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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5389 produtos de "Neurociência"

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  • CI 75300

    CAS:
    <p>CI 75300 targets the P2X purinoceptor 7 (human).</p>
    Fórmula:C21H20O6
    Pureza:99.07%
    Cor e Forma:Solid
    Peso molecular:368.38
  • Tandospirone citrate

    CAS:
    Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)
    Fórmula:C27H37N5O9
    Pureza:97.84% - 99.90%
    Cor e Forma:Solid
    Peso molecular:575.61
  • Umeclidinium bromide

    CAS:
    <p>Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.</p>
    Fórmula:C29H34BrNO2
    Pureza:98.4% - 99.89%
    Cor e Forma:Solid
    Peso molecular:508.49
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Fórmula:C4H10N2O2
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:118.13
  • β-Amyloid 15-21 acetate


    β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.
    Fórmula:C45H69N9O11
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:912.1
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:335.47
  • 6-fluoro-DL-Tryptophan

    CAS:
    <p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>
    Fórmula:C11H11FN2O2
    Pureza:99.25%
    Cor e Forma:Off-White Powder
    Peso molecular:222.22
  • Syk Inhibitor II dihydrochloride

    CAS:
    <p>Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.</p>
    Fórmula:C14H17Cl2F3N6O
    Pureza:98.53%
    Cor e Forma:Solid
    Peso molecular:413.22
  • SSR504734

    CAS:
    <p>SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.</p>
    Fórmula:C20H20ClF3N2O
    Cor e Forma:Solid
    Peso molecular:396.83
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Cor e Forma:Solid
    Peso molecular:446.95
  • β-amyloid 1-11 acetate(190436-05-6 free base)


    <p>β-amyloid 1-11 acetate is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.</p>
    Fórmula:C58H80N16O24
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1385.37
  • Spiperone hydrochloride

    CAS:
    <p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>
    Fórmula:C23H27ClFN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:431.93
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Cor e Forma:Solid
    Peso molecular:433.57
  • Zosuquidar

    CAS:
    <p>Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.</p>
    Fórmula:C32H31F2N3O2
    Cor e Forma:Solid
    Peso molecular:527.6
  • Melitracen

    CAS:
    <p>Melitracen is a tricyclic antidepressant.</p>
    Fórmula:C21H25N
    Cor e Forma:Solid
    Peso molecular:291.43
  • ML 10302

    CAS:
    <p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>
    Fórmula:C15H21ClN2O3
    Cor e Forma:Solid
    Peso molecular:312.79
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Fórmula:C10H12ClNO2
    Pureza:97.20% - 98.94%
    Cor e Forma:Solid
    Peso molecular:213.66
  • Jatrorrhizine

    CAS:
    Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.
    Fórmula:C20H20NO4
    Pureza:97.18% - 99.06%
    Cor e Forma:Solid
    Peso molecular:338.38
  • PHA 568487

    CAS:
    <p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress &amp; neuroinflammation.</p>
    Fórmula:C20H24N2O7
    Cor e Forma:Solid
    Peso molecular:404.419
  • TCS 1102

    CAS:
    TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).
    Fórmula:C27H26N4O2S
    Pureza:99.35% - 99.52%
    Cor e Forma:Solid
    Peso molecular:470.59
  • Verubecestat TFA

    CAS:
    <p>Verubecestat (MK-8931/SCH 900931), a potent BACE1 inhibitor, shows promise for Alzheimer's, cuts Aβ CSF levels by 92%.</p>
    Fórmula:C19H18F5N5O5S
    Cor e Forma:Solid
    Peso molecular:523.435
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Cor e Forma:Solid
    Peso molecular:538.64
  • Pikamilone

    CAS:
    Pikamilone (Picamilon) is an intelligent medicine.
    Fórmula:C10H12N2O3
    Pureza:99.38%
    Cor e Forma:White Crystalline Powder
    Peso molecular:208.21
  • Naftopidil dihydrochloride

    CAS:
    <p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>
    Fórmula:C24H28N2O3·2HCl
    Pureza:99.76%
    Cor e Forma:White Solid
    Peso molecular:465.41
  • Ilmetropium iodide

    CAS:
    <p>Ilmetropium iodide is a bronchodilator.</p>
    Fórmula:C20H30INO3
    Pureza:98.45%
    Cor e Forma:Solid
    Peso molecular:459.36
  • LY900009

    CAS:
    <p>LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.</p>
    Fórmula:C23H27N3O4
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:409.48
  • BRL-15572 hydrochloride

    CAS:
    <p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>
    Fórmula:C25H28Cl2N2O
    Cor e Forma:Solid
    Peso molecular:443.41
  • Sepimostat

    CAS:
    <p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>
    Fórmula:C21H19N5O2
    Pureza:97.75%
    Cor e Forma:Solid
    Peso molecular:373.41
  • Piperidolate

    CAS:
    <p>Piperidolate inhibits intestinal cramp induced by acetylcholine</p>
    Fórmula:C21H25NO2
    Pureza:98.45%
    Cor e Forma:Solid
    Peso molecular:323.43
  • BRL-15572 dihydrochloride

    CAS:
    <p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:479.87
  • Benzetimide hydrochloride

    CAS:
    <p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>
    Fórmula:C23H27ClN2O2
    Pureza:99.32%
    Cor e Forma:Off-White Powder
    Peso molecular:398.93
  • β-Amyloid (31-35)

    CAS:
    <p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>
    Fórmula:C25H47N5O6S
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:545.74
  • Gadoteridol

    CAS:
    <p>Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.</p>
    Fórmula:C17H29GdN4O7
    Pureza:99.77% - 99.91%
    Cor e Forma:Solid
    Peso molecular:558.69
  • Naluzotan

    CAS:
    <p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:450.64
  • Mivacurium dichloride

    CAS:
    Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.
    Fórmula:C58H80Cl2N2O14
    Pureza:99.2% - 99.48%
    Cor e Forma:Off-White Solid
    Peso molecular:1100.17
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Fórmula:C16H22FNO
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:263.35
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:359.89
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Fórmula:C22H33Cl2N3O3
    Pureza:97.32% - 99.08%
    Cor e Forma:Solid
    Peso molecular:458.42
  • Urapidil

    CAS:
    <p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3
    Pureza:99.85% - >99.99%
    Cor e Forma:Solid
    Peso molecular:387.48
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Fórmula:C4H10N2
    Cor e Forma:Solid
    Peso molecular:86.14
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Fórmula:C18H15BrF2N4O2
    Pureza:98.42% - 99.88%
    Cor e Forma:Solid
    Peso molecular:437.24
  • Ansofaxine

    CAS:
    <p>Ansofaxine, an SNRI compound, is commonly utilized in depression research as a serotonin-norepinephrine reuptake inhibitor.</p>
    Fórmula:C24H31NO3
    Cor e Forma:Solid
    Peso molecular:381.516
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Cor e Forma:Solid
    Peso molecular:386.37
  • lavendustin C

    CAS:
    <p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>
    Fórmula:C14H13NO5
    Pureza:98.06%
    Cor e Forma:Yellow To Tan Powder
    Peso molecular:275.26
  • Teriflunomide impurity 3

    CAS:
    <p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>
    Fórmula:C14H11F3N2O
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:280.25
  • Oxyphencyclimine

    CAS:
    <p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>
    Fórmula:C20H28N2O3
    Cor e Forma:Solid
    Peso molecular:344.45
  • Solifenacin hydrochloride

    CAS:
    <p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>
    Fórmula:C23H27ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:398.93
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Cor e Forma:Solid
    Peso molecular:379.36
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:248.75