
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.024 produtos)
- ACK(1 produtos)
- AChR(624 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.029 produtos)
- BACE(36 produtos)
- Beta Amilóide(224 produtos)
- CaMK(73 produtos)
- COX(600 produtos)
- Receptor de Dopamina(443 produtos)
- Receptor GABA(365 produtos)
- Gama-secretase(62 produtos)
- GluR(263 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(326 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5559 produtos de "Neurociência"
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Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Fórmula:C11H18Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:265.18Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Cor e Forma:SolidPeso molecular:386.37Demecarium bromide
CAS:<p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>Fórmula:C32H52Br2N4O4Pureza:98%Cor e Forma:White Powder SolidPeso molecular:716.59JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.72%Cor e Forma:SolidPeso molecular:358.84Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Fórmula:C16H17ClN2OS·HClPureza:98.34% - 99.85%Cor e Forma:SolidPeso molecular:357.3Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Fórmula:C17H24O4Pureza:98.22%Cor e Forma:SolidPeso molecular:292.37Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Fórmula:C30H18O10Pureza:98.21% - 99.22%Cor e Forma:Odourless Whitish SolidPeso molecular:538.46Ref: TM-T3417
2mg35,00€5mg52,00€10mg85,00€25mg133,00€50mg227,00€100mg369,00€200mg540,00€1mL*10mM (DMSO)63,00€5-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Fórmula:C11H16ClNOPureza:98.5%Cor e Forma:SolidPeso molecular:213.7pep2-SVKI acetate
Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.Fórmula:C62H97N13O20Pureza:97.14%Cor e Forma:SolidPeso molecular:1344.51Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Fórmula:C24H46N6O14Pureza:99.8%Cor e Forma:Crystals IndicationPeso molecular:642.65EUK-134
CAS:EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.Fórmula:C18H18ClMnN2O4Pureza:98.39%Cor e Forma:SolidPeso molecular:416.74LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Fórmula:C24H27FN2O2·HClPureza:99.8%Cor e Forma:SolidPeso molecular:430.94MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C23H21N5O3SPureza:97.69% - 98.15%Cor e Forma:SolidPeso molecular:447.51Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Cor e Forma:Off-White PowderPeso molecular:298.29Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Fórmula:C20H25NO2S2Pureza:99.25% - 99.67%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55Clomipramine
CAS:Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.Fórmula:C19H23ClN2Pureza:99.31% - 99.71%Cor e Forma:SolidPeso molecular:314.85DNQX
CAS:<p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C8H4N4O6Pureza:97.27% - 99.1%Cor e Forma:Off-White Powder With A Yellow TingePeso molecular:252.14AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Cor e Forma:SolidPeso molecular:354.38ADX88178
CAS:ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.Fórmula:C12H12N6SPureza:99.55%Cor e Forma:SolidPeso molecular:272.33Ref: TM-T4500
2mg38,00€5mg58,00€10mg96,00€25mg156,00€50mg243,00€100mg354,00€200mg505,00€1mL*10mM (DMSO)60,00€Verubecestat
CAS:Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.Fórmula:C17H17F2N5O3SPureza:94.64% - 99.55%Cor e Forma:SolidPeso molecular:409.41Ref: TM-T7011
2mg40,00€5mg60,00€10mg88,00€25mg153,00€50mg216,00€100mg354,00€500mg825,00€1mL*10mM (DMSO)66,00€VU0364770
CAS:VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGluFórmula:C12H9ClN2OPureza:99.65% - >99.99%Cor e Forma:SolidPeso molecular:232.67GW791343 dihydrochloride
CAS:GW791343 dihydrochloride (GW791343 (HCl)) is a P2X7 allosteric modulator.Fórmula:C20H26Cl2F2N4OPureza:>99.99%Cor e Forma:SolidPeso molecular:447.35pyridostigmine
CAS:Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.Fórmula:C9H13N2O2Pureza:98.10%Cor e Forma:SolidPeso molecular:181.21Ref: TM-T8631
1mg88,00€5mg170,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)167,00€Lu AF21934
CAS:<p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>Fórmula:C14H16Cl2N2O2Pureza:99.79%Cor e Forma:SolidPeso molecular:315.2GALANTHAMINONE
CAS:<p>Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairments</p>Fórmula:C17H19NO3Pureza:99.93%Cor e Forma:White To Off-White ChemicalPeso molecular:285.34A-867744
CAS:A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).Fórmula:C20H19ClN2O3SPureza:95.66%Cor e Forma:SolidPeso molecular:402.89PNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFórmula:C13H17ClN2Pureza:97.83%Cor e Forma:SolidPeso molecular:236.74N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Fórmula:C12H14N2OPureza:98.79%Cor e Forma:PowderPeso molecular:202.25GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52Ref: TM-T8737
1mg43,00€2mg56,00€5mg88,00€10mg119,00€25mg235,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)87,00€Intepirdine
CAS:Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:344.88Acotiamide monohydrochloride trihydrate
CAS:Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.Fórmula:C21H37ClN4O8SPureza:98% - 99.54%Cor e Forma:SolidPeso molecular:541.06Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Cor e Forma:White PowderPeso molecular:614.021-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide
CAS:<p>1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.</p>Fórmula:C20H30Br2N2Pureza:98.17%Cor e Forma:SolidPeso molecular:458.275-BDBD
CAS:5-BDBD is a potent and selective P2X4 receptor antagonist.Fórmula:C17H11BrN2O2Pureza:97.78%Cor e Forma:SolidPeso molecular:355.19Ref: TM-T22518
1mg43,00€2mg57,00€5mg92,00€10mg144,00€25mg305,00€50mg543,00€100mg775,00€1mL*10mM (DMSO)93,00€Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Fórmula:C15H18BrN3O3Pureza:98.51% - 99.24%Cor e Forma:SolidPeso molecular:368.23Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Fórmula:C6H10ClNO2Pureza:98.42%Cor e Forma:SolidPeso molecular:163.602Edonerpic maleate
CAS:Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).Fórmula:C20H25NO6SPureza:98.24%Cor e Forma:SolidPeso molecular:407.48NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Fórmula:C25H25N3O2SPureza:98%Cor e Forma:SolidPeso molecular:431.55Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Fórmula:C22H28FNO3Pureza:98.94% - 99.95%Cor e Forma:SolidPeso molecular:373.46Ref: TM-T5389
1mg42,00€5mg88,00€10mg124,00€25mg233,00€50mg301,00€100mg393,00€200mg560,00€1mL*10mM (DMSO)96,00€Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Fórmula:C20H24O9Pureza:98.76% - 99.81%Cor e Forma:White PowderPeso molecular:408.4Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:440.94NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Fórmula:C14H9Cl2F3N2O2Pureza:99.11%Cor e Forma:SolidPeso molecular:365.13A-582941 dihydrochloride
CAS:A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFórmula:C17H22Cl2N4Pureza:99.55%Cor e Forma:SolidPeso molecular:353.29Ref: TM-T22016
1mg42,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg533,00€200mg743,00€1mL*10mM (DMSO)87,00€Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Fórmula:C20H26N2O7SPureza:99.86% - 99.99%Cor e Forma:SolidPeso molecular:438.49m-Chlorophenylbiguanide hydrochloride
CAS:m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Fórmula:C8H11Cl2N5Pureza:99.43% - 99.87%Cor e Forma:SolidPeso molecular:248.11Donepezil
CAS:<p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>Fórmula:C24H29NO3Pureza:99.69%Cor e Forma:White Or Almost White Crystal PowderPeso molecular:379.49
