
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(647 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.023 produtos)
- BACE(37 produtos)
- Beta Amilóide(230 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(373 produtos)
- Gama-secretase(62 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5637 produtos de "Neurociência"
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α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Pureza:98%Cor e Forma:LiquidPeso molecular:N/AGinkgolide A
CAS:Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Fórmula:C20H24O9Pureza:98.76% - 99.81%Cor e Forma:White PowderPeso molecular:408.40Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Fórmula:C17H21ClN4SCor e Forma:SolidPeso molecular:348.89Glypromate acetate(32302-76-4 free base)
Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.Fórmula:C14H23N3O8Pureza:99.94%Cor e Forma:SolidPeso molecular:361.35Ref: TM-T7778L
2mg37,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg74,00€25mg119,00€50mg160,00€100mg225,00€200mg314,00€Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFórmula:C28H33ClN2·2HClPureza:98.05%Cor e Forma:Off-White PowderPeso molecular:505.95Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Fórmula:C22H24ClN3O3SCor e Forma:SolidPeso molecular:445.96Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Fórmula:C20H24ClN3O2Cor e Forma:SolidPeso molecular:373.88NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Fórmula:C20H23Cl2F2N3O2Pureza:99.59%Cor e Forma:SolidPeso molecular:446.32Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Fórmula:C6H9ClN2O2Pureza:99.39%Peso molecular:176.601Flutriafol
CAS:Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist
Fórmula:C16H13F2N3OPureza:98.75%Cor e Forma:SolidPeso molecular:301.29Niaprazine
CAS:Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.72%Cor e Forma:SolidPeso molecular:358.84Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Fórmula:C15H21N5O4SCor e Forma:SolidPeso molecular:367.42Norfluoxetine Hydrochloride
CAS:Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Fórmula:C16H17ClF3NOPureza:99.71%Cor e Forma:SolidPeso molecular:331.76Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Fórmula:C24H25ClFN3O2Cor e Forma:SolidPeso molecular:441.93Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Cor e Forma:SolidPeso molecular:575.61RU 24969 free base
CAS:RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29VU10010
CAS:VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.
Fórmula:C17H16ClN3OSPureza:99.36%Cor e Forma:SolidPeso molecular:345.85Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Cor e Forma:White SolidPeso molecular:414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Fórmula:C22H28FNO3Pureza:98.94% - 99.95%Cor e Forma:SolidPeso molecular:373.46Ref: TM-T5389
1mg39,00€5mg84,00€1mL*10mM (DMSO)92,00€10mg117,00€25mg220,00€50mg285,00€100mg371,00€200mg530,00€Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Fórmula:C35H43N5O4Pureza:98.12%Cor e Forma:SolidPeso molecular:597.75NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H25N3O2SPureza:98%Cor e Forma:SolidPeso molecular:431.55Edonerpic maleate
CAS:Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).Fórmula:C20H25NO6SPureza:98.24%Cor e Forma:SolidPeso molecular:407.48Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Fórmula:C6H10ClNO2Pureza:98.42%Cor e Forma:SolidPeso molecular:163.602Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Fórmula:C15H18BrN3O3Pureza:98.51% - 99.24%Cor e Forma:SolidPeso molecular:368.23Org 25543 hydrochloride
CAS:Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2).Fórmula:C24H33ClN2O4Pureza:99.26%Cor e Forma:SolidPeso molecular:448.983idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Fórmula:C20H19F5N2OPureza:99.73%Cor e Forma:SolidPeso molecular:398.37Ref: TM-T7103
1mg88,00€2mg118,00€1mL*10mM (DMSO)187,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Fórmula:C67H119F3N22O22Pureza:98%Cor e Forma:SolidPeso molecular:1641.79Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Cor e Forma:SolidPeso molecular:485.961-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide
CAS:1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.
