
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(636 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.030 produtos)
- BACE(37 produtos)
- Beta Amilóide(226 produtos)
- CaMK(73 produtos)
- COX(601 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(369 produtos)
- Gama-secretase(62 produtos)
- GluR(264 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(325 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5488 produtos de "Neurociência"
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EMD 56551
CAS:EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Cor e Forma:SolidPeso molecular:393.522Sultroponium
CAS:Sultroponium may be used as an anticholinergic agent or antispasmodic.Fórmula:C20H29NO6SCor e Forma:SolidPeso molecular:411.51(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFórmula:C6H12ClNO2Pureza:99.69%Cor e Forma:SolidPeso molecular:165.62CB-7921220
CAS:CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.Fórmula:C14H12N2O2Pureza:99.59%Cor e Forma:SolidPeso molecular:240.26Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48sEH/AChE-IN-2
CAS:sEH/AChE-IN-2 targets sEH & AChE, may reduce neuroinflammation & memory loss, potential in Alzheimer's research.Fórmula:C30H33ClF3N5O3Cor e Forma:SolidPeso molecular:604.06mGluR2 modulator 2
CAS:mGluR2 modulator 2: potent, selective, oral, EC50 = 0.13 μM, for antipsychotic research.Fórmula:C20H22FN3Cor e Forma:SolidPeso molecular:323.418-M-PDOT
CAS:8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.Fórmula:C14H19NO2Pureza:99.54% - 99.54%Cor e Forma:SolidPeso molecular:233.31Iferanserin
CAS:Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Fórmula:C23H28N2OCor e Forma:SolidPeso molecular:348.48NO 711
CAS:NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Fórmula:C21H22N2O3Pureza:99.70%Cor e Forma:SolidPeso molecular:350.41Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47JI051
CAS:JI051 has anti-tumor effects and can interact with PHB2 to inhibit the proliferation of HEK293 cells and pancreatic cancer cells.Fórmula:C22H24N2O3Pureza:≥98% - ≥98.0%Cor e Forma:SolidPeso molecular:364.44PF-06455943
CAS:PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK & Parkinson's research.Fórmula:C17H14FN5OCor e Forma:SolidPeso molecular:323.32Talaglumetad hydrochloride
CAS:Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.Fórmula:C11H17ClN2O5Cor e Forma:SolidPeso molecular:292.72AZD 0328
CAS:AZD 0328 is a nicotinic receptor agonist for α7 neurons.Fórmula:C13H16N2OCor e Forma:SolidPeso molecular:216.28AChE/BChE/MAO-B-IN-4
AChE/BChE/MAO-B-IN-4 inhibits MAO-B (IC50: 0.0393 µM), AChE (IC50: 0.0458 µM), BChE (IC50: 0.075 µM), and fights AD with antioxidant action.Fórmula:C26H33N3O4Cor e Forma:SolidPeso molecular:451.56Ambenonium dichloride
CAS:AChE inhibitorFórmula:C28H42Cl3N4O2Pureza:98%Cor e Forma:SolidPeso molecular:573.02Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Fórmula:C32H44N4O3Pureza:98%Cor e Forma:SolidPeso molecular:532.72RX 67668
CAS:RX 67668: Muscle relaxant, relieves fatigue; cholinesterase inhibitor (IC50: 5 μM); reverses D-tubocurarine effects.Fórmula:C16H24ClNPureza:98%Cor e Forma:SolidPeso molecular:265.82Adenylyl cyclase type 2 agonist-1
CAS:Potent AC2 agonist with an EC50 of 90 nM, potential for respiratory disease treatment.Fórmula:C27H17BrClNO5Cor e Forma:SolidPeso molecular:550.78RO5488608
CAS:RO5488608 is a new type of high-efficiency mGlu2/3 NAM.Fórmula:C23H17F3N2O4SCor e Forma:SolidPeso molecular:474.45Aβ-IN-5
CAS:Aβ-IN-5 (Compound e12) is an orally active Aβ aggregation inhibitor that also inhibits AChE and BuChE with IC50 values of 21.29 μM and 1.32 μM, respectively.Fórmula:C21H20N2O3Cor e Forma:SolidPeso molecular:348.4A 841720
CAS:Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.Fórmula:C17H21N5OSCor e Forma:SolidPeso molecular:343.45BChE-IN-11
CAS:BChE-IN-11: potent, selective, non-competitive BChE inhibitor; IC50=2.1μM; used in AD research.Fórmula:C22H18O4Cor e Forma:SolidPeso molecular:346.38NPEC-caged-LY379268
CAS:NPEC-caged-LY379268 is a type II mGluR agonist [1].Fórmula:C16H16N2O9Cor e Forma:SolidPeso molecular:380.31Anabasine hydrochloride
CAS:neuronal nicotinic ACh receptor partial agonistFórmula:C10H15ClN2Pureza:98%Cor e Forma:White To Off-White SolidPeso molecular:198.693Pheniprazine
CAS:Pheniprazine, a potent and long-acting monoamine oxidase inhibitor, shows promise for depression research.Fórmula:C9H14N2Cor e Forma:SolidPeso molecular:150.22Ethybenztropine
CAS:Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.
