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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5389 produtos de "Neurociência"

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  • Syk Inhibitor II dihydrochloride dihydrate

    CAS:
    <p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>
    Fórmula:C14H21Cl2F3N6O3
    Cor e Forma:Solid
    Peso molecular:449.26
  • Tacrine hydrochloride (hydrate)

    CAS:
    <p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>
    Fórmula:C13H14N2·XHCl·XH2O
    Pureza:99.01% - 99.89%
    Cor e Forma:Solid
    Peso molecular:234.72
  • Acotiamide

    CAS:
    <p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>
    Fórmula:C21H30N4O5S
    Cor e Forma:Solid
    Peso molecular:450.55
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:315.37
  • Isocarboxazid

    CAS:
    <p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>
    Fórmula:C12H13N3O2
    Pureza:98.32% - 99.94%
    Cor e Forma:Solid
    Peso molecular:231.25
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Cor e Forma:Solid
    Peso molecular:446.95
  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Fórmula:C23H23F3N2O4
    Pureza:99.66% - ≥95%
    Cor e Forma:Solid
    Peso molecular:448.43
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Cor e Forma:Solid
    Peso molecular:394.85
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Fórmula:C7H6O2
    Pureza:99.05% - 99.86%
    Cor e Forma:Solid
    Peso molecular:122.12
  • Cinanserin

    CAS:
    <p>Cinanserin is a serotonin 5-HT2 antagonist.</p>
    Fórmula:C20H24N2OS
    Cor e Forma:Solid
    Peso molecular:340.48
  • Azeliragon HCl

    CAS:
    <p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>
    Fórmula:C32H40Cl3N3O2
    Cor e Forma:Solid
    Peso molecular:605.04
  • Autocamtide 2 TFA(129198-88-5 free base)


    <p>Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.</p>
    Fórmula:C67H119F3N22O22
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1641.79
  • Alosetron (Hydrochloride(1:X))

    CAS:
    <p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>
    Fórmula:C17H18ClN4O
    Cor e Forma:Solid
    Peso molecular:329.11691
  • Prucalopride Succinate

    CAS:
    Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).
    Fórmula:C18H26ClN3O3·C4H6O4
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:485.96
  • Pimavanserin tartrate

    CAS:
    <p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>
    Fórmula:C50H68F2N6O4·C4H6O6
    Pureza:99.24% - 99.98%
    Cor e Forma:Solid
    Peso molecular:1005.2
  • (S)-Flurbiprofen

    CAS:
    <p>Esflurbiprofen is an inhibitor of COX-1 and COX-2.</p>
    Fórmula:C15H13FO2
    Pureza:99.99%
    Cor e Forma:White To Yellowish Crystalline Powder
    Peso molecular:244.26
  • Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Fórmula:C20H20ClF5N2O
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:434.83
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:281.33
  • S 14506 HCl

    CAS:
    <p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), &lt;6.0 (5-HT3).</p>
    Fórmula:C24H26FN3O2
    Cor e Forma:Solid
    Peso molecular:407.48
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:420.48
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Cor e Forma:Solid
    Peso molecular:427.41
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:335.47
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Fórmula:C16H23Cl2N5O2
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:388.29
  • Flibanserin

    CAS:
    <p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>
    Fórmula:C20H21F3N4O
    Pureza:99.37% - 99.93%
    Cor e Forma:White Powder
    Peso molecular:390.4
  • Mavacoxib

    CAS:
    <p>Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.</p>
    Fórmula:C16H11F4N3O2S
    Pureza:99.90%
    Cor e Forma:Solid
    Peso molecular:385.34
  • Arecaidine hydrochloride

    CAS:
    Arecaidine hydrochloride may have carcinogenesis.
    Fórmula:C7H12ClNO2
    Pureza:99.69% - ≥95%
    Cor e Forma:Solid
    Peso molecular:177.63
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Fórmula:C19H15Cl2N3O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:388.25
  • LY2886721

