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One of the most relevant brands among our more than 25 partners is TargetMol

One of the most relevant brands among our more than 25 partners is TargetMol

We have reached an agreement with TargetMol: CymitQuimica clients will benefit for a 20% discount on all TargetMol products until the end of the year.On our website you can find the products offered by this partner, which has become one of the world's most recognised compound libraries and small molecule inhibitors supplier. TargetMol offers approximately 120 compound libraries and a wide range of chemical products and kits for life sciences.

Ends on Dec 31( 7 days left )

products per page.Found 111935 products on this promotion.
  • hCAIX-IN-16

    CAS:
    hCAIX-IN-16 (Compound 12d), an inhibitor of hCA IX, exhibits inhibition constants (K i) of 190.0 nM for hCA IX and 187.9 nM for hCA XII.
    Formula:C20H20N8O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.49
  • hCAIX-IN-15

    CAS:
    hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancer
    Formula:C18H14FN7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.41
  • LIXIVAPTAN

    CAS:
    Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
    Formula:C27H21ClFN3O2
    Purity:98.36%
    Color and Shape:Solid
    Molecular weight:473.93
  • hCAIX-IN-14

    CAS:
    hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .
    Formula:C11H17ClN6O2S
    Color and Shape:Solid
    Molecular weight:332.81
  • HDAC6-IN-14


    HDAC6-IN-14, an inhibitor of HDAC6 (HDAC), exhibits high selectivity with an IC50 value of 42 nM, demonstrating over 100-fold selectivity compared to HDAC1,
    Formula:C24H30FN3O4
    Color and Shape:Solid
    Molecular weight:443.51
  • MtInhA-IN-1


    MtInhA-IN-1: an oral selective MtInhA inhibitor, IC50 0.23 μM, effective against M. tuberculosis with MIC 0.4 μM.
    Formula:C21H22BrN3
    Color and Shape:Solid
    Molecular weight:396.32
  • TRK II-IN-1

    CAS:
    <p>TRK II-IN-1: potent type II TRK inhibitor; IC50s: TRKA (3.3 nM), TRKB (6.4 nM), TRKC (4.3 nM), TRKA G667C (9.4 nM); also targets FLT3, RET, VEGFR2.</p>
    Formula:C29H31F3N8O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:564.6
  • NLRP3-IN-12


    NLRP3-IN-12 inhibits NLRP3 inflammasome, curbing IL-1β release with 0.45 μM IC50, for inflammatory bowel disease research.
    Formula:C27H32ClNO7
    Color and Shape:Solid
    Molecular weight:518
  • STAT3-IN-15


    STAT3-IN-15: Potent, oral STAT3 inhibitor for IPF, blocks STAT3 phosphorylation, cell migration, and EMT.
    Formula:C20H17F3N2O3S
    Color and Shape:Solid
    Molecular weight:422.42
  • hCA IX-IN-2


    hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative
    Formula:C23H24N2O4STe
    Color and Shape:Solid
    Molecular weight:552.11
  • HSP90-IN-18


    HSP90-IN-18 inhibits Hsp90 with 0.39 μM IC50, useful for viral, neurodegenerative, and inflammatory research.
    Formula:C25H33FO3
    Color and Shape:Solid
    Molecular weight:400.53
  • HSP90-IN-19

    CAS:
    HSP90-IN-19: potent Hsp90 inhibitor, IC50 = 0.27 μM, used in research on viral diseases, neurodegeneration, inflammation.
    Formula:C29H38O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.61
  • CYP1B1-IN-3

    CAS:
    CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.
    Formula:C20H16FN3O2S2
    Color and Shape:Solid
    Molecular weight:413.49
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Formula:C8H4N4O6
    Purity:97.27% - 99.1%
    Color and Shape:Off-White Powder With A Yellow Tinge
    Molecular weight:252.14
  • CYP1B1-IN-4

    CAS:
    <p>CYP1B1-IN-4: 2,4-diarylthiazole, selective CYP1B1 inhibitor (IC50=0.2 nM), low cytotoxicity, stable in liver microsomes.</p>
    Formula:C18H14N2O2S
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:322.38
  • CYP1B1-IN-5

    CAS:
    CYP1B1-IN-5: selective CYP1B1 inhibitor, IC50 = 4.7 nM, useful for metabolism disease research.
    Formula:C14H8INO2
    Purity:97.66%
    Color and Shape:Solid
    Molecular weight:349.12
  • HDAC6-IN-15


