
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(576 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.949 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor GABA(337 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(26 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5389 produtos de "Neurociência"
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A-867744
CAS:<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Fórmula:C20H19ClN2O3SPureza:95.66%Cor e Forma:SolidPeso molecular:402.89NS-398
CAS:<p>NS-398 (N-(2-cyclohexyloxy-4-nitrophenyl)methane sulfonamide) is a COX-2 inhibitor wih anti-inflammatory activity.</p>Fórmula:C13H18N2O5SPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:314.36PNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFórmula:C13H17ClN2Pureza:97.83%Cor e Forma:SolidPeso molecular:236.74N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Fórmula:C12H14N2OPureza:98.79%Cor e Forma:PowderPeso molecular:202.25GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:344.88Acotiamide monohydrochloride trihydrate
CAS:<p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>Fórmula:C21H37ClN4O8SPureza:98% - 99.54%Cor e Forma:SolidPeso molecular:541.06Mosapride Citrate
CAS:<p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Cor e Forma:White PowderPeso molecular:614.021-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide
CAS:<p>1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.</p>Fórmula:C20H30Br2N2Pureza:98.17%Cor e Forma:SolidPeso molecular:458.275-BDBD
CAS:<p>5-BDBD is a potent and selective P2X4 receptor antagonist.</p>Fórmula:C17H11BrN2O2Pureza:97.78%Cor e Forma:SolidPeso molecular:355.19Gabazine
CAS:<p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>Fórmula:C15H18BrN3O3Pureza:98.51% - 99.24%Cor e Forma:SolidPeso molecular:368.23Guvacine hydrochloride
CAS:<p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>Fórmula:C6H10ClNO2Pureza:98.42%Cor e Forma:SolidPeso molecular:163.602Edonerpic maleate
CAS:Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).Fórmula:C20H25NO6SPureza:98.24%Cor e Forma:SolidPeso molecular:407.48NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H25N3O2SPureza:98%Cor e Forma:SolidPeso molecular:431.55Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Fórmula:C22H28FNO3Pureza:98.94% - 99.95%Cor e Forma:SolidPeso molecular:373.46Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Fórmula:C20H24O9Pureza:98.76% - 99.81%Cor e Forma:White PowderPeso molecular:408.4Rapastinel Trifluoroacetate
CAS:<p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>Fórmula:C20H32F3N5O8Pureza:99.01% - 99.77%Cor e Forma:SolidPeso molecular:527.49Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:440.94NS 1738
CAS:<p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>Fórmula:C14H9Cl2F3N2O2Pureza:99.11%Cor e Forma:SolidPeso molecular:365.13A-582941 dihydrochloride
CAS:<p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>Fórmula:C17H22Cl2N4Pureza:99.55%Cor e Forma:SolidPeso molecular:353.29Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Cor e Forma:SolidPeso molecular:438.49m-Chlorophenylbiguanide hydrochloride
CAS:<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Fórmula:C8H11Cl2N5Pureza:99.43% - 99.87%Cor e Forma:SolidPeso molecular:248.11Donepezil
CAS:<p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>Fórmula:C24H29NO3Pureza:99.69%Cor e Forma:White Or Almost White Crystal PowderPeso molecular:379.49CNQX disodium
CAS:<p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>Fórmula:C9H2N4Na2O4Pureza:97.77%Cor e Forma:SolidPeso molecular:276.12Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Cor e Forma:SolidPeso molecular:477.57Frentizole
CAS:<p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>Fórmula:C15H13N3O2SPureza:99.82%Cor e Forma:SolidPeso molecular:299.35α-Conotoxin MII acetate
<p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Cor e Forma:SolidPeso molecular:1770.99TAE-1
CAS:<p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>Fórmula:C39H51I3N6O9Pureza:94.58%Cor e Forma:SolidPeso molecular:1128.57CALP2 acetate(261969-04-4 free base)
<p>CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.</p>Fórmula:C68H104N14O13SPureza:97.43%Cor e Forma:SolidPeso molecular:1357.7Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:White SolidPeso molecular:506.47Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Fórmula:C17H25N3O2S·HClPureza:99.17% - 99.93%Cor e Forma:Beige SolidPeso molecular:371.934BP-TQS
CAS:<p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>Fórmula:C18H17BrN2O2SPureza:99.96%Cor e Forma:SolidPeso molecular:405.31Syntide 2 acetate(108334-68-5 free base)
<p>Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).</p>Fórmula:C70H126N20O20Pureza:99.74%Cor e Forma:SolidPeso molecular:1567.85Aftin-4
CAS:<p>Aftin-4, an amyloid forty-two inducer, activates γ-secretase, promoting the generation of amyloid-β-1-42 (Aβ1-42) from amyloid-β protein precursor.</p>Fórmula:C20H28N6OPureza:98.51%Cor e Forma:SolidPeso molecular:368.486-(4-Methoxyphenyl)-3-pyridazinamine
CAS:<p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>Fórmula:C11H11N3OPureza:99.03%Cor e Forma:SolidPeso molecular:201.22Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Cor e Forma:SolidPeso molecular:552.72'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Fesoterodine
CAS:<p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>Fórmula:C26H37NO3Pureza:97.1%Cor e Forma:SolidPeso molecular:411.58DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Fórmula:C19H23Cl2N3Pureza:99.91%Cor e Forma:SolidPeso molecular:364.31Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:99.55%Cor e Forma:SolidPeso molecular:250.122Darifenacin
CAS:<p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>Fórmula:C28H30N2O2Pureza:99.78%Cor e Forma:SolidPeso molecular:426.55Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Fórmula:C22H21O2PPureza:97.985%Cor e Forma:White Or Slight Yellow PowderPeso molecular:348.37Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Fórmula:C19H21NO2Pureza:98.76% - 99.79%Cor e Forma:SolidPeso molecular:295.38Ro0711401
CAS:<p>Ro0711401 is an agonist of mGlu1 receptor.</p>Fórmula:C18H11F3N2O3Pureza:97.57%Cor e Forma:SolidPeso molecular:360.296-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Fórmula:C16H12O2Pureza:99.69%Cor e Forma:SolidPeso molecular:236.27Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Fórmula:C19H20N2O3Pureza:99.84% - 99.86%Cor e Forma:White PowderPeso molecular:324.37
