
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(647 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.027 produtos)
- BACE(37 produtos)
- Beta Amilóide(230 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(373 produtos)
- Gama-secretase(62 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5639 produtos de "Neurociência"
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Glypromate acetate(32302-76-4 free base)
Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.Fórmula:C14H23N3O8Pureza:99.94%Cor e Forma:SolidPeso molecular:361.35Ref: TM-T7778L
2mg37,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg74,00€25mg119,00€50mg160,00€100mg225,00€200mg314,00€Pitofenone
CAS:Pitofenone is an inhibitor of the acetylcholinesterase activity from bovine erythrocytes and electric eel.Fórmula:C22H25NO4Cor e Forma:SolidPeso molecular:367.44Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Fórmula:C23H24FN3O2Pureza:99.2%Cor e Forma:SolidPeso molecular:393.457-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16Mivacurium dichloride
CAS:Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Cor e Forma:Off-White SolidPeso molecular:1100.17Ref: TM-T22371
2mg46,00€5mg65,00€1mL*10mM (DMSO)90,00€10mg94,00€25mg123,00€50mg188,00€100mg286,00€200mg434,00€Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFórmula:C28H33ClN2·2HClPureza:98.05%Cor e Forma:Off-White PowderPeso molecular:505.95Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Fórmula:C22H24ClN3O3SCor e Forma:SolidPeso molecular:445.96FPS-ZM1
CAS:FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.Fórmula:C20H22ClNOPureza:99.32% - 99.52%Cor e Forma:SolidPeso molecular:327.85Ref: TM-T3259
5mg48,00€1mL*10mM (DMSO)50,00€10mg54,00€25mg96,00€50mg140,00€100mg207,00€200mg333,00€500mg560,00€Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Fórmula:C20H24ClN3O2Cor e Forma:SolidPeso molecular:373.88NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Fórmula:C20H23Cl2F2N3O2Pureza:99.59%Cor e Forma:SolidPeso molecular:446.32Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Fórmula:C6H9ClN2O2Pureza:99.39%Peso molecular:176.601GSK-1034702 HCl
CAS:GSK-1034702 HCl is a potent M1 receptor allosteric agonist.Fórmula:C18H25ClFN3O2Cor e Forma:SolidPeso molecular:369.87Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Fórmula:C15H21N5O4SCor e Forma:SolidPeso molecular:367.42Norfluoxetine Hydrochloride
CAS:Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Fórmula:C16H17ClF3NOPureza:99.71%Cor e Forma:SolidPeso molecular:331.76Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Fórmula:C24H25ClFN3O2Cor e Forma:SolidPeso molecular:441.93Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Cor e Forma:SolidPeso molecular:575.61RU 24969 free base
CAS:RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29VU10010
CAS:VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.
Fórmula:C17H16ClN3OSPureza:99.36%Cor e Forma:SolidPeso molecular:345.85Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Fórmula:C10H13ClN2SCor e Forma:SolidPeso molecular:228.74Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.28%Cor e Forma:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Oxotremorine sesquifumarate
CAS:Oxotremorine sesquifumarate is a muscarinic agonist.
