
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(993 produtos)
- ACK(1 produtos)
- AChR(612 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.004 produtos)
- BACE(36 produtos)
- Beta Amilóide(216 produtos)
- CaMK(71 produtos)
- COX(592 produtos)
- Receptor de Dopamina(433 produtos)
- Receptor GABA(355 produtos)
- Gama-secretase(63 produtos)
- GluR(261 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(381 produtos)
- LRRK2(41 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(15 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(310 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5516 produtos de "Neurociência"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Cor e Forma:Yellow Crystalline SolidPeso molecular:312.8RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Cor e Forma:SolidPeso molecular:228.29IC87201
CAS:<p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>Fórmula:C13H10Cl2N4OPureza:97.44%Cor e Forma:SolidPeso molecular:309.15Verubecestat tosylate
CAS:Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.Fórmula:C25H26N4O4S2Cor e Forma:SolidPeso molecular:510.627Drofenine
CAS:Drofenin: anticonvulsant, anticholinergic, neurotropic, musculotropic, FIASMA.Fórmula:C20H31NO2Cor e Forma:SolidPeso molecular:317.47Polmacoxib
CAS:<p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>Fórmula:C18H16FNO4SPureza:97.88%Cor e Forma:SolidPeso molecular:361.39Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Fórmula:C20H24N2OSCor e Forma:SolidPeso molecular:340.48NMDAR antagonist 1
CAS:<p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>Fórmula:C20H20BrN3O2Pureza:98%Cor e Forma:SolidPeso molecular:414.3Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Fórmula:C21H28BrNO3Pureza:99.29%Cor e Forma:SolidPeso molecular:422.36Fluralaner
CAS:<p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.90%Cor e Forma:Solid PowderPeso molecular:556.29Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Fórmula:C53H90O22Pureza:98.83% - 99.56%Cor e Forma:White PowderPeso molecular:1079.27Dinotefuran
CAS:<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Fórmula:C7H14N4O3Pureza:99.89%Cor e Forma:White Crystalline PowderPeso molecular:202.21Colivelin
CAS:<p>Colivelin is a neuroprotective peptide and activator of STAT3. Colivelin is a hybrid peptide synthesized to enhance the neuroprotective effects of humanin (HN).</p>Fórmula:C119H206N32O35Pureza:96.56%Cor e Forma:SolidPeso molecular:2645.1Abaperidone Hydrochloride
CAS:<p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>Fórmula:C25H26ClFN2O5Cor e Forma:SolidPeso molecular:488.94Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Fórmula:C19H22O2Pureza:99.22% - 99.66%Cor e Forma:SolidPeso molecular:282.38AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Fórmula:C23H31ClN2O2Pureza:99.71%Cor e Forma:SolidPeso molecular:402.96Methiothepin mesylate
CAS:Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:452.65Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Cor e Forma:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Cor e Forma:SolidPeso molecular:288.34XAP044
CAS:XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.Fórmula:C15H9IO4Pureza:97.41%Cor e Forma:SolidPeso molecular:380.13CZC-54252
CAS:CZC-54252 is a potent inhibitor of LRRK2.Fórmula:C22H25ClN6O4SPureza:99.39%Cor e Forma:SolidPeso molecular:504.99Firocoxib
CAS:<p>Firocoxib (ML 1785713) is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.</p>Fórmula:C17H20O5SPureza:99.84%Cor e Forma:SolidPeso molecular:336.4Temgicoluril
CAS:<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Fórmula:C8H14N4O2Pureza:99.8%Cor e Forma:SolidPeso molecular:198.22Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Fórmula:C9H12Cl2N2OPureza:91.74% - 98.71%Cor e Forma:SolidPeso molecular:235.11lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7Cyclopentolate Hydrochloride
CAS:<p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>Fórmula:C17H26ClNO3Pureza:99.91%Cor e Forma:SolidPeso molecular:327.85VU 0357121
CAS:VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.Fórmula:C17H17F2NO2Pureza:99% - >99.99%Cor e Forma:SolidPeso molecular:305.32Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21Myristicin
CAS:<p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>Fórmula:C11H12O3Pureza:99.828%Cor e Forma:LiquidPeso molecular:192.21CaM kinase II inhibitor TFA salt
<p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>Fórmula:C66H117F3N22O21Pureza:>99.99%Cor e Forma:SolidPeso molecular:1611.77MPEP
CAS:MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.Fórmula:C14H11NPureza:99.54%Cor e Forma:SolidPeso molecular:193.24Hypidone hydrochloride
CAS:<p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>Fórmula:C18H23ClN2O2Pureza:99.82% - 99.93%Cor e Forma:SolidPeso molecular:334.84EUK-134
CAS:EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.Fórmula:C18H18ClMnN2O4Pureza:98.39%Cor e Forma:SolidPeso molecular:416.74Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Fórmula:C24H29ClN4O4Cor e Forma:SolidPeso molecular:472.97LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Fórmula:C24H27FN2O2·HClPureza:99.8%Cor e Forma:SolidPeso molecular:430.94MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C23H21N5O3SPureza:97.69% - 98.15%Cor e Forma:SolidPeso molecular:447.51BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Fórmula:C14H18N2OPureza:98.07%Cor e Forma:SolidPeso molecular:230.31Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Cor e Forma:Off-White PowderPeso molecular:298.29Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Fórmula:C20H25NO2S2Pureza:99.25% - 99.67%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Fórmula:C10H22ClNCor e Forma:SolidPeso molecular:191.74Clomipramine
CAS:<p>Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.</p>Fórmula:C19H23ClN2Pureza:99.31% - 99.71%Cor e Forma:SolidPeso molecular:314.85(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Fórmula:C14H14O3Pureza:97% - ≥95%Cor e Forma:White Fine PowderPeso molecular:230.26Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Fórmula:C20H24O9Pureza:98.76% - 99.81%Cor e Forma:White PowderPeso molecular:408.4DNQX
CAS:<p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C8H4N4O6Pureza:97.27% - 99.1%Cor e Forma:Off-White Powder With A Yellow TingePeso molecular:252.14AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Cor e Forma:SolidPeso molecular:354.38Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Fórmula:C25H27N3O2S·xHClPureza:99.05%Cor e Forma:SolidPeso molecular:433.63-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Cor e Forma:SolidPeso molecular:215.23Aminooxyacetic acid hemihydrochloride
CAS:<p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>Fórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Cor e Forma:SolidPeso molecular:394.85Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44
