Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(196 produits)
- Caséine Kinase(138 produits)
- DHFR(32 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(85 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(134 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(86 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(22 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(45 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9182 produits trouvés pour "Métabolisme"
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Colesevelam Hydrochloride
CAS :Colesevelam HCl is a bile acid sequestrant that reduces cholesterol by inhibiting bile reabsorption.Formule :C31H67Cl3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :618.25Enoximone
CAS :Enoximone is a selective inhibitor of phosphodiesterase III (PDE3), with treatment of congestive heart failure.Formule :C12H12N2O2SDegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :248.3THPP-1
CAS :THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 nM for human and rat PDE10A, respectively).Formule :C23H21ClN6O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :464.9Tetrindole mesylate
CAS :Tetrindole mesylate is a MAO-A inhibitor.Formule :C21H30N2O3SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :390.54NCT-505
CAS :NCT-505 is a potent and selective inhibitor of aldehyde dehydrogenase (ALDH1A1, IC50 = 7 nM) and a weak inhibitor of hALDH1A2, hALDH1A3, hALDH2, hALDH3A1 withFormule :C27H28FN5O3SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :521.61Ref: TM-T12196
1mg115,00€5mg235,00€10mg353,00€25mg562,00€50mg758,00€100mg1.017,00€200mg1.359,00€1mL*10mM (DMSO)270,00€1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine
CAS :1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.Formule :C46H84NO8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :810.13AGI-6780
CAS :AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.Formule :C21H18F3N3O3S2Degré de pureté :98.19% - 99.7%Couleur et forme :SolidMasse moléculaire :481.51Ref: TM-T1809
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg220,00€50mg393,00€100mg587,00€500mg1.264,00€1mL*10mM (DMSO)85,00€MAGL-IN-4
CAS :MAGL-IN-4 (His121 ARG57) is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.Formule :C18H21ClN2O4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :364.82Ref: TM-T9687
1mg140,00€5mg344,00€10mg512,00€25mg848,00€50mg1.121,00€100mg1.510,00€1mL*10mM (DMSO)373,00€Dichlorphenamide disodium
CAS :Dichlorphenamide disodium: an oral carbonic anhydrase inhibitor that lowers eye pressure, promising for glaucoma study.Formule :C6H6Cl2N2Na2O4S2Couleur et forme :SolidMasse moléculaire :351.12NP118809
CAS :NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).
Formule :C32H32N2ODegré de pureté :97.74% - 98.68%Couleur et forme :SolidMasse moléculaire :460.61Tienilic Acid
CAS :Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
Formule :C13H8Cl2O4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :331.17PFK-015
CAS :PFK-015 (PFK15) is an effective inhibitor of PFKFB3 (IC50: 110 nM) and inhibits PFKFB3 activity in Y cells (IC50: 20 nM).Formule :C17H12N2ODegré de pureté :99.7% - 99.85%Couleur et forme :SolidMasse moléculaire :260.29Ref: TM-T2455
2mg40,00€5mg57,00€10mg88,00€25mg159,00€50mg250,00€100mg376,00€200mg550,00€1mL*10mM (DMSO)57,00€GSK805
CAS :GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.
Formule :C23H18Cl2F3NO4SDegré de pureté :98% - ≥95%Couleur et forme :SolidMasse moléculaire :532.367-Hydroxy-3,4-dihydro-2(1H)-quinolinone
CAS :7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .Formule :C9H9NO2Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :163.17MCU-i4
CAS :MCU-i4 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formule :C23H27N3O2Degré de pureté :99.45% - 99.98%Couleur et forme :SolidMasse moléculaire :377.48FEMA 4774
CAS :FEMA 4774 (S9632) is a positive allosteric modulator of T1R2/T1R3. FEMA4774 shows obvious enhancement of the sweetness of sucrose in sensory evaluation tests
Formule :C19H25N3O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :359.42Fluvastatin potassium
CAS :Fluvastatin, a synthetic statin, lowers cholesterol and prevents heart disease.Formule :C24H25FKNO4Couleur et forme :SolidMasse moléculaire :449.56PNU-100440
CAS :PNU-100440 is a biologically active compound. It is an intermediate in the synthesis of linezolid dimers, an impurity of the antibacterial agent Linezolid.Formule :C14H17FN2O4Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :296.292-Bromo-4'-hydroxyacetophenone
CAS :2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).
Formule :C8H7BrO2Degré de pureté :98.64%Couleur et forme :Clear Colorless To Light Yellow LiquidMasse moléculaire :215.04Telaglenastat
CAS :Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.Formule :C26H24F3N7O3SDegré de pureté :97.57% - 99.89%Couleur et forme :SolidMasse moléculaire :571.57Ref: TM-T6797
1g1.130,00€2mg38,00€5mg51,00€10mg79,00€25mg126,00€50mg210,00€100mg350,00€500mg825,00€1mL*10mM (DMSO)65,00€NCC007
CAS :NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.Formule :C22H28F3N7Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :447.5Rolipram
CAS :Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Formule :C16H21NO3Degré de pureté :99.22% - >99.99%Couleur et forme :SolidMasse moléculaire :275.34Nampt-IN-1
CAS :Nampt-IN-1 (LSN3154567) (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM.Formule :C20H25N3O5SDegré de pureté :99.28% - 99.4%Couleur et forme :SolidMasse moléculaire :419.49Ref: TM-T4376
1mg37,00€2mg49,00€5mg79,00€10mg130,00€25mg245,00€50mg409,00€100mg605,00€1mL*10mM (DMSO)87,00€TBA-7371
CAS :TBA-7371 (DprE1-IN-1) is a potent inhibitor of DprE1 and PDE6.Formule :C18H21N5O3Degré de pureté :99% - 99.54%Couleur et forme :SolidMasse moléculaire :355.39BMS-986242
CAS :BMS-986242 is an orally active, potent and selective inhibitor of indoleamine-2,3-dioxygenase 1 (IDO1), and it can be used for the research of cancer.Formule :C24H24ClFN2ODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :410.91PQ-10
CAS :PQ-10 (A-844337) is a PDE-10 inhibitor. PQ-10 induces brain glucose metabolism patterns, which may be a potential translational biomarker.
