
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(648 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.028 produtos)
- BACE(37 produtos)
- Beta Amilóide(231 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(373 produtos)
- Gama-secretase(63 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5639 produtos de "Neurociência"
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5-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31Sulfoxaflor
CAS:Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.Fórmula:C10H10F3N3OSPureza:99.56% - 99.98%Cor e Forma:SolidPeso molecular:277.27Ref: TM-T19940
1mg100,00€1mL*10mM (DMSO)245,00€5mg275,00€10mg384,00€25mg572,00€50mg780,00€100mg1.018,00€250mg2.080,00€(-)-Donepezil
CAS:(-)-Donepezil is an isomer of Donepezil -- a nootropic acting as an inhibitor of acetylcholinesterase.Fórmula:C24H29NO3Cor e Forma:SolidPeso molecular:379.49SV5
CAS:SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.Fórmula:C21H30N2O4S2Cor e Forma:SolidPeso molecular:438.6MAO-B-IN-15
CAS:MAO-B-IN-15 selectively inhibits MAO-B, targeting Tyr 326 (IC50 = 13.5 μM), useful for Parkinson's research.Fórmula:C17H18FNO2Cor e Forma:SolidPeso molecular:287.335-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Fórmula:C20H21ClN2O3Cor e Forma:SolidPeso molecular:372.85PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Cor e Forma:SolidPeso molecular:267.37AChE/BuChE-IN-1
CAS:AChE/BuChE-IN-1: BuChE inhibitor (IC50=0.48µM), weaker AChE blocker (IC50=7.16µM), ·OH scavenger (IC50=0.1674µM), may aid in AD research.Fórmula:C19H19NO4Cor e Forma:SolidPeso molecular:325.36Pralidoxime
CAS:Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.Fórmula:C7H9N2OCor e Forma:SolidPeso molecular:137.16VU6001966
CAS:VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.Fórmula:C17H15FN4O2Pureza:98%Cor e Forma:SolidPeso molecular:326.33Aβ Fibrillization modulator 1
CAS:Aβ Fibrillization Modulator 1 stabilizes amyloid-beta (Aβ) monomers, preventing their aggregation into fibrils.Fórmula:C17H12N4O3SSeCor e Forma:SolidPeso molecular:431.33BMS-911172
CAS:BMS-911172 is an adaptor associated kinase 1 (AAK1 kinase) inhibitor with an IC 50 of 35 nM.Fórmula:C16H19F2N3O3Cor e Forma:SolidPeso molecular:339.34FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Fórmula:C22H19N5Cor e Forma:SolidPeso molecular:353.42γ-Secretase modulator 12
CAS:γ-Secretase modulator 12 (Compound 1a) is a selective compound that effectively reduces amyloid-β42 (Aβ42) levels with an IC50 of 0.39 μM.Fórmula:C25H23N3O2Cor e Forma:SolidPeso molecular:397.47SSAO inhibitor-2
CAS:SSAO inhibitor-2 targets human SSAO (<10 nM) and MAO-A (10-100 μM); useful in various diseases research.Fórmula:C14H21FN4O2Cor e Forma:SolidPeso molecular:296.34Sultroponium
CAS:Sultroponium may be used as an anticholinergic agent or antispasmodic.Fórmula:C20H29NO6SCor e Forma:SolidPeso molecular:411.51Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.485-HT6/5-HT2A receptor ligand-2
CAS:Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.Fórmula:C20H18FN3O2Cor e Forma:SolidPeso molecular:351.37Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Fórmula:C32H44N4O3Pureza:98%Cor e Forma:SolidPeso molecular:532.72RX 67668
CAS:RX 67668: Muscle relaxant, relieves fatigue; cholinesterase inhibitor (IC50: 5 μM); reverses D-tubocurarine effects.Fórmula:C16H24ClNPureza:98%Cor e Forma:SolidPeso molecular:265.82Bornaprine
CAS:Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.Fórmula:C21H31NO2Cor e Forma:SolidPeso molecular:329.48CP-809101
