Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(196 produits)
- Caséine Kinase(138 produits)
- DHFR(32 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(301 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(85 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(133 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(86 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(20 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(44 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9158 produits trouvés pour "Métabolisme"
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FPH2
CAS :FPH2 (BRD-9424) (BRD-9424) is a small molecule promoting differentiation of iPS-derived hepatocytes.Formule :C14H16ClN5O2SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :353.83Milrinone Lactate
CAS :Milrinone Lactate is a positive inotropic cardiotonic compound. Milrinone Lactate has vasodilator properties, inhibiting cAMP phosphodiesterase type 3 activity in the myocardium and vascular smooth muscle.Formule :C15H15N3O4Couleur et forme :White Or Whitish Crystalline PowderMasse moléculaire :301.31-phenyl-3,4-dihydroisochinoline
CAS :1-phenyl-3,4-dihydroisochinoline: dopamine analog, interacts with CNS receptors, studied for Parkinson's, Alzheimer's, and Huntington's.Formule :C15H13NDegré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :207.27FR054
CAS :FR054 inhibits PGM3, a key enzyme in the HBP, significantly reducing breast cancer cell growth and survival.Formule :C14H19NO8Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :329.3PAL-4
CAS :PAL-4 stimulates the activity of LYPLAL1, a poorly characterized serine hydrolase with complex genetic links to human metabolic traits.
Formule :C17H15ClN4O3S2Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :422.916-Hydroxy-4-methylcoumarin
CAS :6-Hydroxy-4-methylcoumarin (6-Hydroxy-4-Methyl-2H-Chromen-2-One) is a secondary metabolite of coumarin, which has anticancer effects.Formule :C10H8O3Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :176.17ACTH (18-39) TFA (human)
CAS :Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) is a corticotropinlike intermediate lobe peptide, produced by melanotropic cells.Formule :C114H166F3N27O38Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :2579.69Ref: TM-TP1240
1mg84,00€2mg110,00€5mg177,00€10mg268,00€25mg442,00€50mg645,00€100mg889,00€200mg1.198,00€Methyl 13-cis-4-Oxoretinoate
CAS :Methyl 13-cis-4-Oxoretinoate (13-cis-4-Oxo-retinoic acid Methyl Ester) is a retinoic acid metabolite in neuroblastoma.Formule :C21H28O3Degré de pureté :99.08% - 99.7%Couleur et forme :SolidMasse moléculaire :328.45Ref: TM-T3203
1mg54,00€2mg96,00€5mg158,00€10mg225,00€25mg404,00€50mg593,00€100mg845,00€500mg1.693,00€1mL*10mM (DMSO)154,00€Genz-123346 free base
CAS :Genz 123346 is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1.Formule :C24H38N2O4Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :418.57BAY-1436032
CAS :BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).Formule :C26H30F3N3O3Degré de pureté :99.65% - 99.71%Couleur et forme :SolidMasse moléculaire :489.53Ivosidenib
CAS :Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.Formule :C28H22ClF3N6O3Degré de pureté :98.71% - 99.98%Couleur et forme :SolidMasse moléculaire :582.96Calcifediol monohydrate
CAS :Calcifediol monohydrate (25-hydroxy Vitamin D3 monohydrate), the main circulating metabolite of vitamin D3, is a potent VDR inhibitor.Formule :C27H46O3Degré de pureté :99.31%Couleur et forme :Brownish Fine PowderMasse moléculaire :418.65[11C]MP 10
CAS :[11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.Formule :C25H20N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :391.45FPH1
CAS :FPH1 (BRD-6125) (BRD-6125) can promote the expansion of iPS-derived hepatocytes.Formule :C16H15ClF2N2O3SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :388.82Ref: TM-T6506
2mg38,00€5mg57,00€10mg90,00€25mg177,00€50mg264,00€100mg394,00€200mg582,00€1mL*10mM (DMSO)67,00€Tiplaxtinin
CAS :Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.
Formule :C24H16F3NO4Degré de pureté :99.16% - 99.93%Couleur et forme :SolidMasse moléculaire :439.38Tolfenpyrad
CAS :Tolfenpyrad is an effective insecticide[1], used against pests that are resistant to existing insecticides such as organophosphates and carbamates.[2]Formule :C21H22ClN3O2Degré de pureté :97%Couleur et forme :SolidMasse moléculaire :383.87XEN445
CAS :XEN445, a potent and selective endothelial lipase(EL) inhibitor (IC50=0.237 uM), exhibitis good ADME and PK properties.Formule :C18H17F3N2O3Degré de pureté :99.47% - 99.6%Couleur et forme :SolidMasse moléculaire :366.33Cilobradine
CAS :Cilobradine is an HCN Channel blocker; an open channel blocker of neuronal Ih and related cardiac If channels.Formule :C28H38N2O5Couleur et forme :SolidMasse moléculaire :482.612-Ketoglutaric acid
CAS :2-Ketoglutaric acid is a reversible inhibitor of tyrosinase (IC50=15 mM). 2-Ketoglutaric acid is an intermediate of the Krebs cycle. High-Quality, Low-Cost!Formule :C5H6O5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :146.1Olprinone
CAS :Olprinone (Loprinone)(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and attenuateFormule :C14H10N4ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :250.26Firibastat
CAS :Firibastat (RB150) is a glutamyl aminopeptidase antagonist and an orally active brain penetrating prodrug of EC33.