Formule :C22H21N5O3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :403.43SR1001
CAS :SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).Formule :C15H13F6N3O4S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :477.4CP-640186 hydrochloride
CAS :CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat
Formule :C30H36ClN3O3Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :522.08Edoxaban Tosylate Monohydrate
CAS :Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.Formule :C31H40ClN7O8S2Degré de pureté :99.86% - 99.91%Couleur et forme :SolidMasse moléculaire :738.27Pargyline
CAS :Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.Formule :C11H13NDegré de pureté :95.64% - 97.21%Couleur et forme :SolidMasse moléculaire :159.23Fondaparinux sodium
CAS :Fondaparinux sodium (SR-90107A) is an antithrombin-dependent factor Xa inhibitor with antithrombotic activity.Formule :C31H43N3Na10O49S8Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :1728.08HNHA
CAS :HNHA is an inhibitor of HDAC.Formule :C17H21NO2SDegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :303.42Ref: TM-T21806
1mg44,00€5mg84,00€10mg135,00€25mg279,00€50mg445,00€100mg640,00€200mg879,00€1mL*10mM (DMSO)90,00€FOY 251
CAS :FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.Formule :C17H19N3O7SDegré de pureté :97.11% - 99.33%Couleur et forme :SolidMasse moléculaire :409.41Ref: TM-T8676
1mg51,00€5mg110,00€10mg177,00€25mg300,00€50mg424,00€100mg605,00€500mg1.198,00€1mL*10mM (DMSO)126,00€Dimethylfraxetin
CAS :Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki：0.0097 μM)Formule :C12H12O5Degré de pureté :99.96% - ≥95%Couleur et forme :SolidMasse moléculaire :236.22EMD638683
CAS :EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).Formule :C18H18F2N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.34Ref: TM-T6635
1mg74,00€2mg92,00€5mg150,00€10mg233,00€25mg358,00€50mg517,00€100mg737,00€200mg982,00€1mL*10mM (DMSO)120,00€Rosiptor
CAS :Rosiptor (AQX-1125) (AQX-1125) is an orally-active and specific phosphatase SHIP1 activator with anti-inflammatory effects.Formule :C20H35NO2Degré de pureté :99.53% - 99.73%Couleur et forme :SolidMasse moléculaire :321.5HA 155
CAS :HA 155 (Autotaxin Inhibitor IV) is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.Formule :C24H19BFNO5SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :463.29Roflumilast N-oxide
CAS :Roflumilast N-oxide is an inhibitor of PDE type 4.Formule :C17H14Cl2F2N2O4Degré de pureté :98.19% - 99.69%Couleur et forme :SolidMasse moléculaire :419.21Ref: TM-T4462
1mg35,00€2mg52,00€5mg74,00€10mg99,00€25mg170,00€50mg274,00€100mg350,00€500mg840,00€1mL*10mM (DMSO)69,00€Melilotic acid
CAS :3-(2-Hydroxyphenyl)propanoic acid, aka melilotic acid, found in cytoplasm, in foods like herbs, beetroot, cinnamon.Formule :C9H10O3Degré de pureté :99.65% - 99.83%Couleur et forme :SolidMasse moléculaire :166.17PD 128042
CAS :PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formule :C23H39NO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.56KML29
CAS :KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.Formule :C24H21F6NO7Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :549.42PfDHODH-IN-2
CAS :PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.Formule :C13H12ClNO3SDegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :297.76Ref: TM-T8767
1mg46,00€5mg92,00€10mg138,00€25mg245,00€50mg363,00€100mg515,00€200mg702,00€1mL*10mM (DMSO)100,00€BI-0115
CAS :BI-0115 inhibits LOX-1, preventing oxLDL uptake by triggering receptor inhibition and dimer formation.Formule :C15H14ClN3ODegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :287.74Minaprine dihydrochloride
CAS :Minaprine dihydrochloride: reversible MAO-A inhibitor, mild on acetylcholinesterase, used for depression.Formule :C17H24Cl2N4ODegré de pureté :99.43% - 99.99%Couleur et forme :SolidMasse moléculaire :371.3Tipifarnib
CAS :Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Formule :C27H22Cl2N4ODegré de pureté :97.1% - 99.22%Couleur et forme :Off-White To Pale Beige SolidMasse moléculaire :489.4Thiorphan
CAS :Thiorphan is an neprilysin inhibitor (NEP; IC50 : 0.007 μM).Formule :C12H15NO3SDegré de pureté :99.33%Couleur et forme :Off-White SolidMasse moléculaire :253.32Ref: TM-T7693
2mg35,00€5mg52,00€10mg93,00€25mg170,00€50mg255,00€100mg379,00€500mg870,00€1mL*10mM (DMSO)58,00€Pentamidine isethionate
CAS :Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.
Formule :C23H36N4O10S2Degré de pureté :98% - 99.83%Couleur et forme :Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)Masse moléculaire :592.68UCPH-101
CAS :UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Formule :C27H22N2O3Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :422.48Ref: TM-T4138
1mg50,00€2mg75,00€5mg130,00€10mg203,00€25mg409,00€50mg655,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)142,00€Evacetrapib
CAS :Evacetrapib (LY2484595) inhibits CETP strongly (IC50=5.5 nM), raises HDL cholesterol, no rise in aldosterone/blood pressure. Phase 3.Formule :C31H36F6N6O2Degré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :638.65AGI-5198
CAS :AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).Formule :C27H31FN4O2Degré de pureté :97.37% - 99.23%Couleur et forme :SolidMasse moléculaire :462.56Copper tripeptide
CAS :GHK-Cu is a copper complex with the peptide glycyl-L-histidyl-L-lysine, found in human plasma, saliva, and urine.Formule :C14H22CuN6O4Degré de pureté :99.94% - >99.99%Couleur et forme :SolidMasse moléculaire :401.91Ethyl 3,4-dihydroxybenzoate
CAS :Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.Formule :C9H10O4Degré de pureté :99.88%Couleur et forme :White Crystal Or PowderMasse moléculaire :182.17JNJ-42165279
CAS :JNJ-42165279 selectively inactivates FAAH without notably affecting other enzymes, ion channels, receptors, or CYPs/hERG at 10 μM.Formule :C18H17ClF2N4O3Degré de pureté :99.67% - 99.88%Couleur et forme :SolidMasse moléculaire :410.8Ref: TM-T3215
2mg46,00€5mg65,00€10mg96,00€25mg170,00€50mg246,00€100mg363,00€200mg512,00€1mL*10mM (DMSO)75,00€Nequinate
CAS :Nequinate is an anticoccidial agent, preventing coccidiosis .
