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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5400 produtos de "Neurociência"

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  • Lensiprazine

    CAS:
    <p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>
    Fórmula:C24H27FN4O2
    Pureza:98.04%
    Cor e Forma:Solid
    Peso molecular:422.5
  • NS-2710

    CAS:
    <p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Fórmula:C22H20N4O
    Pureza:99.7% - 99.82%
    Cor e Forma:Solid
    Peso molecular:356.42
  • ADR-851 free base

    CAS:
    <p>ADR-851 free base is an antagonist of the HT3 receptor.</p>
    Fórmula:C14H18ClN3O2
    Pureza:97.88% - 98.39%
    Cor e Forma:Solid
    Peso molecular:295.77
  • SB 699551 dihydrochloride

    CAS:
    <p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>
    Fórmula:C34H47Cl2N3O
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:584.66
  • Adoprazine

    CAS:
    <p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>
    Fórmula:C24H24FN3O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:405.46
  • Nexopamil

    CAS:
    <p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>
    Fórmula:C24H40N2O3
    Pureza:97.87% - >99.99%
    Cor e Forma:Solid
    Peso molecular:404.59
  • PAT-1251

    CAS:
    <p>PAT-1251 is an inhibitor of LOXL2 with IC50s of 10, 0.12, and 0.16 μM for the mouse, rat, and dog and can be used in studies about fibrotic diseases.</p>
    Fórmula:C18H17F4N3O3
    Pureza:97.27% - 98.46%
    Cor e Forma:Solid
    Peso molecular:399.34
  • LM-1685

    CAS:
    <p>LM-1685是一种有效且具有选择性的人单核细胞和全血中COX-2抑制剂,IC50分别为0.65 µM 和IC50 = 4.3 μM,是治疗炎症的潜在化合物。</p>
    Fórmula:C18H16ClNO4S
    Pureza:98.16%
    Cor e Forma:Solid
    Peso molecular:377.84
  • Aplindore Fumarate

    CAS:
    <p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>
    Fórmula:C22H22N2O7
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:426.42
  • Roxindole

    CAS:
    <p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>
    Fórmula:C23H26N2O
    Pureza:98.03% - 98.93%
    Cor e Forma:Solid
    Peso molecular:346.47
  • Repinotan

    CAS:
    <p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>
    Fórmula:C21H24N2O4S
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:400.49
  • ATC 0175 hydrochloride

    CAS:
    <p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>
    Fórmula:C23H26ClF2N5O
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:461.93
  • SPD-473 citrate

    CAS:
    <p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>
    Fórmula:C23H31Cl2NO8S
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:552.47
  • Mibampator

    CAS:
    <p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>
    Fórmula:C21H30N2O4S2
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:438.6
  • MK-3328

    CAS:
    <p>MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.</p>
    Fórmula:C14H9FN4O
    Pureza:99.70% - >99.99%
    Cor e Forma:Solid
    Peso molecular:268.25
  • ABP688

    CAS:
    <p>ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.</p>
    Fórmula:C15H16N2O
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:240.3
  • BPDBA

    CAS:
    <p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>
    Fórmula:C19H20Cl2N2O
    Pureza:99.37% - 99.95%
    Cor e Forma:Solid
    Peso molecular:363.28
  • Otenzepad

    CAS:
    <p>Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.</p>
    Fórmula:C24H31N5O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:421.54
  • Ezeprogind disulfate

    CAS:
    <p>Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.</p>
    Fórmula:C25H48N6O8S2
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:624.81
  • Lesopitron

    CAS:
    <p>Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.</p>
    Fórmula:C15H21ClN6
    Pureza:99.15% - 99.38%
    Cor e Forma:Solid
    Peso molecular:320.82
  • 8-OH-Dpat

    CAS:
    <p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>
    Fórmula:C16H25NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.38
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Fórmula:C17H17Cl2NO
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:322.23
  • Sudoxicam

    CAS:
    <p>Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema</p>
    Fórmula:C13H11N3O4S2
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:337.37
  • Sarmazenil

    CAS:
    <p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>
    Fórmula:C15H14ClN3O3
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:319.74
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Cor e Forma:Off-White Powder
    Peso molecular:195.01
  • NB001

    CAS:
    <p>NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.</p>
    Fórmula:C12H20N6O
    Pureza:99.69%
    Cor e Forma:Off-White To Pale Pink Solid
    Peso molecular:264.33
  • DA-6886

