
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(639 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.031 produtos)
- BACE(37 produtos)
- Beta Amilóide(221 produtos)
- CaMK(73 produtos)
- COX(600 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(369 produtos)
- Gama-secretase(57 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(325 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5459 produtos de "Neurociência"
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3-AQC
CAS:3-AQC is a competitive antagonist of 5-HT3.Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28Ref: TM-T8007
2mg34,00€5mg50,00€10mg81,00€25mg137,00€50mg215,00€100mg340,00€500mg795,00€1mL*10mM (DMSO)55,00€SB-334867 free base
CAS:SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:319.32Ref: TM-T6140
2mg42,00€5mg70,00€10mg99,00€25mg160,00€50mg226,00€100mg338,00€200mg502,00€1mL*10mM (DMSO)78,00€Aclidinium bromide
CAS:Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.
Fórmula:C26H30NO4S2·BrPureza:99.53% - 99.69%Cor e Forma:SolidPeso molecular:564.55Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Cor e Forma:SolidPeso molecular:495.58Mosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFórmula:C21H25ClFN3O3Pureza:99.56%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:421.89α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Cor e Forma:SolidPeso molecular:1770.99Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Fórmula:C15H17N3O3Cor e Forma:SolidPeso molecular:287.31Duloxetine
CAS:Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.Fórmula:C18H19NOSPureza:99.71% - 99.89%Cor e Forma:SolidPeso molecular:297.41STO-609
CAS:STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.
Fórmula:C19H10N2O3Pureza:97.14% - 98.8%Cor e Forma:SolidPeso molecular:314.29Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Fórmula:C20H33NO7Pureza:99.26%Cor e Forma:White Crystalline PowdePeso molecular:399.48Frovatriptan Succinate
CAS:Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.Fórmula:C18H25N3O6Cor e Forma:SolidPeso molecular:379.41Temanogrel
CAS:Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).Fórmula:C24H28N4O4Pureza:99.24%Cor e Forma:SolidPeso molecular:436.5Ref: TM-T17033
1mg49,00€5mg103,00€10mg154,00€25mg250,00€50mg354,00€100mg480,00€200mg622,00€1mL*10mM (DMSO)112,00€MK-0752 Sodium
CAS:Sodium MK-0752 is a novel and potent gamma-secretase inhibitor that has been evaluated in clinical trials for the treatment of various types of cancer.Fórmula:C21H21ClF2NaO4SCor e Forma:SolidPeso molecular:465.89GNE-7915
CAS:GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.Fórmula:C19H21F4N5O3Pureza:98% - ≥95%Cor e Forma:SolidPeso molecular:443.4Ref: TM-T1945
5mg44,00€10mg58,00€25mg108,00€50mg177,00€100mg299,00€200mg389,00€500mg645,00€1mL*10mM (DMSO)48,00€MK-0752
CAS:MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).
