
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(647 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.028 produtos)
- BACE(37 produtos)
- Beta Amilóide(231 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(373 produtos)
- Gama-secretase(62 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(42 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5638 produtos de "Neurociência"
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Opiranserin
CAS:Opiranserin is a development as an injectable agent for the treatment of postoperative pain.Fórmula:C21H34N2O5Pureza:98%Cor e Forma:SolidPeso molecular:394.51U-101017
CAS:U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.Fórmula:C23H27ClN4O3Pureza:98%Cor e Forma:SolidPeso molecular:442.94TPA-023B
CAS:TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.Fórmula:C21H15F2N5OPureza:98%Cor e Forma:SolidPeso molecular:391.37ELN318463
CAS:ELN 318463 selectively inhibits γ-secretase; EC50: 12 nM (PS1), 656 nM (PS2); 51x more selective for PS1; targets APP.Fórmula:C19H20BrClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:471.8TC299423
CAS:TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.Fórmula:C11H15N3Cor e Forma:SolidPeso molecular:189.26BTM-1086
CAS:BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.Fórmula:C21H25N3OSPureza:98%Cor e Forma:SolidPeso molecular:367.51(S)-Rasagiline mesylate
CAS:(S)-Rasagiline mesylate is rasagiline S-isomer, and is an agent of anti-Parkinson.Fórmula:C13H17NO3SPureza:98%Cor e Forma:SolidPeso molecular:267.34SL-25.1188
CAS:SL-25.1188: Reversible MAO-B inhibitor with high brain uptake & slow plasma metabolism.Fórmula:C16H17F3N2O5Cor e Forma:SolidPeso molecular:374.31SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFórmula:C19H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:348.44CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFórmula:C19H32O2Pureza:98%Cor e Forma:SolidPeso molecular:292.46ACPT-II
CAS:metabotropic receptor antagonistFórmula:C8H11NO6Pureza:98%Cor e Forma:SolidPeso molecular:217.18AChE-IN-15
CAS:AChE-IN-15 is a reversible inhibitor of huAChE and huBChE (IC50: 6.8 μM, 16.1 μM), with antioxidant activity, used in Alzheimer's research.Fórmula:C23H24N2O7Cor e Forma:SolidPeso molecular:440.45LY 393558
CAS:Dual 5-HT1B/1D receptor antagonistFórmula:C26H31FN4O4S2Pureza:98%Cor e Forma:SolidPeso molecular:546.68AChE/BChE-IN-9
CAS:Compound 7a inhibits AChE/BChE (IC50: 5.74/14.05 μM), has antioxidant effects (IC50: 57.35 μM), chelates iron, and affects amyloid β 1-42 aggregation.Fórmula:C20H19N3O4Cor e Forma:SolidPeso molecular:365.38Z164597606
CAS:Z164597606 inhibits BChE (1.3 μM equine, 1.7 μM human), binds Trp82 via π-π, potential in Alzheimer's research.Fórmula:C20H19N3O4Cor e Forma:SolidPeso molecular:365.38Quifenadine
CAS:Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.Fórmula:C20H23NOPureza:98%Cor e Forma:SolidPeso molecular:293.4AChE-IN-6
CAS:AChE-IN-6: inhibits EeAChE (IC50=0.20μM), HuAChE (IC50=37.02nM), and modulates Aβ1-42 aggregation (IC50=~1.86μM). Potential Alzheimer's research.Fórmula:C29H41N5O2Cor e Forma:SolidPeso molecular:491.67VU0652835
CAS:VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).Fórmula:C16H19N3O3SPureza:98%Cor e Forma:SolidPeso molecular:333.41Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Fórmula:C19H28N2Pureza:99.54%Cor e Forma:SolidPeso molecular:284.44Ref: TM-T37015
2mg34,00€5mg50,00€10mg75,00€1mL*10mM (DMSO)79,00€25mg145,00€50mg253,00€100mg432,00€200mg618,00€PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Fórmula:C23H21ClFN5O4SPureza:97.59%Cor e Forma:SolidPeso molecular:517.96Ref: TM-T6959
1mg79,00€5mg168,00€10mg220,00€1mL*10mM (DMSO)380,00€25mg398,00€50mg587,00€100mg835,00€200mg1.134,00€UB 165 fumarate
CAS:UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.Fórmula:C17H19ClN2O4Pureza:99.72%Cor e Forma:SolidPeso molecular:350.8Metixene hydrochloride
