
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(648 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.028 produtos)
- BACE(37 produtos)
- Beta Amilóide(231 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(372 produtos)
- Gama-secretase(63 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5637 produtos de "Neurociência"
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Fluoroclorgyline
CAS:Fluoroclorgyline is a specific inhibitor of monoamine oxidase A (MAO-A).Fórmula:C13H15ClFNOPureza:98%Cor e Forma:SolidPeso molecular:255.72RS-0466
CAS:RS-0466 is an β-amyloid-induced cytotoxicity inhibitor.Fórmula:C17H17N5O2Pureza:98%Cor e Forma:SolidPeso molecular:323.35Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Fórmula:C16H13ClN2O4SPureza:98%Cor e Forma:SolidPeso molecular:364.8SIB 1508Y maleate
CAS:neuronal nicotinic ACh receptor agonistFórmula:C16H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:302.33HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Fórmula:C10H12N2O3SPureza:98%Cor e Forma:SolidPeso molecular:240.28AL-37350A
CAS:AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.Fórmula:C14H18N2OCor e Forma:SolidPeso molecular:230.31L 858051
CAS:L 858051 activates adenylate cyclase. It also inhibits glucose transport in rat adipocytes.Fórmula:C29H48N2O7Cor e Forma:SolidPeso molecular:536.7Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Fórmula:C13H19NO2H2O4SPureza:98%Cor e Forma:SolidPeso molecular:270.34Amitifadine hydrochloride
CAS:Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Fórmula:C11H12Cl3NPureza:98%Cor e Forma:SolidPeso molecular:264.58KMS88009
CAS:KMS88009 is an amyloid-β aggregation inhibitor that acts by ameliorating neurodegenerative disorder.Fórmula:C19H19NO2Cor e Forma:SolidPeso molecular:293.36LEK 8841
CAS:LEK 8841 is an ergoline derivative that is a potential antipsychotic.Fórmula:C21H24BrN3O4SPureza:98%Cor e Forma:SolidPeso molecular:494.4GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Fórmula:C16H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:315.37SB 272183
CAS:SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Fórmula:C29H28ClN5OPureza:98%Cor e Forma:SolidPeso molecular:498.02PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Fórmula:C18H23ClN6Pureza:98%Cor e Forma:SolidPeso molecular:358.87Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Fórmula:C17H26N4OPureza:98%Cor e Forma:SolidPeso molecular:302.41S(-)-8-Hydroxy-DPAT hydrobromide
CAS:S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.Fórmula:C16H26BrNOPureza:98%Cor e Forma:SolidPeso molecular:328.29Pivalylbenzhydrazine
CAS:Pivhydrazine: strong MAO inhibitor, stunts rat cartilage growth, used in depression research.Fórmula:C12H18N2OCor e Forma:SolidPeso molecular:206.28E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Fórmula:C20H27Cl2N3O2Pureza:98.88% - 98.88%Cor e Forma:SolidPeso molecular:412.35LY 334370 hydrochloride
CAS:5-HT1F receptor agonistFórmula:C21H23ClFN3OPureza:98%Cor e Forma:SolidPeso molecular:387.88GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFórmula:C15H23N5O2SPureza:99.92%Cor e Forma:SolidPeso molecular:337.44mAChr-in-1
CAS:mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).Fórmula:C23H25IN2O2Pureza:98%Cor e Forma:SolidPeso molecular:488.36Aβ42-IN-1 free base
CAS:Aβ42-IN-1 free base (compound 1v), an orally active γ-secretase modulator with high brain exposure, effectively lowers Aβ42 levels, exhibiting an IC 50 of 0.091Fórmula:C29H26N4O2Pureza:98%Cor e Forma:SolidPeso molecular:462.54PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Fórmula:C20H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:366.41SZV558
CAS:SZV558: Strong MAO-B inhibitor, non-mutagenic, hERG-safe, high-dose tolerant, neuroprotective in PD model.Fórmula:C13H16ClNPureza:98%Cor e Forma:SolidPeso molecular:221.73KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Fórmula:C12H21N5O2Pureza:99.21%Cor e Forma:SolidPeso molecular:267.33Ref: TM-T29038
1mg264,00€1mL*10mM (DMSO)590,00€5mg650,00€10mg888,00€25mg1.369,00€50mg1.783,00€100mg2.250,00€Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Fórmula:C18H14N4O3Pureza:98%Cor e Forma:SolidPeso molecular:334.334-Chloro Trazodone hydrochloride
CAS:4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Fórmula:C19H23Cl2N5OCor e Forma:SolidPeso molecular:408.32Esoxybutynin Chloride
CAS:(S)-oxybutynin, with antimuscarinic effects, is being developed for urinary incontinence.Fórmula:C22H32ClNO3Cor e Forma:SolidPeso molecular:393.95Z-Cyclopentyl-AP4
CAS:Group III mGlu receptor agonistFórmula:C6H12NO5PPureza:98%Cor e Forma:SolidPeso molecular:209.14Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C19H26ClN3O2S2Cor e Forma:SolidPeso molecular:428.01RR-11a
CAS:RR-11a is a synthetic enzyme Legumain inhibitor.