Formule :C8H20N2O6S4Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :368.51Trichlormethiazide sodium
CAS :Trichlormethiazide sodium: oral thiazide diuretic, antihypertensive, boosts urine, Na/K excretion, may enhance renal clearance.Formule :C8H8Cl3N3NaO4S2Couleur et forme :SolidMasse moléculaire :403.63Maltoheptaose
CAS :Maltoheptaose is an activator of phosphorylase B for the preparation of heptulose-2-phosphate.Formule :C42H72O36Degré de pureté :99.43% - 99.81%Couleur et forme :SolidMasse moléculaire :1153.00Darexaban maleate
CAS :Darexaban maleate is a derivative used in the preparation of inhibitors of activated blood coagulation factor X.Formule :C31H34N4O8Couleur et forme :SolidMasse moléculaire :590.63SMS2-IN-2
CAS :SMS2-IN-2: potent, selective oral SMS2 inhibitor with IC50s 100 μM for SMS2, 56 μM for SMS1, anti-inflammatory.Formule :C19H13ClFN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.78Ref: TM-T7263
1mg108,00€2mg158,00€5mg259,00€10mg404,00€25mg665,00€50mg888,00€100mg1.251,00€1mL*10mM (DMSO)265,00€Lifirafenib HCl
CAS :Lifirafenib (Beigene-283/BGB-283): a potent, selective RAF/EGFR inhibitor effective against B-RAF mutated colorectal cancers.Formule :C26H19ClF3N3O3Couleur et forme :SolidMasse moléculaire :513.9012IDO-IN-1
CAS :IDO-IN-1: potent IDO inhibitor, IC50 of 59 nM (enzyme), 12 nM (HeLa cells).Formule :C9H7BrFN5O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :316.09Ref: TM-T7181
1mg49,00€5mg96,00€10mg155,00€25mg269,00€50mg404,00€100mg567,00€200mg763,00€1mL*10mM (DMSO)110,00€Tauro-Obeticholic acid
CAS :Tauro-Obeticholic acid is an active Obeticholic acid metabolite. Obeticholic acid is an orally bioavailable agonist of farnesoid-X receptor (FXR).Formule :C28H49NO6SDegré de pureté :99.74% - 99.82%Couleur et forme :SolidMasse moléculaire :527.76Ref: TM-T13092
1mg111,00€5mg260,00€10mg393,00€25mg650,00€50mg888,00€100mg1.243,00€1mL*10mM (DMSO)331,00€MSDC 0160
CAS :MSDC 0160 (CAY10415) is a prototype mTOT-modulating insulin sensitizer being used in trials studying the treatment of Type 2 Diabetes and Alzheimer's Disease.Formule :C19H18N2O4SDegré de pureté :98.11% - 99.53%Couleur et forme :SolidMasse moléculaire :370.42Ref: TM-T2607
1mg34,00€2mg48,00€5mg73,00€10mg94,00€25mg145,00€50mg187,00€100mg333,00€1mL*10mM (DMSO)78,00€Tetrahydropapaverine hydrochloride
CAS :Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.Formule :C20H26ClNO4Degré de pureté :99.08%Couleur et forme :White Crystal PowderMasse moléculaire :379.878U-73343
CAS :U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.Formule :C29H42N2O3Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :466.66Phenprocoumon
CAS :Phenprocoumon is an antagonist of vitamin K(IC50:1 μM).Formule :C18H16O3Degré de pureté :95.79% - 97.98%Couleur et forme :Fine White Crystalline Powder SolidMasse moléculaire :280.32Cycloguanil hydrochloride
CAS :Cycloguanil hydrochloride, proguanil's metabolite, inhibits Plasmodium/human dihydrofolate reductase (Ki: 0.3/1.5 nM).Formule :C11H14ClN5·ClHDegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :288.18NSC 4810
CAS :NSC 4810: an amide used with cytochrome P450 in vivo and acetylcholinesterase in vitro.Formule :C13H18ClNODegré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :239.74Carbasalate calcium
CAS :Carbasalate calcium (Rheomin) is an analgesic, antipyretic, and anti-inflammatory drug, as well as a platelet aggregation inhibitor.Formule :C19H18CaN2O9Degré de pureté :98%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :458.436Udenafil
CAS :Udenafil is an inhibitor of PDE5 .Formule :C25H36N6O4SDegré de pureté :99.90%Couleur et forme :Off-White SolidMasse moléculaire :516.66Ref: TM-T17199
5mg50,00€10mg80,00€25mg140,00€50mg219,00€100mg319,00€200mg457,00€1mL*10mM (DMSO)52,00€Pentamidine dihydrochloride
CAS :Pentamidine dihydrochloride (MP-601205 dihydrochloride) is an aromatic diamidine agent with activity against a number of microorganisms including protozoa (Formule :C19H26Cl2N4O2Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :413.34Ref: TM-T23132
5mg52,00€10mg78,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€500mg642,00€1mL*10mM (DMSO)52,00€16α-Hydroxyprednisolone
16α-Hydroxyprednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonideFormule :C21H28O6Degré de pureté :99.75% - 99.97%Couleur et forme :White SolidMasse moléculaire :376.44Fabomotizole dihydrochloride
CAS :Fabomotizole (Afobazole, Obenoxazine, CM346) is a non-sedative anxiolytic with neuroprotective properties, launched in Russia 2000s; exact mechanism unclear.Formule :C15H23Cl2N3O2SCouleur et forme :SolidMasse moléculaire :380.33CP-91149
CAS :CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence ofFormule :C21H22ClN3O3Degré de pureté :99.66% - 99.81%Couleur et forme :SolidMasse moléculaire :399.87Ref: TM-T6455
2mg35,00€5mg51,00€10mg84,00€25mg137,00€50mg197,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)57,00€Potassium 2-hydroxy-2-methylsuccinate
CAS :Potassium 2-hydroxy-2-methylsuccinate ((±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt) is a type of endogenous metabolite.Formule :C5H6K2O5Degré de pureté :99.96% - ≥98%Couleur et forme :SolidMasse moléculaire :224.296-Phosphogluconic acid
CAS :6-Phosphogluconic acid competitively inhibits PGI with Ki: 0.048 mM for glucose 6-P, 0.042 mM for fructose 6-P.Formule :C6H13O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :276.14Gabapentin hydrochloride
CAS :Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.Formule :C9H17NO2·HClDegré de pureté :99.71%Couleur et forme :Off-White SolidMasse moléculaire :207.7Alagebrium chloride
CAS :Alagebrium chloride (ALT711) inhibits AGEs, lowers systolic blood pressure, and benefits diastolic patients.Formule :C13H14ClNOSDegré de pureté :99.65% - 99.77%Couleur et forme :SolidMasse moléculaire :267.77RHC 80267
CAS :RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Formule :C20H34N4O4Degré de pureté :99.54%Couleur et forme :White SolidMasse moléculaire :394.51A 922500
CAS :A 922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse DGAT-1, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.Formule :C26H24N2O4Degré de pureté :97.34% - 97.66%Couleur et forme :SolidMasse moléculaire :428.48Enecadin HCl
CAS :Enecadin HCl is a voltage-dependent sodium and calcium channel blocker.Formule :C21H29ClFN3OCouleur et forme :SolidMasse moléculaire :393.93AGI-6780
CAS :AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.Formule :C21H18F3N3O3S2Degré de pureté :98.19% - 99.7%Couleur et forme :SolidMasse moléculaire :481.51Ref: TM-T1809
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg220,00€50mg393,00€100mg587,00€500mg1.264,00€1mL*10mM (DMSO)85,00€Tienilic Acid
CAS :Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
Formule :C13H8Cl2O4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :331.177-Hydroxy-3,4-dihydro-2(1H)-quinolinone
CAS :7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .Formule :C9H9NO2Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :163.17Fluvastatin potassium
CAS :Fluvastatin, a synthetic statin, lowers cholesterol and prevents heart disease.Formule :C24H25FKNO4Couleur et forme :SolidMasse moléculaire :449.56N-Glycolylneuraminic acid
CAS :N-Glycolylneuraminic acid (GcNeu) is a nonhuman sialic acid molecule synthesized in pigs. N-Glycolylneuraminic acid is a receptor of human and animal IAVs.Formule :C11H19NO10Degré de pureté :99.94%Couleur et forme :White To Off-White PowderMasse moléculaire :325.27Nampt-IN-1
CAS :Nampt-IN-1 (LSN3154567) (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM.Formule :C20H25N3O5SDegré de pureté :99.28% - 99.4%Couleur et forme :SolidMasse moléculaire :419.49Ref: TM-T4376
1mg37,00€2mg49,00€5mg79,00€10mg130,00€25mg245,00€50mg409,00€100mg605,00€1mL*10mM (DMSO)87,00€Y-29794 Tosylate
CAS :Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.Formule :C30H42N2O4S3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :590.86IDO-IN-7
CAS :IDO-IN-7 (NLG-919 analogue) is a potent IDO (indoleamine-(2, 3)-dioxygenase) pathway inhibitor.Formule :C18H22N2ODegré de pureté :99.32% - 99.9%Couleur et forme :SolidMasse moléculaire :282.38Tetradecylthioacetic acid
CAS :Synthetic fatty acid TTA has β-sulfur, resists β-oxidation, and activates PPARs, especially PPARα.
