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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5389 produtos de "Neurociência"

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  • Dehydrodiscretamine chloride

    CAS:
    <p>Dehydrodiscretamine chloride, a dual inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), exhibits IC50 values of 17.8 μM and 118.8 μM,</p>
    Fórmula:C19H18ClNO4
    Cor e Forma:Solid
    Peso molecular:359.8
  • VU6028418

    CAS:
    <p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>
    Cor e Forma:Solid
  • Bis-(-)-8-demethylmaritidine


    <p>Bis-(-)-8-demethylmaritidine, a natural alkaloid, serves as a potent inhibitor of acetylcholinesterase (AChE) and is utilized in Alzheimer's disease research [1</p>
    Cor e Forma:Odour Solid
  • BChE-IN-12

    CAS:
    <p>BChE-IN-12, non-competitive BChE inhibitor from Bletilla striata, IC50=2.3μM; potential Alzheimer’s research.</p>
    Fórmula:C31H30O5
    Cor e Forma:Solid
    Peso molecular:482.57
  • 1H-Indole-3-carboxylic acid, 5-[2-hydroxy-3-[[2-hydroxy-1,1-bis(hydroxymethyl)ethyl]amino]propoxy]-2-methyl-1-(4-methylphenyl)-, ethyl ester

    CAS:
    <p>Compound 5936-0108对β-淀粉样蛋白可能具有调节作用。</p>
    Fórmula:C26H34N2O7
    Pureza:99.44%
    Cor e Forma:Soild
    Peso molecular:486.56
  • Heliosupine


    <p>Heliosupine is a useful organic compound for research related to life sciences and the catalog number is T125038.</p>
    Fórmula:C20H31NO7
    Cor e Forma:Solid
    Peso molecular:397.468
  • β-Amyloid (1-11)

    CAS:
    <p>Anionic interaction of Beta-amyloid (1-11) with Factor XII is suspected to cause massive activation of the C4 (complement 4) system in the cerebrospinal fluid</p>
    Fórmula:C56H76N16O22
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1325.3
  • LP 12 hydrochloride

    CAS:
    <p>LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).</p>
    Fórmula:C32H40ClN3O
    Cor e Forma:Solid
    Peso molecular:518.14
  • RuBi-GABA

    CAS:
    <p>Ruthenium-bipyridine-triphenylphosphine caged GABA</p>
    Fórmula:C42H39F6N5O2P2Ru
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:922.8
  • 4-Methoxyphenyl isothiocyanate

    CAS:
    <p>4-Methoxyphenyl isothiocyanate (4-Methylphenyl ITC) is recognized as an antioxidant demonstrating an IC50 of 1.25 mM for scavenging DPPH free radicals. Its antioxidant capacity, as shown by the ORAC test, is 11.7 mM TE, equivalent to the efficacy of 11.7 mmol Trolox under similar conditions. Additionally, it extends the oxidation process in the Briggs–Rauscher reaction by approximately 9180 seconds. The compound also exhibits moderate cholinesterase inhibitory activity, with an inhibition rate of 30.4% for acetylcholinesterase (AChE) and 17.9% for butyrylcholinesterase (BChE). Research suggests 4-Methoxyphenyl isothiocyanate holds promise for applications in antioxidant and neurological disorder studies.</p>
    Fórmula:C8H7NOS
    Cor e Forma:Solid
    Peso molecular:165.21
  • AHN-683

    CAS:
    AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.
    Fórmula:C42H32FN3O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:709.72
  • nAChR agonist 2

    CAS:
    <p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>
    Fórmula:C11H16N2
    Cor e Forma:Solid
    Peso molecular:176.263
  • Anabaseine

    CAS:
    <p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>
    Fórmula:C10H12N2
    Cor e Forma:Solid
    Peso molecular:160.22
  • JF-NP-26


    <p>Releases pain-blocking raseglurant under 405 nm light. Inhibits Quisqualate. Analgesic in vivo. Quantum yield: 0.18.</p>
    Cor e Forma:Solid
  • β-Amyloid (1-15)

    CAS:
    <p>β-Amyloid (1-15) (Amyloid β-Protein (1-15)) is a fragment of β-amyloid protein used in the study of Alzheimer's disease.</p>
    Fórmula:C78H107N25O27
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:1826.84
  • LY3027788 hydrochloride

    CAS:
    <p>LY3027788 HCl, potent oral prodrug of LY3020371, targets mGlu2/3 with antidepressant effects.</p>
    Fórmula:C25H32ClF2NO11S
    Cor e Forma:Solid
    Peso molecular:628.03
  • Syk Inhibitor II hydrochloride

    CAS:
    <p>Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.</p>
    Fórmula:C14H16ClF3N6O
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:376.77
  • (S)-AMPA HCl


    <p>(S)-AMPA HCl (L-AMPA HCl) is a selective AMPA receptor agonist with potential antidepressant activity. It can be used in research on Parkinson's disease.</p>
    Fórmula:C7H11ClN2O4
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:222.63
  • Deoxynojirimycin Tetrabenzyl Ether

    CAS:
    <p>Deoxynojirimycin tetrabenzyl ether aids in making 1-dNM, a strong α-glucosidase I &amp; II blocker.</p>
    Fórmula:C34H37NO4
    Cor e Forma:Solid
    Peso molecular:523.673
  • LY3027788

    CAS:
    <p>LY3027788, potent oral prodrug of LY3020371, is a strong mGlu2/3 antagonist with notable antidepressant effects.</p>
    Fórmula:C25H31F2NO11S
    Cor e Forma:Solid
    Peso molecular:591.58