Fórmula:C24H28N6O10Pureza:98%Cor e Forma:SolidPeso molecular:560.51UH-AH 37
CAS:UH-AH 37 is a antagonist of human muscarinic acetylcholine receptor.Fórmula:C21H23Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:420.33NW-1772 free base
CAS:NW-1772 free base is a monoamine oxidase B inhibitor.Fórmula:C18H16ClNO3Cor e Forma:SolidPeso molecular:329.78Tropatepine
CAS:Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.Fórmula:C22H23NSCor e Forma:SolidPeso molecular:333.49Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Fórmula:C15H17Cl2NO2Pureza:99.77%Cor e Forma:SolidPeso molecular:314.21Asoxime dichloride
CAS:Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.Fórmula:C14H16Cl2N4O3Pureza:99.75% - 99.86%Cor e Forma:SolidPeso molecular:359.21Milacemide HCl
CAS:Milacemide HCl is an MAO-B inhibitor and glycine prodrug.Fórmula:C7H17ClN2OPureza:98%Cor e Forma:SolidPeso molecular:180.68PNU-282987 S enantiomer hydrochloride
CAS:(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.Fórmula:C14H18Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:301.21Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Fórmula:C23H29ClN2OCor e Forma:SolidPeso molecular:384.95RJR-2429
CAS:RJR-2429 is a potent AChR agonist.Fórmula:C12H16N2Cor e Forma:SolidPeso molecular:188.27Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Fórmula:C16H17BrN2Pureza:98%Cor e Forma:SolidPeso molecular:317.22Octamylamine sulfamate
CAS:Octamylamine sulfamate is a P450 inhibitor.Fórmula:C13H32N2O3SCor e Forma:SolidPeso molecular:296.47LC kinetic stabilizer-2
CAS:LC Kinetic Stabilizer-2 is a powerful stabilizer for amyloidogenic immunoglobulin light chains (LC), demonstrating significant efficacy with an EC50 of 24 nM.Fórmula:C28H31N3O3Cor e Forma:SolidPeso molecular:457.56Metanicotine
CAS:Metanicotine is a selective nicotinic agonist with antinociceptive properties.Fórmula:C10H14N2Cor e Forma:SolidPeso molecular:162.23AZD-9164 bromide
CAS:AMG-221, a selective 11β-HSD1 inhibitor, suppresses enzyme activity, lowers glucose/insulin, and reduces weight in obese mice.Fórmula:C29H38BrFN2O2Cor e Forma:SolidPeso molecular:545.53CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Fórmula:C5H14NO2PPureza:98%Cor e Forma:SolidPeso molecular:151.14YM-58790
CAS:YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.Fórmula:C27H31N3O2Pureza:99.87%Cor e Forma:SoildPeso molecular:429.55Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Fórmula:C18H12Cl2N2OCor e Forma:SolidPeso molecular:343.21AS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Fórmula:C18H25N3Pureza:98%Cor e Forma:SolidPeso molecular:283.41ASP2535
CAS:ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 can improve cognitiveFórmula:C22H18N6OPureza:98%Cor e Forma:SolidPeso molecular:382.42ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Fórmula:C13H17ClN2Pureza:98%Cor e Forma:SolidPeso molecular:236.74Ref: TM-T23396
1mg44,00€5mg111,00€1mL*10mM (DMSO)123,00€10mg178,00€25mg316,00€50mg470,00€100mg682,00€200mg954,00€Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Fórmula:C37H61BrN2O4Pureza:98%Cor e Forma:SolidPeso molecular:677.8Donitriptan
CAS:Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。Fórmula:C23H25N5O2Pureza:98.76%Cor e Forma:SolidPeso molecular:403.48Aβ42-IN-2
CAS:Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].Fórmula:C24H26N6O2Pureza:98.09% - 99.87%Cor e Forma:SolidPeso molecular:430.5Ref: TM-T9641
1mg42,00€1mL*10mM (DMSO)93,00€5mg94,00€10mg134,00€25mg215,00€50mg304,00€100mg420,00€200mg582,00€LRE1
