
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(942 produtos)
- ACK(1 produtos)
- AChR(575 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.946 produtos)
- BACE(36 produtos)
- Beta Amilóide(205 produtos)
- CaMK(69 produtos)
- COX(562 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor GABA(336 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(359 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(28 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5400 produtos de "Neurociência"
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Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Fórmula:C24H27FN4O2Pureza:98.04%Cor e Forma:SolidPeso molecular:422.5NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C22H20N4OPureza:99.7% - 99.82%Cor e Forma:SolidPeso molecular:356.42ADR-851 free base
CAS:<p>ADR-851 free base is an antagonist of the HT3 receptor.</p>Fórmula:C14H18ClN3O2Pureza:97.88% - 98.39%Cor e Forma:SolidPeso molecular:295.77SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Fórmula:C34H47Cl2N3OPureza:99.83%Cor e Forma:SolidPeso molecular:584.66Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Fórmula:C24H24FN3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:405.46Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Fórmula:C24H40N2O3Pureza:97.87% - >99.99%Cor e Forma:SolidPeso molecular:404.59PAT-1251
CAS:<p>PAT-1251 is an inhibitor of LOXL2 with IC50s of 10, 0.12, and 0.16 μM for the mouse, rat, and dog and can be used in studies about fibrotic diseases.</p>Fórmula:C18H17F4N3O3Pureza:97.27% - 98.46%Cor e Forma:SolidPeso molecular:399.34LM-1685
CAS:<p>LM-1685是一种有效且具有选择性的人单核细胞和全血中COX-2抑制剂,IC50分别为0.65 µM 和IC50 = 4.3 μM,是治疗炎症的潜在化合物。</p>Fórmula:C18H16ClNO4SPureza:98.16%Cor e Forma:SolidPeso molecular:377.84Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:426.42Roxindole
CAS:<p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>Fórmula:C23H26N2OPureza:98.03% - 98.93%Cor e Forma:SolidPeso molecular:346.47Repinotan
CAS:<p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>Fórmula:C21H24N2O4SPureza:99%Cor e Forma:SolidPeso molecular:400.49ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Fórmula:C23H26ClF2N5OPureza:99.98%Cor e Forma:SolidPeso molecular:461.93SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Fórmula:C23H31Cl2NO8SPureza:99.37%Cor e Forma:SolidPeso molecular:552.47Mibampator
CAS:<p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>Fórmula:C21H30N2O4S2Pureza:99.34%Cor e Forma:SolidPeso molecular:438.6MK-3328
CAS:<p>MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.</p>Fórmula:C14H9FN4OPureza:99.70% - >99.99%Cor e Forma:SolidPeso molecular:268.25ABP688
CAS:<p>ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.</p>Fórmula:C15H16N2OPureza:98.63%Cor e Forma:SolidPeso molecular:240.3BPDBA
CAS:<p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>Fórmula:C19H20Cl2N2OPureza:99.37% - 99.95%Cor e Forma:SolidPeso molecular:363.28Otenzepad
CAS:<p>Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.</p>Fórmula:C24H31N5O2Pureza:99.79%Cor e Forma:SolidPeso molecular:421.54Ezeprogind disulfate
CAS:<p>Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.</p>Fórmula:C25H48N6O8S2Pureza:99.72%Cor e Forma:SolidPeso molecular:624.81Lesopitron
CAS:<p>Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.</p>Fórmula:C15H21ClN6Pureza:99.15% - 99.38%Cor e Forma:SolidPeso molecular:320.828-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Fórmula:C17H17Cl2NOPureza:99%Cor e Forma:SolidPeso molecular:322.23Sudoxicam
CAS:<p>Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema</p>Fórmula:C13H11N3O4S2Pureza:99.93%Cor e Forma:SolidPeso molecular:337.37Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Fórmula:C15H14ClN3O3Pureza:99.46%Cor e Forma:SolidPeso molecular:319.74Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Fórmula:C4H7BrN2O2Pureza:98.13%Cor e Forma:Off-White PowderPeso molecular:195.01NB001