Formule :C22H23NO4Degré de pureté :96.43%Couleur et forme :Light Yellow Odorless PowderMasse moléculaire :365.42amflutizole
CAS :Amflutizole used for the treatment of gout, and is a Xanthine oxidase inhibitor
Formule :C11H7F3N2O2SDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :288.246Dorzolamide hydrochloride
CAS :Dorzolamide hydrochloride (MK507 hydrochloride) is the hydrochloride salt form of dorzolamide, an inhibitor of carbonic anhydrase, a zinc-containing enzyme thatFormule :C10H17ClN2O4S3Degré de pureté :99.48% - 99.67%Couleur et forme :White Off-White Crystalline PowderMasse moléculaire :360.9DG051
CAS :DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).Formule :C21H25Cl2NO4Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :426.33Ref: TM-TQ0047
2mg37,00€5mg74,00€10mg116,00€25mg239,00€50mg380,00€100mg610,00€200mg815,00€1mL*10mM (DMSO)84,00€FG-2216
CAS :FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.Formule :C12H9ClN2O4Degré de pureté :97.1% - >99.99%Couleur et forme :SolidMasse moléculaire :280.66Eprobemide
CAS :Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).Formule :C14H19ClN2O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :282.77D-Histidine
CAS :D-Histidine is an enantiomer of L-histidine. L-Histidine is an inhibitor of mitochondrial glutamine transport and also an essential amino acid for infants.
Formule :C6H9N3O2Degré de pureté :99.57%Couleur et forme :White Crystalline PowderMasse moléculaire :155.15JZL 184
CAS :JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.Formule :C27H24N2O9Degré de pureté :97.56% - 99.31%Couleur et forme :SolidMasse moléculaire :520.49LMPTP INHIBITOR 1 dihydrochloride
CAS :LMPTP Inhibitor 1 Dihydrochloride is a compound selectively targeting low molecular weight protein tyrosine phosphatase (LMPTP), exhibiting potent inhibitoryFormule :C28H38Cl2N4ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :517.53Ref: TM-T41298
1mg73,00€5mg160,00€10mg250,00€25mg465,00€50mg673,00€100mg945,00€200mg1.251,00€1mL*10mM (DMSO)178,00€2-Phenylglycine
CAS :2-Phenylglycine (DL-α-Phenylglycine) is a metabolite in breast milk during the lactation period.Formule :C8H9NO2Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :151.16RP-64477
CAS :RP-64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.Formule :C29H42N2O3SDegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :498.72Vardenafil hydrochloride
CAS :Vardenafil hydrochloride is a New Phosphodiesterase Type 5(PDE5) Inhibitor, in the Treatment of Erectile Dysfunction in Men With DiabetesFormule :C23H33ClN6O4SDegré de pureté :99.76% - 99.94%Couleur et forme :White To Off-White Cyrstalline SolidMasse moléculaire :525.068-Azaadenosine
CAS :8-Azaadenosine inhibits ADAR1, blocks RNA editing, and reduces thyroid cancer cell proliferation and spread.Formule :C9H12N6O4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :268.234-Nonylphenylboronic acid
CAS :4-Nonylphenylboronic acid is a inhibitor of FAAH.
Formule :C15H25BO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :248.174-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
CAS :4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-Formule :C7H8F3N3O4S2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :319.28Tropifexor
CAS :Tropifexor (LJN452) is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM.
Formule :C29H25F4N3O5SDegré de pureté :99.3% - 99.85%Couleur et forme :SolidMasse moléculaire :603.58Ref: TM-T4379
1mg87,00€5mg166,00€10mg248,00€25mg437,00€50mg665,00€100mg1.008,00€200mg1.520,00€500mg2.252,00€RGX-104
CAS :RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)Formule :C34H33ClF3NO3Degré de pureté :98.79% - 99.53%Couleur et forme :SolidMasse moléculaire :596.08Ref: TM-T7768
1mg38,00€5mg92,00€10mg145,00€25mg281,00€50mg447,00€100mg688,00€200mg964,00€1mL*10mM (DMSO)119,00€WIN 18446
CAS :inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)Formule :C12H20Cl4N2O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :366.11YM-750
CAS :YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.Formule :C31H36N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :452.63Ref: TM-T23550
2mg38,00€5mg52,00€10mg90,00€25mg164,00€50mg259,00€100mg374,00€200mg545,00€1mL*10mM (DMSO)62,00€Lomitapide
CAS :Lomitapide (AEGR-733) blocks MTP, a key enzyme in dietary lipid absorption and VLDL assembly.Formule :C39H37F6N3O2Degré de pureté :98.91% - 99.40%Couleur et forme :SolidMasse moléculaire :693.72Ref: TM-T6267
2mg62,00€5mg89,00€10mg138,00€25mg219,00€50mg314,00€100mg472,00€200mg678,00€500mg1.044,00€1mL*10mM (DMSO)153,00€2-Hydroxy-3-methylbutanoic acid
CAS :2-Hydroxy-3-methylbutanoic acid ((±)-2-Hydroxyisopentanoic Acid) is a metabolite found in the urine of patients with phenylketonuria, methylmalonic acidemia.Formule :C5H10O3Degré de pureté :98% - 98.63%Couleur et forme :SolidMasse moléculaire :118.13Epacadostat
CAS :Epacadostat (INCB 024360) is an oral, potent and selective IDO1 inhibitor with IC50 value of 71.8 nM.Cost-effective and quality-assured.Formule :C11H13BrFN7O4SDegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :438.23Ref: TM-T3548
1g757,00€2g1.035,00€5mg47,00€10mg70,00€25mg87,00€50mg111,00€100mg187,00€200mg311,00€500mg525,00€1mL*10mM (DMSO)50,00€MY-5445
CAS :MY-5445 (N-(3-chlorophenyl)-4-phenylphthalazin-1-amine) is a specific inhibitor of phosphodiesterase type 5 (PDE5).
