
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(648 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.029 produtos)
- BACE(37 produtos)
- Beta Amilóide(231 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(372 produtos)
- Gama-secretase(63 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5636 produtos de "Neurociência"
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Y 23684
CAS:Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.Fórmula:C18H13ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:356.83Tarafenacin
CAS:Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Fórmula:C21H20F4N2O2Pureza:98%Cor e Forma:SolidPeso molecular:408.39AChE-IN-7
CAS:AChE-IN-7 inhibits eeAChE (IC50: 0.045μM), eeBuChE (19.68μM), crosses the blood-brain barrier, safe, with good pharmacokinetics and 55.5% bioavailability.Fórmula:C26H28N2O2Cor e Forma:SolidPeso molecular:400.51Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Cor e Forma:SolidPeso molecular:255.74AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Fórmula:C19H29NO5Pureza:98.19% - 99.55%Cor e Forma:SolidPeso molecular:351.44RS 64459-193
CAS:RS 64459-193 has a high affinity for the 5-HT1A binding site.Fórmula:C26H36Cl2N2O2Cor e Forma:SolidPeso molecular:479.48S-(+)-Mecamylamine hydrochloride
CAS:Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.Fórmula:C11H22ClNCor e Forma:SolidPeso molecular:203.75Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Fórmula:C13H25NO2Cor e Forma:SolidPeso molecular:227.34Ref: TM-T72977
1mg37,00€5mg72,00€1mL*10mM (DMSO)79,00€10mg99,00€25mg169,00€50mg229,00€100mg320,00€200mg479,00€ACPT-I
CAS:Agonist for group III mGlu receptorsFórmula:C8H11NO6Pureza:98%Cor e Forma:SolidPeso molecular:217.18Mebanazine
CAS:Mebanazine, a potent monoamine oxidase (MAO) inhibitor, is utilized in depression research.Fórmula:C8H12N2Cor e Forma:SolidPeso molecular:136.19(S)-Venlafaxine
CAS:(S)-Venlafaxine: oral antidepressant, potent dual serotonin/norepinephrine reuptake inhibitor.Fórmula:C17H27NO2Cor e Forma:SolidPeso molecular:277.4DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Fórmula:C18H10Br2ClN3OSCor e Forma:SolidPeso molecular:511.62(R)-Viloxazine Hydrochloride
CAS:(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.Fórmula:C13H20ClNO3Pureza:99.88% - 99.94%Cor e Forma:SolidPeso molecular:273.76Ref: TM-T22413
1mg52,00€1mL*10mM (DMSO)101,00€5mg111,00€10mg162,00€25mg235,00€50mg330,00€100mg452,00€200mg607,00€Iloperidone hydrochloride
CAS:Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.Fórmula:C24H28ClFN2O4Pureza:98%Cor e Forma:SolidPeso molecular:462.95JNJ-46356479
CAS:JNJ-46356479: Selective, oral mGlu2 receptor PAM, EC50=78 nM, Emax=256%.Fórmula:C22H22F5N5Cor e Forma:SolidPeso molecular:451.44SB 258719 hydrochloride
CAS:Selective 5-HT7 receptor antagonistFórmula:C18H31ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:374.97Alaproclate hydrochloride, (S)-
CAS:Alaproclate hydrochloride, (S)- is a selective inhibitor of serotonin reuptake.Fórmula:C13H19Cl2NO2Pureza:98%Cor e Forma:SolidPeso molecular:292.2OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Fórmula:C23H28ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:413.94NFPS
CAS:NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion.Fórmula:C24H24FNO3Pureza:98%Cor e Forma:SolidPeso molecular:393.45LY320135
CAS:CB1 receptor antagonist/inverse agonistFórmula:C24H17NO4Pureza:98%Cor e Forma:SolidPeso molecular:383.4CV-159
CAS:CV-159 is a unique dihydropyridine Ca2+ antagonist with antiinflammatory activities. It has an anti-calmodulin (CaM) action.Fórmula:C31H34N4O7Pureza:98%Cor e Forma:SolidPeso molecular:574.62Cimoxatone
CAS:Cimoxatone is used as a Monoamine Oxidase Inhibitor.Fórmula:C19H18N2O4Cor e Forma:SolidPeso molecular:338.36YIAD-0205
CAS:YIAD-0205, an orally administered inhibitor of Aβ(1-42) aggregation, has exhibited in vivo efficacy in a 5XFAD transgenic mouse model that harbors five familialFórmula:C26H16Br2ClN3Cor e Forma:SolidPeso molecular:565.69Org-12962 hydrochloride
