
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(575 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.948 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor GABA(336 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(27 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5390 produtos de "Neurociência"
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PNU-282987 S enantiomer free base
CAS:<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Fórmula:C14H17ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:264.75Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21Serotonin
CAS:<p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>Fórmula:C10H12N2OPureza:97.47% - 99.92%Cor e Forma:SolidPeso molecular:176.22(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
CAS:<p>(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).</p>Fórmula:C6H8Cl2N2Pureza:97.23%Cor e Forma:SolidPeso molecular:179.05Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Fórmula:C22H23N3O3SPureza:98.77%Cor e Forma:SolidPeso molecular:409.5VU-29
CAS:<p>VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.</p>Fórmula:C22H16N4O3Pureza:99.63%Cor e Forma:SolidPeso molecular:384.39Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Cor e Forma:White SolidPeso molecular:397.34Eliapixant
CAS:<p>Eliapixant (BAY 1817080) is a selective P2X3 antagonist with an 8 nM IC50, used for refractory chronic cough research.</p>Fórmula:C22H21F3N4O3SPureza:99.86%Cor e Forma:SolidPeso molecular:478.49RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29Encenicline
CAS:<p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>Fórmula:C16H17ClN2OSPureza:99.20%Cor e Forma:SolidPeso molecular:320.84Ipratropium Bromide
CAS:<p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>Fórmula:C20H30BrNO3Pureza:99.92%Cor e Forma:SolidPeso molecular:412.37SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Cor e Forma:SolidPeso molecular:324.24Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83VU0155094
CAS:<p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>Fórmula:C24H24N2O4SPureza:97.21%Cor e Forma:SolidPeso molecular:436.52Norfluoxetine Hydrochloride
CAS:<p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>Fórmula:C16H17ClF3NOPureza:99.71%Cor e Forma:SolidPeso molecular:331.76Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35AMN082 free base
CAS:<p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>Fórmula:C28H28N2Pureza:97.75% - 97.79%Cor e Forma:SolidPeso molecular:392.54Coluracetam
CAS:<p>Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.</p>Fórmula:C19H23N3O3Pureza:99.96%Cor e Forma:SolidPeso molecular:341.4Atracurium besylate
CAS:<p>Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.</p>Fórmula:C65H82N2O18S2Pureza:98.94% - 99.71%Cor e Forma:SolidPeso molecular:1243.49GSK3i XIII
CAS:<p>GSK3i XIII (GSK3 inhibitor XIII) is a GSK-3 ATP-binding site inhibitor.</p>Fórmula:C18H19N5Pureza:98.87%Cor e Forma:SolidPeso molecular:305.38Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:463Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Cor e Forma:SolidPeso molecular:423.53MDL 72527
CAS:<p>MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) is a polyamine oxidase (POA) inhibitor</p>Fórmula:C12H22Cl2N2Pureza:98.98%Cor e Forma:SolidPeso molecular:265.22RAGE antagonist peptide acetate
<p>RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.</p>Fórmula:C59H105N13O19SPureza:97.17%Cor e Forma:SolidPeso molecular:1332.61Colivelin
CAS:<p>Colivelin is a neuroprotective peptide and activator of STAT3. Colivelin is a hybrid peptide synthesized to enhance the neuroprotective effects of humanin (HN).</p>Fórmula:C119H206N32O35Pureza:96.56%Cor e Forma:SolidPeso molecular:2645.1FTIDC
CAS:FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.Fórmula:C18H23FN6OPureza:94.58%Cor e Forma:SolidPeso molecular:358.41Basmisanil
CAS:<p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>Fórmula:C21H20FN3O5SPureza:99.21% - 99.42%Cor e Forma:SolidPeso molecular:445.46Sepimostat
CAS:<p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>Fórmula:C21H19N5O2Pureza:97.75%Cor e Forma:SolidPeso molecular:373.41Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Fórmula:C13H15ClN4Pureza:99.66%Cor e Forma:SolidPeso molecular:262.74α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Fórmula:C12H16O3Pureza:99.64% - 99.64%Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.25Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Cor e Forma:SolidPeso molecular:386.37Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Fórmula:C14H22ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:299.80Firocoxib
CAS:<p>Firocoxib (ML 1785713) is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.</p>Fórmula:C17H20O5SPureza:99.84%Cor e Forma:SolidPeso molecular:336.44-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16Azeliragon
CAS:<p>Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-</p>Fórmula:C32H38ClN3O2Pureza:96.7% - 98.33%Cor e Forma:SolidPeso molecular:532.12Umibecestat HCl
CAS:<p>Umibecestat HCl (CNP520 HCl) is an efficient β-secretase (BACE1/BACE2) inhibitor that reduces Aβ levels in mice and rats.</p>Fórmula:C19H16Cl2F7N5O2Pureza:99.92%Cor e Forma:SolidPeso molecular:550.26Suritozole
CAS:<p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>Fórmula:C10H10FN3SPureza:99.25%Cor e Forma:SolidPeso molecular:223.27Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95Azeliragon HCl
CAS:<p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>Fórmula:C32H40Cl3N3O2Cor e Forma:SolidPeso molecular:605.04Tebanicline hydrochloride
CAS:<p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>Fórmula:C9H12Cl2N2OPureza:91.74% - 98.71%Cor e Forma:SolidPeso molecular:235.11(RS)-3-Hydroxyphenylglycine
CAS:<p>(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.</p>Fórmula:C8H9NO3Pureza:99.29%Cor e Forma:SolidPeso molecular:167.16(2S)-6-Prenylnaringenin
CAS:<p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>Fórmula:C20H20O5Pureza:99.47%Cor e Forma:SolidPeso molecular:340.37Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Fórmula:C41H72O2Pureza:99.65%Cor e Forma:SolidPeso molecular:597.01JNJ16259685
CAS:<p>JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19</p>Fórmula:C20H23NO3Pureza:98.31%Cor e Forma:SolidPeso molecular:325.4Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97AZD-6280
CAS:<p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>Fórmula:C20H22N4O3Pureza:98.99%Cor e Forma:SolidPeso molecular:366.41PHCCC
CAS:<p>PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.</p>Fórmula:C17H14N2O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:294.34i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Fórmula:C16H12ClN3OPureza:99.49%Cor e Forma:SolidPeso molecular:297.74VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28