CAS:LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.Fórmula:C12H13ClN4SPureza:>99.99%Cor e Forma:SolidPeso molecular:280.78ML375
CAS:ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).Fórmula:C23H15ClF2N2O2Cor e Forma:SolidPeso molecular:424.83ML169
CAS:ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).Fórmula:C21H17BrFN3O4SPureza:98%Cor e Forma:SolidPeso molecular:506.34LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.13AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Fórmula:C20H19ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:402.89Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Fórmula:C24H28N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:472.62ML289
CAS:ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.Fórmula:C22H23NO3Pureza:99.54%Cor e Forma:SolidPeso molecular:349.42Ref: TM-T23000
5mg48,00€1mL*10mM (DMSO)49,00€10mg75,00€25mg138,00€50mg212,00€100mg320,00€200mg445,00€TC-N 22A
CAS:TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.Fórmula:C14H13N5SPureza:99.95%Cor e Forma:SolidPeso molecular:283.35SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Fórmula:C18H28N2O3SPureza:98%Cor e Forma:SolidPeso molecular:352.49MAO-B-IN-21
CAS:MAO-B-IN-21: MAO-B inhibitor with antioxidant, anti-amyloid aggregation, neuroprotective properties, BBB permeable, improves memory in Alzheimer's mice.Fórmula:C24H25ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:440.92LRRK2-IN-10
CAS:LRRK2-IN-10 (compound 34) is a potent, mutation-selective, brain-penetrant inhibitor targeting G2019S-LRRK2 kinase with IC50 values of 11 nM for G2019S-LRRK2Fórmula:C20H15N5OPureza:98%Cor e Forma:SolidPeso molecular:341.37Piperilate HCl
CAS:Piperilate HCl is an antispasmodic, antimuscarinic agent. It is a muscarinic cholinergic receptor antagonist.Fórmula:C21H26ClNO3Cor e Forma:SolidPeso molecular:375.89Nexopamil racemate
CAS:Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.Fórmula:C24H40N2O3Pureza:98.61%Cor e Forma:SolidPeso molecular:404.59OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4SLV-310
CAS:SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Fórmula:C25H24FN3O2Pureza:99.39%Cor e Forma:SolidPeso molecular:417.48Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Fórmula:C11H16N2OPureza:98%Cor e Forma:SolidPeso molecular:192.26Chlorisondamine chloride
CAS:Chlorisondamine chloride: a nicotinic antagonist, mainly for animal research, former antihypertensive.Fórmula:C14H20Cl6N2Cor e Forma:SolidPeso molecular:429.03BuChE-IN-6
CAS:BuChE-IN-6 inhibits BuChE (IC50: 0.46 μM eqBuChE, 0.51 μM hBuChE) and prevents Aβ 42 self-aggregation.Fórmula:C21H26N4O2Cor e Forma:SolidPeso molecular:366.46AChE/BChE/MAO-B-IN-3
AChE/BChE/MAO-B-IN-3: potent MAO-B, AChE & BChE inhibitor; IC50: 0.0359μM (MAO-B), 0.0473/0.0782μM (AChE/BChE); possible Alzheimer's research use.Fórmula:C25H31N3O3Cor e Forma:SolidPeso molecular:421.53AChE-IN-20
CAS:AChE-IN-20: AChE inhibitor (IC50: 397.32 nM), hCA-I/II blocker (IC50: ~77 nM avg), α GLY suppressor (IC50: 52.08 nM).Fórmula:C22H20N8O6S2Cor e Forma:SolidPeso molecular:556.57Territrem B
CAS:Territrem B: A mycotoxin that irreversibly blocks AChE, causes tremors in mice at 0.21 mg/kg.Fórmula:C29H34O9Cor e Forma:SolidPeso molecular:526.57BMS-902483
CAS:BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.Fórmula:C18H20N4OPureza:98%Cor e Forma:SolidPeso molecular:308.38AC-42
CAS:AC-42 is an allosteric agonist of M1 muscarinic receptor.
Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Fórmula:C22H19N5Cor e Forma:SolidPeso molecular:353.42AChE/BChE-IN-8
CAS:AChE/BChE-IN-8 inhibits AChE (Ki=0.788 μM) & BChE (Ki=2.364 μM), crosses the blood-brain barrier, and is low in cytotoxicity.Fórmula:C26H32N2O2Cor e Forma:SolidPeso molecular:404.54γ-Secretase modulator 12
CAS:γ-Secretase modulator 12 (Compound 1a) is a selective compound that effectively reduces amyloid-β42 (Aβ42) levels with an IC50 of 0.39 μM.Fórmula:C25H23N3O2Cor e Forma:SolidPeso molecular:397.47Oxybutynin R-isomer HCl
CAS:Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.Fórmula:C22H32ClNO3Cor e Forma:SolidPeso molecular:393.95GR-55562 dihydrobromide
CAS:GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93Alvameline maleate
CAS:Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.Fórmula:C13H19N5O4Cor e Forma:SolidPeso molecular:309.32BACE1-IN-12
CAS:BACE1-IN-12: potent BACE1 and BuChE inhibitor, IC50s - 8.9 μM and 3.2 μM, blood-brain barrier permeable, anti-Alzheimer's potential.Fórmula:C29H28Cl2N6OCor e Forma:SolidPeso molecular:547.48Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48Befloxatone
CAS:Befloxatone is a potent, selective and reversible inhibitor of monoamine oxidase A.Fórmula:C15H18F3NO5Cor e Forma:SolidPeso molecular:349.3SD-6
CAS:SD-6, oral hAChE/hBChE inhibitor (IC50: 0.907/1.579 µM), crosses BBB, non-toxic, for Alzheimer's research.Fórmula:C20H22N4OSCor e Forma:SolidPeso molecular:366.48Belaperidone
CAS:Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.Fórmula:C22H22FN3O2Cor e Forma:SolidPeso molecular:379.43sEH inhibitor-5
CAS:sEH inhibitor-5 is a potent inhibitor of sEH (soluble epoxide hydrolase) (IC50: 0.1 nM).Fórmula:C27H26Cl2N6O3SCor e Forma:SolidPeso molecular:585.5Yhhu-3792
CAS:Yhhu-3792 activates Notch, boosts Hes3/Hes5, enhances NSC renewal, expands NSC pool, and may improve memory.Fórmula:C24H24N4O2Cor e Forma:SolidPeso molecular:400.47GABAA receptor agent 7
CAS:Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.Fórmula:C18H13ClN4OCor e Forma:SolidPeso molecular:336.77Caroxazone
CAS:Caroxazone is an antidepressant drug, monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective meanwhile.Fórmula:C10H10N2O3Cor e Forma:SolidPeso molecular:206.2(R)-Oxybutynin
CAS:(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.Fórmula:C22H31NO3Cor e Forma:SolidPeso molecular:357.49BACE2-IN-1
CAS:BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.Fórmula:C36H38F3N3O3Cor e Forma:SolidPeso molecular:617.7LSP4-2022
CAS:LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.Fórmula:C13H18NO8PPureza:100%Cor e Forma:SolidPeso molecular:347.26UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Fórmula:C6H12NaO3Cor e Forma:SolidPeso molecular:155.149(RS)-4-Carboxy-3-hydroxyphenylglycine
CAS:broad spectrum EAA agonist/antagonistFórmula:C9H9NO5Pureza:98%Cor e Forma:SolidPeso molecular:211.17Chlorpyrifos-oxon
CAS:Chlorpyrifos-oxon, an active metabolite of Chlorpyrifos, is a potent phosphorylating agent that significantly inhibits AChE activity and induces cross-linking between tubulin subunits, thereby disrupting microtubule function [4].Fórmula:C9H11Cl3NO4PCor e Forma:SolidPeso molecular:334.52sEH/AChE-IN-1
CAS:Compound 12a is a dual sEH/AChE inhibitor with potential for treating Alzheimer's-related neuroinflammation and memory loss.Fórmula:C29H31ClF3N5O3Cor e Forma:SolidPeso molecular:590.04Phenglutarimid
CAS:Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.Fórmula:C17H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:288.38

