
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(576 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.949 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(565 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor GABA(337 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(26 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5389 produtos de "Neurociência"
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SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Fórmula:C16H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:302.33MAO-B-IN-11
CAS:<p>MAO-B-IN-11 (Compound 8c) is a strong MAO-B blocker with a 1.3 μM IC50 and neuroprotective effects.</p>Fórmula:C22H32O3Cor e Forma:SolidPeso molecular:344.49NRA-0160
CAS:<p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>Fórmula:C24H23F2N3OSPureza:98%Cor e Forma:SolidPeso molecular:439.52VU0366248
CAS:<p>VU0366248 is a mGlu5 negative allosteric modulator.</p>Fórmula:C14H7ClF2N2OPureza:98%Cor e Forma:SolidPeso molecular:292.67BGT1-IN-9
CAS:<p>BGT1-IN-9 is an M1 muscarinic agonist.</p>Fórmula:C5H10ClN3O2Cor e Forma:SolidPeso molecular:179.605GABAA receptor agent 5
CAS:<p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>Fórmula:C21H25N3O2SCor e Forma:SolidPeso molecular:383.51PF-3246799
CAS:<p>PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.</p>Fórmula:C15H17N3Pureza:98%Cor e Forma:SolidPeso molecular:239.32Amitriptylinoxide
CAS:<p>Amitriptylinoxide is an antidepressant.</p>Fórmula:C20H23NOPureza:98%Cor e Forma:SolidPeso molecular:293.4BGC 20-761
CAS:<p>BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.</p>Fórmula:C19H22N2OCor e Forma:SolidPeso molecular:294.39PF-03463275
CAS:<p>PF-03463275 is an orally active and selective reversible inhibitor of competitive glycine transporter protein-1 (GlyT1) with a Ki of 11.6 nM.PF-03463275 has CNS</p>Fórmula:C19H22ClFN4OPureza:99.86%Cor e Forma:SolidPeso molecular:376.86Way 100289
CAS:<p>Way 100289 is a selective 5-HT3 receptor antagonist.</p>Fórmula:C20H27N3O3Cor e Forma:SolidPeso molecular:357.453,3'-Difluorobenzaldazine
CAS:<p>allosteric potentiator of mGlu5</p>Fórmula:C14H10F2N2Pureza:98%Cor e Forma:SolidPeso molecular:244.24CGP 46381
CAS:<p>CGP 46381 is a GABAB receptor antagonist.</p>Fórmula:C10H22NO2PPureza:98%Cor e Forma:White SolidPeso molecular:219.26GAT107
CAS:<p>GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.</p>Fórmula:C18H17BrN2O2SPureza:99.33%Cor e Forma:SolidPeso molecular:405.31Sofiniclin
CAS:<p>Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).</p>Fórmula:C10H11Cl2N3Pureza:98%Cor e Forma:SolidPeso molecular:244.12SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Fórmula:C25H31N3O2SPureza:99.12% - 99.69%Cor e Forma:SolidPeso molecular:437.6(RS)-MCPG disodium salt
CAS:group I/group II metabotropic glutamate receptor antagonistFórmula:C10H11NNaO4Pureza:98%Cor e Forma:SolidPeso molecular:232.19Masupirdine mesylate
CAS:<p>Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease</p>Fórmula:C23H32BrN3O9S3Pureza:99.57%Cor e Forma:SolidPeso molecular:670.61Zimelidine dihydrochloride
CAS:<p>5-HT re-uptake inhibitor</p>Fórmula:C16H18BrClN2Pureza:98%Cor e Forma:SolidPeso molecular:353.69GSK-215083
CAS:<p>GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.</p>Fórmula:C20H20FN3O2SCor e Forma:SolidPeso molecular:385.46(+)-Donepezil
CAS:<p>(+)-Donepezil is an isomer of Donepezil -- a nootropic acting as an inhibitor of acetylcholinesterase.</p>Fórmula:C24H29NO3Cor e Forma:SolidPeso molecular:379.49Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Fórmula:C23H32Cl2FN3Pureza:98%Cor e Forma:SolidPeso molecular:440.42ELND006
CAS:<p>ELND006, an oral Alzheimer's drug, has improved bioavailability as a nanosuspension, and food doesn't affect it.</p>Fórmula:C20H14F5N3O2SCor e Forma:SolidPeso molecular:455.4mGluR2 modulator 1
CAS:<p>Potent mGluR2 modulator 1 crosses blood-brain barrier, EC50: 0.03 μM, useful for psychiatric research.</p>Fórmula:C21H20F3N3O3Cor e Forma:SolidPeso molecular:419.4RO4988546