Fórmula:C12H18N2OC4H4O4Pureza:97.94%Cor e Forma:SolidPeso molecular:380.39SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Fórmula:C22H25NO2Cor e Forma:SolidPeso molecular:335.44Hemicholinium 3
CAS:Hemicholinium 3 is a potent and selective choline uptake blocker.Fórmula:C24H34Br2N2O4Pureza:98% - 99.95%Cor e Forma:SolidPeso molecular:574.35MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Fórmula:C22H28FNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:373.46Ref: TM-T22359
1mg99,00€5mg187,00€1mL*10mM (DMSO)222,00€10mg280,00€25mg434,00€50mg585,00€100mg775,00€200mg1.054,00€Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Cor e Forma:White SolidPeso molecular:414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Fórmula:C7H14N4O3Pureza:99.89%Cor e Forma:White Crystalline PowderPeso molecular:202.21Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Fórmula:C22H32BrNO5Pureza:98.85%Cor e Forma:SolidPeso molecular:470.4Ref: TM-T28827
1mg74,00€5mg160,00€1mL*10mM (DMSO)165,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€TAT-GluA2 3Y acetate(1404188-93-7 free base)
TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blockedFórmula:C115H185N43O29Pureza:99.43%Cor e Forma:SolidPeso molecular:2634.02Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Fórmula:C35H43N5O4Pureza:98.12%Cor e Forma:SolidPeso molecular:597.75SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFórmula:C22H26ClNO2Pureza:98.02%Cor e Forma:SolidPeso molecular:371.9Ref: TM-T12930
1mg34,00€5mg65,00€1mL*10mM (DMSO)71,00€10mg89,00€25mg167,00€50mg264,00€100mg409,00€200mg590,00€Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Fórmula:C19H22O2Pureza:99.22% - 99.66%Cor e Forma:SolidPeso molecular:282.38PNU-282987 S enantiomer free base
CAS:PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Fórmula:C14H17ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:264.75Ref: TM-T7695
1mg71,00€5mg161,00€1mL*10mM (DMSO)180,00€10mg219,00€25mg338,00€50mg460,00€100mg623,00€200mg837,00€Org 25543 hydrochloride
CAS:Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2).Fórmula:C24H33ClN2O4Pureza:99.26%Cor e Forma:SolidPeso molecular:448.983Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Fórmula:C67H119F3N22O22Pureza:98%Cor e Forma:SolidPeso molecular:1641.79Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Cor e Forma:SolidPeso molecular:485.96Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Cor e Forma:White PowderPeso molecular:390.4Tacrine hydrochloride (hydrate)
CAS:Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.Fórmula:C13H14N2·XHCl·XH2OPureza:99.01% - 99.89%Cor e Forma:SolidPeso molecular:234.72AMN082 free base
CAS:AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.Fórmula:C28H28N2Pureza:97.75% - 97.79%Cor e Forma:SolidPeso molecular:392.54Ref: TM-T21935L
5mg50,00€1mL*10mM (DMSO)52,00€10mg74,00€25mg135,00€50mg212,00€100mg340,00€200mg475,00€NS3861
CAS:NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Fórmula:C12H14BrNSPureza:99.853%Cor e Forma:SolidPeso molecular:284.224F 4PP oxalate
CAS:4F 4PP oxalate is a 5-HT2A antagonist.Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Cor e Forma:SolidPeso molecular:429.49Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.99%Cor e Forma:Solid PowderPeso molecular:556.29Serotonin
CAS:Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Fórmula:C10H12N2OPureza:97.47% - 99.92%Cor e Forma:SolidPeso molecular:176.22(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
CAS:(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).Fórmula:C6H8Cl2N2Pureza:97.23%Cor e Forma:SolidPeso molecular:179.05NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Fórmula:C23H19N3OPureza:99.44% - 99.86%Cor e Forma:SolidPeso molecular:353.42Ref: TM-T2067
2mg34,00€5mg50,00€1mL*10mM (DMSO)58,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€Melatonin
CAS:Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Fórmula:C13H16N2O2Pureza:98% - 99.89%Cor e Forma:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28VU-29
CAS:VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.Fórmula:C22H16N4O3Pureza:99.63%Cor e Forma:SolidPeso molecular:384.39Ref: TM-T23515