CAS:CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Fórmula:C15H17ClN4OPureza:98%Cor e Forma:SolidPeso molecular:304.77Org-13011 fumarate
CAS:Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.Fórmula:C22H29F3N4O5Pureza:98.92%Cor e Forma:SolidPeso molecular:486.48Enciprazine
CAS:Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Fórmula:C23H32N2O6Pureza:98.63%Cor e Forma:SolidPeso molecular:432.51Dihydro Donepezil
CAS:Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).Fórmula:C24H31NO3Cor e Forma:SolidPeso molecular:381.51UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Fórmula:C6H12NaO3Cor e Forma:SolidPeso molecular:155.149ENS-163 phosphate
CAS:Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.Fórmula:C11H19N2O5PSPureza:98%Cor e Forma:SolidPeso molecular:322.32S 14063
CAS:S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Fórmula:C22H22FN3O5SCor e Forma:SolidPeso molecular:459.49RS 56812 hydrochloride
CAS:5-HT3 partial agonistFórmula:C18H22ClN3O2Pureza:98.62%Cor e Forma:SolidPeso molecular:347.84A-794282
CAS:A-794282 is a selective antagonist of mGluR1.Fórmula:C19H18N4OSPureza:99.87%Cor e Forma:SolidPeso molecular:350.44Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Fórmula:C24H32N4O2SPureza:99.74%Cor e Forma:SolidPeso molecular:440.6Ref: TM-T24885
1mg123,00€5mg293,00€1mL*10mM (DMSO)354,00€10mg537,00€25mg863,00€50mg1.161,00€100mg1.558,00€ABP688
CAS:ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.Fórmula:C15H16N2OPureza:98.63%Cor e Forma:SolidPeso molecular:240.3Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Fórmula:C15H21ClN6Pureza:99.33% - 99.46%Cor e Forma:SolidPeso molecular:320.82Ref: TM-T25672
1mg133,00€1mL*10mM (DMSO)323,00€5mg324,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€500mg2.872,00€5HT6-ligand-1
CAS:5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Fórmula:C20H22BrN3O2SPureza:99.24% - 99.93%Cor e Forma:SolidPeso molecular:448.38DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Fórmula:C14H12FNOPureza:99.51% - 99.56%Cor e Forma:SolidPeso molecular:229.25Ref: TM-T11106
1mg109,00€2mg163,00€1mL*10mM (DMSO)208,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€Panadiplon
CAS:Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment ofFórmula:C18H17N5O2Pureza:98.30% - 98.94%Cor e Forma:SolidPeso molecular:335.36Nexopamil
CAS:Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Fórmula:C24H40N2O3Pureza:97.87% - >99.99%Cor e Forma:SolidPeso molecular:404.59Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Fórmula:C18H19FN2O3SPureza:97.61% - 99.99%Cor e Forma:SolidPeso molecular:362.42Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Fórmula:C10H17IN2O2Pureza:99.81%Cor e Forma:SolidPeso molecular:324.16Ref: TM-T25538
1mg50,00€5mg106,00€1mL*10mM (DMSO)117,00€10mg168,00€25mg339,00€50mg512,00€100mg748,00€200mg1.026,00€LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Fórmula:C21H25ClN2O2Pureza:99.47%Cor e Forma:SolidPeso molecular:372.89LY-2624803
CAS:LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Fórmula:C22H25N3O3Pureza:99.78% - 99.97%Cor e Forma:SolidPeso molecular:379.45MK-3328
CAS:MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.Fórmula:C14H9FN4OPureza:99.77% - >99.99%Cor e Forma:SolidPeso molecular:268.25Ref: TM-T16094
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Fórmula:C21H31NO2Pureza:99.90% - 99.99%Cor e Forma:SolidPeso molecular:329.48NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C22H20N4OPureza:99.7% - 99.82%Cor e Forma:SolidPeso molecular:356.42Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Fórmula:C23H26N2OPureza:98.03% - 98.93%Cor e Forma:SolidPeso molecular:346.47MM 77 dihydrochloride
