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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5390 produtos de "Neurociência"

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  • PNU-282987 S enantiomer free base

    CAS:
    <p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>
    Fórmula:C14H17ClN2O
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:264.75
  • Pikamilone

    CAS:
    <p>Pikamilone (Picamilon) is an intelligent medicine.</p>
    Fórmula:C10H12N2O3
    Pureza:99.38%
    Cor e Forma:White Crystalline Powder
    Peso molecular:208.21
  • Serotonin

    CAS:
    <p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>
    Fórmula:C10H12N2O
    Pureza:97.47% - 99.92%
    Cor e Forma:Solid
    Peso molecular:176.22
  • (2-Chloropyridin-4-yl)MethanaMine Hydrochloride

    CAS:
    <p>(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).</p>
    Fórmula:C6H8Cl2N2
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:179.05
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Fórmula:C22H23N3O3S
    Pureza:98.77%
    Cor e Forma:Solid
    Peso molecular:409.5
  • VU-29

    CAS:
    <p>VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.</p>
    Fórmula:C22H16N4O3
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:384.39
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Fórmula:C14H30N2O4·2Cl·2H2O
    Pureza:99.87%
    Cor e Forma:White Solid
    Peso molecular:397.34
  • Eliapixant

    CAS:
    <p>Eliapixant (BAY 1817080) is a selective P2X3 antagonist with an 8 nM IC50, used for refractory chronic cough research.</p>
    Fórmula:C22H21F3N4O3S
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:478.49
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Fórmula:C14H16N2O
    Pureza:97.38%
    Cor e Forma:Solid
    Peso molecular:228.29
  • Encenicline

    CAS:
    <p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>
    Fórmula:C16H17ClN2OS
    Pureza:99.20%
    Cor e Forma:Solid
    Peso molecular:320.84
  • Ipratropium Bromide

    CAS:
    <p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>
    Fórmula:C20H30BrNO3
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:412.37
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Cor e Forma:Solid
    Peso molecular:324.24
  • Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Fórmula:C20H20ClF5N2O
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:434.83
  • VU0155094

    CAS:
    <p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>
    Fórmula:C24H24N2O4S
    Pureza:97.21%
    Cor e Forma:Solid
    Peso molecular:436.52
  • Norfluoxetine Hydrochloride

    CAS:
    <p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>
    Fórmula:C16H17ClF3NO
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:331.76
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Fórmula:C16H22FNO
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:263.35
  • AMN082 free base

    CAS:
    <p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>
    Fórmula:C28H28N2
    Pureza:97.75% - 97.79%
    Cor e Forma:Solid
    Peso molecular:392.54
  • Coluracetam

    CAS:
    <p>Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.</p>
    Fórmula:C19H23N3O3
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:341.4
  • Atracurium besylate

    CAS:
    <p>Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.</p>
    Fórmula:C65H82N2O18S2
    Pureza:98.94% - 99.71%
    Cor e Forma:Solid
    Peso molecular:1243.49
  • GSK3i XIII

    CAS:
    <p>GSK3i XIII (GSK3 inhibitor XIII) is a GSK-3 ATP-binding site inhibitor.</p>
    Fórmula:C18H19N5
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:305.38
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Cor e Forma:White Solid
    Peso molecular:463
  • Dihydroergotoxine mesylate

    CAS:
    Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.
    Fórmula:C20H29N3O5S
    Pureza:99.39% - ≥95%
    Cor e Forma:Solid
    Peso molecular:423.53
  • MDL 72527

    CAS:
    <p>MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) is a polyamine oxidase (POA) inhibitor</p>
    Fórmula:C12H22Cl2N2
    Pureza:98.98%
    Cor e Forma:Solid
    Peso molecular:265.22
  • RAGE antagonist peptide acetate


    <p>RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.</p>
    Fórmula:C59H105N13O19S
    Pureza:97.17%
    Cor e Forma:Solid
    Peso molecular:1332.61
  • Colivelin