2mg33,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg86,00€25mg161,00€50mg259,00€100mg371,00€200mg530,00€Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Fórmula:C58H94O26Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:1207.35NAN-190 hydrobromide
CAS:NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Fórmula:C23H28BrN3O3Pureza:95.20%Cor e Forma:SolidPeso molecular:474.39Medetomidine hydrochloride
CAS:Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.Fórmula:C13H16N2·HClPureza:99.96%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.74JH-II-127
CAS:JH-II-127 is an oral LRRK2 inhibitor with IC50s: 6.6 nM (WT), 2.2 nM (G2019S), 47.7 nM (A2016T).Fórmula:C19H21ClN6O3Pureza:98.32%Cor e Forma:SolidPeso molecular:416.86Ref: TM-T7155
2mg43,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg96,00€25mg166,00€50mg259,00€100mg366,00€200mg520,00€3-AQC
CAS:3-AQC is a competitive antagonist of 5-HT3.Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28Ref: TM-T8007
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg81,00€25mg137,00€50mg215,00€100mg340,00€500mg795,00€Ipratropium Bromide
CAS:Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Fórmula:C20H30BrNO3Pureza:99.92%Cor e Forma:SolidPeso molecular:412.37SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Fórmula:C17H19Cl2NOPureza:98% - 99.83%Cor e Forma:SolidPeso molecular:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€1mL*10mM (DMSO)78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€Mosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFórmula:C21H25ClFN3O3Pureza:99.56%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:421.89(RS)-3-Hydroxyphenylglycine
CAS:(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.Fórmula:C8H9NO3Pureza:99.29%Cor e Forma:SolidPeso molecular:167.16Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Fórmula:C24H23ClF3NPureza:99.99%Cor e Forma:SolidPeso molecular:417.89Ref: TM-T9272
1mg38,00€5mg80,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg222,00€50mg356,00€100mg512,00€200mg735,00€GNE-7915
CAS:GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.Fórmula:C19H21F4N5O3Pureza:98% - ≥95%Cor e Forma:SolidPeso molecular:443.4Ref: TM-T1945
5mg44,00€1mL*10mM (DMSO)48,00€10mg58,00€25mg108,00€50mg177,00€100mg299,00€200mg389,00€500mg645,00€MK-0752
CAS:MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).Fórmula:C21H21ClF2O4SPureza:98% - 99.55%Cor e Forma:SolidPeso molecular:442.9Tianeptine sodium salt
CAS:Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H24ClN2NaO4SPureza:99.82%Cor e Forma:SolidPeso molecular:458.93RO4929097
CAS:RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).Fórmula:C22H20F5N3O3Pureza:98.5% - 99.51%Cor e Forma:SolidPeso molecular:469.4E4CPG
CAS:E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.Fórmula:C11H13NO4Pureza:99.96%Cor e Forma:SolidPeso molecular:223.23CZC-25146
CAS:CZC-25146, a stable LRRK2 inhibitor, IC50: 4.76 nM (wild-type), 6.87 nM (G2019S).Fórmula:C22H25FN6O4SPureza:97.68%Cor e Forma:SolidPeso molecular:488.54KN-92 hydrochloride
CAS:KN-92 hydrochloride is an inactive derivative of KN-93.Fórmula:C24H26Cl2N2O3SPureza:99.68%Cor e Forma:SolidPeso molecular:493.45Tinoridine hydrochloride
CAS:Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.Fórmula:C17H21ClN2O2SPureza:97.49%Cor e Forma:SolidPeso molecular:352.88PBD-150
CAS:PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)Fórmula:C15H20N4O2SPureza:99.68%Cor e Forma:SolidPeso molecular:320.41Venlafaxine
CAS:Venlafaxine (Wy 45030), an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), is used to treat major generalised anxiety disorder (GAD),Fórmula:C17H27NO2Pureza:99.2%Cor e Forma:White Solid CrystallinePeso molecular:277.4Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Fórmula:C20H21N3OPureza:99.17%Cor e Forma:SolidPeso molecular:319.4Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Cor e Forma:SolidPeso molecular:423.53Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Fórmula:C19H15BrClF3N2O3SPureza:99.76%Cor e Forma:SolidPeso molecular:523.75Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Fórmula:C12H17ClN2O2Pureza:99.35%Cor e Forma:SolidPeso molecular:256.73VU-1545