Formule :C20H14ClN3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :331.8GOT1 inhibitor-1
CAS :GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.Formule :C19H19ClN4ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :354.83Ref: TM-T8766
1mg87,00€5mg177,00€10mg295,00€25mg502,00€50mg710,00€100mg1.009,00€1mL*10mM (DMSO)203,00€Genz-123346 free base
CAS :Genz 123346 is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1.Formule :C24H38N2O4Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :418.57(2R)-3-(((2-Aminoethoxy)(hydroxy)phosphoryl)oxy)propane-1,2-diyl ditetradecanoate
CAS :(2R)-3-(((2-Aminoethoxy)(hydroxy)phosphoryl)oxy)propane-1,2-diyl ditetradecanoate (DMPE) is a phosphatidylethanolamine (PE or GPEtn).Formule :C33H66NO8PDegré de pureté :99.46% - ≥95%Couleur et forme :SolidMasse moléculaire :635.85Paricalcitol
CAS :Paricalcitol is a vitamin D receptor agonist.Formule :C27H44O3Degré de pureté :98.59% - 99.84%Couleur et forme :SolidMasse moléculaire :416.64Sacubitrilat
CAS :Sacubitrilat (LBQ-657) (LBQ657) is an effective inhibitor of active neprilysin (NEP).Formule :C22H25NO5Degré de pureté :99.17% - 99.89%Couleur et forme :SolidMasse moléculaire :383.44Ref: TM-TQ0106
1mg48,00€2mg63,00€5mg96,00€10mg160,00€25mg344,00€50mg550,00€100mg792,00€500mg1.605,00€1mL*10mM (DMSO)96,00€AMG-208
CAS :AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.Formule :C22H17N5O2Degré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :383.4BAY-1436032
CAS :BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).Formule :C26H30F3N3O3Degré de pureté :99.65% - 99.71%Couleur et forme :SolidMasse moléculaire :489.53JNJ-42041935
CAS :JNJ-42041935 (HIF-PHD Inhibitor II) is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes.Formule :C12H6ClF3N4O3Degré de pureté :99.58% - ≥95%Couleur et forme :SolidMasse moléculaire :346.65Ref: TM-T3180
1mg40,00€2mg52,00€5mg88,00€10mg119,00€25mg210,00€50mg354,00€100mg567,00€500mg1.198,00€1mL*10mM (DMSO)87,00€Clorgyline
CAS :Clorgyline,M&B 9302, an irreversible and selective MAO-A inhibitor with the advantages of oral activity and blood-brain barrier permeability, antidepressant.Formule :C13H15Cl2NODegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :272.17O-Succinylhomoserine
CAS :O-Succinylhomoserine (O-Succinyl-L-homoserine) is an intermediate in the synthesis of cystathionine by E coli..
Formule :C8H13NO6Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :219.19Dansylglycine
CAS :Dansylglycine is a fluorescent probe for specific determination of halogenating activity of myeloperoxidase and eosinophil peroxidase[1].Formule :C14H16N2O4SDegré de pureté :99.1%Couleur et forme :SolidMasse moléculaire :308.35SR3335
CAS :SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).Formule :C13H9F6NO3S2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :405.34Ref: TM-T5160
1mg34,00€5mg74,00€10mg119,00€25mg233,00€50mg371,00€100mg595,00€200mg833,00€1mL*10mM (DMSO)82,00€ML-211
CAS :ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)
Formule :C25H30N4O2Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :418.53AA26-9
CAS :AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Formule :C7H10N4ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :166.18Ref: TM-T3990
1mg34,00€2mg49,00€5mg74,00€10mg113,00€25mg200,00€50mg333,00€100mg495,00€1mL*10mM (DMSO)82,00€UDP-GlcNAc Disodium Salt
CAS :UDP-GlcNAc Disodium Salt (UDP-α-D-N-Acetylglucosamine Disodium Salt) is a nucleotide sugar.Formule :C17H25N3Na2O17P2Degré de pureté :97.11% - 99.22%Couleur et forme :White PowderMasse moléculaire :651.32Fmoc-N-Me-Ala-OH
CAS :Fmoc-N-Me-Ala-OH is available for the peptide-coupling reaction.Formule :C19H19NO4Degré de pureté :99.45%Couleur et forme :Cream-Colored PowderMasse moléculaire :325.36AZ876
CAS :AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.Formule :C24H29N3O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :439.57Zinc Phytate
CAS :Zinc Phytate, present in food, plays a crucial role in human nutrient absorption.Formule :C6H6O24P6Zn6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :10405-Nitro-1,10-phenanthroline
CAS :5-Nitro-1,10-phenanthroline (5-NP)(5-NP) is a potent bactericidal agent and inhibiting Clostridium difficile.Formule :C12H7N3O2Degré de pureté :97.42% - 99.5%Couleur et forme :Pale Yellow Or Brown SolidMasse moléculaire :225.2Zolamide
CAS :Zolamide (CL 5343) may be used to prevent altitude sickness and reduce the symptoms.Formule :C2H4N4O2S2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :180.21Nifursol
CAS :Nifursol is a livestock feed additive and antiobiotic used to prevent the growth of histomonas.Formule :C12H7N5O9Degré de pureté :97.18%Masse moléculaire :365.21Piclamilast
CAS :Piclamilast (RP 73401) is a PDE4 inhibitor.Formule :C18H18Cl2N2O3Degré de pureté :98.28% - 99.57%Couleur et forme :SolidMasse moléculaire :381.25FMoc-Arg(Tos)-OH
CAS :FMoc-Arg(Tos)-OH: Synthetic amino acid for solid-phase peptide synthesis, biochemistry, and molecular biology.Formule :C28H30N4O6SDegré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :550.63Amino Tadalafil
CAS :Amino tadalafil is a potent phosphodiesterase 5 (PDE5) inhibitor.Formule :C21H18N4O4Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :390.39Emtricitabine
CAS :Emtricitabine is a nucleoside reverse transcriptase inhibitor with anti-human immunodeficiency virus (HIV) and hepatitis B virus activity.Cost-effective and quality-assured.Formule :C8H10FN3O3SDegré de pureté :99.15% - 99.78%Couleur et forme :White PowderMasse moléculaire :247.25Navoximod
CAS :Navoximod (GDC-0919) (NLG- 919, GDC-0919) is a potent indoleamine-(2,3)-dioxygenase (IDO) pathway inhibitor (Ki/EC50: 7 nM/75 nM).Formule :C18H21FN2O2Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :316.37Ref: TM-TQ0071
1mg150,00€5mg313,00€10mg470,00€25mg600,00€50mg745,00€100mg1.044,00€1mL*10mM (DMSO)318,00€Phenprocoumon
CAS :Phenprocoumon is an antagonist of vitamin K(IC50:1 μM).Formule :C18H16O3Degré de pureté :95.79% - 97.98%Couleur et forme :Fine White Crystalline Powder SolidMasse moléculaire :280.32ST271
CAS :ST271 is an effective protein tyrosine kinase (PTK) inhibitor.
