
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(645 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.022 produtos)
- BACE(37 produtos)
- Beta Amilóide(228 produtos)
- CaMK(73 produtos)
- COX(600 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(372 produtos)
- Gama-secretase(61 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5574 produtos de "Neurociência"
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(RS)-3-Hydroxyphenylglycine
CAS:(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.Fórmula:C8H9NO3Pureza:99.29%Cor e Forma:SolidPeso molecular:167.16BRL-15572 hydrochloride
CAS:BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.Fórmula:C25H28Cl2N2OCor e Forma:SolidPeso molecular:443.41SB-203186 hydrochloride
CAS:SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Fórmula:C17H21F3O3Pureza:99.69% - >99.99%Cor e Forma:SolidPeso molecular:330.34Ref: TM-T4176
2mg43,00€5mg60,00€1mL*10mM (DMSO)71,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€LPYFD-NH2 acetate
LPYFD-NH2 acetate shows some inhibitory effect on the aggregation of Abeta(1-42).Fórmula:C35H48N6O10Pureza:96.51%Cor e Forma:SolidPeso molecular:712.79Ref: TM-T22932L
1mg66,00€5mg130,00€10mg187,00€1mL*10mM (DMSO)188,00€25mg309,00€50mg439,00€100mg590,00€200mg793,00€Sevoflurane
CAS:Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Fórmula:C4H3F7OPureza:98%Cor e Forma:Less Oil Colorless OilPeso molecular:200.05Ref: TM-T22425
2mg39,00€5mg54,00€1mL*10mM (DMSO)56,00€10mg75,00€25mg110,00€50mg158,00€100mg226,00€200mg339,00€γ-Mangostin
CAS:Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Fórmula:C23H24O6Pureza:98.55% - 99.08%Cor e Forma:SolidPeso molecular:396.43Oxyphenonium bromide
CAS:Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.
Fórmula:C21H34BrNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:428.404Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Fórmula:C18H27ClN2O4Pureza:99.74%Cor e Forma:SolidPeso molecular:370.87Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.28%Cor e Forma:Colorless - Light Yellow Clear LiquidPeso molecular:155.28GNE-7915
CAS:GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.Fórmula:C19H21F4N5O3Pureza:98% - ≥95%Cor e Forma:SolidPeso molecular:443.4Ref: TM-T1945
5mg44,00€1mL*10mM (DMSO)48,00€10mg58,00€25mg108,00€50mg177,00€100mg299,00€200mg389,00€500mg645,00€Miridesap
CAS:Miridesap (GSK2315698) rapidly depletes SAP in blood, cerebrospinal fluid, and amyloid deposits via liver clearance.Fórmula:C16H24N2O6Pureza:≥95%Cor e Forma:SolidPeso molecular:340.37Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Fórmula:C10H22ClNCor e Forma:SolidPeso molecular:191.74FPS-ZM1
CAS:FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.Fórmula:C20H22ClNOPureza:99.32% - 99.52%Cor e Forma:SolidPeso molecular:327.85Ref: TM-T3259
5mg48,00€1mL*10mM (DMSO)50,00€10mg54,00€25mg96,00€50mg140,00€100mg207,00€200mg333,00€500mg560,00€MK-0752 Sodium
CAS:Sodium MK-0752 is a novel and potent gamma-secretase inhibitor that has been evaluated in clinical trials for the treatment of various types of cancer.Fórmula:C21H21ClF2NaO4SCor e Forma:SolidPeso molecular:465.89MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Fórmula:C22H28FNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:373.46Ref: TM-T22359
1mg99,00€5mg187,00€1mL*10mM (DMSO)222,00€10mg280,00€25mg434,00€50mg585,00€100mg775,00€200mg1.054,00€Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Fórmula:C6H11NO2Pureza:99.82%Cor e Forma:White To Faint Pink-Beige PowderPeso molecular:129.16Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Fórmula:C23H29F2N3OPureza:99.68%Cor e Forma:SolidPeso molecular:401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€1mL*10mM (DMSO)321,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€MPEP
CAS:MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.Fórmula:C14H11NPureza:99.54%Cor e Forma:SolidPeso molecular:193.24Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Fórmula:C35H43N5O4Pureza:98.12%Cor e Forma:SolidPeso molecular:597.75F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Fórmula:C19H21ClF2N4OPureza:98.72%Cor e Forma:SolidPeso molecular:394.85Ref: TM-T7281
1mg49,00€5mg92,00€1mL*10mM (DMSO)104,00€10mg152,00€25mg295,00€50mg477,00€100mg715,00€200mg982,00€Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Fórmula:C19H22O2Pureza:99.22% - 99.66%Cor e Forma:SolidPeso molecular:282.38GNE-9605