CAS:VU-1545 is mGlu5 positive allosteric modulator.Fórmula:C22H15FN4O3Pureza:98.8%Cor e Forma:SolidPeso molecular:402.38Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Fórmula:C20H17NO6Pureza:98% - 99.99%Cor e Forma:Light Yellow PowderPeso molecular:367.35Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Fórmula:C10H6Cl3N3Pureza:99.78%Cor e Forma:SolidPeso molecular:274.53MK-1064
CAS:MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).Fórmula:C24H20ClN5O3Pureza:99.19% - 99.82%Cor e Forma:SolidPeso molecular:461.9Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.36Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Fórmula:C11H18Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:265.18Gadoteridol
CAS:Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.Fórmula:C17H29GdN4O7Pureza:99.77% - 99.91%Cor e Forma:SolidPeso molecular:558.69Azaphen dihydrochloride monohydrate
CAS:Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Fórmula:C16H23Cl2N5O2Pureza:99.85%Cor e Forma:SolidPeso molecular:388.29(-)-(S)-B-973B
CAS:(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.Fórmula:C24H26F2N6OPureza:99.52%Cor e Forma:SolidPeso molecular:452.5Umibecestat HCl
CAS:Umibecestat HCl (CNP520 HCl) is an efficient β-secretase (BACE1/BACE2) inhibitor that reduces Aβ levels in mice and rats.Fórmula:C19H16Cl2F7N5O2Pureza:99.92%Cor e Forma:SolidPeso molecular:550.26CaM kinase II inhibitor TFA salt
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
Fórmula:C66H117F3N22O21Pureza:>99.99%Cor e Forma:SolidPeso molecular:1611.77Ramosetron hydrochloride
CAS:Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Fórmula:C17H18ClN3OPureza:99.95%Cor e Forma:SolidPeso molecular:315.8Syk Inhibitor II dihydrochloride
CAS:Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Fórmula:C14H17Cl2F3N6OPureza:98.53%Cor e Forma:SolidPeso molecular:413.22Ref: TM-T4391
1mg123,00€2mg200,00€5mg432,00€1mL*10mM (DMSO)432,00€10mg613,00€25mg897,00€50mg1.198,00€100mg1.611,00€γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Fórmula:C6H9NO2Cor e Forma:SolidPeso molecular:127.143Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Cor e Forma:SolidPeso molecular:359.89PF-06447475
CAS:PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.Fórmula:C17H15N5OPureza:98.61% - 99.62%Cor e Forma:SolidPeso molecular:305.33Ralmitaront
CAS:Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).Fórmula:C17H22N4O2Pureza:99.71% - 99.79%Cor e Forma:SolidPeso molecular:314.38Ref: TM-T9183
1mg105,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg401,00€25mg668,00€50mg897,00€100mg1.243,00€200mg1.693,00€BRL-15572 dihydrochloride
CAS:BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Fórmula:C25H27ClN2O·2HClPureza:99.74%Cor e Forma:SolidPeso molecular:479.87(S)-3-Hydroxyphenylglycine
CAS:(S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).Fórmula:C8H9NO3Pureza:99.65%Cor e Forma:SolidPeso molecular:167.16Oxyphencyclimine Hydrochloride
CAS:Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Fórmula:C20H29ClN2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:380.91STO-609
CAS:STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.
Fórmula:C19H10N2O3Pureza:97.14% - 98.8%Cor e Forma:SolidPeso molecular:314.29Ref: TM-T8862
1mg34,00€5mg75,00€1mL*10mM (DMSO)87,00€10mg110,00€25mg245,00€50mg363,00€100mg515,00€200mg702,00€(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Fórmula:C13H17NO2Cor e Forma:SolidPeso molecular:219.284Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Fórmula:C16H19N3O5Pureza:99.76%Cor e Forma:SolidPeso molecular:333.34Ref: TM-T25146
1mg84,00€5mg168,00€1mL*10mM (DMSO)172,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€SB-203186 hydrochloride
CAS:SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81Quipazine
CAS:Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.Fórmula:C13H15N3Cor e Forma:SolidPeso molecular:213.28Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Fórmula:C18H22N2SPureza:99.34% - 99.34%Cor e Forma:SolidPeso molecular:298.45Ref: TM-T2395
1mL*10mM (DMSO)46,00€10mg48,00€25mg65,00€50mg90,00€100mg117,00€200mg203,00€500mg333,00€1g477,00€Eltoprazine dihydrochloride
CAS:Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Fórmula:C12H18Cl2N2O2Pureza:99.64%Cor e Forma:SolidPeso molecular:293.19SSR504734
CAS:SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.Fórmula:C20H20ClF3N2OCor e Forma:SolidPeso molecular:396.83