    CAS:
    <p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>
    Fórmula:C19H28Cl2N6O2
    Pureza:99.28% - 99.91%
    Cor e Forma:Solid
    Peso molecular:443.37
  • GSK233705

    CAS:
    <p>GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.</p>
    Fórmula:C24H29BrN2
    Pureza:99.87% - 99.98%
    Cor e Forma:Solid
    Peso molecular:425.4
  • R 59-022 hydrochloride

    CAS:
    <p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>
    Fórmula:C27H27ClFN3OS
    Pureza:97.7%
    Cor e Forma:Solid
    Peso molecular:496.04
  • Perphenazine dihydrochloride

    CAS:
    <p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>
    Fórmula:C21H28Cl3N3OS
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:476.89
  • UK-240455

    CAS:
    <p>UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.</p>
    Fórmula:C11H11Cl2N3O5S
    Pureza:98.34% - 99.84%
    Cor e Forma:Solid
    Peso molecular:368.19
  • Desformylflustrabromine hydrochloride

    CAS:
    <p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>
    Fórmula:C17H12INO5
    Pureza:98.12%
    Cor e Forma:Solid
    Peso molecular:437.19
  • 5HT6-ligand-1

    CAS:
    <p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>
    Fórmula:C20H22BrN3O2S
    Pureza:99.24% - 99.93%
    Cor e Forma:Solid
    Peso molecular:448.38
  • AZD6538

    CAS:
    <p>AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.</p>
    Fórmula:C15H6FN5O
    Pureza:98.68%
    Cor e Forma:Solid
    Peso molecular:291.24
  • Tribendimidine

    CAS:
    <p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>
    Fórmula:C28H32N6
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:452.59
  • Cilansetron

    CAS:
    <p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>
    Fórmula:C20H21N3O
    Pureza:99.82% - 99.98%
    Cor e Forma:Solid
    Peso molecular:319.4
  • Selurampanel

    CAS:
    <p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>
    Fórmula:C16H19N5O4S
    Pureza:99.60% - 99.78%
    Cor e Forma:Solid
    Peso molecular:377.42
  • Fenlean

    CAS:
    <p>"Fenlean (FLZ) in phase I trial at Chinese Academy's Institute of Pharmacy for Parkinson's treatment."</p>
    Fórmula:C26H27NO6
    Pureza:98.99%
    Cor e Forma:Solid
    Peso molecular:449.5
  • (E/Z)-SIB-1893

    CAS:
    <p>(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.</p>
    Fórmula:C14H13N
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:195.26
  • Femoxetine hydrochloride

    CAS:
    <p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>
    Fórmula:C20H26ClNO2
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:347.88
  • BL-1020 Mesylate

    CAS:
    <p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>
    Fórmula:C28H45ClN4O11S4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:777.39
  • Tiospirone

    CAS:
    <p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>
    Fórmula:C24H32N4O2S
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:440.6
  • Eltenac

    CAS:
    <p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>
    Fórmula:C12H9Cl2NO2S
    Pureza:98.53%
    Cor e Forma:Solid
    Peso molecular:302.18
  • Golexanolone

    CAS:
    <p>Golexanolone can be used to study neurological diseases.</p>
    Fórmula:C21H31NO2
    Pureza:99.90% - 99.99%
    Cor e Forma:Solid
    Peso molecular:329.48
  • Ru-32514

    CAS:
    <p>Ru-32514 is a benzodiazepine receptor agonist.</p>
    Fórmula:C18H17N3O2
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:307.35
  • SB-215505

    CAS:
    <p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>
    Fórmula:C19H16ClN3O
    Pureza:98.33%
    Cor e Forma:Solid
    Peso molecular:337.8
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Fórmula:C28H30ClN5O3
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:520.02
  • Itasetron

    CAS:
    <p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>
    Fórmula:C16H20N4O2
    Pureza:98.58% - 99.33%
    Cor e Forma:Solid
    Peso molecular:300.36
  • McN-A 343

    CAS:
    <p>McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.</p>
    Fórmula:C14H18Cl2N2O2
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:317.21
  • cis-Urocanic acid

    CAS:
    <p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>
    Fórmula:C6H6N2O2
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:138.12