Formule :C16H32O2SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :288.49CP-640186 hydrochloride
CAS :CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat
Formule :C30H36ClN3O3Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :522.08Epiblastin A
CAS :Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.Formule :C12H10ClN7Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :287.71Pradefovir mesylate
CAS :Pradefovir mesylate (Hepavir B) is converted to 9-(2-phosphonylmethoxyethyl)adenine (PMEA) in human liver microsomes with Km of 60 μM.Formule :C18H23ClN5O7PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :519.9HNHA
CAS :HNHA is an inhibitor of HDAC.Formule :C17H21NO2SDegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :303.42Ref: TM-T21806
1mg44,00€5mg84,00€10mg135,00€25mg279,00€50mg445,00€100mg640,00€200mg879,00€1mL*10mM (DMSO)90,00€LH846
CAS :LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and 2.5 uM for CK1δ, ε and α); exhibits no inhibitory activity at CK2.Formule :C16H13ClN2OSDegré de pureté :90% - 98.26%Couleur et forme :SolidMasse moléculaire :316.81EMD638683
CAS :EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).Formule :C18H18F2N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.34Ref: TM-T6635
1mg74,00€2mg92,00€5mg150,00€10mg233,00€25mg358,00€50mg517,00€100mg737,00€200mg982,00€1mL*10mM (DMSO)120,00€Melilotic acid
CAS :3-(2-Hydroxyphenyl)propanoic acid, aka melilotic acid, found in cytoplasm, in foods like herbs, beetroot, cinnamon.Formule :C9H10O3Degré de pureté :99.65% - 99.83%Couleur et forme :SolidMasse moléculaire :166.17PD 128042
CAS :PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formule :C23H39NO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.56K-Ras-PDEδ-IN-1
CAS :K-Ras-PDEδ-IN-1 is a potent inhibitor of competitive K-Ras-PDEδ.It binds to the farnesyl binding pocket of PDEδ(Kd of 8 nM).
Formule :C25H26FN5O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :447.5BI-0115
CAS :BI-0115 inhibits LOX-1, preventing oxLDL uptake by triggering receptor inhibition and dimer formation.Formule :C15H14ClN3ODegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :287.74UCPH-101
CAS :UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Formule :C27H22N2O3Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :422.48Ref: TM-T4138
1mg50,00€2mg75,00€5mg130,00€10mg203,00€25mg409,00€50mg655,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)142,00€Ethyl 3,4-dihydroxybenzoate
CAS :Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.Formule :C9H10O4Degré de pureté :99.88%Couleur et forme :White Crystal Or PowderMasse moléculaire :182.17ML-030
CAS :ML-030 is a potent PDE4 inhibitor, selective for subtypes (A1, B1, B2, C1, D2) with IC50 ranging from 6.7 to 452 nM.Formule :C20H20N4O4SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :412.46ICI 63197
CAS :ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.Formule :C9H13N5ODegré de pureté :99.70%Couleur et forme :White SolidMasse moléculaire :207.23Orthanilamide
CAS :Orthanilamide (Orthanilamide) is a molecule containing the sulfonamide functional group attached to an aniline.Formule :C6H8N2O2SDegré de pureté :99.72% - 99.96%Couleur et forme :White To Pale Cream Crystalline Powder Or CrystalsMasse moléculaire :172.2Fraxinellone
CAS :1.Formule :C14H16O3Degré de pureté :99.35% - 99.92%Couleur et forme :SolidMasse moléculaire :232.27Ref: TM-T6S0071
2mg34,00€5mg50,00€10mg84,00€25mg152,00€50mg222,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)81,00€Tebufenpyrad
CAS :Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicantFormule :C18H24ClN3ODegré de pureté :98.63% - 99.16%Couleur et forme :SolidMasse moléculaire :333.864-Nonylphenylboronic acid
CAS :4-Nonylphenylboronic acid is a inhibitor of FAAH.
Formule :C15H25BO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :248.17Nifurtimox
CAS :Nifurtimox (BAY-A-2502) is an antiprotozoal agent (IC50s = 9.91, 12.28, and 10.44 μM against Taluahuén, LQ, and Brener strains of T.Formule :C10H13N3O5SDegré de pureté :99.87% - 99.89%Couleur et forme :SolidMasse moléculaire :287.29Tropifexor
CAS :Tropifexor (LJN452) is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM.