CAS:<p>RO4988546 is a potent negative allosteric modulator of mGlu₂/₃.</p>Fórmula:C21H10F6N4O3SPureza:98%Cor e Forma:SolidPeso molecular:512.38Isamoltane hemifumarate
CAS:<p>5-HT1B antagonist</p>Fórmula:C16H22N202C4H404Pureza:98%Cor e Forma:SolidPeso molecular:332.4LSN2814617
CAS:<p>LSN2814617: oral, brain-penetrant mGlu5 PAM, EC50 = 52 nM (human), 42 nM (rat). Promotes wakefulness, useful in schizophrenia study.</p>Fórmula:C18H20FN5OPureza:98%Cor e Forma:SolidPeso molecular:341.38UCSF648
CAS:<p>UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].</p>Fórmula:C15H19ClN2O2SCor e Forma:SolidPeso molecular:326.84Milameline
CAS:<p>Milameline is a muscarinic receptor agonist that improves cognition.</p>Fórmula:C8H14N2OCor e Forma:SolidPeso molecular:154.21CP-409092 hydrochloride
CAS:<p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>Fórmula:C17H20ClN3O2Cor e Forma:SolidPeso molecular:333.81Rispenzepine
CAS:<p>Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.</p>Fórmula:C19H20N4O2Pureza:98%Cor e Forma:SolidPeso molecular:336.39CK59
CAS:<p>CK59 inhibits CaMKII and several voltage-gated calcium channels, with an IC50 of ~50 μM.</p>Fórmula:C21H37N7O3Pureza:98%Cor e Forma:SolidPeso molecular:435.56(S)-4C3HPG
CAS:<p>group I mGlu1a/1a receptor antagonist and mGluR2 agonist</p>Fórmula:C9H9NO5Pureza:98%Cor e Forma:SolidPeso molecular:211.17Arbaclofen placarbil
CAS:<p>Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.</p>Fórmula:C19H26ClNO6Cor e Forma:SolidPeso molecular:399.87TC-E 5006
CAS:γ-secretase modulatorFórmula:C29H29F4NO2Pureza:98%Cor e Forma:SolidPeso molecular:499.54LY 344864 S-enantiomer
CAS:<p>LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.</p>Fórmula:C21H22FN3OPureza:98%Cor e Forma:SolidPeso molecular:351.42Ethyl dirazepate
CAS:Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Fórmula:C18H14Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:377.22VU0364289
CAS:<p>VU0364289 is a positive allosteric modulator of mGlu5.</p>Fórmula:C20H21N3O2Cor e Forma:SolidPeso molecular:335.4Revatropate
CAS:<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Fórmula:C19H27NO4SCor e Forma:SolidPeso molecular:365.49Bopindolol fumarate
CAS:<p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>Fórmula:C27H32N2O7Cor e Forma:SolidPeso molecular:496.56AChE/BChE/BACE-1-IN-2
CAS:<p>Compound 4o, an oral AChE, BChE, & BACE-1 inhibitor, has potent antioxidant, neuroprotective qualities & breaks down Aβ aggregates.</p>Fórmula:C18H20F2N2Cor e Forma:SolidPeso molecular:302.36U-7524
CAS:<p>U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.</p>Fórmula:C2H5NO3Cor e Forma:SolidPeso molecular:91.07Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Cor e Forma:SolidPeso molecular:255.74AZD 3043
CAS:<p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>Fórmula:C19H29NO5Pureza:98.19% - 99.55%Cor e Forma:SolidPeso molecular:351.445-HT6/5-HT2A receptor ligand-1
CAS:<p>Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.</p>Fórmula:C21H19FN2O2Cor e Forma:SolidPeso molecular:350.39Y 23684
CAS:<p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>Fórmula:C18H13ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:356.83Tarafenacin
CAS:<p>Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.</p>Fórmula:C21H20F4N2O2Pureza:98%Cor e Forma:SolidPeso molecular:408.39AChE-IN-7
CAS:<p>AChE-IN-7 inhibits eeAChE (IC50: 0.045μM), eeBuChE (19.68μM), crosses the blood-brain barrier, safe, with good pharmacokinetics and 55.5% bioavailability.</p>Fórmula:C26H28N2O2Cor e Forma:SolidPeso molecular:400.51RS 64459-193
CAS:<p>RS 64459-193 has a high affinity for the 5-HT1A binding site.</p>Fórmula:C26H36Cl2N2O2Cor e Forma:SolidPeso molecular:479.48S-(+)-Mecamylamine hydrochloride
CAS:<p>Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.</p>Fórmula:C11H22ClNCor e Forma:SolidPeso molecular:203.75