Formule :C16H20N2O2Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :272.34Tipifarnib (S enantiomer)
CAS :Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Formule :C27H22Cl2N4ODegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :489.4Ref: TM-T17102
1mg49,00€5mg102,00€10mg163,00€25mg284,00€50mg409,00€100mg577,00€200mg778,00€1mL*10mM (DMSO)109,00€trans-4-Hydroxycyclohexanecarboxylic Acid
CAS :trans-4-Hydroxycyclohexanecarboxylic Acid is an organic intermediate.Formule :C7H12O3Degré de pureté :96.24%Couleur et forme :SolidMasse moléculaire :144.17Isavuconazole
CAS :Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.Formule :C22H17F2N5OSDegré de pureté :99.74% - >99.99%Couleur et forme :SolidMasse moléculaire :437.47Ref: TM-T2305
1mg34,00€5mg73,00€10mg90,00€25mg166,00€50mg260,00€100mg356,00€200mg535,00€1mL*10mM (DMSO)81,00€LXR-623
CAS :LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.Formule :C21H12ClF5N2Degré de pureté :97.91% - 99.24%Couleur et forme :SolidMasse moléculaire :422.78Umbralisib
CAS :Umbralisib (TGR 1202) is a PI3Kδ inhibitor.Formule :C31H24F3N5O3Degré de pureté :99.56% - 99.56%Couleur et forme :White SolidMasse moléculaire :571.55Ref: TM-T4976
1mg48,00€2mg65,00€5mg96,00€10mg170,00€25mg343,00€50mg449,00€100mg658,00€1mL*10mM (DMSO)120,00€Inosine
CAS :Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!Formule :C10H12N4O5Degré de pureté :99.51% - 99.89%Couleur et forme :SolidMasse moléculaire :268.23LOX-IN-3 dihydrochloride
CAS :LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).Formule :C13H15Cl2FN2O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :353.24Ref: TM-T39986
1mg57,00€5mg120,00€10mg188,00€25mg354,00€50mg588,00€100mg938,00€200mg1.320,00€1mL*10mM (DMSO)127,00€Cobicistat
CAS :Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.Formule :C40H53N7O5S2Degré de pureté :97.36% - 99.62%Couleur et forme :SolidMasse moléculaire :776.02Ref: TM-T6246
1mg43,00€2mg56,00€5mg88,00€10mg117,00€25mg200,00€50mg333,00€100mg477,00€1mL*10mM (DMSO)105,00€Fomepizole
CAS :Fomepizole (4-Methylpyrazole), a competitive inhibitor of alcohol dehydrogenase, is used as an antidote in methanol or ethylene glycol poisoning.Formule :C4H6N2Degré de pureté :98.1% - 99.94%Couleur et forme :Yellow <13°C Solid >13°C LiquidMasse moléculaire :82.1Methyclothiazide
CAS :Methyclothiazide (Aquatensen) is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions includingFormule :C9H11Cl2N3O4S2Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :360.24H-Ser-His-OH acetate
H-Ser-His-OH acetate is an endogenous metabolite hydrolysis cleavage activity.Formule :C11H18N4O6Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :302.28Ref: TM-T11527L
5mg49,00€10mg63,00€25mg89,00€50mg130,00€100mg177,00€200mg281,00€500mg475,00€1mL*10mM (DMSO)56,00€ABX-1431
CAS :ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).Formule :C20H22F9N3O2Degré de pureté :99.8% - 99.96%Couleur et forme :SolidMasse moléculaire :507.39ML355
CAS :ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.
Formule :C21H19N3O4S2Degré de pureté :98.02% - 98.2%Couleur et forme :SolidMasse moléculaire :441.52RS-25344
CAS :RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.Formule :C19H13N5O4Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :375.34Ref: TM-T9239
1mg84,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€1mL*10mM (DMSO)177,00€ML351
CAS :ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).Formule :C15H11N3ODegré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :249.27Ref: TM-T21902
1mg50,00€5mg105,00€10mg167,00€25mg334,00€50mg505,00€100mg713,00€1mL*10mM (DMSO)117,00€Osoresnontrine
CAS :Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.Formule :C16H17N5O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :311.34Ref: TM-T8515
1mg38,00€2mg50,00€5mg81,00€10mg119,00€25mg188,00€50mg350,00€100mg522,00€200mg748,00€1mL*10mM (DMSO)89,00€VAS2870
CAS :VAS2870 is an inhibitor of NADPH oxidase (NOX).Formule :C18H12N6OSDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :360.39WWL70
CAS :WWL70 is a selective alpha/beta hydrolase domain 6 inhibitors (IC50: 70 nM).Formule :C27H23N3O3Degré de pureté :98.38% - 98.53%Couleur et forme :SolidMasse moléculaire :437.49Tuna AI acetate
Tuna AI acetate is an inhibitor of angiotensin-converting enzyme (ACE) in non-competitive manner derived from tuna muscle.Formule :C46H68N12O14Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :1013.1Ref: TM-T24906L
1mg115,00€2mg162,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)437,00€Imidazole-5-propionic acid
CAS :Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination.Formule :C6H8N2O2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :140.14Tryptophan, N-indol-3-ylacetyl- (6CI)
CAS :Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiologicalFormule :C21H19N3O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :361.42,3-dihydro-1H-indene-5-sulfonamide
CAS :2,3-dihydro-1H-indene-5-sulfonamide is Carbonic anhydrase 12 (human) inhibitor.Formule :C9H11NO2SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :197.25Ref: TM-T8611
1mg62,00€5mg123,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)104,00€Hydroxy Dimetridazole
CAS :Hydroxy Dimetridazole is a hydroxy metabolite of Dimetridazole which combats protozoan infections.
