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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5516 produtos de "Neurociência"

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  • N-Desmethylclozapine

    CAS:
    N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.
    Fórmula:C17H17ClN4
    Pureza:97.25% - 99.83%
    Cor e Forma:Yellow Crystalline Solid
    Peso molecular:312.8
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Fórmula:C14H16N2O
    Pureza:97.38%
    Cor e Forma:Solid
    Peso molecular:228.29
  • IC87201

    CAS:
    <p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>
    Fórmula:C13H10Cl2N4O
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:309.15
  • Verubecestat tosylate

    CAS:
    Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.
    Fórmula:C25H26N4O4S2
    Cor e Forma:Solid
    Peso molecular:510.627
  • Drofenine

    CAS:
    Drofenin: anticonvulsant, anticholinergic, neurotropic, musculotropic, FIASMA.
    Fórmula:C20H31NO2
    Cor e Forma:Solid
    Peso molecular:317.47
  • Polmacoxib

    CAS:
    <p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>
    Fórmula:C18H16FNO4S
    Pureza:97.88%
    Cor e Forma:Solid
    Peso molecular:361.39
  • Cinanserin

    CAS:
    Cinanserin is a serotonin 5-HT2 antagonist.
    Fórmula:C20H24N2OS
    Cor e Forma:Solid
    Peso molecular:340.48
  • NMDAR antagonist 1

    CAS:
    <p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>
    Fórmula:C20H20BrN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:414.3
  • Methylbenactyzium Bromide

    CAS:
    Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.
    Fórmula:C21H28BrNO3
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:422.36
  • Fluralaner

    CAS:
    <p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>
    Fórmula:C22H17Cl2F6N3O3
    Pureza:99.72% - 99.90%
    Cor e Forma:Solid Powder
    Peso molecular:556.29
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Fórmula:C53H90O22
    Pureza:98.83% - 99.56%
    Cor e Forma:White Powder
    Peso molecular:1079.27
  • Dinotefuran

    CAS:
    <p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>
    Fórmula:C7H14N4O3
    Pureza:99.89%
    Cor e Forma:White Crystalline Powder
    Peso molecular:202.21
  • Colivelin

    CAS:
    <p>Colivelin is a neuroprotective peptide and activator of STAT3. Colivelin is a hybrid peptide synthesized to enhance the neuroprotective effects of humanin (HN).</p>
    Fórmula:C119H206N32O35
    Pureza:96.56%
    Cor e Forma:Solid
    Peso molecular:2645.1
  • Abaperidone Hydrochloride

    CAS:
    <p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>
    Fórmula:C25H26ClFN2O5
    Cor e Forma:Solid
    Peso molecular:488.94
  • Miltirone

    CAS:
    Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.
    Fórmula:C19H22O2
    Pureza:99.22% - 99.66%
    Cor e Forma:Solid
    Peso molecular:282.38
  • AC-90179 HCl

    CAS:
    AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.
    Fórmula:C23H31ClN2O2
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:402.96
  • Methiothepin mesylate

    CAS:
    Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
    Fórmula:C21H28N2O3S3
    Pureza:98% - 99.92%
    Cor e Forma:Solid
    Peso molecular:452.65
  • Melatonin

    CAS:
    <p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>
    Fórmula:C13H16N2O2
    Pureza:98% - 99.89%
    Cor e Forma:Pale Yellow Leaflets From Benzene Solid
    Peso molecular:232.28
  • PHA 568487 free base

    CAS:
    <p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>
    Fórmula:C16H20N2O3
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:288.34
  • XAP044

    CAS:
    XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.
    Fórmula:C15H9IO4
    Pureza:97.41%
    Cor e Forma:Solid
    Peso molecular:380.13
  • CZC-54252

    CAS:
    CZC-54252 is a potent inhibitor of LRRK2.
    Fórmula:C22H25ClN6O4S
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:504.99
  • Firocoxib

    CAS:
    <p>Firocoxib (ML 1785713) is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.</p>
    Fórmula:C17H20O5S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:336.4
  • Temgicoluril