Formule :C29H25F4N3O5SDegré de pureté :99.3% - 99.85%Couleur et forme :SolidMasse moléculaire :603.58Ref: TM-T4379
1mg87,00€5mg166,00€10mg248,00€25mg437,00€50mg665,00€100mg1.008,00€200mg1.520,00€500mg2.252,00€Bepridil hydrochloride
CAS :Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channelsFormule :C24H35ClN2ODegré de pureté :99.45% - 99.68%Couleur et forme :SolidMasse moléculaire :403WIN 18446
CAS :inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)Formule :C12H20Cl4N2O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :366.11ABX-1431
CAS :ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).Formule :C20H22F9N3O2Degré de pureté :99.8% - 99.96%Couleur et forme :SolidMasse moléculaire :507.39Milacemide
CAS :Milacemide is a glycine prodrug and MAO-B inhibitor.Formule :C7H16N2ODegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :144.21Ref: TM-T50055
2mg39,00€5mg60,00€10mg86,00€25mg138,00€50mg200,00€100mg289,00€200mg405,00€1mL*10mM (DMSO)49,00€PF-9601N
CAS :PF-9601N: potent, selective MAO-BI with neuroprotection in PD models.Formule :C19H18N2ODegré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :290.36Mitochondrial fusion promoter M1
CAS :Mitochondrial fusion promoter M1, a modulator of mitochondrial dynamics, enhances mitochondrial function and cellular respiration, and has shown efficacy inFormule :C14H10Cl4N2ODegré de pureté :99.54% - 99.54%Couleur et forme :SolidMasse moléculaire :364.05Panaxadiol
CAS :Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng.Formule :C30H52O3Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :460.73Darexaban
CAS :Darexaban (YM-150) selectively inhibits Factor Xa, reducing clotting and risk of heart/stroke events.Formule :C27H30N4O4Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :474.55Ref: TM-T31206
1mg48,00€5mg95,00€10mg144,00€25mg235,00€50mg354,00€100mg512,00€200mg727,00€1mL*10mM (DMSO)92,00€Oroxylin A
CAS :Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion and enhances leukemia treatment.Formule :C16H12O5Degré de pureté :98.72% - 99.55%Couleur et forme :SolidMasse moléculaire :284.26Ref: TM-T6S1315
1mg37,00€5mg71,00€10mg90,00€25mg147,00€50mg208,00€100mg309,00€200mg447,00€1mL*10mM (DMSO)84,00€CP671305
CAS :CP671305 is an orally active, potent and selective inhibitor of phosphodiesterase-4-D.Formule :C23H19FN2O7Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :454.4Imidazole-5-propionic acid
CAS :Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination.Formule :C6H8N2O2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :140.14Sacubitril hemicalcium salt
CAS :Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.Formule :C48H56CaN2O10Degré de pureté :99.86% - 99.93%Couleur et forme :SolidMasse moléculaire :861.06Ref: TM-T4200
2mg39,00€5mg52,00€10mg64,00€25mg94,00€50mg106,00€100mg155,00€200mg207,00€1mL*10mM (DMSO)64,00€Glyco-Obeticholic acid
CAS :Glyco-Obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is an agonist of the farnesoid X receptor (FXR).Formule :C28H47NO5Degré de pureté :99.77% - 99.95%Couleur et forme :SolidMasse moléculaire :477.68Ref: TM-T11428
1mg49,00€2mgÀ demander5mg105,00€10mg160,00€25mg313,00€50mg1.320,00€1mL*10mM (DMSO)126,00€Hydroxy Dimetridazole
CAS :Hydroxy Dimetridazole is a hydroxy metabolite of Dimetridazole which combats protozoan infections.
Formule :C5H7N3O3Degré de pureté :99.83% - 99.85%Couleur et forme :SolidMasse moléculaire :157.13trans-AUCB
CAS :trans-AUCB (t-AUCB) is an effective and selective soluble epoxide hydrolase inhibitor (IC50s: 1.3 nM, 8 nM, 8 nM for hsEH, mouse sEH and rat sEH, respectively).Formule :C24H32N2O4Degré de pureté :99.27% - 99.66%Couleur et forme :SolidMasse moléculaire :412.52TMS
CAS :TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).Formule :C18H20O4Degré de pureté :99.17% - 99.73%Couleur et forme :SolidMasse moléculaire :300.35Calcitriol
CAS :Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM).
Formule :C27H44O3Degré de pureté :98.81% - 99.64%Couleur et forme :Colorless Crystalline Solid SolidMasse moléculaire :416.64(R)-GNE-140
CAS :(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.Formule :C25H23ClN2O3S2Degré de pureté :98.25% - 98.91%Couleur et forme :SolidMasse moléculaire :499.04AG-120 (racemic)
CAS :AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.Formule :C28H22ClF3N6O3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :582.96PDE10-IN-1
CAS :PDE10-IN-1 (SEP-0372814) is used for treating CNS and metabolic disorders.Formule :C21H19N7Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :369.42IOX4
CAS :IOX4 is a potent PHD2 inhibitor (IC50 = 1.6 nM)Formule :C15H16N6O3Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :328.33Amifostine trihydrate
CAS :Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formule :C5H15N2O3PS·3H2ODegré de pureté :99.71% - 99.80%Couleur et forme :SolidMasse moléculaire :268.27DMU-2139
CAS :DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).Formule :C19H15NO2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :289.33Ref: TM-T8728
1mg38,00€5mg80,00€10mg116,00€25mg226,00€50mg334,00€100mg497,00€200mg720,00€1mL*10mM (DMSO)80,00€PSB-1434
CAS :PSB-1434 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 1.59 nM, selectivity versus MAO-A>6000-fold.Formule :C14H9F2N3ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :273.24Ref: TM-T24679
1mg86,00€5mg177,00€10mg268,00€25mg439,00€50mg628,00€100mg870,00€200mg1.153,00€1mL*10mM (DMSO)167,00€Eliglustat
CAS :Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.Formule :C23H36N2O4Degré de pureté :99% - 99.70%Couleur et forme :SolidMasse moléculaire :404.54Ref: TM-T3663
1mg54,00€2mg71,00€5mg89,00€10mg117,00€25mg173,00€50mg226,00€100mg421,00€500mg945,00€1mL*10mM (DMSO)88,00€RMC-4550
CAS :RMC-4550 is an effective and allosteric inhibitor of SHP2 (IC50: 0.583 nM).Formule :C21H26Cl2N4O2Degré de pureté :98.95% - 99.65%Couleur et forme :SolidMasse moléculaire :437.36Ref: TM-T16762
1mg58,00€5mg113,00€10mg178,00€25mg409,00€50mg605,00€100mg860,00€1mL*10mM (DMSO)124,00€ATP disodium salt hydrate