Fórmula:C20H30Br2N2Pureza:98.17%Cor e Forma:SolidPeso molecular:458.27Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Cor e Forma:White PowderPeso molecular:390.4CCMI
CAS:CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Fórmula:C19H15Cl2N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:388.25LY2886721
CAS:LY2886721, a BACE inhibitor, is used for the therapy of Alzheimer's Disease.Fórmula:C18H16F2N4O2SPureza:99% - 99.75%Cor e Forma:SolidPeso molecular:390.41AF-353
CAS:AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).Fórmula:C14H17IN4O2Pureza:92.98% - 99.356%Cor e Forma:SolidPeso molecular:400.21Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Cor e Forma:White PowderPeso molecular:614.02Amitriptyline
CAS:Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Fórmula:C20H23NPureza:98.24% - 99.64%Cor e Forma:Crystals SolidPeso molecular:277.4Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Fórmula:C10H14ClNO2Pureza:99.93%Cor e Forma:White Crystalline PowderPeso molecular:215.68Jagged-1 (188-204) TFA(219127-21-6 free base)
Jagged-1 (188-204) TFA, a JAG-1 skin protein fragment, induces epidermal maturation and keratinocyte stratification.Fórmula:C95H128F3N25O28S3Pureza:99.48%Cor e Forma:SolidPeso molecular:2221.37Acotiamide monohydrochloride trihydrate
CAS:Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.Fórmula:C21H37ClN4O8SPureza:98% - 99.54%Cor e Forma:SolidPeso molecular:541.06Crenigacestat
CAS:Crenigacestat (LY3039478) is an orally bioavailable Notch inhibitor with an IC50 of ~1 nM in most of the tumor cell lines tested.Fórmula:C22H23F3N4O4Pureza:97.27% - 98.99%Cor e Forma:SolidPeso molecular:464.44Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFórmula:C21H35ClN2O5Pureza:99.33%Cor e Forma:SolidPeso molecular:430.97Ref: TM-T9833
1mg90,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Fórmula:C23H31ClN2O2Pureza:99.71%Cor e Forma:SolidPeso molecular:402.96AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Fórmula:C17H21N5O2SPureza:99.81%Cor e Forma:SolidPeso molecular:359.45Ref: TM-T5179
1mg37,00€2mg50,00€5mg77,00€1mL*10mM (DMSO)85,00€10mg114,00€25mg225,00€50mg335,00€100mg484,00€Avagacestat
CAS:Avagacestat (BMS-708163) (BMS-708163) is a potent, selective, orally bioavailable γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM,Fórmula:C20H17ClF4N4O4SPureza:98.87% - 99.73%Cor e Forma:SolidPeso molecular:520.89Ref: TM-T6249
1mg38,00€5mg77,00€1mL*10mM (DMSO)88,00€10mg116,00€25mg215,00€50mg310,00€100mg450,00€200mg605,00€γ-Mangostin
CAS:Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Fórmula:C23H24O6Pureza:98.55% - 99.08%Cor e Forma:SolidPeso molecular:396.434-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Fórmula:C13H15ClN4Pureza:99.66%Cor e Forma:SolidPeso molecular:262.74SR 57227 hydrochloride
CAS:SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Fórmula:C10H14ClN3·HClPureza:99.89%Cor e Forma:SolidPeso molecular:248.15LOX-IN-3 dihydrochloride monohydrate
CAS:LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.Fórmula:C13H17Cl2FN2O3SCor e Forma:SolidPeso molecular:371.25Ladostigil hydrochloride
CAS:Ladostigil hydrochloride: oral dual cholinesterase and MAO-B/AChE inhibitor; IC50s: 37.1 & 31.8 μM; potential for depression and Alzheimer's research.Fórmula:C16H21ClN2O2Cor e Forma:SolidPeso molecular:308.8Verubecestat TFA
CAS:Verubecestat (MK-8931/SCH 900931), a potent BACE1 inhibitor, shows promise for Alzheimer's, cuts Aβ CSF levels by 92%.Fórmula:C19H18F5N5O5SCor e Forma:SolidPeso molecular:523.435PHA 568487
CAS:PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.Fórmula:C20H24N2O7Cor e Forma:SolidPeso molecular:404.419Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFórmula:C23H27ClFN3O2Pureza:98%Cor e Forma:SolidPeso molecular:431.93Paroxetine maleate
CAS:Paroxetine maleate is a selective inhibitor of serotonin reuptake and an antidepressant.Fórmula:C23H24FNO7Cor e Forma:SolidPeso molecular:445.4433,5-Bis(4-nitrophenoxy)benzoic acid
CAS:3,5-Bis(4-nitrophenoxy)benzoic acid (Compound W) is an inhibitor of γ-secretase. It decreases the released levels of Aβ42 and notch-1 Aβ-like peptide 25.Fórmula:C19H12N2O8Pureza:99.14%Cor e Forma:SolidPeso molecular:396.31JNJ-40411813
CAS:JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).
Fórmula:C20H25ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:344.88Intepirdine
CAS:Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Fórmula:C35H47FN10O8Pureza:97.97%Cor e Forma:SolidPeso molecular:754.85Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Fórmula:C80H122F3N21O22Pureza:99.41%Cor e Forma:SolidPeso molecular:1786.98GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52Ref: TM-T8737
1mg40,00€2mg52,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg113,00€25mg222,00€50mg333,00€100mg495,00€N-ACETYLTRYPTAMINE
CAS:N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Fórmula:C12H14N2OPureza:98.79%Cor e Forma:PowderPeso molecular:202.25PNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFórmula:C13H17ClN2Pureza:97.83%Cor e Forma:SolidPeso molecular:236.74CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Fórmula:C15H24Cl2NO4PPureza:98.75%Cor e Forma:SolidPeso molecular:384.24GALANTHAMINONE
CAS:Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairmentsFórmula:C17H19NO3Pureza:99.93%Cor e Forma:White To Off-White ChemicalPeso molecular:285.34Ref: TM-T7114
2mg39,00€5mg58,00€1mL*10mM (DMSO)84,00€10mg93,00€25mg144,00€50mg200,00€100mg290,00€200mg414,00€Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Fórmula:C18H19ClN4OPureza:98.65% - 99.94%Cor e Forma:SolidPeso molecular:342.82Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Fórmula:C20H30N2O3S2Pureza:99.70%Cor e Forma:White To Off-White SolidPeso molecular:410.59TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.