CAS:MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.Fórmula:C19H29Cl2N3O3Pureza:99.91%Cor e Forma:SolidPeso molecular:418.36Ref: TM-T23007
1mg86,00€5mg157,00€10mg215,00€1mL*10mM (DMSO)281,00€25mg472,00€50mg687,00€100mg938,00€500mg1.882,00€Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Fórmula:C15H14ClN3O3Pureza:99.46%Cor e Forma:SolidPeso molecular:319.74amyloid P-IN-1
CAS:amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer's disease, amyloidosis, osteoarthritis, andFórmula:C30H44N2O14Pureza:99.76%Cor e Forma:SolidPeso molecular:656.68ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Fórmula:C14H16ClN3OPureza:>99.99%Cor e Forma:SolidPeso molecular:277.75ML 10302 hydrochloride
CAS:ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Fórmula:C15H22Cl2N2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:349.25GSK233705
CAS:GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.Fórmula:C24H29BrN2Pureza:99.87% - 99.98%Cor e Forma:SolidPeso molecular:425.4SB228357
CAS:SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Fórmula:C22H17F4N3O2Pureza:99.82%Cor e Forma:SolidPeso molecular:431.38Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Fórmula:C21H24N2Pureza:99.77%Cor e Forma:SolidPeso molecular:304.43(E/Z)-SIB-1893
CAS:(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.Fórmula:C14H13NPureza:99.96%Cor e Forma:SolidPeso molecular:195.26Aβ-IN-1
CAS:Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).Fórmula:C35H49NPureza:99.1%Cor e Forma:SoildPeso molecular:483.77Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFórmula:C13H19NO3Pureza:99.65%Cor e Forma:SolidPeso molecular:237.29Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Fórmula:C24H31N5O2Pureza:99.79%Cor e Forma:SolidPeso molecular:421.54Ref: TM-T16411
1mg44,00€5mg79,00€1mL*10mM (DMSO)87,00€10mg114,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Fórmula:C8H6ClF3N2OSPureza:99.76%Cor e Forma:SolidPeso molecular:270.66CT-179
CAS:CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.Fórmula:C17H22Cl2N6OPureza:98.67%Cor e Forma:SolidPeso molecular:397.3NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Fórmula:C21H23ClN2O3Pureza:99.92%Cor e Forma:SolidPeso molecular:386.87BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFórmula:C19H20Cl2N2OPureza:99.43% - 99.95%Cor e Forma:SolidPeso molecular:363.28RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Fórmula:C21H19F2N3O3Pureza:99.57% - 99.95%Cor e Forma:SolidPeso molecular:399.39Ref: TM-T16811
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Fórmula:C19H27N3OPureza:99.52%Cor e Forma:SolidPeso molecular:313.44E6801
CAS:E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Fórmula:C17H18ClN5O2S2Pureza:96.32% - 97.24%Cor e Forma:SolidPeso molecular:423.94ATC 0175
CAS:ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Fórmula:C23H26ClF2N5OPureza:99.98%Cor e Forma:SolidPeso molecular:461.93Xanomeline
CAS:Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Fórmula:C14H23N3OSPureza:99.61%Cor e Forma:SolidPeso molecular:281.42Goxalapladib
CAS:Goxalapladib(GSK 677116) is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Fórmula:C40H39F5N4O3Pureza:99.64% - 99.93%Cor e Forma:SolidPeso molecular:718.75Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Fórmula:C22H22N2O7Pureza:99.66%Cor e Forma:SolidPeso molecular:426.42Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Fórmula:C18H21NSPureza:99.76% - >99.99%Cor e Forma:SolidPeso molecular:283.43LY266097 hydrochloride
CAS:LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.