    HDAC6-IN-15: selective HDAC6 inhibitor, IC50 of 38.2 nM, for cancer and neurodegenerative research.
    Formula:C25H28FFeN3O2
    Color and Shape:Solid
    Molecular weight:477.35
  • Urease-IN-4


    <p>Urease-IN-4 inhibits urease (IC50: 1.64 µM), targets P. vulgaris (IC50: 15.27 µg/mL), and is low in cytotoxicity.</p>
    Formula:C16H20N2O3S
    Color and Shape:Solid
    Molecular weight:320.41
  • Urease-IN-5


    Urease-IN-5: urease inhibitor, IC50 1.473 µM, low cytotoxicity, IC50 17.78 µg/mL on P. vulgaris.
    Formula:C16H20N2O3S
    Color and Shape:Solid
    Molecular weight:320.41
  • KIF18A-IN-6

    CAS:
    KIF18A-IN-6 (Compound 134) is an orally active KIF18A inhibitor that suppresses KIF18A microtubule-dependent ATPase activity with an IC50 of 0.016 μM.
    Formula:C28H37N3O5S2
    Purity:97.59%
    Molecular weight:559.74
  • JQEZ5

    CAS:
    JQEZ5 is an inhibitor of EZH2 lysine methyltransferase (IC50 = 11.1 nM).
    Formula:C30H38N8O2
    Purity:98.14% - ≥98%
    Color and Shape:Solid
    Molecular weight:542.68
  • KIF18A-IN-7

    CAS:
    KIF18A-IN-7 is an orally active inhibitor targeting KIF18A, demonstrating potent inhibition with an IC50 value of 9.4 nM against the microtubule-dependent
    Formula:C27H35N3O5S2
    Color and Shape:Soild
    Molecular weight:545.71
  • Leritrelvir

    CAS:
    <p>Dermatan sulphate sodium (Chondroitin sulfate B sodium salt) is a linear sulfated polysaccharide, a glycosaminoglycan component of important proteoglycans.</p>
    Formula:C31H44F3N5O6
    Purity:97.42%
    Color and Shape:Solid
    Molecular weight:639.71
  • Pomotrelvir

    CAS:
    <p>Pomotrelvir (PBI-0451) is an oral SARS-CoV-2 3CL protease inhibitor with antiviral properties for COVID-19 research.</p>
    Formula:C23H26ClN5O3
    Color and Shape:Solid
    Molecular weight:455.94
  • BAY 2965501

    CAS:
    BAY 2965501 is a potent and selective diacylglycerol kinase zeta (DGKζ) inhibitor that induces pERK activation.BAY 2965501 can be used in the study of cancer.
    Formula:C20H19FN4O3S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:414.45
  • Moiramide B

    CAS:
    Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.
    Formula:C25H31N3O5
    Purity:98.53% - 99.90%
    Color and Shape:Solid
    Molecular weight:453.53
  • (S)-VQW-765


    (S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39
  • Tiludronate

    CAS:
    Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.
    Formula:C7H9ClO6P2S
    Color and Shape:Solid
    Molecular weight:318.61
  • Cloxacillin

    CAS:
    Cloxacillin, a β-lactamase inhibitor, tackles S. aureus inflammation and has an IC50 of 0.04 µM.
    Formula:C19H18ClN3O5S
    Color and Shape:Solid
    Molecular weight:435.88
  • Acamprosate

    CAS:
    Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust
    Formula:C5H11NO4S
    Purity:98.30%
    Color and Shape:Solid
    Molecular weight:181.21
  • Valorphin

    CAS:
    Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
    Formula:C44H61N9O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:892.01
  • Pralidoxime

    CAS:
    Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.
    Formula:C7H9N2O
    Color and Shape:Solid
    Molecular weight:137.16
  • Amakusamine

    CAS:
    Amakusamine is an indole alkaloid from the sponge of Psammocinia sp. that inhibits RANKL-induced isolation of multinucleated osteoclast formation.
    Formula:C9H5Br2NO2
    Purity:98.37% - 98.42%
    Color and Shape:Solid
    Molecular weight:318.95
  • Rostratin A

    CAS:
    Rostratin A, a disulfide from Exserohilum rostratum, is cytotoxic to HCT-116 cells with an IC50 of 8.5 μg/mL.
    Formula:C18H24N2O6S2
    Color and Shape:Solid
    Molecular weight:428.52
  • Rostratin B

