
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(576 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.949 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor GABA(337 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(26 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5389 produtos de "Neurociência"
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Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Fórmula:C14H21Cl2F3N6O3Cor e Forma:SolidPeso molecular:449.26Tacrine hydrochloride (hydrate)
CAS:<p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>Fórmula:C13H14N2·XHCl·XH2OPureza:99.01% - 99.89%Cor e Forma:SolidPeso molecular:234.72Acotiamide
CAS:<p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>Fórmula:C21H30N4O5SCor e Forma:SolidPeso molecular:450.55A-804598
CAS:<p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>Fórmula:C19H17N5Pureza:99.57%Cor e Forma:SolidPeso molecular:315.37Isocarboxazid
CAS:<p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>Fórmula:C12H13N3O2Pureza:98.32% - 99.94%Cor e Forma:SolidPeso molecular:231.25Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Cor e Forma:SolidPeso molecular:394.85p-Hydroxybenzaldehyde
CAS:1.Fórmula:C7H6O2Pureza:99.05% - 99.86%Cor e Forma:SolidPeso molecular:122.12Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSCor e Forma:SolidPeso molecular:340.48Azeliragon HCl
CAS:<p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>Fórmula:C32H40Cl3N3O2Cor e Forma:SolidPeso molecular:605.04Autocamtide 2 TFA(129198-88-5 free base)
<p>Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.</p>Fórmula:C67H119F3N22O22Pureza:98%Cor e Forma:SolidPeso molecular:1641.79Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Fórmula:C17H18ClN4OCor e Forma:SolidPeso molecular:329.11691Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Cor e Forma:SolidPeso molecular:485.96Pimavanserin tartrate
CAS:<p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>Fórmula:C50H68F2N6O4·C4H6O6Pureza:99.24% - 99.98%Cor e Forma:SolidPeso molecular:1005.2(S)-Flurbiprofen
CAS:<p>Esflurbiprofen is an inhibitor of COX-1 and COX-2.</p>Fórmula:C15H13FO2Pureza:99.99%Cor e Forma:White To Yellowish Crystalline PowderPeso molecular:244.26Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Fórmula:C17H16FN3Pureza:99.32%Cor e Forma:SolidPeso molecular:281.33S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Cor e Forma:SolidPeso molecular:407.48Ocaperidone
CAS:<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Fórmula:C24H25FN4O2Pureza:99.33%Cor e Forma:SolidPeso molecular:420.48Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.41Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Cor e Forma:SolidPeso molecular:335.47Azaphen dihydrochloride monohydrate
CAS:<p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C16H23Cl2N5O2Pureza:99.85%Cor e Forma:SolidPeso molecular:388.29Flibanserin
CAS:<p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>Fórmula:C20H21F3N4OPureza:99.37% - 99.93%Cor e Forma:White PowderPeso molecular:390.4Mavacoxib
CAS:<p>Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.</p>Fórmula:C16H11F4N3O2SPureza:99.90%Cor e Forma:SolidPeso molecular:385.34Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Cor e Forma:SolidPeso molecular:177.63CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Fórmula:C19H15Cl2N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:388.25LY2886721
CAS:<p>LY2886721, a BACE inhibitor, is used for the therapy of Alzheimer's Disease.</p>Fórmula:C18H16F2N4O2SPureza:99% - 99.75%Cor e Forma:SolidPeso molecular:390.41HG-10-102-01
CAS:<p>HG-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (LRRK2, IC50 of 20.3 nM).</p>Fórmula:C17H20ClN5O3Pureza:99.59%Cor e Forma:SolidPeso molecular:377.83Syn-Ake acetate
CAS:<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Cor e Forma:SolidPeso molecular:495.58CNQX
CAS:<p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C9H4N4O4Pureza:99.70%Cor e Forma:Pale Yellow SolidPeso molecular:232.15(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Fórmula:C13H15NO2Pureza:99.58% - 99.87%Cor e Forma:SolidPeso molecular:217.26PF3274167
CAS:PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Fórmula:C19H19ClFN5O3Pureza:99.67% - 99.88%Cor e Forma:SolidPeso molecular:419.84AF-353
CAS:AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).Fórmula:C14H17IN4O2Pureza:92.98% - 99.356%Cor e Forma:SolidPeso molecular:400.21QNZ46
CAS:<p>QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.</p>Fórmula:C24H17N3O6Pureza:99.65%Cor e Forma:SolidPeso molecular:443.41EUK-134
CAS:EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.Fórmula:C18H18ClMnN2O4Pureza:98.39%Cor e Forma:SolidPeso molecular:416.74Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Fórmula:C20H22ClF3N4OCor e Forma:SolidPeso molecular:426.87SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFórmula:C15H14N4OPureza:99.61%Cor e Forma:SolidPeso molecular:266.3Amitriptyline
CAS:<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Fórmula:C20H23NPureza:98.24% - 99.64%Cor e Forma:Crystals SolidPeso molecular:277.4Demecarium bromide
CAS:<p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>Fórmula:C32H52Br2N4O4Pureza:98%Cor e Forma:White Powder SolidPeso molecular:716.59OXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Fórmula:C79H125N23O22Pureza:98.52%Cor e Forma:SolidPeso molecular:1748.98CZC-25146 hydrochloride
CAS:<p>CZC-25146 is a selective LRRK2 inhibitor with IC50 of 4.76 nM/6.87 nM for wild type LRRK2 and G2019S LRRK2, respectively.</p>Fórmula:C22H26ClFN6O4SPureza:98.76%Cor e Forma:SolidPeso molecular:525(R)-baclofen
CAS:<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Fórmula:C10H12ClNO2Pureza:97.20% - 98.94%Cor e Forma:SolidPeso molecular:213.66Edrophonium chloride
CAS:Edrophonium chloride is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by bindingFórmula:C10H16ClNOPureza:97.41%Cor e Forma:LiquidPeso molecular:201.69Phenibut (hydrochloride)
CAS:<p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>Fórmula:C10H14ClNO2Pureza:99.93%Cor e Forma:White Crystalline PowderPeso molecular:215.683-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Cor e Forma:SolidPeso molecular:215.23CaM kinase II inhibitor TFA salt
<p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>Fórmula:C66H117F3N22O21Pureza:>99.99%Cor e Forma:SolidPeso molecular:1611.77Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Cor e Forma:Pale Yellow SolidPeso molecular:469.55A 438079 hydrochloride
CAS:<p>A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.</p>Fórmula:C13H10Cl3N5Pureza:99.74% - >99.99%Cor e Forma:SolidPeso molecular:342.61W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Fórmula:C32H44Br2N4O4Pureza:95.56%Cor e Forma:SolidPeso molecular:708.52