    CAS:
    <p>Colivelin is a neuroprotective peptide and activator of STAT3. Colivelin is a hybrid peptide synthesized to enhance the neuroprotective effects of humanin (HN).</p>
    Fórmula:C119H206N32O35
    Pureza:96.56%
    Cor e Forma:Solid
    Peso molecular:2645.1
  • FTIDC

    CAS:
    FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.
    Fórmula:C18H23FN6O
    Pureza:94.58%
    Cor e Forma:Solid
    Peso molecular:358.41
  • Basmisanil

    CAS:
    <p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>
    Fórmula:C21H20FN3O5S
    Pureza:99.21% - 99.42%
    Cor e Forma:Solid
    Peso molecular:445.46
  • Sepimostat

    CAS:
    <p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>
    Fórmula:C21H19N5O2
    Pureza:97.75%
    Cor e Forma:Solid
    Peso molecular:373.41
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Fórmula:C18H20N4
    Pureza:99.15% - 99.82%
    Cor e Forma:Solid
    Peso molecular:292.38
  • VUF 10166

    CAS:
    <p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>
    Fórmula:C13H15ClN4
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:262.74
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Fórmula:C12H16O3
    Pureza:99.64% - 99.64%
    Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From Water
    Peso molecular:208.25
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Cor e Forma:Solid
    Peso molecular:386.37
  • Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Fórmula:C14H22ClN3O2
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:299.80
  • Firocoxib

    CAS:
    <p>Firocoxib (ML 1785713) is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.</p>
    Fórmula:C17H20O5S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:336.4
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Fórmula:C6H11NO3
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:145.16
  • Azeliragon

    CAS:
    <p>Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-</p>
    Fórmula:C32H38ClN3O2
    Pureza:96.7% - 98.33%
    Cor e Forma:Solid
    Peso molecular:532.12
  • Umibecestat HCl

    CAS:
    <p>Umibecestat HCl (CNP520 HCl) is an efficient β-secretase (BACE1/BACE2) inhibitor that reduces Aβ levels in mice and rats.</p>
    Fórmula:C19H16Cl2F7N5O2
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:550.26
  • Suritozole

    CAS:
    <p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>
    Fórmula:C10H10FN3S
    Pureza:99.25%
    Cor e Forma:Solid
    Peso molecular:223.27
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Cor e Forma:Solid
    Peso molecular:446.95
  • Azeliragon HCl

    CAS:
    <p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>
    Fórmula:C32H40Cl3N3O2
    Cor e Forma:Solid
    Peso molecular:605.04
  • Tebanicline hydrochloride

    CAS:
    <p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>
    Fórmula:C9H12Cl2N2O
    Pureza:91.74% - 98.71%
    Cor e Forma:Solid
    Peso molecular:235.11
  • (RS)-3-Hydroxyphenylglycine

    CAS:
    <p>(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.</p>
    Fórmula:C8H9NO3
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:167.16
  • (2S)-6-Prenylnaringenin

    CAS:
    <p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>
    Fórmula:C20H20O5
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:340.37
  • Cholesterol myristate

    CAS:
    <p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>
    Fórmula:C41H72O2
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:597.01
  • JNJ16259685

    CAS:
    <p>JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19</p>
    Fórmula:C20H23NO3
    Pureza:98.31%
    Cor e Forma:Solid
    Peso molecular:325.4
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • AZD-6280

    CAS:
    <p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>
    Fórmula:C20H22N4O3
    Pureza:98.99%
    Cor e Forma:Solid
    Peso molecular:366.41
  • PHCCC

    CAS:
    <p>PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.</p>
    Fórmula:C17H14N2O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:294.3
  • 4i

    CAS:
    <p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>
    Fórmula:C16H12ClN3O
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:297.74
  • VU 0238429

    CAS:
    <p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>
    Fórmula:C17H12F3NO4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:351.28