Fórmula:C22H27NOPureza:98%Cor e Forma:SolidPeso molecular:321.46Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Fórmula:C22H27ClN2Cor e Forma:SolidPeso molecular:354.925-HT7 agonist 2
CAS:Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.Fórmula:C23H29N3OCor e Forma:SolidPeso molecular:363.5Memoquin
CAS:Memoquin is a multi-target-directed ligand for the therapy of Alzheimer's disease.Fórmula:C38H56N4O4Cor e Forma:SolidPeso molecular:632.88IEM 1925 dihydrobromide
CAS:AMPA receptor antagonistFórmula:C17H30Br2N2Pureza:98%Cor e Forma:SolidPeso molecular:422.24BChE-IN-7
CAS:BChE-IN-7 inhibits AChE/BChE selectively and reversibly; IC50 for BChE: 0.06 μM; crosses blood-brain barrier, protects neurons from Aβ toxicity.Fórmula:C21H24N2O2Cor e Forma:SolidPeso molecular:336.43Ambutonium bromide
CAS:Ambutonium bromide is an antagonist of acetylcholine.Fórmula:C20H27BrN2OPureza:98%Cor e Forma:SolidPeso molecular:391.35SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Fórmula:C19H27IN2O4Cor e Forma:SolidPeso molecular:474.33MAO-B-IN-12
CAS:MAO-B-IN-12 (16c) is a potent MAO-B inhibitor with an IC50 of 1.3 μM and has neuroprotective properties.Fórmula:C22H30O4Cor e Forma:SolidPeso molecular:358.47Antioxidant agent-2
CAS:Antioxidant agent-2 (3c), BBB-permeable, selectively chelates metals; shows neuroprotection, fights liver damage in Alzheimer's research.Fórmula:C23H26N2O7Cor e Forma:SolidPeso molecular:442.46VU0455691
CAS:VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.Fórmula:C24H25N5O3SPureza:98%Cor e Forma:SolidPeso molecular:463.55LY314228
CAS:LY314228 is an antagonist of 5-HT2A receptor.Fórmula:C20H24N4O3Cor e Forma:SolidPeso molecular:368.43SERT-IN-2
SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.Cor e Forma:SolidNAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Fórmula:C20H18ClNO2Cor e Forma:SolidPeso molecular:339.82FG-5893
CAS:FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.Fórmula:C27H29F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:465.53Trimedoxime bromide
CAS:Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.Fórmula:C15H18Br2N4O2Cor e Forma:SolidPeso molecular:446.14Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53MAO-B-IN-16
CAS:MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.Fórmula:C18H19NO3Cor e Forma:SolidPeso molecular:297.35BACE1/2-IN-1
CAS:BACE1/2-IN-1 inhibits BACE1/2 with IC50s of 0.01μM/0.0053μM, has better permeability and lower Pgp efflux but reduced metabolic stability.Fórmula:C21H31N5OSCor e Forma:SolidPeso molecular:401.57TMPH hydrochloride
CAS:neuronal nicotinic ACh receptors (nAChRs) antagonistFórmula:C16H32ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:305.88Hexafluronium Bromide
CAS:Hexafluronium bromide enhances muscle relaxation in surgery by blocking acetylcholine receptors.Fórmula:C36H42BrN2Cor e Forma:SolidPeso molecular:582.649Rivanicline oxalate
CAS:Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).Fórmula:C12H16N2O4Pureza:98%Cor e Forma:SolidPeso molecular:252.27ENS-163 phosphate
CAS:Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.Fórmula:C11H19N2O5PSPureza:98%Cor e Forma:SolidPeso molecular:322.32