Fórmula:C25H32N4OPureza:97.87% - 99.9%Cor e Forma:SolidPeso molecular:404.55L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Fórmula:C18H22Cl4N4Pureza:97.52%Cor e Forma:SolidPeso molecular:436.21Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Fórmula:C14H22ClN3O2SCor e Forma:SolidPeso molecular:331.86Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Fórmula:C18H18ClNSPureza:98.77% - 99.756%Cor e Forma:Pale Yellow Crystals SolidPeso molecular:315.86NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Fórmula:C28H29Cl2N3OPureza:98.79%Cor e Forma:SolidPeso molecular:494.46Ref: TM-T28167
500mgA consultar2mg38,00€5mg55,00€1mL*10mM (DMSO)72,00€10mg86,00€25mg155,00€50mg264,00€100mg374,00€Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Fórmula:C79H125N23O22Pureza:98.52%Cor e Forma:SolidPeso molecular:1748.98MPEP hydrochloride
CAS:MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).Fórmula:C14H12ClNPureza:99.87% - >99.99%Cor e Forma:SolidPeso molecular:229.7SSR504734
CAS:SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.Fórmula:C20H20ClF3N2OCor e Forma:SolidPeso molecular:396.836-fluoro-DL-Tryptophan
CAS:6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Fórmula:C11H11FN2O2Pureza:99.25%Cor e Forma:Off-White PowderPeso molecular:222.22β-Amyloid 15-21 acetate
β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.Fórmula:C45H69N9O11Pureza:99.62%Cor e Forma:SolidPeso molecular:912.1Loxapine hydrochloride
CAS:Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Fórmula:C18H19Cl2N3OCor e Forma:SolidPeso molecular:364.27Dicyclomine
CAS:Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.Fórmula:C19H35NO2Cor e Forma:SolidPeso molecular:309.49Lu AF21934
CAS:Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).Fórmula:C14H16Cl2N2O2Pureza:99.79%Cor e Forma:SolidPeso molecular:315.2Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Fórmula:C17H25N3O2SPureza:99.85%Cor e Forma:Light Yellow Or White PowerPeso molecular:335.46VU0467154
CAS:VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Fórmula:C17H15F3N4O3S2Pureza:99.51% - 99.53%Cor e Forma:SolidPeso molecular:444.45Ref: TM-T17244
1mg47,00€2mg63,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg126,00€25mg236,00€50mg400,00€100mg695,00€200mg945,00€pyridostigmine
CAS:Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.Fórmula:C9H13N2O2Pureza:98.10%Cor e Forma:SolidPeso molecular:181.21Ref: TM-T8631
1mg84,00€1mL*10mM (DMSO)159,00€5mg167,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€VU0364770
CAS:VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGluFórmula:C12H9ClN2OPureza:99.65% - >99.99%Cor e Forma:SolidPeso molecular:232.67Succinylcholine Chloride Dihydrate
CAS:Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Cor e Forma:White SolidPeso molecular:397.34Bitopertin
CAS:Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nMFórmula:C21H20F7N3O4SPureza:98.57% - 98.71%Cor e Forma:SolidPeso molecular:543.46PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Fórmula:C16H12N4SPureza:99.35%Cor e Forma:SolidPeso molecular:292.36Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFórmula:C22H25N5O2Pureza:99% - 99.79%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:391.47Ref: TM-T1512
10mg44,00€1mL*10mM (DMSO)48,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Fórmula:C30H34N4OPureza:98.65%Cor e Forma:SolidPeso molecular:466.62Ref: TM-T5387
2mg44,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg170,00€50mg289,00€100mg462,00€200mg658,00€Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Fórmula:C13H12N2OPureza:98.29% - 99.92%Cor e Forma:Off-White SolidPeso molecular:212.25Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Fórmula:C14H22ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:299.80Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83p-Hydroxybenzaldehyde
CAS:1.Fórmula:C7H6O2Pureza:99.05% - 99.86%Cor e Forma:SolidPeso molecular:122.12TG6-10-1
CAS:TG6-10-1 is an EP2 antagonist.Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43Isocarboxazid
CAS:Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.Fórmula:C12H13N3O2Pureza:98.32% - 99.94%Cor e Forma:SolidPeso molecular:231.25Ref: TM-T4559
1mg34,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg90,00€25mg164,00€50mg235,00€100mg350,00€500mg795,00€Tacrine hydrochloride (hydrate)
CAS:Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.Fórmula:C13H14N2·XHCl·XH2OPureza:99.01% - 99.89%Cor e Forma:SolidPeso molecular:234.72Puerarin
CAS:Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.Fórmula:C21H20O9Pureza:98.90% - 99.21%Cor e Forma:Yellow Brown Fine PowderPeso molecular:416.38NS3861
CAS:NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Fórmula:C12H14BrNSPureza:99.853%Cor e Forma:SolidPeso molecular:284.224F 4PP oxalate
CAS:4F 4PP oxalate is a 5-HT2A antagonist.Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Cor e Forma:SolidPeso molecular:429.49