    CAS:
    Rostratin B, a cytotoxic disulfide, demonstrates in vitro cytotoxicity against human colon carcinoma (HCT-116), exhibiting an IC50 value of 1.9 μg/mL.
    Formula:C18H20N2O6S2
    Color and Shape:Solid
    Molecular weight:424.49
  • Rostratin C

    CAS:
    Rostratin C, a cytotoxic disulfide, exhibits in vitro cytotoxicity against human colon carcinoma (HCT-116), demonstrating an IC50 value of 0.76 μg/mL.
    Formula:C20H24N2O8S2
    Color and Shape:Solid
    Molecular weight:484.54
  • Thielavin B

    CAS:
    Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.
    Formula:C31H34O10
    Color and Shape:Solid
    Molecular weight:566.6
  • Isodispar B

    CAS:
    Isodispar B: an anticancer drug, halts many cancer types' growth, triggers cell death.
    Formula:C20H18O5
    Color and Shape:Solid
    Molecular weight:338.35
  • Mammea A/BA

    CAS:
    Mammea A/BA combats T. cruzi by causing mitochondrial damage, ROS, DNA fragmentation, and vacuolization, leading to cell death. Useful for Chagas research.
    Formula:C25H26O5
    Color and Shape:Solid
    Molecular weight:406.47
  • Kurzipene D

    CAS:
    Kurzipene D: anticancer, induces apoptosis, halts HepG2 at S phase, anti-tumor in zebrafish, inhibits tumor growth and spread.
    Formula:C26H36O8
    Color and Shape:Solid
    Molecular weight:476.56
  • Vorasidenib

    CAS:
    Vorasidenib (PVM/MA) is an inhibitor of mutant isocitrate dehydrogenase (IDH; IC50s = 31.9 and 31.7 nM for IDH1R132H and IDH2R140Q, respectively)
    Formula:C14H13ClF6N6
    Purity:98.28% - 99.57%
    Color and Shape:Solid
    Molecular weight:414.74
  • STAT3-IN-14

    CAS:
    <p>STAT3-IN-14 is a STAT3 inhibitor and has STAT3 phosphorylation inhibitory activity. STAT3-IN-14 can directly bind to the hinge region of STAT3 .</p>
    Formula:C14H10O5
    Color and Shape:Solid
    Molecular weight:258.23
  • PTP1B-IN-20


    PTP1B-IN-20: Selective PTP1B inhibitor, IC50=1.05μM; less effective on TCPTP (IC50=78μM), targets type 2 diabetes.
    Formula:C26H28O15
    Color and Shape:Solid
    Molecular weight:580.49
  • PTP1B-IN-21


    PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.
    Formula:C22H22O11
    Color and Shape:Solid
    Molecular weight:462.4
  • Phanginin A

    CAS:
    Phanginin A, a natural product, activates SIK1 and inhibits gluconeogenesis in mouse primary hepatocytes, can be used in studies of type 2 diabetes.
    Formula:C21H28O5
    Purity:95.54%
    Color and Shape:Solid
    Molecular weight:360.44
  • BACE1-IN-10

    CAS:
    <p>BACE1-IN-10 is a potent inhibitor of BACE1, demonstrating sub-micromolar activity against recombinant BACE1 (rBACE1) [1].</p>
    Formula:C33H49N5O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:675.84
  • Nomifensine

    CAS:
    Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.
    Formula:C16H18N2
    Purity:99.83% - ≥95%
    Color and Shape:Solid
    Molecular weight:238.33
  • (R)-V-0219


    (R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.
    Formula:C20H25F3N4O2
    Color and Shape:Solid
    Molecular weight:410.43
  • (S)-V-0219


    (S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.
    Formula:C20H25F3N4O2
    Color and Shape:Solid
    Molecular weight:410.43
  • TES Sodium

    CAS:
    TES sodium is an amphoteric ion buffer with an effective pH range of 6.8 to 8.2, commonly used in cell culture and enzyme studies.
    Formula:C6H15NNaO6S
    Color and Shape:Solid
    Molecular weight:252.24
  • Nipradolol

    CAS:
    Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.
    Formula:C15H22N2O6
    Color and Shape:Solid
    Molecular weight:326.35
  • BMS 310705

    CAS:
    BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.
    Formula:C27H42N2O6S
    Color and Shape:Solid
    Molecular weight:522.70
  • Talotrexin

