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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5400 produtos de "Neurociência"

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  • Furosemide

    CAS:
    <p>Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chronic renal insufficiency.</p>
    Fórmula:C12H11ClN2O5S
    Pureza:99.32% - 99.89%
    Cor e Forma:Crystals From Aqueous Ethanol Tasteless (Ntp 1992)
    Peso molecular:330.744
  • NMDA receptor antagonist 6


    <p>NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotective</p>
    Fórmula:C25H23NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:369.46
  • TC-2216

    CAS:
    <p>TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.</p>
    Fórmula:C12H17N3
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:203.28
  • 3-Chloroamphetamine hydrochloride

    CAS:
    <p>3-Chloroamphetamine hydrochloride is a derivative of amphetamine that acts as a central nervous system stimulant by releasing serotonin and dopamine.</p>
    Fórmula:C9H13Cl2N
    Cor e Forma:Solid
    Peso molecular:206.11
  • 5-HT2A receptor agonist-6

    CAS:
    <p>5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.</p>
    Fórmula:C18H19N3O3
    Cor e Forma:Solid
    Peso molecular:325.36
  • 4-Hydroxy MPT

    CAS:
    <p>4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.</p>
    Fórmula:C14H20N2O
    Cor e Forma:Solid
    Peso molecular:232.32
  • Methalthiazide

    CAS:
    <p>Methalthiazide enhances the activity of natural agonists of AMPA receptors and can be utilized in schizophrenia research.</p>
    Fórmula:C12H16ClN3O4S3
    Cor e Forma:Solid
    Peso molecular:397.92
  • γ-DGG TFA

    CAS:
    <p>Gamma-DGG TFA is an antagonist of excitatory amino acids that can inhibit depolarization induced by NMDA, Kainate, and Quisqualate. In addition, it counteracts excitatory postsynaptic potentials (e.p.s.p.) in rat hippocampal slices.</p>
    Fórmula:C9H13F3N2O7
    Cor e Forma:Solid
    Peso molecular:318.2
  • Pridinol hydrochloride

    CAS:
    <p>Pridinolhydrochloride is the hydrochloride form of Pridinol. Pridinol hydrochloride is an orally active anticholinergic agent, which can also be used as a muscle relaxant.</p>
    Fórmula:C20H26ClNO
    Cor e Forma:Solid
    Peso molecular:331.88
  • Timegadine hydrochloride

    CAS:
    <p>Timegadine hydrochloride (SR1368 hydrochloride) is the hydrochloride salt form of Timegadine. It is an orally active inhibitor of COX and lipo-oxygenase, effectively suppressing COX in rabbit platelets and rat brain with IC50 values of 5 nM and 20 μM, respectively, and inhibiting lipo-oxygenase in horse and rabbit platelets with an IC50 of 100 μM. Timegadine hydrochloride also exhibits anti-arthritis activity.</p>
    Fórmula:C20H24ClN5S
    Cor e Forma:Solid
    Peso molecular:401.96
  • (-)-2-Phenylpropylamine

    CAS:
    <p>(-)-2-Phenylpropylamine ((S)-2-Phenylpropylamine) (compound 3b) functions as an inhibitor for both MAO-A and MAO-B, with Ki values of 584 μM and 156 μM, respectively.</p>
    Fórmula:C9H13N
    Cor e Forma:Solid
    Peso molecular:135.21
  • SIB 1553A

    CAS:
    <p>SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.</p>
    Fórmula:C13H19NOS
    Pureza:99.79%
    Cor e Forma:Soild
    Peso molecular:237.36
  • mHTT-IN-1

    CAS:
    <p>mHTT-IN-1 is a potent inhibitor of toxic mHTT, linked to Huntington's disease, with an EC50 of 46 nM.</p>
    Fórmula:C18H19N7OS
    Cor e Forma:Solid
    Peso molecular:381.45
  • LY3020371

    CAS:
    <p>LY3020371: potent, selective mGlu 2/3 receptor antagonist with Ki of 5.26 nM (hmGluR2) and 2.50 nM (hmGluR3); key in depression studies.</p>
    Fórmula:C15H15F2NO5S
    Cor e Forma:Solid
    Peso molecular:359.34
  • (-)-Eseroline fumarate

    CAS:
    <p>(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.</p>
    Fórmula:C17H22N2O5
    Cor e Forma:Solid
    Peso molecular:334.37
  • CVN417


    <p>CVN417 is an orally active antagonist of nAChR containing the α6 subunit, modulating phasic dopaminergic neurotransmission in an impulse-dependent fashion.</p>
    Cor e Forma:Odour Solid
  • Ro60-0175

    CAS:
    <p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>
    Fórmula:C11H12ClFN2
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:226.68
  • Desfesoterodine

    CAS:
    <p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>
    Fórmula:C22H31NO2
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:341.49
  • CZC-54252 hydrochloride

    CAS:
    <p>CZC-54252 hydrochloride: selective LRRK2 inhibitor; IC50 = 1.85/1.28 nM (wild-type/G2019S); neuroprotective; EC50 = 1 nM for G2019S injury.</p>
    Fórmula:C22H26Cl2N6O4S
    Pureza:98.21%
    Cor e Forma:Solid
    Peso molecular:541.45
  • Tiquizium

    CAS:
    <p>Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.</p>
    Fórmula:C19H24NS2
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:330.53