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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5389 produtos de "Neurociência"

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  • A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Fórmula:C20H19ClN2O3S
    Pureza:95.66%
    Cor e Forma:Solid
    Peso molecular:402.89
  • NS-398

    CAS:
    <p>NS-398 (N-(2-cyclohexyloxy-4-nitrophenyl)methane sulfonamide) is a COX-2 inhibitor wih anti-inflammatory activity.</p>
    Fórmula:C13H18N2O5S
    Pureza:99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:314.36
  • PNU 22394 hydrochloride

    CAS:
    PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
    Fórmula:C13H17ClN2
    Pureza:97.83%
    Cor e Forma:Solid
    Peso molecular:236.74
  • N-ACETYLTRYPTAMINE

    CAS:
    <p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>
    Fórmula:C12H14N2O
    Pureza:98.79%
    Cor e Forma:Powder
    Peso molecular:202.25
  • GR 125743

    CAS:
    GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
    Fórmula:C25H28N4O2
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:416.52
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Fórmula:C19H19N3O2S
    Pureza:98% - 98.63%
    Cor e Forma:Solid
    Peso molecular:353.44
  • JNJ-40411813

    CAS:
    <p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:344.88
  • Acotiamide monohydrochloride trihydrate

    CAS:
    <p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>
    Fórmula:C21H37ClN4O8S
    Pureza:98% - 99.54%
    Cor e Forma:Solid
    Peso molecular:541.06
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Fórmula:C21H25ClFN3O3·C6H8O7
    Pureza:99.70%
    Cor e Forma:White Powder
    Peso molecular:614.02
  • 1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide

    CAS:
    <p>1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.</p>
    Fórmula:C20H30Br2N2
    Pureza:98.17%
    Cor e Forma:Solid
    Peso molecular:458.27
  • 5-BDBD

    CAS:
    <p>5-BDBD is a potent and selective P2X4 receptor antagonist.</p>
    Fórmula:C17H11BrN2O2
    Pureza:97.78%
    Cor e Forma:Solid
    Peso molecular:355.19
  • Gabazine

    CAS:
    <p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>
    Fórmula:C15H18BrN3O3
    Pureza:98.51% - 99.24%
    Cor e Forma:Solid
    Peso molecular:368.23
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Fórmula:C6H10ClNO2
    Pureza:98.42%
    Cor e Forma:Solid
    Peso molecular:163.602
  • Edonerpic maleate

    CAS:
    Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).
    Fórmula:C20H25NO6S
    Pureza:98.24%
    Cor e Forma:Solid
    Peso molecular:407.48
  • NPS ALX Compound 4a

    CAS:
    NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)
    Fórmula:C25H25N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:431.55
  • Tianeptine

    CAS:
    Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。
    Fórmula:C21H25ClN2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:436.95
  • Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Fórmula:C22H28FNO3
    Pureza:98.94% - 99.95%
    Cor e Forma:Solid
    Peso molecular:373.46
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Fórmula:C20H25FN4O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:356.44
  • Ginkgolide A

    CAS:
    <p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>
    Fórmula:C20H24O9
    Pureza:98.76% - 99.81%
    Cor e Forma:White Powder
    Peso molecular:408.4
  • Rapastinel Trifluoroacetate

    CAS:
    <p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>
    Fórmula:C20H32F3N5O8
    Pureza:99.01% - 99.77%
    Cor e Forma:Solid
    Peso molecular:527.49
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Cor e Forma:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • NS 1738

    CAS:
    <p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>
    Fórmula:C14H9Cl2F3N2O2
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:365.13
  • A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:353.29
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Fórmula:C20H26N2O7S
    Pureza:99.86% - 99.9%
    Cor e Forma:Solid
    Peso molecular:438.49
  • m-Chlorophenylbiguanide hydrochloride

    CAS:
    <p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>
    Fórmula:C8H11Cl2N5
    Pureza:99.43% - 99.87%
    Cor e Forma:Solid
    Peso molecular:248.11
  • Donepezil

    CAS:
    <p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>
    Fórmula:C24H29NO3
    Pureza:99.69%
    Cor e Forma:White Or Almost White Crystal Powder
    Peso molecular:379.49
  • CNQX disodium

    CAS:
    <p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>
    Fórmula:C9H2N4Na2O4
    Pureza:97.77%
    Cor e Forma:Solid
    Peso molecular:276.12
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Cor e Forma:Solid
    Peso molecular:477.57
  • Frentizole

    CAS:
    <p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>
    Fórmula:C15H13N3O2S
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:299.35
  • α-Conotoxin MII acetate


    <p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>
    Fórmula:C69H107N23O24S4
    Pureza:94.82% - 97.79%
    Cor e Forma:Solid
    Peso molecular:1770.99
  • TAE-1

    CAS:
    <p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>
    Fórmula:C39H51I3N6O9
    Pureza:94.58%
    Cor e Forma:Solid
    Peso molecular:1128.57
  • CALP2 acetate(261969-04-4 free base)


    <p>CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.</p>
    Fórmula:C68H104N14O13S
    Pureza:97.43%
    Cor e Forma:Solid
    Peso molecular:1357.7
  • Nefazodone hydrochloride

    CAS:
    <p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>
    Fórmula:C25H33Cl2N5O2
    Pureza:99% - 99.86%
    Cor e Forma:White Solid
    Peso molecular:506.47
  • Naratriptan hydrochloride

    CAS:
    <p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>
    Fórmula:C17H25N3O2S·HCl
    Pureza:99.17% - 99.93%
    Cor e Forma:Beige Solid
    Peso molecular:371.93
  • 4BP-TQS

    CAS:
    <p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>
    Fórmula:C18H17BrN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:405.31
  • Syntide 2 acetate(108334-68-5 free base)


    <p>Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).</p>
    Fórmula:C70H126N20O20
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:1567.85
  • Aftin-4

    CAS:
    <p>Aftin-4, an amyloid forty-two inducer, activates γ-secretase, promoting the generation of amyloid-β-1-42 (Aβ1-42) from amyloid-β protein precursor.</p>
    Fórmula:C20H28N6O
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:368.48
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Fórmula:C11H11N3O
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:201.22
  • Cannabigerol

    CAS:
    Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Cor e Forma:Solid
    Peso molecular:316.48
  • Ursulcholic acid

    CAS:
    Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
    Fórmula:C24H40O10S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:552.7
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Fórmula:C16H14O4
    Pureza:98.75%
    Cor e Forma:Solid
    Peso molecular:270.28
  • Fesoterodine

    CAS:
    <p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>
    Fórmula:C26H37NO3
    Pureza:97.1%
    Cor e Forma:Solid
    Peso molecular:411.58
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Fórmula:C19H23Cl2N3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:364.31
  • Baclofen hydrochloride

    CAS:
    Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.
    Fórmula:C10H13Cl2NO2
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:250.122
  • Darifenacin

    CAS:
    <p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>
    Fórmula:C28H30N2O2
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:426.55
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Fórmula:C22H21O2P
    Pureza:97.985%
    Cor e Forma:White Or Slight Yellow Powder
    Peso molecular:348.37
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Fórmula:C19H21NO2
    Pureza:98.76% - 99.79%
    Cor e Forma:Solid
    Peso molecular:295.38
  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:360.29
  • 6-Methylflavone

    CAS:
    6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
    Fórmula:C16H12O2
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:236.27
  • Dolasetron

    CAS:
    <p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>
    Fórmula:C19H20N2O3
    Pureza:99.84% - 99.86%
    Cor e Forma:White Powder
    Peso molecular:324.37