CAS :ATP disodium salt hydrate (Adenosine disodium triphosphate) is a nucleoside triphosphate used in cells as a coenzyme.Formule :C10H16N5Na2O14P3Degré de pureté :98.79% - >99.99%Couleur et forme :SolidMasse moléculaire :569.16PRL-3 Inhibitor I
CAS :PRL-3 Inhibitor I (BR-1) is a phosphatase of regenerating liver 3 (PRL-3) inhibitor which blocks the migration and invasion of metastatic cancer cells.Formule :C17H11Br2NO2S2Degré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :485.21Belzutifan
CAS :"Belzutifan (MK-6482) is an oral HIF-2α inhibitor for ccRCC, with enhanced potency (IC50: 9 nM)."Formule :C17H12F3NO4SDegré de pureté :99.34% - 99.88%Couleur et forme :SolidMasse moléculaire :383.34Ref: TM-T16679
1mg66,00€5mg144,00€10mg205,00€25mg389,00€50mg625,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)158,00€TPPU
CAS :TPPU is a potent inhibitor of both human and mouse sEH (IC50 of 3.7 and 2.8 nM, respectively)Formule :C16H20F3N3O3Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :359.34Enpp-1-IN-1
CAS :Enpp-1-IN-1 is an inhibitor of Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1)Formule :C17H17N3O3SDegré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :343.4Ref: TM-T7888
1mg126,00€5mg260,00€10mg394,00€25mg677,00€50mg954,00€100mg1.288,00€1mL*10mM (DMSO)286,00€Vorasidenib
CAS :Vorasidenib (PVM/MA) is an inhibitor of mutant isocitrate dehydrogenase (IDH; IC50s = 31.9 and 31.7 nM for IDH1R132H and IDH2R140Q, respectively)Formule :C14H13ClF6N6Degré de pureté :98.28% - 99.57%Couleur et forme :SolidMasse moléculaire :414.74Ref: TM-T7307
1mg50,00€2mg74,00€5mg113,00€10mg178,00€25mg340,00€50mg512,00€100mg733,00€1mL*10mM (DMSO)102,00€SN 6
CAS :SN 6 (SN6) is a selective Na+/Ca2+ exchanger (NCX) inhibitor (IC50s of NCX1: 2.9 μM , NCX2: 16 μM ,NCX3: 8.6 μM)Formule :C20H22N2O5SDegré de pureté :97.28%Couleur et forme :SolidMasse moléculaire :402.46U-73122
CAS :U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.Formule :C29H40N2O3Degré de pureté :97.50%Couleur et forme :Solid Off-WhiteMasse moléculaire :464.64CAY10698
CAS :CAY10698 is a 12-lipoxygenase inhibitor (12-LO; IC50 of 5.1 μM).Formule :C17H17N3O4S2Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :391.46Ref: TM-T8950
2mg38,00€5mg52,00€10mg88,00€25mg161,00€50mg243,00€100mg355,00€200mg502,00€1mL*10mM (DMSO)62,00€LMPTP INHIBITOR 1 dihydrochloride
CAS :LMPTP Inhibitor 1 Dihydrochloride is a compound selectively targeting low molecular weight protein tyrosine phosphatase (LMPTP), exhibiting potent inhibitoryFormule :C28H38Cl2N4ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :517.53Ref: TM-T41298
1mg73,00€5mg160,00€10mg250,00€25mg465,00€50mg673,00€100mg945,00€200mg1.251,00€1mL*10mM (DMSO)178,00€Mitapivat sulfate hydrate
CAS :Mitapivat sulfate hydrate (AG 348 sulfate hydrate) is a pyruvate kinase (PK) allosteric activator, used to study pyruvate kinase deficiency.Formule :C24H26N4O3S1H2SO43H2ODegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :526.66PGD-IN-S3
CAS :6PGD-IN-S3 (6PGD Inhibitor S3) is an inhibitor of 6-phosphogluconate dehydrogenase (6PGD).Formule :C15H10O4Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :254.24Enasidenib
CAS :Enasidenib (AG-221) is an orally available inhibitor of specific mutant forms of the mitochondrial enzyme isocitrate dehydrogenase type 2 (IDH2), with potentialFormule :C19H17F6N7ODegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :473.38Ref: TM-T2346
5mg44,00€10mg66,00€25mg87,00€50mg105,00€100mg137,00€200mg197,00€500mg333,00€1mL*10mM (DMSO)48,00€CHIKV-IN-2
CAS :CHIKV-IN-2 inhibits DHODH to thwart viruses like CHIKV by depleting pyrimidine, showing strong antiviral action (EC90=270 nM) and liver stability.Formule :C23H26N2O2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :362.46Ref: TM-T9394
1mg42,00€5mg94,00€10mg129,00€25mg221,00€50mg334,00€100mg485,00€200mg622,00€1mL*10mM (DMSO)94,00€Benzolamide
CAS :Benzolamide (CL 11366) inhibits carbonic anhydrase effectively and low-threshold calcium currents in hippocampal pyramidal neurons.Formule :C8H8N4O4S3Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :320.37Ref: TM-T23782
5mg49,00€10mg84,00€25mg152,00€50mg222,00€100mg331,00€200mg489,00€1mL*10mM (DMSO)54,00€Lofemizole
CAS :Lofemizole is an antagonist of CYP1A2.Formule :C10H9ClN2Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :192.64Ref: TM-T50053
1mg34,00€5mg71,00€10mg95,00€25mg161,00€50mg234,00€100mg331,00€200mg455,00€1mL*10mM (DMSO)60,00€amflutizole
CAS :Amflutizole used for the treatment of gout, and is a Xanthine oxidase inhibitor
Formule :C11H7F3N2O2SDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :288.246L(+)-Leucinol
CAS :L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase.Formule :C6H15NODegré de pureté :98%Couleur et forme :Clear Colorless To Slightly Yellow LiquidMasse moléculaire :117.19RGX-104 hydrochloride
CAS :RGX-104 hydrochloride (SB742881) is a small molecule LXR agonist that regulates innate immunity using transcriptional activation of the ApoE gene.Formule :C34H34Cl2F3NO3Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :632.54BMS-986242
CAS :BMS-986242 is an orally active, potent and selective inhibitor of indoleamine-2,3-dioxygenase 1 (IDO1), and it can be used for the research of cancer.Formule :C24H24ClFN2ODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :410.91SU0268
CAS :SU0268 is a potent and specific 8-Oxoguanine DNA glycosylase 1 (OGG1) inhibitor.Formule :C26H25N3O4SDegré de pureté :99.97% - 99.98%Couleur et forme :SolidMasse moléculaire :475.56Polmacoxib
CAS :Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.Formule :C18H16FNO4SDegré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :361.39Ref: TM-T21294
2mg47,00€5mg70,00€10mg107,00€25mg173,00€50mg259,00€100mg378,00€200mg563,00€1mL*10mM (DMSO)77,00€DMOG
CAS :DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.
Formule :C6H9NO5Degré de pureté :80.23% - 99.98%Couleur et forme :SolidMasse moléculaire :175.14MK-8617
CAS :MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).