    CAS:
    Talotrexin (PT523), a nonpolyglutamatable antifolate analog of Aminopterin, inhibits DHFR and RFC, targeting tumor growth.
    Formula:C27H27N9O6
    Color and Shape:Solid
    Molecular weight:573.56
  • Mavodelpar

    CAS:
    Mavodelpar (REN001), a PPARδ agonist, may treat PMM and LC-FAOD by reducing renal damage.
    Formula:C31H29FNNaO5
    Color and Shape:Solid
    Molecular weight:537.55
  • TAS-103 dihydrochloride

    CAS:
    <p>TAS-103 dihydrochloride (BMS-247615 dihydrochloride) is a novel anticancer agent targeting both topoisomerase (Topo) I and Topo II.</p>
    Formula:C20H21Cl2N3O2
    Purity:97.78%
    Color and Shape:Solid
    Molecular weight:406.31
  • EphB1-IN-1

    CAS:
    EphB1-IN-1 is a potent inhibitor of EphB1, exhibiting IC50 values of 3.0 nM for EphB1 G703C, 15 nM for EphB1 T697G, and 220 nM for EphB1 WT.
    Formula:C16H12Cl2N4O2
    Color and Shape:Solid
    Molecular weight:363.2
  • NBI-921352

    CAS:
    NBI-921352 (XEN901) is a potent NaV1.6 sodium channel inhibitor, effectively treating epilepsy without severe side effects.
    Formula:C22H25FN4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.59
  • Udifitimod

    CAS:
    Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.
    Formula:C25H33NO2
    Color and Shape:Solid
    Molecular weight:379.54
  • Z-VRPR-FMK

    CAS:
    Z-VRPR-FMK: irreversible MALT1 inhibitor, halts growth/invasion of diffused B-cell lymphoma by blocking NF-κB activation and MMP expression.
    Formula:C31H49FN10O6
    Color and Shape:Solid
    Molecular weight:676.78
  • Adhesamine

    CAS:
    Adhesamine, a dumbbell molecule, enhances cell adhesion, growth, neuron differentiation, and survival via MAPK/FAK.
    Formula:C24H32Cl4N8O2S2
    Color and Shape:Solid
    Molecular weight:670.51
  • PNU-101603

    CAS:
    <p>PNU-101603, a Sutezolid metabolite, effective against TB including drug-resistant strains, works solo or with SQ109.</p>
    Formula:C16H20FN3O4S
    Color and Shape:Solid
    Molecular weight:369.41
  • Z-LEVD-FMK

    CAS:
    Z-LEVD-FMK is a caspase-4 inhibitor with anti-cancer activity, capable of eliminating LPS-induced GCLC protein degradation.
    Formula:C31H45FN4O10
    Color and Shape:Solid
    Molecular weight:652.71
  • SID-852843

    CAS:
    SID-852843, WNV NS2B-NS3 protease inhibitor, IC50: 0.105 μM, useful in viral infection studies.
    Formula:C17H15N3O5S
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:373.38
  • BACE2-IN-1

    CAS:
    <p>BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.</p>
    Formula:C36H38F3N3O3
    Color and Shape:Solid
    Molecular weight:617.7
  • Etbicyphat

    CAS:
    Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.
    Formula:C6H11O4P
    Color and Shape:Solid
    Molecular weight:178.12
  • Paquinimod

    CAS:
    Paquinimod (ABR 25757) is a S100A9 inhibitor preventing S100A9 binding to TLR-4.
    Formula:C21H22N2O3
    Purity:98.04% - 99.79%
    Color and Shape:Solid
    Molecular weight:350.41
  • ACT-606559


    ACT-606559, a metabolite of ACT451840, is a novel chemical compound exhibiting antimalarial properties. It is utilized in malaria research.
    Formula:C47H52N6O3
    Color and Shape:Solid
    Molecular weight:748.95
  • EGFR-IN-25

    CAS:
    EGFR-IN-25, an efficacious EGFR inhibitor, demonstrates IC50 values of 9 nM for BaF3 cells (EGFR DEL19/T790M/C797S) and 60 nM for A431 cells (WT), respectively.
    Formula:C34H43N9O2
    Color and Shape:Solid
    Molecular weight:609.76
  • EGFR-IN-21

    CAS:
    EGFR-IN-21, a potent EGFR inhibitor, exhibits an IC50 of 0.38 nM, demonstrating significant antitumor activity.
    Formula:C36H44BrN10O2P
    Color and Shape:Solid
    Molecular weight:759.68
  • EGFR-IN-23

