
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(641 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(2.997 produtos)
- BACE(37 produtos)
- Beta Amilóide(217 produtos)
- CaMK(73 produtos)
- COX(598 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(370 produtos)
- Gama-secretase(57 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(325 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5450 produtos de "Neurociência"
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ML380
CAS:ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).Fórmula:C23H25F3N4O3SPureza:99.69%Cor e Forma:SolidPeso molecular:494.53Ref: TM-T28069
2mg47,00€5mg71,00€10mg113,00€25mg178,00€50mg334,00€100mg500,00€500mg1.099,00€1mL*10mM (DMSO)78,00€PF-06454589
CAS:PF-06454589 is a potent inhibitor of LRRK2.Fórmula:C14H16N6OPureza:99.06%Cor e Forma:SolidPeso molecular:284.32Ref: TM-T7729
2mg34,00€5mg52,00€10mg75,00€25mg128,00€50mg187,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)52,00€Flutriafol
CAS:Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist
Fórmula:C16H13F2N3OPureza:98.75%Cor e Forma:SolidPeso molecular:301.29VU 0238429
CAS:VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28Ref: TM-T8007
2mg34,00€5mg50,00€10mg81,00€25mg137,00€50mg215,00€100mg340,00€500mg795,00€1mL*10mM (DMSO)55,00€Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Fórmula:C17H11N5OPureza:99.81%Cor e Forma:SolidPeso molecular:301.3Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Cor e Forma:SolidPeso molecular:177.63Ref: TM-T5799
2mg34,00€5mg48,00€10mg67,00€25mg100,00€50mg149,00€100mg213,00€200mg316,00€1mL*10mM (DMSO)49,00€GSK2578215A
CAS:GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Fórmula:C24H18FN3O2Pureza:99.57% - 99.94%Cor e Forma:SolidPeso molecular:399.42Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Fórmula:C17H19N3O4Cor e Forma:SolidPeso molecular:329.356N-ACETYLTRYPTAMINE
CAS:N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Fórmula:C12H14N2OPureza:98.79%Cor e Forma:PowderPeso molecular:202.25TA-03
CAS:TA-03 (7-Meota) is a potent inhibitor of AChE in treatment of cognitive manifestation of AD.Fórmula:C14H16N2OPureza:99.22%Cor e Forma:SolidPeso molecular:228.29Ref: TM-T8585
1mg58,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€1mL*10mM (DMSO)104,00€pep2-EVKI acetate(1315378-67-6 free base)
Pep2-EVKI acetate, a cell-permeable peptide, disrupts PICK1-GluR2 AMPA receptor binding.Fórmula:C64H99N13O21Pureza:97.63%Cor e Forma:SolidPeso molecular:1386.551-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple
Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.756-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFórmula:C11H11N3OPureza:99.03%Cor e Forma:SolidPeso molecular:201.22Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Fórmula:C10H20CaN2O8S2Pureza:98% - 99.93%Cor e Forma:White Odorless Or Nearly Odorless PowderPeso molecular:400.48CALP1 acetate
CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.
Fórmula:C42H79N9O12Pureza:99.63%Cor e Forma:SolidPeso molecular:902.13JI130
CAS:JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.Fórmula:C23H24N2O3Pureza:99.61%Cor e Forma:SolidPeso molecular:376.45Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Fórmula:C20H25NO2Cor e Forma:SolidPeso molecular:311.42Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Fórmula:C21H25NO4Pureza:99.8% - 99.91%Cor e Forma:Off-White SolidPeso molecular:355.43Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
Fórmula:C53H90O22Pureza:98.83% - 99.56%Cor e Forma:White PowderPeso molecular:1079.27Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Fórmula:C18H18ClNSPureza:98.77% - 99.756%Cor e Forma:Pale Yellow Crystals SolidPeso molecular:315.86Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Fórmula:C16H14FN3OPureza:99.72%Cor e Forma:SolidPeso molecular:283.3Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48Ref: TM-TN1465
1mg138,00€2mg203,00€5mg298,00€10mg449,00€25mg765,00€50mg1.054,00€100mg1.423,00€1mL*10mM (DMSO)306,00€VU0361737
CAS:VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.Fórmula:C13H11ClN2O2Pureza:99.60% - 99.85%Cor e Forma:SolidPeso molecular:262.69NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Fórmula:C28H29Cl2N3OPureza:98.79%Cor e Forma:SolidPeso molecular:494.46Ref: TM-T28167