Formule :C5H7N3O3Degré de pureté :99.83% - 99.85%Couleur et forme :SolidMasse moléculaire :157.13Nicardipine
CAS :Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.Formule :C26H29N3O6Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :479.52Vorasidenib
CAS :Vorasidenib (PVM/MA) is an inhibitor of mutant isocitrate dehydrogenase (IDH; IC50s = 31.9 and 31.7 nM for IDH1R132H and IDH2R140Q, respectively)Formule :C14H13ClF6N6Degré de pureté :98.28% - 99.57%Couleur et forme :SolidMasse moléculaire :414.74Ref: TM-T7307
1mg50,00€2mg74,00€5mg113,00€10mg178,00€25mg340,00€50mg512,00€100mg733,00€1mL*10mM (DMSO)102,00€Enpp-1-IN-1
CAS :Enpp-1-IN-1 is an inhibitor of Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1)Formule :C17H17N3O3SDegré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :343.4Ref: TM-T7888
1mg126,00€5mg260,00€10mg394,00€25mg677,00€50mg954,00€100mg1.288,00€1mL*10mM (DMSO)286,00€Glutamyl-glutamic acid
CAS :Glutamyl-glutamic acid (Glu-glu) is an Interpeptide Bridge in the Murein of Some Micrococci and Arthrobacter sp..Formule :C10H16N2O7Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :276.24Calcineurin Autoinhibitory Peptide acetate
Calcineurin Autoinhibitory Peptide acetate is a selectivecalcineurin phosphatase inhibitor(IC50 ~ 10 μM).Formule :C252H417N78O82S4Degré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :5979.74Lotamilast
CAS :Lotamilast (RVT-501) is a phosphodiesterase 4 (PDE-4) inhibitor (IC50: 2.8 nM) potentially for the treatment of atopic dermatitis.Formule :C26H24N4O5Degré de pureté :97.03% - 99.29%Couleur et forme :SolidMasse moléculaire :472.49TMS
CAS :TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).Formule :C18H20O4Degré de pureté :99.17% - 99.73%Couleur et forme :SolidMasse moléculaire :300.35Calcitriol
CAS :Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM).
Formule :C27H44O3Degré de pureté :98.81% - 99.64%Couleur et forme :Colorless Crystalline Solid SolidMasse moléculaire :416.64(R)-GNE-140
CAS :(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.Formule :C25H23ClN2O3S2Degré de pureté :98.25% - 98.91%Couleur et forme :SolidMasse moléculaire :499.04DG172 dihydrochloride
CAS :DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).
Formule :C20H22BrCl2N3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :455.2Barnidipine
CAS :Barnidipine (YM-09730-5(Free base)) is a calcium channel blocker.Formule :C27H29N3O6Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :491.54Ref: TM-T7550
1mg46,00€2mg57,00€5mg89,00€10mg123,00€25mg230,00€50mg344,00€100mg520,00€1mL*10mM (DMSO)97,00€Firsocostat
CAS :Firsocostat (GS-0976) is an inhibitor of acetyl-CoA carboxylase (ACC) dimerization that inhibits human ACC1 and ACC2 activity (IC50s of 2.1 and 6.1 nM).Formule :C28H31N3O8SDegré de pureté :98% - 99.39%Couleur et forme :SolidMasse moléculaire :569.63Ref: TM-T7184
1mg96,00€2mg127,00€5mg210,00€10mg354,00€25mg510,00€50mg655,00€100mg908,00€500mg1.795,00€1mL*10mM (DMSO)265,00€Benzolamide
CAS :Benzolamide (CL 11366) inhibits carbonic anhydrase effectively and low-threshold calcium currents in hippocampal pyramidal neurons.Formule :C8H8N4O4S3Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :320.37Ref: TM-T23782
5mg51,00€10mg88,00€25mg160,00€50mg235,00€100mg349,00€200mg515,00€1mL*10mM (DMSO)57,00€Lofemizole
CAS :Lofemizole is an antagonist of CYP1A2.Formule :C10H9ClN2Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :192.64Ref: TM-T50053
1mg35,00€5mg74,00€10mg100,00€25mg170,00€50mg246,00€100mg349,00€200mg480,00€1mL*10mM (DMSO)64,00€PDE10-IN-1
CAS :PDE10-IN-1 (SEP-0372814) is used for treating CNS and metabolic disorders.Formule :C21H19N7Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :369.42IOX4
CAS :IOX4 is a potent PHD2 inhibitor (IC50 = 1.6 nM)Formule :C15H16N6O3Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :328.33Zegocractin
CAS :Zegocractin (CM-4620) is a calcium-release activated calcium-channel (CRAC channel) inhibitor.Formule :C19H11ClF3N3O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :421.76Ref: TM-TQ0033
1mg126,00€5mg259,00€10mg432,00€25mg715,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)283,00€Amifostine trihydrate
CAS :Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formule :C5H15N2O3PS·3H2ODegré de pureté :99.71% - 99.80%Couleur et forme :SolidMasse moléculaire :268.27SR0987
CAS :SR0987 is a RORγt agonist,Formule :C16H10ClF6NO2Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :397.7PX-478
CAS :PX-478 is a HIF-1α inhibitor with selectivity, oral activity, and blood-brain barrier permeability.Formule :C13H20Cl4N2O3Degré de pureté :97% - 99.79%Couleur et forme :SolidMasse moléculaire :394.12Ref: TM-T6961
1mg42,00€5mg88,00€10mg137,00€25mg205,00€50mg276,00€100mg434,00€200mg638,00€1mL*10mM (DMSO)88,00€PF-8380 hydrochloride
CAS :PF-8380 hydrochloride is a powerful inhibitor of autotaxin, exhibiting an IC(50) of 2.8 nM in isolated enzyme assays and 101 nM in human whole blood.Formule :C22H22Cl3N3O5Couleur et forme :SolidMasse moléculaire :514.79U-104
CAS :U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).