    CAS:
    EGFR-IN-23, identified as compound 8 in WO2021244502A1, is a potent EGFR tyrosine kinase inhibitor (TKI) demonstrating an inhibitory concentration (IC50) of 8.
    Formula:C36H44BrN10O3P
    Color and Shape:Solid
    Molecular weight:775.68
  • EGFR-IN-28

    CAS:
    EGFR-IN-28 is a potent EGFR inhibitor. EGFR-IN-28 has antitumor activity .
    Formula:C31H39BrN10O3S
    Color and Shape:Solid
    Molecular weight:711.68
  • EGFR-IN-29

    CAS:
    EGFR-IN-29 is a potent EGFR inhibitor.
    Formula:C36H46BrN8O2P
    Color and Shape:Solid
    Molecular weight:733.68
  • RAD51-IN-4

    CAS:
    RAD51-IN-4, a potent RAD51 inhibitor, may be useful in researching mitochondrial defect-related conditions.
    Formula:C31H34FN5O5S2
    Color and Shape:Solid
    Molecular weight:639.76
  • EGFR-IN-30

    CAS:
    EGFR-IN-30 is an EGFR inhibitor (IC50: 1-10 nM, <1 nM WT/mutants) with potential in cancer research.
    Formula:C28H33BrN7O2P
    Color and Shape:Solid
    Molecular weight:610.49
  • JNK-1-IN-1

    CAS:
    JNK-1-IN-1 is an inhibitor specifically targeting JNK-1, also exhibiting inhibition of MKK7 with an IC50 value of 7.8μM.
    Formula:C24H22N6S
    Color and Shape:Solid
    Molecular weight:426.54
  • Oxyphenisatin acetate

    CAS:
    <p>Oxyphenisatin acetate inhibits the growth of the breast cancer cell lines MCF7, T47D, HS578T, and MDA-MB-468.</p>
    Formula:C24H19NO5
    Purity:98% - 99.35%
    Color and Shape:Solid
    Molecular weight:401.41
  • PI3Ka-IN-5

    CAS:
    PI3Ka-IN-5 is a potent PI3Kα/mTOR inhibitor, with an IC 50 of 0.7 nM and 3.3 nM, respectively. PI3Ka-IN-5 can be used for the research of colorectal cancer .
    Formula:C30H35N9O5
    Color and Shape:Solid
    Molecular weight:601.66
  • IDO1-IN-17

    CAS:
    IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .
    Formula:C28H32BrClFN5O2
    Color and Shape:Solid
    Molecular weight:604.94
  • STAT3-IN-7

    CAS:
    STAT3-IN-7, an orally active aryl sulfonamido azetidine compound, serves as a STAT3 inhibitor with anticancer activities.
    Formula:C30H26F5N5O4S
    Color and Shape:Solid
    Molecular weight:647.62
  • (S)-HH2853

    CAS:
    (S)-HH2853 is a potent EZH1/2 inhibitor, aromatic, <100 nM IC50 for EZH2_Y641F, promising for anti-tumor/autoimmune research.
    Formula:C31H36F3N7O3
    Purity:97.18% - 99.74%
    Color and Shape:Solid
    Molecular weight:611.66
  • (R)-HH2853

    CAS:
    (R)-HH2853, a mutant EZH2 inhibitor, IC50 <100 nM for EZH2-Y641F, targets cancer/autoimmune diseases.
    Formula:C31H36F3N7O3
    Purity:97.53% - 98.85%
    Color and Shape:Solid
    Molecular weight:611.66
  • ROCK2-IN-5


    ROCK2-IN-5, a compound blending fasudil, caffeic, and ferulic acids, shows promise for ALS research involving SOD1 mutations.
    Formula:C23H25N3O5S
    Color and Shape:Solid
    Molecular weight:455.53
  • PI3K-IN-28

    CAS:
    PI3K-IN-28, a potent PI3K inhibitor with low toxicity in MCF-10a, has IC50 values of 5.8, 2.3, 7.9 μM and high selectivity index of 39.
    Formula:C26H16F9N3O3S2
    Color and Shape:Solid
    Molecular weight:653.54
  • AX20017

    CAS:
    AX20017 is a small-molecule protein kinase G (PknG) inhibitor(IC50 : 0.39 μM). It acts by blocking the proliferation of M. tuberculosis.
    Formula:C13H16N2O2S
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:264.34
  • MptpB-IN-1