Fórmula:C21H21ClF2O4SPureza:98% - 99.55%Cor e Forma:SolidPeso molecular:442.9Tianeptine sodium salt
CAS:Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H24ClN2NaO4SPureza:99.82%Cor e Forma:SolidPeso molecular:458.93Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Cor e Forma:SolidPeso molecular:552.7Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Fórmula:C17H19N3O4Cor e Forma:SolidPeso molecular:329.356RO4929097
CAS:RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).Fórmula:C22H20F5N3O3Pureza:98.5% - 99.51%Cor e Forma:SolidPeso molecular:469.4Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Cor e Forma:SolidPeso molecular:463.87Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Fórmula:C21H28BrNO3Pureza:99.29%Cor e Forma:SolidPeso molecular:422.36Frentizole
CAS:Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interactionFórmula:C15H13N3O2SPureza:99.82%Cor e Forma:SolidPeso molecular:299.35CZC-54252
CAS:CZC-54252 is a potent inhibitor of LRRK2.Fórmula:C22H25ClN6O4SPureza:99.39%Cor e Forma:SolidPeso molecular:504.99Miridesap
CAS:Miridesap (GSK2315698) rapidly depletes SAP in blood, cerebrospinal fluid, and amyloid deposits via liver clearance.Fórmula:C16H24N2O6Pureza:≥95%Cor e Forma:SolidPeso molecular:340.37Clomipramine
CAS:Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.Fórmula:C19H23ClN2Pureza:99.31% - 99.71%Cor e Forma:SolidPeso molecular:314.85Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Fórmula:C20H25NO2S2Pureza:99.25% - 99.67%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7Oxyphencyclimine Hydrochloride
CAS:Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Fórmula:C20H29ClN2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:380.91KN-92 hydrochloride
CAS:KN-92 hydrochloride is an inactive derivative of KN-93.Fórmula:C24H26Cl2N2O3SPureza:99.68%Cor e Forma:SolidPeso molecular:493.45Chelidamic acid
CAS:Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.Fórmula:C7H5NO5Pureza:98.11%Cor e Forma:Pale Yellow PowderPeso molecular:183.12Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Cor e Forma:SolidPeso molecular:477.57Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Cor e Forma:Off-White PowderPeso molecular:298.29Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Fórmula:C19H23N3O3Pureza:99.96%Cor e Forma:SolidPeso molecular:341.4Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFórmula:C21H20FN3O5SPureza:99.21% - 99.42%Cor e Forma:SolidPeso molecular:445.46Ref: TM-T7165
2mg35,00€5mg52,00€10mg74,00€25mg116,00€50mg187,00€100mg356,00€500mg802,00€1mL*10mM (DMSO)49,00€A-484954
CAS:A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.Fórmula:C13H15N5O3Pureza:97.47% - 99.86%Cor e Forma:SolidPeso molecular:289.29Ref: TM-TQ0137
1mg43,00€2mg56,00€5mg88,00€10mg144,00€25mg305,00€50mg543,00€100mg775,00€1mL*10mM (DMSO)103,00€Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Fórmula:C12H16N2O4Pureza:98%Cor e Forma:SolidPeso molecular:207.23Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Fórmula:C23H29F2N3OPureza:99.68%Cor e Forma:SolidPeso molecular:401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€1mL*10mM (DMSO)321,00€JI130
CAS:JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.Fórmula:C23H24N2O3Pureza:99.61%Cor e Forma:SolidPeso molecular:376.45Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Fórmula:C19H15BrClF3N2O3SPureza:99.76%Cor e Forma:SolidPeso molecular:523.75Ref: TM-T8946
1mg42,00€5mg82,00€10mg116,00€25mg188,00€50mg260,00€100mg366,00€200mg497,00€1mL*10mM (DMSO)95,00€Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Fórmula:C12H17ClN2O2Pureza:99.35%Cor e Forma:SolidPeso molecular:256.73CRANAD 2
CAS:CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.Fórmula:C23H25BF2N2O2Pureza:99.44%Cor e Forma:Dark Blue To Black PowderPeso molecular:410.27VU-1545
CAS:VU-1545 is mGlu5 positive allosteric modulator.Fórmula:C22H15FN4O3Pureza:98.8%Cor e Forma:SolidPeso molecular:402.38Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Fórmula:C22H32ClN3O2Cor e Forma:SolidPeso molecular:405.96Cyclopiazonic acid
CAS:Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Cor e Forma:SolidPeso molecular:336.38Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Fórmula:C20H17NO6Pureza:98% - 99.99%Cor e Forma:Light Yellow PowderPeso molecular:367.35LY 2886721 Hydrochloride
CAS:Potent, selective BACE inhibitor; IC50 of 10.2 nM (BACE2) & 20.3 nM (BACE1). >5000x selectivity vs. other proteases. Lowers Aβ & sAPPβ in Alzheimer's mice.Fórmula:C18H17ClF2N4O2SCor e Forma:SolidPeso molecular:426.87Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48Ref: TM-TN1465
1mg138,00€2mg203,00€5mg298,00€10mg449,00€25mg765,00€50mg1.054,00€100mg1.423,00€1mL*10mM (DMSO)306,00€