Formule :C24H21N5O4Degré de pureté :99.38% - >99.99%Couleur et forme :SolidMasse moléculaire :443.45Trandolapril
CAS :Trandolapril is an orally administered angiotensin converting enzyme (ACE) inhibitor that is hydrolysed to the active diacid trandolaprilat.Formule :C24H34N2O5Degré de pureté :99.70% - 99.83%Couleur et forme :White PowderMasse moléculaire :430.54Ref: TM-T5329
5mg44,00€10mg66,00€25mg107,00€50mg177,00€100mg281,00€200mg421,00€500mg677,00€1mL*10mM (DMSO)73,00€(E)-3PO
CAS :(E)-3PO is a PFKFB3 (6-phosphofructo-2-kinase/fructose-2, 6-bisphosphatase) inhibitor.Formule :C13H10N2ODegré de pureté :98.8% - 98.92%Couleur et forme :SolidMasse moléculaire :210.23TOFA
CAS :TOFA (MDL14514) is an allosteric inhibitor of acetyl-CoA carboxylase-α (ACCA).Formule :C19H32O4Degré de pureté :97.52% - 98.98%Couleur et forme :SolidMasse moléculaire :324.45Imidapril
CAS :Imidapril: oral ACE & MMP-9 inhibitor, lowers blood pressure, useful in hypertension, diabetic nephropathy, heart failure.Formule :C20H27N3O6Couleur et forme :SolidMasse moléculaire :405.44CALP2 acetate(261969-04-4 free base)
CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.Formule :C68H104N14O13SDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :1357.7Des(benzylpyridyl) Atazanavi
CAS :The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.Formule :C26H43N5O7Degré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :537.65ND-646
CAS :ND-646 is an orally bioavailable and allosteric inhibitor of the ACC enzymes ACC1 and ACC2(IC50s of 3.5 nM and 4.1 nM for recombinant hACC1 and hACC2,Formule :C28H32N4O7SDegré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :568.64Ref: TM-TQ0243
1mg62,00€5mg177,00€10mg289,00€25mg492,00€50mg708,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)222,00€Atglistatin
CAS :Atglistatin: ATGL inhibitor, IC50 ~0.7 μM, inhibits lipolysis, non-toxic up to 50 μM.Formule :C17H21N3ODegré de pureté :97.2% - 99.01%Couleur et forme :SolidMasse moléculaire :283.37Ref: TM-T1875
2mg38,00€5mg57,00€10mg98,00€25mg178,00€50mg333,00€100mg525,00€500mg1.125,00€1mL*10mM (DMSO)63,00€L-Alanine
CAS :L-Alanine (L-2-Aminopropionic acid) is an Amino Acid. Alanine is involved in the metabolism of tryptophan and vitamin pyridoxine.Formule :C3H7NO2Degré de pureté :99.83%Couleur et forme :Orthorhombic Crystals From Water SolidMasse moléculaire :89.09Sephin1
CAS :Sephin1 (IFB-088) is reportedly a selective inhibitor of GADD34 (PPP1R15A), which is a stress-induced regulatory subunit of protein phosphatase 1 complex thatFormule :C8H9ClN4Degré de pureté :99.24% - 99.78%Couleur et forme :SolidMasse moléculaire :196.64AMG-3969
CAS :AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).Formule :C21H20F6N4O3SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :522.46Ref: TM-TQ0055
1mg52,00€5mg111,00€10mg172,00€25mg289,00€50mg399,00€100mg532,00€200mg740,00€1mL*10mM (DMSO)131,00€Fosfructose
CAS :D-fructose-1,6-diphosphate (D-fructose-1,6-diphosphate), also known as Fosfructose, is a cytoprotective natural sugar phosphate.Formule :C6H14O12P2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :340.12MAGL-IN-4
CAS :MAGL-IN-4 (His121 ARG57) is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.Formule :C18H21ClN2O4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :364.82Ref: TM-T9687
1mg140,00€5mg344,00€10mg512,00€25mg848,00€50mg1.121,00€100mg1.510,00€1mL*10mM (DMSO)373,00€MCU-i4
CAS :MCU-i4 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formule :C23H27N3O2Degré de pureté :99.45% - 99.98%Couleur et forme :SolidMasse moléculaire :377.482-Deoxy-2-sulfoamino-D-glucose sodium
CAS :2-Deoxy-2-sulfoamino-D-glucose sodium (GlcN-2S) is possible to effect reaction at arthritis.Formule :C6H12NNaO8SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :281.22GW1929
CAS :GW1929 is a potent PPAR-γ agonist (pKi: 8.84 for human PPAR-γ; pEC50s of 8.56 and 8.27 for human and murine PPAR-γ).
Formule :C30H29N3O4Degré de pureté :98.1% - 98.21%Couleur et forme :SolidMasse moléculaire :495.572-Hydroxy-3-methylbutanoic acid
CAS :2-Hydroxy-3-methylbutanoic acid ((±)-2-Hydroxyisopentanoic Acid) is a metabolite found in the urine of patients with phenylketonuria, methylmalonic acidemia.Formule :C5H10O3Degré de pureté :98% - 98.63%Couleur et forme :SolidMasse moléculaire :118.13KL-11743
CAS :KL-11743 blocks glucose metabolism, collapses NADH, and increases aspartate, shifting cells to oxidative phosphorylation.Formule :C30H30N6O3Degré de pureté :98.46% - 99.57%Couleur et forme :SolidMasse moléculaire :522.6Ref: TM-T9558
1mg113,00€5mg235,00€10mg378,00€25mg630,00€50mg898,00€100mg1.216,00€1mL*10mM (DMSO)269,00€Nifursol
CAS :Nifursol is a livestock feed additive and antiobiotic used to prevent the growth of histomonas.Formule :C12H7N5O9Degré de pureté :97.18%Masse moléculaire :365.21Mephenytoin
CAS :Mephenytoin (Phenantoin) is an anticonvulsant and a substrate of CYP2C19 and CYP2B6.Formule :C12H14N2O2Degré de pureté :99.67% - 99.91%Couleur et forme :Crystals SolidMasse moléculaire :218.25Ref: TM-T21425
1mg43,00€2mg57,00€5mg93,00€10mg131,00€25mg168,00€50mg215,00€100mg320,00€1mL*10mM (DMSO)115,00€Droxicainide hydrochloride
CAS :Tecicani hydrochloride is a new antiarrhythmic drug.Formule :C16H25ClN2O2Couleur et forme :SolidMasse moléculaire :312.83Raphin1 acetate
CAS :Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor.Formule :C10H12Cl2N4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :291.13Olesoxime
CAS :Olesoxime (TRO 19622) (TRO19622), A Mitochondrial-Targeted Neuroprotective Compound,is an experimental neuroprotective drug.Formule :C27H45NODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :399.65HA 155
CAS :HA 155 (Autotaxin Inhibitor IV) is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.Formule :C24H19BFNO5SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :463.29SEP-0372814
CAS :SEP-0372814 is a potent inhibitor of PDE10.Formule :C21H19N7Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :369.42Ref: TM-T8454
1mg62,00€5mg123,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)136,00€(E/Z)-GO289
CAS :(E/Z)-GO289, which strongly lengthened circadian period, is a potent and selective inhibitor of CK2.Formule :C17H15BrN4O2SDegré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :419.3Ref: TM-T9356
2mg34,00€5mg52,00€10mg86,00€25mg170,00€50mg250,00€100mg354,00€200mg482,00€1mL*10mM (DMSO)54,00€KML29
CAS :KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.Formule :C24H21F6NO7Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :549.42UNC6934
CAS :UNC6934 is a chemical probe targeting the N-terminal PWWP (PWWP1) domain of NSD2.Formule :C24H21N5O4Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :443.45Ref: TM-T9584
1mg47,00€5mg92,00€10mg152,00€25mg326,00€50mg485,00€100mg670,00€200mg888,00€1mL*10mM (DMSO)101,00€γ-Glu-Phe TFA(7432-24-8 free base)
γ-Glu-Phe TFA(7432-24-8 free base) is a dipeptide composed of gamma-glutamate and phenylalanine and is a proteolytic breakdown product of larger proteins.
