p>Formula:C26H33FNNaO5Purity:Min. 98 Area-%Color and Shape:PowderMolecular weight:481.53 g/molSU 11274
CAS:<p>MET tyrosine kinase inhibitor; anti-proliferative; pro-apoptotic</p>Formula:C28H30ClN5O4SPurity:Min. 95%Color and Shape:Yellow To Orange SolidMolecular weight:568.09 g/molOmeprazole - Bio-X ™
CAS:<p>Omeprazole is a proton pump inhibitor (PPI) that inhibits the production of gastric acid in the stomach. This is due to Omeprazole binding through a stable disulphide bond to the H+/K+ ATPase enzyme found on parietal cells, and preventing hydrogen ion transport. Consequently, gastric acid secretion is supressed. As a PPI, Omerprazole can be used to treat disorders where gastric acid is over-secreted. Examples of these disorders are gastroesophageal reflux disease (GERD) and peptic ulcer disease.</p>Formula:C17H19N3O3SPurity:Min. 95%Color and Shape:PowderMolecular weight:345.42 g/molAceclofenac - Bio-X ™
CAS:<p>Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.</p>Formula:C16H13Cl2NO4Purity:Min. 95%Color and Shape:PowderMolecular weight:354.18 g/molRivastigmine tartrate - Bio-X ™
CAS:Controlled Product<p>Rivastigmine is a cholinergic agent that is used in the treatment of dementia in Parkinson’s and Alzheimer’s disease. This drug is a carbamate derivative that binds to and inactivates cholinesterase such as acetylcholinesterase and butyrylcholinesterase. This leads to an increase concentration of acetylcholine at cholinergic synapse.</p>Formula:C14H22N2O2•C4H6O6Purity:Min. 95%Color and Shape:PowderMolecular weight:400.42 g/molTideglusib
CAS:<p>An irreversible GSK-3β inhibitor that reduces phosphorylation of tau proteins, protects from neuronal loss and has cognitive and behavioural benefits in murine models. Studied for its potential as a therapeutic agent in Alzheimer’s disease and other neurodegenerative diseases. Tideglusib was also shown to inhibit the main protease Mpro from the SARS-CoV-2 virus with IC50 of 1.55 μM.</p>Formula:C19H14N2O2SPurity:Min. 95%Color and Shape:White To Off-White SolidMolecular weight:334.39 g/molChymostatin
CAS:<p>Inhibitor of chymotrypsin</p>Formula:C31H41N7O6Color and Shape:White To Yellowish SolidMolecular weight:607.7 g/molBAY 607550
CAS:<p>A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.</p>Formula:C27H32N4O4Purity:Min. 95%Color and Shape:PowderMolecular weight:476.24236Zotarolimus
CAS:<p>Inhibitor of immunophilin FKBP12 and mTOR signalling with immunosuppressant activity. Zotarolimus inhibits proliferation of endothelial cells and smooth muscle cells and is employed in vascular interventional therapies.</p>Formula:C52H79N5O12Purity:Min. 95%Color and Shape:White PowderMolecular weight:966.21 g/molRebamipide - Bio-X ™
CAS:<p>Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.</p>Formula:C19H15ClN2O4Purity:Min. 95%Color and Shape:PowderMolecular weight:370.79 g/molAG 120
CAS:<p>Inhibits isocitrate dehydrogenase 1 (IDH-1) harbouring a gain of function mutation at R132, which causes impaired cellular differentiation via epigenetic modulation. By inhibiting mutant IDH1, synthesis of oncometabolite 2-hydroxyglutarate is reduced. This compound therefore has therapeutic potential in solid and haematological malignancies, such as acute myeloid leukemia (AML).</p>Formula:C28H22ClF3N6O3Purity:Min. 95%Color and Shape:White To Off-White SolidMolecular weight:582.96 g/molGilteritinib
CAS:<p>Inhibitor of FLT3 and AXL tyrosine kinases</p>Formula:C29H44N8O3Purity:Min. 95%Color and Shape:PowderMolecular weight:552.71 g/molXMU MP 2
CAS:<p>BRK tyrosine kinase (PTK6) inhibitor; anti-proliferative in breast cancer cells</p>Formula:C32H33F3N8O2Purity:Min. 95%Color and Shape:PowderMolecular weight:618.65 g/molCZC 25146
CAS:<p>Inhibitor of leucine-rich repeat kinase LRRK2Â</p>Formula:C22H25FN6O4SPurity:Min. 98 Area-%Color and Shape:PowderMolecular weight:488.54 g/molLovastatin - Bio-X ™
CAS:<p>Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.</p>Formula:C24H36O5Purity:Min. 95%Color and Shape:PowderMolecular weight:404.54 g/molMRK 560
CAS:<p>γ-secretase inhibitor; reduces amyloid-β in brainÂ</p>Formula:C19H17ClF5NO4S2Purity:Min. 95%Molecular weight:517.92 g/molApremilast - Bio-X ™
CAS:<p>Apremilast is the commercial name of a phosphodiesterase-4 (PDE4) inhibitor developed to treat chronic inflammatory disorders. Similarly to thalidomide, the apremilast molecule carries a phthalimide ring, but it lacks however the glutarimide ring needed to bind to cereblon, specifically targeted by thalidomide. As a drug, apremilast is indicated for the treatment of psoriasis and psoriatic arthritis.</p>Formula:C22H24N2O7SPurity:Min. 99 Area-%Color and Shape:White/Off-White SolidMolecular weight:460.5 g/mol