    CAS:
    <p>Temgicoluril (mebikar) acts on GABA Receptor.</p>
    Fórmula:C8H14N4O2
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:198.22
  • Tebanicline hydrochloride

    CAS:
    Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.
    Fórmula:C9H12Cl2N2O
    Pureza:91.74% - 98.71%
    Cor e Forma:Solid
    Peso molecular:235.11
  • lumateperone Tosylate

    CAS:
    lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.
    Fórmula:C31H36FN3O4S
    Pureza:95.83% - 99.95%
    Cor e Forma:Solid
    Peso molecular:565.7
  • Cyclopentolate Hydrochloride

    CAS:
    <p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>
    Fórmula:C17H26ClNO3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:327.85
  • VU 0357121

    CAS:
    VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.
    Fórmula:C17H17F2NO2
    Pureza:99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:305.32
  • Pikamilone

    CAS:
    Pikamilone (Picamilon) is an intelligent medicine.
    Fórmula:C10H12N2O3
    Pureza:99.38%
    Cor e Forma:White Crystalline Powder
    Peso molecular:208.21
  • Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Fórmula:C11H12O3
    Pureza:99.828%
    Cor e Forma:Liquid
    Peso molecular:192.21
  • CaM kinase II inhibitor TFA salt


    <p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>
    Fórmula:C66H117F3N22O21
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1611.77
  • MPEP

    CAS:
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
    Fórmula:C14H11N
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:193.24
  • Hypidone hydrochloride

    CAS:
    <p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>
    Fórmula:C18H23ClN2O2
    Pureza:99.82% - 99.93%
    Cor e Forma:Solid
    Peso molecular:334.84
  • EUK-134

    CAS:
    EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.
    Fórmula:C18H18ClMnN2O4
    Pureza:98.39%
    Cor e Forma:Solid
    Peso molecular:416.74
  • Temanogrel hydrochloride

    CAS:
    Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.
    Fórmula:C24H29ClN4O4
    Cor e Forma:Solid
    Peso molecular:472.97
  • LY310762

    CAS:
    LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.
    Fórmula:C24H27FN2O2·HCl
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:430.94
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Cor e Forma:Solid
    Peso molecular:447.51
  • BRL 54443

    CAS:
    BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
    Fórmula:C14H18N2O
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:230.31
  • Metadoxine

    CAS:
    Metadoxine (Metadoxil) is a neurotransmitter stimulant.
    Fórmula:C8H11NO3·C5H7NO3
    Pureza:99.19%
    Cor e Forma:Off-White Powder
    Peso molecular:298.29
  • Tiagabine

    CAS:
    Tiagabine (NO050328) is an Anti-epileptic Agent.
    Fórmula:C20H25NO2S2
    Pureza:99.25% - 99.67%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:375.55
  • Pempidine HCl

    CAS:
    Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.
    Fórmula:C10H22ClN
    Cor e Forma:Solid
    Peso molecular:191.74
  • Clomipramine

    CAS:
    <p>Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.</p>
    Fórmula:C19H23ClN2
    Pureza:99.31% - 99.71%
    Cor e Forma:Solid
    Peso molecular:314.85
  • (+)-Kavain

    CAS:
    (+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.
    Fórmula:C14H14O3
    Pureza:97% - ≥95%
    Cor e Forma:White Fine Powder
    Peso molecular:230.26
  • Ginkgolide A

    CAS:
    <p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>
    Fórmula:C20H24O9
    Pureza:98.76% - 99.81%
    Cor e Forma:White Powder
    Peso molecular:408.4
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C8H4N4O6
    Pureza:97.27% - 99.1%
    Cor e Forma:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:354.38
  • Brexpiprazole HCl

    CAS:
    Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.
    Fórmula:C25H27N3O2S·xHCl
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:433.6
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Cor e Forma:Solid
    Peso molecular:215.23
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Cor e Forma:Light Beige Crystalline Powder
    Peso molecular:109.3
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Cor e Forma:Solid
    Peso molecular:394.85
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Fórmula:C20H25FN4O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:356.44