    CAS:
    <p>LY2886721, a BACE inhibitor, is used for the therapy of Alzheimer's Disease.</p>
    Fórmula:C18H16F2N4O2S
    Pureza:99% - 99.75%
    Cor e Forma:Solid
    Peso molecular:390.41
  • HG-10-102-01

    CAS:
    <p>HG-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (LRRK2, IC50 of 20.3 nM).</p>
    Fórmula:C17H20ClN5O3
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:377.83
  • Syn-Ake acetate

    CAS:
    <p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>
    Fórmula:C19H29N5O3·2(C2H4O2)
    Pureza:99.60%
    Cor e Forma:Solid
    Peso molecular:495.58
  • CNQX

    CAS:
    <p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C9H4N4O4
    Pureza:99.70%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:232.15
  • (-)-Securinine

    CAS:
    <p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>
    Fórmula:C13H15NO2
    Pureza:99.58% - 99.87%
    Cor e Forma:Solid
    Peso molecular:217.26
  • PF3274167

    CAS:
    PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
    Fórmula:C19H19ClFN5O3
    Pureza:99.67% - 99.88%
    Cor e Forma:Solid
    Peso molecular:419.84
  • AF-353

    CAS:
    AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).
    Fórmula:C14H17IN4O2
    Pureza:92.98% - 99.356%
    Cor e Forma:Solid
    Peso molecular:400.21
  • QNZ46

    CAS:
    <p>QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.</p>
    Fórmula:C24H17N3O6
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:443.41
  • EUK-134

    CAS:
    EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.
    Fórmula:C18H18ClMnN2O4
    Pureza:98.39%
    Cor e Forma:Solid
    Peso molecular:416.74
  • Flibanserin hydrochloride

    CAS:
    <p>Flibanserin HCl: oral 5-HT1A agonist &amp; 5-HT2A antagonist, Ki values 1 nM &amp; 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>
    Fórmula:C20H22ClF3N4O
    Cor e Forma:Solid
    Peso molecular:426.87
  • SB-200646

    CAS:
    SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
    Fórmula:C15H14N4O
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:266.3
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Fórmula:C20H23N
    Pureza:98.24% - 99.64%
    Cor e Forma:Crystals Solid
    Peso molecular:277.4
  • Demecarium bromide

    CAS:
    <p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>
    Fórmula:C32H52Br2N4O4
    Pureza:98%
    Cor e Forma:White Powder Solid
    Peso molecular:716.59
  • OXA (17-33) acetate


    <p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>
    Fórmula:C79H125N23O22
    Pureza:98.52%
    Cor e Forma:Solid
    Peso molecular:1748.98
  • CZC-25146 hydrochloride

    CAS:
    <p>CZC-25146 is a selective LRRK2 inhibitor with IC50 of 4.76 nM/6.87 nM for wild type LRRK2 and G2019S LRRK2, respectively.</p>
    Fórmula:C22H26ClFN6O4S
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:525
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Fórmula:C10H12ClNO2
    Pureza:97.20% - 98.94%
    Cor e Forma:Solid
    Peso molecular:213.66
  • Edrophonium chloride

    CAS:
    Edrophonium chloride is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by binding
    Fórmula:C10H16ClNO
    Pureza:97.41%
    Cor e Forma:Liquid
    Peso molecular:201.69
  • Phenibut (hydrochloride)

    CAS:
    <p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>
    Fórmula:C10H14ClNO2
    Pureza:99.93%
    Cor e Forma:White Crystalline Powder
    Peso molecular:215.68
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Cor e Forma:Solid
    Peso molecular:215.23
  • CaM kinase II inhibitor TFA salt


    <p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>
    Fórmula:C66H117F3N22O21
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1611.77
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:469.55
  • A 438079 hydrochloride

    CAS:
    <p>A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.</p>
    Fórmula:C13H10Cl3N5
    Pureza:99.74% - >99.99%
    Cor e Forma:Solid
    Peso molecular:342.61
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Fórmula:C32H44Br2N4O4
    Pureza:95.56%
    Cor e Forma:Solid
    Peso molecular:708.52