Fórmula:C21H24Cl2N2O2Pureza:98.58%Cor e Forma:SolidPeso molecular:407.33RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Fórmula:C19H23ClN2OPureza:99.70%Cor e Forma:SolidPeso molecular:330.85Ref: TM-T20739
1mg158,00€1mL*10mM (DMSO)349,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€CP-810123
CAS:CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.Fórmula:C14H18N4OPureza:98.63% - 99.60%Cor e Forma:SolidPeso molecular:258.32CPCCOEt
CAS:CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1bFórmula:C13H13NO4Pureza:99.91%Cor e Forma:SolidPeso molecular:247.25Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFórmula:C9H15NO2Pureza:>99.99%Cor e Forma:SolidPeso molecular:169.22Cilansetron
CAS:Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Fórmula:C20H21N3OPureza:99.82% - 99.98%Cor e Forma:SolidPeso molecular:319.4PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Fórmula:C15H17N3O2Pureza:99.43% - 99.96%Cor e Forma:SolidPeso molecular:271.31Ref: TM-T23145
1mg52,00€1mL*10mM (DMSO)100,00€5mg102,00€10mg166,00€25mg358,00€50mg610,00€100mg895,00€500mg1.945,00€H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Fórmula:C11H15Cl2N3O2SPureza:97.3%Cor e Forma:SolidPeso molecular:324.23Sudoxicam
CAS:Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema
Fórmula:C13H11N3O4S2Pureza:99.93%Cor e Forma:SolidPeso molecular:337.37Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFórmula:C24H27FN4O2Pureza:97.86%Cor e Forma:SolidPeso molecular:422.5Ecopipam
CAS:Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Fórmula:C19H20ClNOPureza:99.68%Cor e Forma:SolidPeso molecular:313.82CBiPES hydrochloride
CAS:CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.Fórmula:C21H20ClN3O2SPureza:99.66%Cor e Forma:SolidPeso molecular:413.92Lecozotan HCl
CAS:Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Fórmula:C28H30ClN5O3Pureza:99.04%Cor e Forma:SolidPeso molecular:520.02Ensaculin
CAS:Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Fórmula:C26H32N2O5Pureza:99.56% - 99.81%Cor e Forma:SolidPeso molecular:452.54Agomelatine hydrochloride
CAS:Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Fórmula:C15H18ClNO2Pureza:99.57%Cor e Forma:SolidPeso molecular:279.76ASM-024
CAS:ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Fórmula:C15H25N2Pureza:99.74%Cor e Forma:SolidPeso molecular:233.37RS 67333 hydrochloride
CAS:RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Fórmula:C19H30Cl2N2O2Pureza:98.78%Cor e Forma:SolidPeso molecular:389.36Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Cor e Forma:SolidPeso molecular:295.34Buntanetap
CAS:Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular diseaseFórmula:C20H23N3O2Pureza:98.2%Cor e Forma:SolidPeso molecular:337.42Ref: TM-T17312
1mg177,00€5mg447,00€1mL*10mM (DMSO)492,00€10mg713,00€25mg1.333,00€50mg1.935,00€100mg2.520,00€LSN2463359
CAS:LSN2463359 is a positive allosteric modulators of the mGlu5 receptor.Fórmula:C16H15N3OPureza:99.26%Cor e Forma:SolidPeso molecular:265.31Ref: TM-T27854
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg80,00€25mg161,00€50mg245,00€100mg363,00€200mg515,00€Sarizotan HCl
CAS:Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Fórmula:C22H22ClFN2OPureza:96%Cor e Forma:SolidPeso molecular:384.87SB-215505
CAS:SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Fórmula:C19H16ClN3OPureza:98.33%Cor e Forma:SolidPeso molecular:337.8Fengabine
CAS:Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Fórmula:C17H17Cl2NOPureza:99.37%Cor e Forma:SolidPeso molecular:322.23Dipraglurant
CAS:Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.Fórmula:C16H12FN3Pureza:98.7%Cor e Forma:SolidPeso molecular:265.29Ref: TM-T15134
1mg92,00€5mg215,00€1mL*10mM (DMSO)260,00€10mg313,00€25mg685,00€50mg1.009,00€100mg1.341,00€Itasetron
CAS:Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.
Fórmula:C16H20N4O2Pureza:98.58% - 99.33%Cor e Forma:SolidPeso molecular:300.36MNI 137
CAS:MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.Fórmula:C15H9BrN4OPureza:97.49%Cor e Forma:SolidPeso molecular:341.16Cianopramine
CAS:Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Fórmula:C20H23N3Pureza:99.92% - 99.92%Cor e Forma:SolidPeso molecular:305.42Piromelatine
CAS:Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFórmula:C17H16N2O4Pureza:99.83%Cor e Forma:SolidPeso molecular:312.32Ref: TM-T34081
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€Glutaminyl Cyclase Inhibitor 1
CAS:Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor (IC50: 0.5 μM) that can be used to study neurological disorders.Fórmula:C21H24FN3O2Pureza:99.81%Cor e Forma:SolidPeso molecular:369.43Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Fórmula:C19H21N3SPureza:97.01%Cor e Forma:SolidPeso molecular:323.46

