
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(636 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.030 produtos)
- BACE(37 produtos)
- Beta Amilóide(226 produtos)
- CaMK(73 produtos)
- COX(601 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(369 produtos)
- Gama-secretase(62 produtos)
- GluR(264 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(325 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5488 produtos de "Neurociência"
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SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Fórmula:C25H31N3O2SPureza:99.12% - 99.69%Cor e Forma:SolidPeso molecular:437.6CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Fórmula:C21H21Cl2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:446.33JNJ-40068782
CAS:JNJ-40068782 is a potent, selective and systemically active positive allosteric modulator of the mGlu2 receptor.Fórmula:C21H23N3OPureza:98%Cor e Forma:SolidPeso molecular:333.43MAO-IN-M30 dihydrochloride
CAS:MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.Fórmula:C14H16Cl2N2OPureza:99.83%Cor e Forma:SolidPeso molecular:299.2Ref: TM-T38034
1mg35,00€2mg46,00€5mg69,00€10mg96,00€25mg170,00€50mg244,00€100mg336,00€500mgA consultarZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Fórmula:C23H22N2O4Cor e Forma:SolidPeso molecular:390.43Afacifenacin
CAS:Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.Fórmula:C27H26F3N3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:481.51Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Fórmula:C13H10N2OPureza:98.66%Cor e Forma:SolidPeso molecular:210.23Piperilate
CAS:Piperilate (Pipethanate), a hetrazepine PAF antagonist and anticholinergic used in asthma studies, counters organophosphate toxicity.Fórmula:C21H25NO3Cor e Forma:SolidPeso molecular:339.43EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Fórmula:C15H22N2OPureza:97.66% - 99.78%Cor e Forma:SolidPeso molecular:246.35Ref: TM-T11183
1mg92,00€2mg125,00€5mg170,00€10mg213,00€25mg474,00€50mg688,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)170,00€Auglurant
CAS:Auglurant is a novel and selective mGlu5 antagonist (IC50: 11 nM (rat) and an IC50: 14 nM (human)). Auglurant has an acceptable CNS penetration.Fórmula:C16H12FN5O2Cor e Forma:SolidPeso molecular:325.3Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Fórmula:C21H25ClN2O4SPureza:99.57%Cor e Forma:SolidPeso molecular:436.95CP 135807
CAS:CP 135807 is a 5-HT1D receptor agonist.Fórmula:C19H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:351.4MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Fórmula:C4H10NO6PPureza:98%Cor e Forma:SolidPeso molecular:199.1GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Fórmula:C19H16N4OCor e Forma:SolidPeso molecular:316.36AChE/MAO-IN-2
Potent AChE/MAO-B inhibitor; IC50: AChE 0.0224 μM, MAO-B 0.0412 μM, MAO-A 0.1116 μM. Antioxidant, anti-β-amyloid, for AD research.Fórmula:C23H26N2O3Cor e Forma:SolidPeso molecular:378.46(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:98%Cor e Forma:SolidPeso molecular:250.12TASP0433864
CAS:TASP0433864 enhances mGlu2 activity; EC50: 199 nM (human), 206 nM (rat); not an agonist.Fórmula:C18H23N3O3Pureza:98%Cor e Forma:SolidPeso molecular:329.39AFDX384
CAS:AFDX384 is potent M2/M4 selective antagonist.Fórmula:C28H42N6O5SCor e Forma:SolidPeso molecular:574.74ZAPA sulfate
CAS:GABAA receptors agonistFórmula:C4H8N2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:244.25VU6010572
CAS:VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.Fórmula:C20H18FNO3Cor e Forma:SolidPeso molecular:339.36VU6001966
CAS:VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.Fórmula:C17H15FN4O2Pureza:98%Cor e Forma:SolidPeso molecular:326.33Aβ Fibrillization modulator 1
CAS:Aβ Fibrillization Modulator 1 stabilizes amyloid-beta (Aβ) monomers, preventing their aggregation into fibrils.Fórmula:C17H12N4O3SSeCor e Forma:SolidPeso molecular:431.33Bisindolylmaleimide VII
CAS:Bisindolylmaleimide VII is a selective inhibitor of protein kinase C.Fórmula:C27H27N5O2Cor e Forma:SolidPeso molecular:453.54DPNB-ABT594
DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.Fórmula:C31H46ClN3O11Cor e Forma:SolidPeso molecular:672.16AChE-IN-12
CAS:AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.Fórmula:C33H41NO7Cor e Forma:SolidPeso molecular:563.68AC-42
CAS:AC-42 is an allosteric agonist of M1 muscarinic receptor.
Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47BMS-911172
CAS:BMS-911172 is an adaptor associated kinase 1 (AAK1 kinase) inhibitor with an IC 50 of 35 nM.Fórmula:C16H19F2N3O3Cor e Forma:SolidPeso molecular:339.34CGS 12066B dimaleate
CAS:5-HT1B full agonistFórmula:C25H25F3N4O8Pureza:98%Cor e Forma:SolidPeso molecular:566.48AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Fórmula:C20H19ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:402.89RX 801077
CAS:RX 801077 is a selective I2R agonist, Ki of 70.1 nM, with anti-inflammatory and neuroprotective properties for TBI research.Fórmula:C11H10N2OCor e Forma:SolidPeso molecular:186.21CP 93129 dihydrochloride
CAS:5-HT1B agonist, potent and highly selectiveFórmula:C12H14ClN3OPureza:98%Cor e Forma:SolidPeso molecular:251.71Parapenzolate bromide
CAS:Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.Fórmula:C21H26BrNO3Cor e Forma:SolidPeso molecular:420.347Prucalopride hydrochloride
CAS:Prucalopride hydrochloride is a selective agonist of the 5-HT4.Fórmula:C18H27Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:404.33ZM 169369
CAS:ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.Fórmula:C19H20N2SCor e Forma:SolidPeso molecular:308.44VU0409106
CAS:VU0409106 is a potent, mGlu5-selective inhibitor.Fórmula:C15H11FN4O2SPureza:98%Cor e Forma:SolidPeso molecular:330.34Cycrimine
CAS:Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.Fórmula:C19H29NOCor e Forma:SolidPeso molecular:287.44Alniditan dihydrochloride
CAS:Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.Fórmula:C17H28Cl2N4OCor e Forma:SolidPeso molecular:375.34Milameline hydrochloride
CAS:Milameline hydrochloride is a Muscarinic receptor agonist.Fórmula:C8H15ClN2OPureza:98%Cor e Forma:SolidPeso molecular:190.67Arecaidine but-2-ynyl ester tosylate
CAS:mAChR M2 agonistFórmula:C18H23NO5SPureza:98%Cor e Forma:SolidPeso molecular:365.44TC-2153
CAS:TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.Fórmula:C7H5ClF3NS5Cor e Forma:SolidPeso molecular:355.89Pimprinine
CAS:Pimprinine: an alkaloid, inhibits MAO, and has anticonvulsant properties.Fórmula:C12H10N2OCor e Forma:SolidPeso molecular:198.22FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Fórmula:C22H19N5Cor e Forma:SolidPeso molecular:353.42γ-Secretase modulator 11
CAS:5-{8-[(3,4'-Difluoro[1,1'-biphenyl]-4-yl)methoxy]-2-methylimidazo[1,2-a]pyridin-3-yl}-N-methylpyridine-2-carboxamide (1o) exhibited high in vitro potency andFórmula:C28H22F2N4O2Cor e Forma:SolidPeso molecular:484.5PCS1055 dihydrochloride
CAS:PCS1055 is a selective M4 antagonist (IC50: 18.1 nM, Ki: 6.5 nM) and potent AChE inhibitor with >100-fold M1/M3/M5 selectivity.Fórmula:C27H34Cl2N4Pureza:98%Cor e Forma:SolidPeso molecular:485.49Tertatolol
CAS:Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.Fórmula:C16H25NO2SPureza:98%Cor e Forma:SolidPeso molecular:295.44SUN-C5174
CAS:"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."Fórmula:C22H29FN4O2Pureza:98%Cor e Forma:SolidPeso molecular:400.49AChE/BChE-IN-8
CAS:AChE/BChE-IN-8 inhibits AChE (Ki=0.788 μM) & BChE (Ki=2.364 μM), crosses the blood-brain barrier, and is low in cytotoxicity.Fórmula:C26H32N2O2Cor e Forma:SolidPeso molecular:404.54Itameline
CAS:RU 47213 can be used to inhibit scopolamine-induced working memory impairment in rats.Fórmula:C14H15ClN2O3Pureza:99.98%Cor e Forma:SolidPeso molecular:294.73Dual AChE-MAO B-IN-2
CAS:Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) & MAO B (0.01 μM); promising for Alzheimer's research.Fórmula:C26H25NO4Cor e Forma:SolidPeso molecular:415.48

