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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5400 produtos de "Neurociência"

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  • TAK-137

    CAS:
    <p>TAK-137 is an AMPA receptor enhancer with antidepressant effects. TAK-137 has the ability to improve cognition and could be used to study schizophrenia.</p>
    Fórmula:C19H16N2O3S
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:352.41
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Fórmula:C17H17N3O2
    Pureza:97.44% - 98.25%
    Cor e Forma:Solid
    Peso molecular:295.34
  • SCH-900271

    CAS:
    <p>SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.</p>
    Fórmula:C14H16N2O4
    Pureza:98.82% - 99.93%
    Cor e Forma:Solid
    Peso molecular:276.29
  • Landipirdine

    CAS:
    <p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>
    Fórmula:C18H19FN2O3S
    Pureza:97.61% - 99.37%
    Cor e Forma:Solid
    Peso molecular:362.42
  • Ezeprogind disulfate

    CAS:
    <p>Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.</p>
    Fórmula:C25H48N6O8S2
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:624.81
  • NB001

    CAS:
    <p>NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.</p>
    Fórmula:C12H20N6O
    Pureza:99.69%
    Cor e Forma:Off-White To Pale Pink Solid
    Peso molecular:264.33
  • Liafensine

    CAS:
    <p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>
    Fórmula:C24H22N4
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:366.46
  • Sarizotan HCl

    CAS:
    <p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>
    Fórmula:C22H22ClFN2O
    Pureza:96%
    Cor e Forma:Solid
    Peso molecular:384.87
  • ALX-1393

    CAS:
    <p>ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a concentration-dependent manner and inhibits the</p>
    Fórmula:C23H22FNO4
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:395.42
  • (Z)-Thiothixene

    CAS:
    <p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>
    Fórmula:C23H29N3O2S2
    Pureza:99.21%
    Cor e Forma:Yellow To Yellow With A Tan Cast Powder
    Peso molecular:443.63
  • LRRK2-IN-7

    CAS:
    <p>LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, &gt;1000x selectivity vs kinases/channels/CYPs.</p>
    Fórmula:C24H26N6O
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:414.5
  • ABP688

    CAS:
    <p>ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.</p>
    Fórmula:C15H16N2O
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:240.3
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Fórmula:C28H30ClN5O3
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:520.02
  • Desformylflustrabromine hydrochloride

    CAS:
    <p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>
    Fórmula:C17H12INO5
    Pureza:98.12%
    Cor e Forma:Solid
    Peso molecular:437.19
  • BPDBA

    CAS:
    <p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>
    Fórmula:C19H20Cl2N2O
    Pureza:99.37% - 99.95%
    Cor e Forma:Solid
    Peso molecular:363.28
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Cor e Forma:Off-White Powder
    Peso molecular:195.01
  • CP 96021

    CAS:
    <p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>
    Fórmula:C29H21FN4OS
    Pureza:97.81% - 99.62%
    Cor e Forma:Soild
    Peso molecular:492.57
  • E6801

    CAS:
    <p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>
    Fórmula:C17H18ClN5O2S2
    Pureza:96.32% - 99.53%
    Cor e Forma:Solid
    Peso molecular:423.94
  • Ecopipam

    CAS:
    <p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>
    Fórmula:C19H20ClNO
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:313.82
  • BL-1020 Mesylate

    CAS:
    <p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>
    Fórmula:C28H45ClN4O11S4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:777.39
  • Cilansetron

    CAS:
    <p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>
    Fórmula:C20H21N3O
    Pureza:99.82% - 99.98%
    Cor e Forma:Solid
    Peso molecular:319.4
  • UK-240455

    CAS:
    <p>UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.</p>
    Fórmula:C11H11Cl2N3O5S
    Pureza:98.34% - 99.84%
    Cor e Forma:Solid
    Peso molecular:368.19
  • LY266097 hydrochloride

    CAS:
    <p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>
    Fórmula:C21H24Cl2N2O2
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:407.33
  • 8-OH-Dpat