Formule :C16H19F3N2O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :408.33Lazabemide hydrochloride
CAS :Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki：7.9nM).Formule :C8H11Cl2N3ODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :236.098KY-226
CAS :KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,)Formule :C27H31NO3S2Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :481.67Vesnarinone
CAS :Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFormule :C22H25N3O4Degré de pureté :96.69% - 98.13%Couleur et forme :SolidMasse moléculaire :395.45Ref: TM-T3465
2mg34,00€5mg50,00€10mg75,00€25mg111,00€100mg296,00€200mg427,00€1mL*5mM (DMSO)47,00€50mg*5mM (DMSO)198,00€Bendazac L-lysine
CAS :Bendazac L-lysine (Bendazaco lisina) is an agent introduced for the management of cataracts, protecting the level of vision in patients.Formule :C22H28N4O5Degré de pureté :99.85%Couleur et forme :WhiteMasse moléculaire :428.48Fluxapyroxad
CAS :Fluxapyroxad is a broad-spectrum fungicide that inhibits the succinate dehydrogenase (SQR) enzyme.Formule :C18H12F5N3ODegré de pureté :99.15% - 99.89%Couleur et forme :SolidMasse moléculaire :381.30JNJ-42041935
CAS :JNJ-42041935 (HIF-PHD Inhibitor II) is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes.Formule :C12H6ClF3N4O3Degré de pureté :99.58% - ≥95%Couleur et forme :SolidMasse moléculaire :346.65Ref: TM-T3180
1mg40,00€2mg52,00€5mg88,00€10mg119,00€25mg210,00€50mg354,00€100mg567,00€500mg1.198,00€1mL*10mM (DMSO)87,00€SPI-112
CAS :SPI-112, the SPI-112 methyl ester analog, can inhibit cellular Shp2 PTP activity.Formule :C22H17FN4O5SDegré de pureté :97.51% - >99.99%Couleur et forme :SolidMasse moléculaire :468.46Bifemelane hydrochloride
CAS :Bifemelane hydrochloride is a MAO inhibitor
Formule :C18H23NO·HClDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :305.84AM-2394
CAS :AM-2394 is an effective and specific Glucokinase agonist (GKA, EC50: 60 nM), which catalyzes the phosphorylation of glucose to glucose-6-phosphate.Formule :C22H25N5O4Degré de pureté :99.01% - 99.62%Couleur et forme :SolidMasse moléculaire :423.46Ref: TM-T3312
2mg34,00€5mg49,00€10mg66,00€25mg105,00€50mg172,00€100mg264,00€200mg394,00€1mL*10mM (DMSO)50,00€RP-64477
CAS :RP-64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.Formule :C29H42N2O3SDegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :498.728-Azaadenosine
CAS :8-Azaadenosine inhibits ADAR1, blocks RNA editing, and reduces thyroid cancer cell proliferation and spread.Formule :C9H12N6O4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :268.23GSK 650394
CAS :GSK 650394 is an inhibitor of serum- and glucocorticoid-regulated kinases (SGK). GSK 650394 has antitumor activity. Cost-effective and quality-assured.Formule :C25H22N2O2Degré de pureté :97.46% - >99.99%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T2622
1mg38,00€2mg50,00€5mg84,00€10mg105,00€25mg197,00€50mg313,00€100mg447,00€200mg623,00€1mL*10mM (DMSO)93,00€4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
CAS :4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-Formule :C7H8F3N3O4S2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :319.28Pheneturide
CAS :Pheneturide (Benuride) is the ureide class, used to treat epilepsy, and is an anticonvulsant.Formule :C11H14N2O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :206.24Haloxyfop
CAS :(±)-Haloxyfop (Haloxyfop Acid) is a herbicide.Formule :C15H11ClF3NO4Degré de pureté :99.96% - >99.99%Couleur et forme :SolidMasse moléculaire :361.7Aramchol
CAS :Aramchol (C20-FABAC), a mix of arachidic & cholic acid, lessens cholesterol crystallization & dissolves crystals in bile.Formule :C44H79NO5Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :702.1CAY10650
CAS :CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Formule :C28H25NO6Degré de pureté :97.33%Couleur et forme :SolidMasse moléculaire :471.5Ref: TM-TQ0105
1mg49,00€5mg114,00€10mg172,00€25mg334,00€50mg467,00€100mg620,00€1mL*10mM (DMSO)118,00€lavendustin B
CAS :Lavendustin B inhibits Tyrosine Kinase and HIV-1 integrase-LEDGF/p75 interaction.Formule :C21H19NO5Degré de pureté :95.72%Couleur et forme :Off-White SolidMasse moléculaire :365.38Tofisopam
CAS :Tofisopam (Grandaxin) is a 2,3-benzodiazepine compound with anxiolytic activity that can be taken orally.Formule :C22H26N2O4Degré de pureté :99.84%Couleur et forme :White SolidMasse moléculaire :382.45Ref: TM-T34896
2mg39,00€5mg58,00€10mg88,00€25mg137,00€50mg200,00€100mg295,00€200mg442,00€1mL*10mM (DMSO)64,00€PSB-1491
CAS :PSB-1491 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 0.386 nM, >25000-fold selective versus MAO-A.Formule :C15H11Cl2N3ODegré de pureté :98.41% - 99.68%Couleur et forme :SolidMasse moléculaire :320.17YM-750
CAS :YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.Formule :C31H36N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :452.63Ref: TM-T23550
2mg38,00€5mg52,00€10mg90,00€25mg164,00€50mg259,00€100mg374,00€200mg545,00€1mL*10mM (DMSO)62,00€Fatostatin
CAS :Fatostatin inhibits SREBP-1/2 by binding to SCAP, blocking their ER-Golgi transport.Formule :C18H18N2SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :294.41Ref: TM-T9266
2mg34,00€5mg48,00€10mg70,00€25mg112,00€50mg182,00€100mg309,00€200mg465,00€1mL*10mM (DMSO)50,00€Enterostatin, human, mouse, rat acetate
Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.Formule :C23H40N8O8Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :556.61Icerguastat
CAS :Icerguastat (IFB-088) is a selective inhibitor of holophosphatase. Icerguastat selectively inhibited a regulatory subunit of protein phosphatase 1 in vivo.Formule :C8H9ClN4Degré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :196.64Amifostine sodium
CAS :Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formule :C5H15N2NaO3PSCouleur et forme :SolidMasse moléculaire :237.21CaMKP Inhibitor
CAS :CaMKP Inhibitor can inhibit CaMKP.Formule :C10H8NNaO7S2Degré de pureté :96.55% - 99.98%Couleur et forme :SolidMasse moléculaire :341.28Ref: TM-T2159
1mg39,00€5mg82,00€10mg120,00€25mg227,00€50mg334,00€100mg460,00€500mg1.035,00€1mL*10mM (DMSO)102,00€L-778123 Dihydrochloride
CAS :L-778123 blocks FPTase/GGPTase-I, halts Ki-Ras prenylation, has acceptable toxicity with radiotherapy in advanced pancreatic cancer.Formule :C22H22Cl3N5OCouleur et forme :SolidMasse moléculaire :478.802LB-60-OF61 hydrochloride
CAS :LB-60-OF61 hydrochloride is a potent NAMPT enzyme inhibitor with cytotoxic effects, targeting MYC-overexpressing cell lines.Formule :C29H31ClN6O2Couleur et forme :SolidMasse moléculaire :531.063,4, 5-trimethoxyphenylacetic acid
CAS :3,4,5-trimethoxyphenylacetic acid: used in organic synthesis, mainly for carboxyl group conversion.Formule :C11H14O5Degré de pureté :99.84%Couleur et forme :White Crystalline PowderMasse moléculaire :226.23ML348
CAS :ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Formule :C18H17ClF3N3O3Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :415.79Ref: TM-T3439
2mg44,00€5mg65,00€10mg92,00€25mg215,00€50mg334,00€100mg537,00€200mg750,00€500mg1.134,00€Liquiritin
CAS :Liquiritin (Liquiritigenin-4'-O-glucoside) (LIQ) is a main component among the licorice flavonoids, and possesses anti-inflammatory and anti-cancer abilities.Formule :C21H22O9Degré de pureté :98.16% - 98.66%Couleur et forme :SolidMasse moléculaire :418.39Fmoc-Gly-Thr(psi(Me,Me)pro)-OH
CAS :Fmoc-Gly-Thr(psi(Me,Me)pro)-OH is a polypeptide composed of two amino acids.Formule :C24H26N2O6Degré de pureté :97.35%Couleur et forme :SolidMasse moléculaire :438.47PT-2385
CAS :PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).Formule :C17H12F3NO4SDegré de pureté :98.91% - 99.55%Couleur et forme :SolidMasse moléculaire :383.34Ref: TM-T7848
1mg63,00€2mg93,00€5mg144,00€10mg222,00€25mg379,00€50mg532,00€100mg740,00€200mg982,00€1mL*10mM (DMSO)119,00€Uniconazole
CAS :Uniconazole is a plant growth regulator that inhibit cytochrome P450 707As (Ki=68 nM).Formule :C15H18ClN3ODegré de pureté :99.94%Couleur et forme :White-Light Brown CrystallineMasse moléculaire :291.782-Phenylglycine
CAS :2-Phenylglycine (DL-α-Phenylglycine) is a metabolite in breast milk during the lactation period.Formule :C8H9NO2Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :151.16Ziritaxestat
CAS :Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.Formule :C30H33FN8O2SDegré de pureté :97% - 99.85%Couleur et forme :SolidMasse moléculaire :588.7Norathiol
CAS :Norathiol (N-methyl-N-dithiocarboxyglucamine) is a metal chelator that promotes the excretion of 109Cd and may be used in the treatment of cadmium poisoning.Formule :C8H17NO5S2Couleur et forme :SolidMasse moléculaire :271.35IBMX
CAS :IBMX (Methylisobutylxanthine) is a broad-spectrum phosphodiesterase (PDE) inhibitor with inhibitory activity against PDE3, PDE4, and PDE5 (IC50=6.5/26.3/31.7 μM
Formule :C10H14N4O2Degré de pureté :98% - >99.99%Couleur et forme :Off-WhiteMasse moléculaire :222.24Taselisib
CAS :Taselisib (GDC-0032) is an oral PI3K alpha inhibitor with potential cancer-treating properties.Formule :C24H28N8O2Degré de pureté :99.62% - 99.79%Couleur et forme :SolidMasse moléculaire :460.53Ref: TM-T1999
2mg46,00€5mg66,00€10mg92,00€25mg157,00€50mg197,00€100mg350,00€200mg522,00€500mg840,00€1mL*10mM (DMSO)66,00€Varespladib
CAS :Varespladib (LY315920) inhibits hnsPLA2 effectively (IC50=7 nM), studied for sickle cell, VOC, and acute coronary syndrome.Formule :C21H20N2O5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :380.39Ref: TM-T2044
1mg46,00€5mg87,00€10mg144,00€25mg227,00€50mg338,00€100mg487,00€200mg705,00€1mL*10mM (DMSO)81,00€Furafylline
CAS :Furafylline is a selective inhibitor of human cytochrome P450 (CYP)1A2 (IC50 : 0.07 μM),Formule :C12H12N4O3Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :260.25Ref: TM-T7410
1mg119,00€5mg235,00€10mg349,00€25mg593,00€50mg832,00€100mg1.159,00€200mg1.568,00€1mL*10mM (DMSO)268,00€SR1001
CAS :SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).Formule :C15H13F6N3O4S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :477.421-deacetyldeflazacort
CAS :21-deacetyldeflazacort is a metabolite of Deflazacort, which is a systemic corticosteroid and a derivative of prednisolone.Formule :C23H29NO5Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :399.48Cyclo(his-pro)
CAS :Cyclo(his-pro) is a cyclic dipeptide that shields against oxidative damage by activating Nrf2.Formule :C11H14N4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :234.25Brinzolamide hydrochloride
Brinzolamide (AL-4862) HCl selectively inhibits carbonic anhydrase II, reducing IOP for glaucoma research. IC50: 3.2 nM.Couleur et forme :Solid
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