Formule :C13H12FN3O3SDegré de pureté :98.76% - 99.88%Couleur et forme :SolidMasse moléculaire :309.324-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid
CAS :4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid is used as a pharmaceutical intermediate.
Formule :C12H8F3NO2SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :287.26Cedirogant
CAS :Cedirogant (ABBV-157) is an orally active retinoid-related orphan receptor-γt(RORγt) inverse agonist that is used for psoriasis study.Formule :C24H20Cl3F3N2O3Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :547.78Ref: TM-T9635
1mg81,00€5mg167,00€10mg259,00€25mg470,00€50mg703,00€100mg1.044,00€200mg1.404,00€1mL*10mM (DMSO)197,00€3-Methylglutaric acid
CAS :Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.Formule :C6H10O4Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :146.14CAY10650
CAS :CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Formule :C28H25NO6Degré de pureté :97.33%Couleur et forme :SolidMasse moléculaire :471.5Ref: TM-TQ0105
1mg49,00€5mg114,00€10mg172,00€25mg334,00€50mg467,00€100mg620,00€1mL*10mM (DMSO)118,00€Enterostatin, human, mouse, rat acetate
Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.Formule :C23H40N8O8Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :556.61Glycerol 3-phosphate biscyclohexylammonium salt
CAS :Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.Formule :C15H35N2O6PDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :370.423PO
CAS :3PO inhibits PFKFB3 (IC50: 22.9 µM) and cancer cell growth (IC50: 1.4-24 µM), reducing glucose uptake and key cellular metabolites.
Formule :C13H10N2ODegré de pureté :99.56% - 99.67%Couleur et forme :SolidMasse moléculaire :210.23ARM1
CAS :ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.Formule :C16H14N2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :266.36(±)-Amiflamine
CAS :(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.Formule :C12H20N2Degré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :192.3Cecropin P1, porcine acetate
Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.Formule :C149H257N45O45Degré de pureté :95.4% - 98%Couleur et forme :SolidMasse moléculaire :3398.91ZM223 hydrochloride
ZM223 hydrochloride is a potent, non-covalent, orally active inhibitor of NEDD8 activase (NAE).Formule :C23H18ClF3N4O2S2Couleur et forme :SolidMasse moléculaire :538.991-Ethynylpyrene
CAS :1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).Formule :C18H10Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :226.27Diflubenzuron
CAS :Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.Formule :C14H9ClF2N2O2Degré de pureté :99.58% - 99.96%Couleur et forme :Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective InsecticideMasse moléculaire :310.68L-778123 free base
CAS :L-778123, an FPTase and GGPTase-I inhibitor, has tolerable toxicity with radiotherapy in advanced pancreatic cancer.Formule :C22H20ClN5OCouleur et forme :SolidMasse moléculaire :405.88SR8278
CAS :SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112Formule :C18H19NO3S2Degré de pureté :99.44% - 99.73%Couleur et forme :SolidMasse moléculaire :361.48Ref: TM-T7837
1mg49,00€5mg97,00€10mg160,00€25mg303,00€50mg437,00€100mg642,00€200mg914,00€1mL*10mM (DMSO)106,00€DHBP dibromide
CAS :DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.Formule :C24H38Br2N2Degré de pureté :99.73%Couleur et forme :Yellow To Yellow-Green Powder Or FlakesMasse moléculaire :514.38Sephin1 Hydrochloride
CAS :Sephin1 HCl selectively inhibits PPP1R15A, enhancing eIF2α phosphorylation to protect cells from proteostatic flaws.Formule :C8H10Cl2N4Couleur et forme :SolidMasse moléculaire :233.1(Rac)-LB-100
CAS :LB-100, a novel Protein Phosphatase 2A (PP2A) inhibitor, sensitizes malignant meningioma cells to the therapeutic effects of radiationFormule :C13H20N2O4Degré de pureté :98.31% - 99.77%Couleur et forme :SolidMasse moléculaire :268.31Ref: TM-T2068
1mg62,00€2mg88,00€5mg124,00€10mg172,00€25mg295,00€50mg442,00€100mg645,00€500mg1.341,00€Pep 2-8 ammonium salt(1541011-97-5 free base)
Pep 2-8 ammonium salt inhibits PCSK9-LDL receptor binding (IC50 = 0.8 μM), boosting LDL uptake in HepG2 cells.Formule :C83H113N17O24Degré de pureté :95.76% - 99.87%Couleur et forme :SolidMasse moléculaire :1732.91Idoxuridine hydrate
CAS :Idoxuridine (5-IUdR) blocks DNA polymerase, treating herpes eye infections, with an IC50 of 4.3 μM against feline herpes.Formule :C9H13IN2O6Couleur et forme :SolidMasse moléculaire :372.115kb NB 142-70
CAS :kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).Formule :C11H9NO2S2Degré de pureté :98.15% - ≥95%Couleur et forme :SolidMasse moléculaire :251.32D-Valine
CAS :D-Valine (H-D-Val-OH) is the enantiomer of L-Valine.Formule :C5H11NO2Degré de pureté :99.93%Couleur et forme :White CrystalsMasse moléculaire :117.15GSK2033
CAS :GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).Formule :C29H28F3NO5S2Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :591.66Efonidipine
CAS :Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Formule :C34H38N3O7PDegré de pureté :98.35% - 99.47%Couleur et forme :SolidMasse moléculaire :631.66IDO5L
CAS :IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).Formule :C9H7ClFN5O2Degré de pureté :99.49% - 99.75%Couleur et forme :SolidMasse moléculaire :271.64Ref: TM-T2647
10mg50,00€25mg86,00€50mg124,00€100mg187,00€200mg321,00€500mg505,00€1mL*10mM (DMSO)35,00€Tedizolid
CAS :Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit ofFormule :C17H15FN6O3Degré de pureté :96.97% - 99.89%Couleur et forme :SolidMasse moléculaire :370.34Calcifediol monohydrate