    CAS:
    <p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>
    Fórmula:C16H25NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.38
  • ASM-024

    CAS:
    <p>ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.</p>
    Fórmula:C15H25N2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:233.37
  • Felcisetrag

    CAS:
    <p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>
    Fórmula:C25H37N5O3
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:455.59
  • CT-179

    CAS:
    <p>CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.</p>
    Fórmula:C17H22Cl2N6O
    Pureza:98.67%
    Cor e Forma:Solid
    Peso molecular:397.3
  • ADR-851 free base

    CAS:
    <p>ADR-851 free base is an antagonist of the HT3 receptor.</p>
    Fórmula:C14H18ClN3O2
    Pureza:97.88% - 98.39%
    Cor e Forma:Solid
    Peso molecular:295.77
  • Quinupramine

    CAS:
    <p>Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.</p>
    Fórmula:C21H24N2
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:304.43
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Fórmula:C14H16ClN3O
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:277.75
  • Sudoxicam

    CAS:
    <p>Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema</p>
    Fórmula:C13H11N3O4S2
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:337.37
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Fórmula:C19H19F2N7O
    Pureza:98.12% - 99.70%
    Cor e Forma:Solid
    Peso molecular:399.4
  • Eltenac

    CAS:
    <p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>
    Fórmula:C12H9Cl2NO2S
    Pureza:98.53%
    Cor e Forma:Solid
    Peso molecular:302.18
  • RS 42358-197

    CAS:
    <p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>
    Fórmula:C19H23ClN2O
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:330.85
  • Xanomeline oxalate

    CAS:
    <p>Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.</p>
    Fórmula:C16H25N3O5S
    Pureza:99.1%
    Cor e Forma:Solid
    Peso molecular:371.45
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Fórmula:C17H14O6
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:314.29
  • Buntanetap

    CAS:
    <p>Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular disease</p>
    Fórmula:C20H23N3O2
    Pureza:98.2%
    Cor e Forma:Solid
    Peso molecular:337.42
  • Tribendimidine

    CAS:
    <p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>
    Fórmula:C28H32N6
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:452.59
  • Oxotremorine M iodide

    CAS:
    <p>Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.</p>
    Fórmula:C11H19IN2O
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:322.19
  • Adoprazine

    CAS:
    <p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>
    Fórmula:C24H24FN3O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:405.46
  • VU 0285683

    CAS:
    <p>VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for the MPEP binding site. VU 0285683 shows anxiolytic-like activity.</p>
    Fórmula:C14H7FN4O
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:266.23
  • Aceclidine

    CAS:
    <p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>
    Fórmula:C9H15NO2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:169.22
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Fórmula:C21H23ClN2O3
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:386.87
  • cis-Urocanic acid

    CAS:
    <p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>
    Fórmula:C6H6N2O2
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:138.12
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Fórmula:C19H20ClN3O
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:341.83
  • CP-810123

    CAS:
    <p>CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.</p>
    Fórmula:C14H18N4O
    Pureza:98.63% - 99.60%
    Cor e Forma:Solid
    Peso molecular:258.32
  • DSS30

    CAS:
    <p>DSS30 is a P25/CDK5 inhibitor that reduces β-amyloid secretion to help prevent Alzheimer's.</p>
    Fórmula:C16H14ClNO3S2
    Pureza:99.19% - 99.4%
    Cor e Forma:Solid
    Peso molecular:367.87
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Fórmula:C20H20ClN5O3S2
    Pureza:99.21% - 99.73%
    Cor e Forma:Solid
    Peso molecular:477.99
  • LSN2463359

    CAS:
    <p>LSN2463359 is a positive allosteric modulators of the mGlu5 receptor.</p>
    Fórmula:C16H15N3O
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:265.31
  • AZD6538

    CAS:
    <p>AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.</p>
    Fórmula:C15H6FN5O
    Pureza:98.68%
    Cor e Forma:Solid
    Peso molecular:291.24