CAS:Metixene hydrochloride is an anticholinergic antiparkinsonian agent.Fórmula:C20H24ClNSPureza:98%Cor e Forma:SolidPeso molecular:345.93Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Fórmula:C21H21N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:347.41Ref: TM-T10961
1mg203,00€5mg404,00€1mL*10mM (DMSO)447,00€10mg567,00€25mg842,00€50mg1.125,00€100mg1.521,00€Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFórmula:C25H36N4O10Pureza:98%Cor e Forma:SolidPeso molecular:552.581Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Fórmula:C10H11ClF3N3Pureza:98.34%Cor e Forma:SolidPeso molecular:265.66(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:98%Cor e Forma:SolidPeso molecular:250.12MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Fórmula:C4H10NO6PPureza:98%Cor e Forma:SolidPeso molecular:199.1Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.Fórmula:C21H25ClN2O4SPureza:99.57%Cor e Forma:SolidPeso molecular:436.95EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Fórmula:C15H22N2OPureza:97.66% - 99.78%Cor e Forma:SolidPeso molecular:246.35Ref: TM-T11183
1mg87,00€2mg118,00€1mL*10mM (DMSO)166,00€5mg167,00€10mg202,00€25mg449,00€50mg652,00€100mg888,00€500mg1.783,00€Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Fórmula:C13H10N2OPureza:98.66%Cor e Forma:SolidPeso molecular:210.23Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Fórmula:C17H20N2O3Pureza:99.62%Cor e Forma:Solid CrystallinePeso molecular:300.35Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Cor e Forma:SolidPeso molecular:328.38CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Fórmula:C19H28ClN5OPureza:99.72%Cor e Forma:SolidPeso molecular:377.91TG41
CAS:TG41 is a GABAA receptors positive modulator.Fórmula:C18H13BrCl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:440.12CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Fórmula:C18H17N3O3Pureza:99.06% - 99.74%Cor e Forma:SolidPeso molecular:323.35FR-188582
CAS:FR-188582 is a highly selective cyclooxygenase (COX)-2 inhibitor (IC50: 17 nM).Fórmula:C16H13ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:332.8PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Fórmula:C15H23NO2SPureza:99.53%Cor e Forma:SolidPeso molecular:281.41Ref: TM-T28435
1mg73,00€1mL*10mM (DMSO)138,00€5mg146,00€10mg210,00€25mg319,00€50mg447,00€100mg600,00€200mg800,00€Chlorisondamine chloride
CAS:Chlorisondamine chloride: a nicotinic antagonist, mainly for animal research, former antihypertensive.Fórmula:C14H20Cl6N2Cor e Forma:SolidPeso molecular:429.03Trelanserin
CAS:Trelanserin (SL-650472) is an antagonist of the serotonin receptor.Fórmula:C24H24FN5O2SCor e Forma:SolidPeso molecular:465.54Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Fórmula:C18H19NCor e Forma:SolidPeso molecular:249.35Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Fórmula:C11H16N2OPureza:98%Cor e Forma:SolidPeso molecular:192.26CDD0102
CAS:CDD0102 is a potent agonist of M1 Muscarinic receptor.Fórmula:C8H12N4OPureza:98%Cor e Forma:SolidPeso molecular:180.21R-PSOP
CAS:R-PSOP, a selective NMUR2 antagonist, binds human/rat receptors with 52/32 nM affinity, useful for CNS-related disorders.Fórmula:C20H22N4O2Cor e Forma:SolidPeso molecular:350.41DCB
CAS:DCB is an mGluR5 allosteric ligand that blocks mGluR modulation, countering DMeOB and DFB effects.Fórmula:C14H10Cl2N2Pureza:99.12% - 99.9%Cor e Forma:SolidPeso molecular:277.15Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Fórmula:C18H14N4O3Pureza:98%Cor e Forma:SolidPeso molecular:334.33Esoxybutynin Chloride
CAS:(S)-oxybutynin, with antimuscarinic effects, is being developed for urinary incontinence.Fórmula:C22H32ClNO3Cor e Forma:SolidPeso molecular:393.95Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFórmula:C16H23ClN2O2Cor e Forma:SolidPeso molecular:310.82KDS2010 mesylate
CAS:KDS2010: potent, reversible MAO-B inhibitor with 12,500x selectivity vs. MAO-A; enhances memory in APP/PS1 mice.Fórmula:C18H21F3N2O4SCor e Forma:SolidPeso molecular:418.43Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Fórmula:C15H14ClN3O3Cor e Forma:SolidPeso molecular:319.74
