
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(576 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.949 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor GABA(337 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(26 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5389 produtos de "Neurociência"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
CI 75300
CAS:<p>CI 75300 targets the P2X purinoceptor 7 (human).</p>Fórmula:C21H20O6Pureza:99.07%Cor e Forma:SolidPeso molecular:368.38Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Cor e Forma:SolidPeso molecular:575.61Umeclidinium bromide
CAS:<p>Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.</p>Fórmula:C29H34BrNO2Pureza:98.4% - 99.89%Cor e Forma:SolidPeso molecular:508.49L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Fórmula:C4H10N2O2Pureza:99.32%Cor e Forma:SolidPeso molecular:118.13β-Amyloid 15-21 acetate
β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.Fórmula:C45H69N9O11Pureza:99.62%Cor e Forma:SolidPeso molecular:912.1Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Cor e Forma:SolidPeso molecular:335.476-fluoro-DL-Tryptophan
CAS:<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Fórmula:C11H11FN2O2Pureza:99.25%Cor e Forma:Off-White PowderPeso molecular:222.22Syk Inhibitor II dihydrochloride
CAS:<p>Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.</p>Fórmula:C14H17Cl2F3N6OPureza:98.53%Cor e Forma:SolidPeso molecular:413.22SSR504734
CAS:<p>SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.</p>Fórmula:C20H20ClF3N2OCor e Forma:SolidPeso molecular:396.83Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95β-amyloid 1-11 acetate(190436-05-6 free base)
<p>β-amyloid 1-11 acetate is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.</p>Fórmula:C58H80N16O24Pureza:>99.99%Cor e Forma:SolidPeso molecular:1385.37Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Fórmula:C23H27ClFN3O2Pureza:98%Cor e Forma:SolidPeso molecular:431.93Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Cor e Forma:SolidPeso molecular:433.57Zosuquidar
CAS:<p>Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.</p>Fórmula:C32H31F2N3O2Cor e Forma:SolidPeso molecular:527.6Melitracen
CAS:<p>Melitracen is a tricyclic antidepressant.</p>Fórmula:C21H25NCor e Forma:SolidPeso molecular:291.43ML 10302
CAS:<p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>Fórmula:C15H21ClN2O3Cor e Forma:SolidPeso molecular:312.79Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97(R)-baclofen
CAS:<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Fórmula:C10H12ClNO2Pureza:97.20% - 98.94%Cor e Forma:SolidPeso molecular:213.66Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Fórmula:C20H20NO4Pureza:97.18% - 99.06%Cor e Forma:SolidPeso molecular:338.38PHA 568487
CAS:<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Fórmula:C20H24N2O7Cor e Forma:SolidPeso molecular:404.419TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Fórmula:C27H26N4O2SPureza:99.35% - 99.52%Cor e Forma:SolidPeso molecular:470.59Verubecestat TFA
CAS:<p>Verubecestat (MK-8931/SCH 900931), a potent BACE1 inhibitor, shows promise for Alzheimer's, cuts Aβ CSF levels by 92%.</p>Fórmula:C19H18F5N5O5SCor e Forma:SolidPeso molecular:523.435WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Cor e Forma:SolidPeso molecular:538.64Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21Naftopidil dihydrochloride
CAS:<p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>Fórmula:C24H28N2O3·2HClPureza:99.76%Cor e Forma:White SolidPeso molecular:465.41Ilmetropium iodide
CAS:<p>Ilmetropium iodide is a bronchodilator.</p>Fórmula:C20H30INO3Pureza:98.45%Cor e Forma:SolidPeso molecular:459.36LY900009
CAS:<p>LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.</p>Fórmula:C23H27N3O4Pureza:97.07%Cor e Forma:SolidPeso molecular:409.48BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Fórmula:C25H28Cl2N2OCor e Forma:SolidPeso molecular:443.41Sepimostat
CAS:<p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>Fórmula:C21H19N5O2Pureza:97.75%Cor e Forma:SolidPeso molecular:373.41Piperidolate
CAS:<p>Piperidolate inhibits intestinal cramp induced by acetylcholine</p>Fórmula:C21H25NO2Pureza:98.45%Cor e Forma:SolidPeso molecular:323.43BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Cor e Forma:SolidPeso molecular:479.87Benzetimide hydrochloride
CAS:<p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>Fórmula:C23H27ClN2O2Pureza:99.32%Cor e Forma:Off-White PowderPeso molecular:398.93β-Amyloid (31-35)
CAS:<p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>Fórmula:C25H47N5O6SPureza:>99.99%Cor e Forma:SolidPeso molecular:545.74Gadoteridol
CAS:<p>Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.</p>Fórmula:C17H29GdN4O7Pureza:99.77% - 99.91%Cor e Forma:SolidPeso molecular:558.69Naluzotan
CAS:<p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>Fórmula:C23H38N4O3SPureza:>99.99%Cor e Forma:SolidPeso molecular:450.64Mivacurium dichloride
CAS:Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Cor e Forma:Off-White SolidPeso molecular:1100.17Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Cor e Forma:SolidPeso molecular:359.89BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Cor e Forma:SolidPeso molecular:458.42Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3Pureza:99.85% - >99.99%Cor e Forma:SolidPeso molecular:387.48Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Cor e Forma:SolidPeso molecular:86.14Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Fórmula:C18H15BrF2N4O2Pureza:98.42% - 99.88%Cor e Forma:SolidPeso molecular:437.24Ansofaxine
CAS:<p>Ansofaxine, an SNRI compound, is commonly utilized in depression research as a serotonin-norepinephrine reuptake inhibitor.</p>Fórmula:C24H31NO3Cor e Forma:SolidPeso molecular:381.516Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Cor e Forma:SolidPeso molecular:386.37lavendustin C
CAS:<p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>Fórmula:C14H13NO5Pureza:98.06%Cor e Forma:Yellow To Tan PowderPeso molecular:275.26Teriflunomide impurity 3
CAS:<p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>Fórmula:C14H11F3N2OPureza:99.62%Cor e Forma:SolidPeso molecular:280.25Oxyphencyclimine
CAS:<p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>Fórmula:C20H28N2O3Cor e Forma:SolidPeso molecular:344.45Solifenacin hydrochloride
CAS:<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Fórmula:C23H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.93Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.361-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.75