2mg38,00€5mg55,00€10mg86,00€25mg155,00€50mg264,00€100mg374,00€500mgA consultar1mL*10mM (DMSO)72,00€Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Cor e Forma:SolidPeso molecular:552.7ST034307
CAS:ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).Fórmula:C10H4Cl4O2Pureza:99.28%Cor e Forma:SolidPeso molecular:297.95Ref: TM-T16938
1mg38,00€2mg49,00€5mg81,00€10mg115,00€25mg235,00€50mg373,00€100mg597,00€200mg842,00€1mL*10mM (DMSO)88,00€Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Fórmula:C20H21N3OPureza:99.17%Cor e Forma:SolidPeso molecular:319.4γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Fórmula:C6H9NO2Cor e Forma:SolidPeso molecular:127.143Serotonin
CAS:Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Fórmula:C10H12N2OPureza:97.47% - 99.92%Cor e Forma:SolidPeso molecular:176.22Ref: TM-TN2437
2mg34,00€5mg52,00€10mg85,00€25mg157,00€50mg250,00€100mg404,00€200mg585,00€1mL*10mM (DMSO)46,00€VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Fórmula:C18H19N3O2SPureza:99.56%Cor e Forma:SolidPeso molecular:341.43Ref: TM-T17238
2mg39,00€5mg58,00€10mg92,00€25mg195,00€50mg325,00€100mg522,00€200mg743,00€1mL*10mM (DMSO)64,00€Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Fórmula:C6H11NO2Pureza:99.82%Cor e Forma:White To Faint Pink-Beige PowderPeso molecular:129.16Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Fórmula:C24H32ClNO6Pureza:99.73%Cor e Forma:Colorless LiquidPeso molecular:465.97VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Fórmula:C15H10BrNO2Pureza:97.56%Cor e Forma:SolidPeso molecular:316.15(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
CAS:(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).Fórmula:C6H8Cl2N2Pureza:97.23%Cor e Forma:SolidPeso molecular:179.05α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Pureza:98%Cor e Forma:LiquidPeso molecular:N/AMosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFórmula:C21H25ClFN3O3Pureza:99.56%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:421.89Temanogrel
CAS:Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).Fórmula:C24H28N4O4Pureza:99.24%Cor e Forma:SolidPeso molecular:436.5Ref: TM-T17033
1mg49,00€5mg103,00€10mg154,00€25mg250,00€50mg354,00€100mg480,00€200mg622,00€1mL*10mM (DMSO)112,00€Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Fórmula:C30H18O10Pureza:98.21% - 99.22%Cor e Forma:Odourless Whitish SolidPeso molecular:538.46Ref: TM-T3417
2mg34,00€5mg50,00€10mg80,00€25mg126,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)59,00€Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Fórmula:C17H21ClN4SCor e Forma:SolidPeso molecular:348.89Glypromate acetate(32302-76-4 free base)
Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.Fórmula:C14H23N3O8Pureza:99.94%Cor e Forma:SolidPeso molecular:361.35Ref: TM-T7778L
2mg37,00€5mg52,00€10mg74,00€25mg119,00€50mg160,00€100mg225,00€200mg314,00€1mL*10mM (DMSO)57,00€Pitofenone
CAS:Pitofenone is an inhibitor of the acetylcholinesterase activity from bovine erythrocytes and electric eel.Fórmula:C22H25NO4Cor e Forma:SolidPeso molecular:367.44ARC-239
CAS:ARC-239 is an agonist of α2-adrenergic receptor.Fórmula:C24H29N3O3Cor e Forma:SolidPeso molecular:407.51Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Fórmula:C23H24FN3O2Pureza:99.2%Cor e Forma:SolidPeso molecular:393.45LP-922761 hydrate
LP-922761 hydrate: selective AAK1 inhibitor; IC50: 4.8 nM (enzyme), 7.6 nM (cellular); also inhibits BIKE (IC50: 24 nM); inert to GAK, opioids, α2, GABAa.Fórmula:C21H28N6O4Cor e Forma:SolidPeso molecular:414.98NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Fórmula:C23H19N3OPureza:99.44% - 99.86%Cor e Forma:SolidPeso molecular:353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€7-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16Ro 67-7476
CAS:Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.Fórmula:C17H18FNO2SPureza:99.69%Cor e Forma:SolidPeso molecular:319.39Ref: TM-T3478
1mg34,00€2mg48,00€5mg88,00€10mg124,00€25mg244,00€50mg442,00€100mg643,00€1mL*10mM (DMSO)78,00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Mivacurium dichloride
CAS:Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Cor e Forma:Off-White SolidPeso molecular:1100.17Ref: TM-T22371
2mg46,00€5mg65,00€10mg94,00€25mg123,00€50mg188,00€100mg286,00€200mg434,00€1mL*10mM (DMSO)90,00€