CAS:<p>NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.</p>Fórmula:C12H20N6OPureza:99.69%Cor e Forma:Off-White To Pale Pink SolidPeso molecular:264.33DA-6886
CAS:<p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>Fórmula:C19H28Cl2N6O2Pureza:99.28% - 99.91%Cor e Forma:SolidPeso molecular:443.37GSK233705
CAS:<p>GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.</p>Fórmula:C24H29BrN2Pureza:99.87% - 99.98%Cor e Forma:SolidPeso molecular:425.4R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Fórmula:C27H27ClFN3OSPureza:97.7%Cor e Forma:SolidPeso molecular:496.04Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Fórmula:C21H28Cl3N3OSPureza:99.67%Cor e Forma:SolidPeso molecular:476.89UK-240455
CAS:<p>UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.</p>Fórmula:C11H11Cl2N3O5SPureza:98.34% - 99.84%Cor e Forma:SolidPeso molecular:368.19Desformylflustrabromine hydrochloride
CAS:<p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>Fórmula:C17H12INO5Pureza:98.12%Cor e Forma:SolidPeso molecular:437.195HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Fórmula:C20H22BrN3O2SPureza:99.24% - 99.93%Cor e Forma:SolidPeso molecular:448.38AZD6538
CAS:<p>AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.</p>Fórmula:C15H6FN5OPureza:98.68%Cor e Forma:SolidPeso molecular:291.24Tribendimidine
CAS:<p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>Fórmula:C28H32N6Pureza:≥98%Cor e Forma:SolidPeso molecular:452.59Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Fórmula:C20H21N3OPureza:99.82% - 99.98%Cor e Forma:SolidPeso molecular:319.4Selurampanel
CAS:<p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>Fórmula:C16H19N5O4SPureza:99.60% - 99.78%Cor e Forma:SolidPeso molecular:377.42Fenlean
CAS:<p>"Fenlean (FLZ) in phase I trial at Chinese Academy's Institute of Pharmacy for Parkinson's treatment."</p>Fórmula:C26H27NO6Pureza:98.99%Cor e Forma:SolidPeso molecular:449.5(E/Z)-SIB-1893
CAS:<p>(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.</p>Fórmula:C14H13NPureza:99.92%Cor e Forma:SolidPeso molecular:195.26Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Fórmula:C20H26ClNO2Pureza:99.63%Cor e Forma:SolidPeso molecular:347.88BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Fórmula:C28H45ClN4O11S4Pureza:>99.99%Cor e Forma:SolidPeso molecular:777.39Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Fórmula:C24H32N4O2SPureza:99.74%Cor e Forma:SolidPeso molecular:440.6Eltenac
CAS:<p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>Fórmula:C12H9Cl2NO2SPureza:98.53%Cor e Forma:SolidPeso molecular:302.18Golexanolone
CAS:<p>Golexanolone can be used to study neurological diseases.</p>Fórmula:C21H31NO2Pureza:99.90% - 99.99%Cor e Forma:SolidPeso molecular:329.48Ru-32514
CAS:<p>Ru-32514 is a benzodiazepine receptor agonist.</p>Fórmula:C18H17N3O2Pureza:99.21%Cor e Forma:SolidPeso molecular:307.35SB-215505
CAS:<p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>Fórmula:C19H16ClN3OPureza:98.33%Cor e Forma:SolidPeso molecular:337.8Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Fórmula:C28H30ClN5O3Pureza:99.04%Cor e Forma:SolidPeso molecular:520.02Itasetron
CAS:<p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>Fórmula:C16H20N4O2Pureza:98.58% - 99.33%Cor e Forma:SolidPeso molecular:300.36McN-A 343
CAS:<p>McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.</p>Fórmula:C14H18Cl2N2O2Pureza:99.65%Cor e Forma:SolidPeso molecular:317.21cis-Urocanic acid
CAS:<p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>Fórmula:C6H6N2O2Pureza:99.81%Cor e Forma:SolidPeso molecular:138.12