CAS:Org-12962 hydrochloride is a 5-HT2C receptor agonist.Fórmula:C10H12Cl2F3N3Pureza:98%Cor e Forma:SolidPeso molecular:302.12CP-601932
CAS:CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.Fórmula:C12H12F3NCor e Forma:SolidPeso molecular:227.233-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Fórmula:C20H30N2O10S2Pureza:98%Cor e Forma:SolidPeso molecular:522.59OAB-14
CAS:OAB-14, a Bexarotene derivative, enhances β-amyloid clearance and cognitive function in APP/PS1 mice, improving Alzheimer's symptoms.Fórmula:C32H46N4O2Cor e Forma:SolidPeso molecular:518.73DR4485 hydrochloride
CAS:5-HT7 antagonistFórmula:C26H29Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:491.88Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Fórmula:C15H14N6O3Pureza:98%Cor e Forma:SolidPeso molecular:326.31(±)-Duloxetine hydrochloride
CAS:(±)-Duloxetine ((Rac)-Duloxetine) hydrochloride is the Duloxetine hydrochloride racemate.Fórmula:C18H20ClNOSCor e Forma:SolidPeso molecular:333.88hMAO-B-IN-3
CAS:hMAO-B-IN-3: potent hMAO-B inhibitor, IC50 of 47.4 nM, good drug properties, safe, ideal for lead optimization.Fórmula:C20H15NO4Cor e Forma:SolidPeso molecular:333.34Ambenonium chloride tetrahydrate
CAS:Ambenonium chloride, a salt with cholinesterase inhibiting properties, treats myasthenia gravis by enhancing acetylcholine activity.Fórmula:C28H50Cl4N4O6Cor e Forma:SolidPeso molecular:680.53T761-0184
CAS:T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].Fórmula:C16H20FN3OCor e Forma:SolidPeso molecular:289.35Echothiophate Iodide
CAS:Echothiophate iodide is an effective long-acting cholinesterase inhibitor for the treatment of glaucoma.Fórmula:C9H23INO3PSCor e Forma:SolidPeso molecular:383.23UPF-523
CAS:group I metabotropic glutamate receptors (mGlu1a) antagonistFórmula:C11H11NO4Pureza:98%Cor e Forma:White SolidPeso molecular:221.21SEP-363856
CAS:SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.Fórmula:C9H13NOSPureza:98%Cor e Forma:SolidPeso molecular:183.27DAU 5884 hydrochloride
CAS:muscarinic M3 receptor antagonistFórmula:C17H22ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:351.83K 01-162
CAS:K 01-162 binds and destabilizes AβO (β-amyloid), with an EC50 of 80 nM.Fórmula:C15H14BrNCor e Forma:SolidPeso molecular:288.18Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Fórmula:C25H26F4N2O8Pureza:99.86%Cor e Forma:SolidPeso molecular:558.48Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Fórmula:C19H21NPureza:99.15% - 99.66%Cor e Forma:SolidPeso molecular:263.38Zaldaride maleate
CAS:Zaldaride maleate blocks Ca2+, Na+, K+ currents, and nAChR; inhibits CaM cAMP PDE (IC50: 3.3 nM) and estrogen signaling.Fórmula:C30H32N4O6Pureza:98%Cor e Forma:SolidPeso molecular:544.6BChE-IN-6
CAS:BChE-IN-6 inhibits BChE with a Ki of 0.182 μM and chelates Zn 2+, useful in AD research.Fórmula:C24H29N3O2Cor e Forma:SolidPeso molecular:391.51Alvameline
CAS:Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.Fórmula:C9H15N5Pureza:98%Cor e Forma:SolidPeso molecular:193.25Lilly 51641
CAS:Lilly 51641 is used as a MAO inhibitor.Fórmula:C11H14ClNOPureza:98%Cor e Forma:SolidPeso molecular:211.69DL-AP4 Sodium salt
CAS:Broad spectrum EAA ligandFórmula:C4H10NNaO5PPureza:98%Cor e Forma:SolidPeso molecular:206.09Trimipramine
CAS:Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.Fórmula:C20H26N2Pureza:98%Cor e Forma:SolidPeso molecular:294.432-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98.56%Cor e Forma:White SolidPeso molecular:265.71VU0090157
CAS:VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.Fórmula:C19H21N3O7Pureza:98%Cor e Forma:SolidPeso molecular:403.39Thiochrome
CAS:Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.Fórmula:C12H14N4OSPureza:98%Cor e Forma:SolidPeso molecular:262.33S-22153
CAS:S22153 is an antagonist of melatonin receptor.Fórmula:C14H17NOSCor e Forma:SolidPeso molecular:247.36