CAS :Calcifediol monohydrate (25-hydroxy Vitamin D3 monohydrate), the main circulating metabolite of vitamin D3, is a potent VDR inhibitor.Formule :C27H46O3Degré de pureté :99.31%Couleur et forme :Brownish Fine PowderMasse moléculaire :418.65Torcetrapib
CAS :Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.Formule :C26H25F9N2O4Degré de pureté :98% - 99.59%Couleur et forme :LipidMasse moléculaire :600.47Pimecrolimus
CAS :Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.Formule :C43H68ClNO11Degré de pureté :99.53% - 99.87%Couleur et forme :White Crystalline PowderMasse moléculaire :810.45[11C]MP 10
CAS :[11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.Formule :C25H20N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :391.45SI-113
CAS :SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.Formule :C23H24N6ODegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :400.48Ref: TM-T9589
1mg43,00€2mg56,00€5mg93,00€10mg133,00€25mg236,00€50mg354,00€100mg518,00€1mL*10mM (DMSO)101,00€BAY-876
CAS :BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.Formule :C24H16F4N6O2Degré de pureté :98.61% - 99.78%Couleur et forme :SolidMasse moléculaire :496.42Ref: TM-T3713
1mg55,00€2mg78,00€5mg95,00€10mg131,00€25mg221,00€50mg334,00€100mg533,00€200mg755,00€1mL*10mM (DMSO)96,00€Benzenesulfonamide
CAS :Benzenesulfonamide (Benzosulfonamide) ia an inhibitor of carbonic anhydrases.Formule :C6H7NO2SDegré de pureté :99.42% - 99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :157.19IDF-11774
CAS :IDF-11774 is a HIF-1 inhibitor.It reduces hif-1α HRE luciferase activity (IC50 = 3.65 μM).Formule :C23H32N2O2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :368.51Z-HA155
CAS :Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.Formule :C24H19BFNO5SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :463.29Ref: TM-T11533
1mg34,00€5mg71,00€10mg101,00€25mg200,00€50mg321,00€100mg475,00€200mg680,00€1mL*10mM (DMSO)73,00€Raphin1
CAS :Raphin1 is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B).Formule :C8H8Cl2N4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :231.08IOX2
CAS :IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.Formule :C19H16N2O5Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :352.34ZINC13466751
CAS :ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).Formule :C20H21N5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :363.41Azumolene
CAS :Azumolene (EU4093 free base)Formule :C13H9BrN4O3Degré de pureté :98.1% - 98.35%Couleur et forme :SolidMasse moléculaire :349.14Ref: TM-T8815
2mg49,00€5mg73,00€10mg116,00€25mg235,00€50mg373,00€100mg562,00€500mg1.216,00€1mL*10mM (DMSO)82,00€Olumacostat Glasaretil
CAS :Olumacostat glasaretil is a small molecule inhibitor of acetyl coenzyme A carboxylase (ACC). It has been used in trials studying the treatment of Acne Vulgaris.Formule :C26H43NO7Degré de pureté :97.79% - 99.34%Couleur et forme :SolidMasse moléculaire :481.62Ref: TM-T3510
1mg52,00€5mg96,00€10mg144,00€25mg265,00€50mg454,00€100mg662,00€200mg943,00€1mL*10mM (DMSO)97,00€2-Aminoethyl diphenylborinate
CAS :2-Aminoethyl diphenylborinate (2-APB) is a chemical that acts to inhibit both IP3 receptors and TRP channels.Formule :C14H16BNODegré de pureté :98.74% - 99.92%Couleur et forme :WhiteMasse moléculaire :225.09MBCQ
CAS :MBCQ is an inhibitor of cGMP-specific phosphodiesterase PDE5.Formule :C16H12ClN3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :313.74Ref: TM-T21965
5mg47,00€10mg80,00€25mg145,00€50mg233,00€100mg335,00€200mg467,00€1mL*10mM (DMSO)49,00€Ingliforib
CAS :Ingliforib (CP 368296) is a novel glycogen phosphorylase inhibitor,has antihyperglycemic and cardioprotective properties.Formule :C23H24ClN3O5Degré de pureté :99.04% - 99.30%Couleur et forme :SolidMasse moléculaire :457.91Ref: TM-T8493
1mg52,00€5mg92,00€10mg155,00€25mg299,00€50mg480,00€100mg772,00€200mg1.035,00€1mL*10mM (DMSO)92,00€Cyfluthrin
CAS :Cyfluthrin binds to voltage-sensitive sodium channel such as Nav 1.8 sodium channel and modify their gating kinetics, thereby disrupting nerve function of pestsFormule :C22H18Cl2FNO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :434.29Biotin sulfone
CAS :Biotin sulfone is an oxidized form of biotin.Formule :C10H16N2O5SDegré de pureté :95.51% - 99.17%Couleur et forme :SolidMasse moléculaire :276.31Lactisole
CAS :Lactisole (na-PMP) is an inhibitor of the glucose-sensing receptorFormule :C10H11NaO4Degré de pureté :99.9%Couleur et forme :White To Pale Cream Crystalline SolidMasse moléculaire :218.18BCI hydrochloride
CAS :BCI hydrochloride ((E)-BCI hydrochloride) is a DUSP6 inhibitor that inhibits RANKL-mediated osteoclastogenesis and attenuates oophorectomy-induced bone loss.Formule :C22H24ClNODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :353.89PKM2-IN-1
CAS :PKM2-IN-1 (compound 3k) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.Formule :C18H19NO2S2Degré de pureté :99.49% - 99.68%Couleur et forme :SolidMasse moléculaire :345.48Glucosamine sulfate
CAS :Glucosamine sulfate (D-Glucosaminesulfate) was extracted from synthetic product;Store the product in sealed, cool and dry condition.Formule :C6H13NO5·H2SO4Degré de pureté :99.64%Couleur et forme :White CrystalMasse moléculaire :277.25GW604714X
CAS :GW604714X (2,4-Thiazolidinedione, 5-[[5-[6-(4-acetyl-1-piperazinyl)-3-nitro-2-pyridinyl]-2-fluorophenyl]methylene]-) were found to be potent inhibitors ofFormule :C21H18FN5O5SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :471.46SDZ285428
CAS :SDZ285428 is a CYP24A1 inhibitor.Formule :C24H20ClN3ODegré de pureté :97.51%Couleur et forme :SolidMasse moléculaire :401.89Ref: TM-T4188
2mg37,00€5mg52,00€10mg90,00€25mg170,00€50mg255,00€100mg375,00€200mg533,00€1mL*10mM (DMSO)58,00€
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