    CAS:
    MptpB-IN-1: orally active, potent MptpB inhibitor; reduces drug-resistant tuberculosis.
    Formula:C17H11Cl2NO4
    Color and Shape:Solid
    Molecular weight:364.18
  • FGFR4-IN-8

    CAS:
    FGFR4-IN-8 is a selective, ATP-competitive FGFR4 inhibitor with IC50s as low as 0.25 nM, halting growth of Hep3B cells at 29 nM and showing in vivo efficacy.
    Formula:C32H34Cl2FN7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.56
  • ThrRS-IN-3


    ThrRS-IN-3: Potent inhibitor of Salmonella enterica ThrRS, IC50 = 19 nM, Kd = 34 nM, with antibacterial effects.
    Formula:C31H30Cl2N6O5
    Color and Shape:Solid
    Molecular weight:637.51
  • SMTIN-T140

    CAS:
    SMTIN-T140: strong TRAP1 inhibitor, IC50=1.646μM, anticancer; disrupts mitochondria, boosts ROS, activates AMPK, shrinks PC3 tumors, no in vivo toxicity.
    Formula:C36H34BrClFN5OP
    Purity:98%
    Color and Shape:Solid
    Molecular weight:718.02
  • C16-K-cBB1


    C16-K-cBB1: potent, selective MRSA killer; MIC 1µg/mL, low hemolysis, works in 120 min at 12.5µg/mL.
    Formula:C33H58ClN5O5S
    Color and Shape:Solid
    Molecular weight:672.36
  • EGFR-IN-61

    CAS:
    EGFR-IN-61 inhibits EGFR kinase (IC50: 42 nM L858R/T790M, 137 nM L858R/T790M/C797S, 743 nM WT) and slows A549 & H1975 cell growth (IC50: 2.14 & 1.82 μM).
    Formula:C33H37ClN8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:629.15
  • STAT6-IN-1

    CAS:
    STAT6-IN-1: STAT6 inhibitor, IC50=0.028 µM, targets SH2 domain, for allergy and cancer research.
    Formula:C33H37IN3O7P
    Color and Shape:Solid
    Molecular weight:745.54
  • Enclomiphene citrate

    CAS:
    Enclomiphene citrate (trans-Clomiphene citrate) is a non-steroidal estrogen receptor antagonist,with antioestrogenic property
    Formula:C32H36ClNO8
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:598.08
  • Mebanazine

    CAS:
    <p>Mebanazine, a potent monoamine oxidase (MAO) inhibitor, is utilized in depression research.</p>
    Formula:C8H12N2
    Color and Shape:Solid
    Molecular weight:136.19
  • DS69910557


    DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism & osteoporosis research.
    Formula:C32H33Cl2FN4O3
    Color and Shape:Solid
    Molecular weight:611.53
  • FGF22-IN-1

    CAS:
    <p>FGF22-IN-1 is a CD4 N-terminal immunoglobulin variable region-like structural domain (CD4 D1) inhibitor that suppresses the immune response.</p>
    Formula:C14H11N3OS
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:269.32
  • EZH2-IN-14

    CAS:
    <p>EZH2-IN-14 selectively inhibits EZH2 at 12 nM IC50, has &gt;200-fold specificity over EZH1, reducing H3K27me3 levels.</p>
    Formula:C31H39N7O2
    Color and Shape:Solid
    Molecular weight:541.69
  • USP7-IN-10

    CAS:
    <p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>
    Formula:C26H29ClN4O3S
    Color and Shape:Solid
    Molecular weight:513.05
  • MAT2A-IN-9

    CAS:
    <p>MAT2A-IN-9, a 2-oxoquinazoline, inhibits MAT2A with antitumor effects on lymphomas and solid cancers.</p>
    Formula:C14H8ClF3N4O
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:340.69
  • GSK1790627

    CAS:
    GSK1790627, the N-deacetylated metabolite of Trametinib, represents an orally active MEK inhibitor that promotes autophagy and triggers apoptosis [1].
    Formula:C24H21FIN5O3
    Color and Shape:Solid
    Molecular weight:573.36
  • FLT3-IN-18

    CAS:
    FLT3-IN-18: potent, selective FLT3 inhibitor, IC50 0.003 μM, induces apoptosis, G1 arrest, blocks FLT3/STAT5, potential in AML research.
    Formula:C26H36N8O
    Color and Shape:Solid
    Molecular weight:476.62