CAS:GNE-9605 is a highly effective, specifical, and brain-penetrant LRRK2 inhibitor (IC50: 19 nM).Fórmula:C17H20ClF4N7OPureza:98.55% - 98.75%Cor e Forma:SolidPeso molecular:449.83AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89Ref: TM-T26690
1mg34,00€5mg75,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg205,00€50mg334,00€100mg557,00€200mg790,00€Ipratropium Bromide
CAS:Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Fórmula:C20H30BrNO3Pureza:99.92%Cor e Forma:SolidPeso molecular:412.37Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Fórmula:C8H11N5Pureza:99.54%Cor e Forma:SolidPeso molecular:177.21(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Fórmula:C20H20O5Pureza:99.47%Cor e Forma:SolidPeso molecular:340.37ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Fórmula:C13H16ClN3O3Pureza:98.15%Cor e Forma:SolidPeso molecular:297.74Ref: TM-T9193
1mg50,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg172,00€25mg304,00€50mg424,00€100mg583,00€200mg785,00€W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Fórmula:C32H44Br2N4O4Pureza:95.56%Cor e Forma:SolidPeso molecular:708.52Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Fórmula:C23H31ClN2O2Pureza:99.71%Cor e Forma:SolidPeso molecular:402.96Avagacestat
CAS:Avagacestat (BMS-708163) (BMS-708163) is a potent, selective, orally bioavailable γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM,Fórmula:C20H17ClF4N4O4SPureza:98.87% - 99.73%Cor e Forma:SolidPeso molecular:520.89Ref: TM-T6249
1mg38,00€5mg77,00€1mL*10mM (DMSO)88,00€10mg116,00€25mg215,00€50mg310,00€100mg450,00€200mg605,00€GSK2578215A
CAS:GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Fórmula:C24H18FN3O2Pureza:99.57% - 99.94%Cor e Forma:SolidPeso molecular:399.42NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Fórmula:C14H8N4OPureza:99.12%Cor e Forma:SolidPeso molecular:248.24SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Fórmula:C18H21ClF3N3OPureza:99.03% - 99.95%Cor e Forma:SolidPeso molecular:387.83Ref: TM-T4522
2mg34,00€1mL*10mM (DMSO)46,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€Ondansetron
CAS:Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.Fórmula:C18H19N3OPureza:99.92%Cor e Forma:White To Yellow CrystalsPeso molecular:293.36FTIDC
CAS:FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.Fórmula:C18H23FN6OPureza:94.58%Cor e Forma:SolidPeso molecular:358.41Ref: TM-T3483
1mg100,00€2mg145,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg565,00€50mg797,00€100mg1.071,00€LRRK2-IN-1
CAS:LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.Fórmula:C31H38N8O3Pureza:98% - 98.82%Cor e Forma:SolidPeso molecular:570.69Semagacestat
CAS:Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).Fórmula:C19H27N3O4Pureza:97.1% - 99.9%Cor e Forma:SolidPeso molecular:361.44(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Fórmula:C12H14O5Pureza:99.83%Cor e Forma:SolidPeso molecular:238.24RAGE antagonist peptide acetate
RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.Fórmula:C59H105N13O19SPureza:97.17%Cor e Forma:SolidPeso molecular:1332.61Amyloid β-Protein 10-20 acetate
Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research ofFórmula:C73H103N17O18Pureza:97.23%Cor e Forma:SolidPeso molecular:1506.65Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Fórmula:C16H23Cl2N3O2Cor e Forma:SolidPeso molecular:360.28Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Fórmula:C80H122F3N21O22Pureza:99.41%Cor e Forma:SolidPeso molecular:1786.98Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:463A 582941 HCl (848591-90-2(free base))
A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing propertiesFórmula:C17H21ClN4Pureza:99.83%Cor e Forma:SolidPeso molecular:316.83Ref: TM-T8725
1mg58,00€1mL*10mM (DMSO)116,00€5mg118,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Nanofin
CAS:Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.Fórmula:C7H15NPureza:97.38% - 99.818%Cor e Forma:Clear Colorless To Slightly Yellow LiquidPeso molecular:113.2Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Fórmula:C28H36N4O2S·HClPureza:99.51%Cor e Forma:SolidPeso molecular:529.14Ref: TM-T1735
5mg39,00€1mL*10mM (DMSO)54,00€10mg59,00€25mg75,00€50mg90,00€100mg137,00€200mg213,00€500mg447,00€
