
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(1.025 produtos)
- ACK(1 produtos)
- AChR(647 produtos)
- ATP Citrato Liase(17 produtos)
- Receptor adrenérgico(3.025 produtos)
- BACE(37 produtos)
- Beta Amilóide(230 produtos)
- CaMK(73 produtos)
- COX(602 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor GABA(373 produtos)
- Gama-secretase(62 produtos)
- GluR(265 produtos)
- GlyT(26 produtos)
- Receptor de Histamina(385 produtos)
- LRRK2(43 produtos)
- Receptor de Melatonina(26 produtos)
- NMDAR(10 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(327 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5639 produtos de "Neurociência"
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LRE1
CAS:LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.Fórmula:C12H13ClN4SPureza:>99.99%Cor e Forma:SolidPeso molecular:280.78Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Fórmula:C24H28N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:472.62Ro 67-4853
CAS:Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the agonist (S)-3,5-dihydroxy-phenylglycine (DHPG).Fórmula:C19H19NO4Pureza:98.57%Cor e Forma:SolidPeso molecular:325.36MAO-IN-M30 dihydrochloride
CAS:MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.Fórmula:C14H16Cl2N2OPureza:99.83%Cor e Forma:SolidPeso molecular:299.2Ref: TM-T38034
500mgA consultar1mg34,00€2mg43,00€5mg65,00€10mg90,00€25mg161,00€50mg230,00€100mg319,00€LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.132-Iodomelatonin
CAS:2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Fórmula:C13H15IN2O2Pureza:99.7%Cor e Forma:SolidPeso molecular:358.17Ref: TM-T10073
500mgA consultar1mL*10mM (DMSO)34,00€10mg43,00€25mg79,00€50mg118,00€100mg178,00€200mg268,00€GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Fórmula:C19H27N3O4SPureza:98.16% - 99.96%Cor e Forma:SolidPeso molecular:393.5Foliglurax
CAS:Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).Fórmula:C23H23N3O3SPureza:98%Cor e Forma:SolidPeso molecular:421.51PRX933 hydrochloride
CAS:PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Fórmula:C16H22ClN5O2Pureza:99.51% - 99.89%Cor e Forma:SolidPeso molecular:351.84Ref: TM-T12565
1mg338,00€5mg538,00€1mL*10mM (DMSO)618,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47JI051
CAS:JI051 has anti-tumor effects and can interact with PHB2 to inhibit the proliferation of HEK293 cells and pancreatic cancer cells.Fórmula:C22H24N2O3Pureza:≥98% - ≥98.0%Cor e Forma:SolidPeso molecular:364.44S 32212 hydrochloride
CAS:S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .Fórmula:C25H29ClN4O2Pureza:97.11% - 99.57%Cor e Forma:SolidPeso molecular:452.98GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Fórmula:C18H17BrN2O2SPureza:99.33%Cor e Forma:SolidPeso molecular:405.31SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Fórmula:C25H31N3O2SPureza:99.12% - 99.69%Cor e Forma:SolidPeso molecular:437.6Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Fórmula:C20H25NOPureza:99.93%Cor e Forma:SolidPeso molecular:295.42Ref: TM-T22964
1mg38,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg259,00€50mg409,00€100mg605,00€500mg1.288,00€Afacifenacin
CAS:Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.Fórmula:C27H26F3N3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:481.51Ampreloxetine
CAS:Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Fórmula:C18H18F3NOPureza:98%Cor e Forma:SolidPeso molecular:321.34TC-N 22A
CAS:TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.Fórmula:C14H13N5SPureza:99.95%Cor e Forma:SolidPeso molecular:283.35WAY208466 dihydrochloride
CAS:WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.Fórmula:C17H20Cl2FN3O2SPureza:98.43% - 99.56%Cor e Forma:SolidPeso molecular:420.33U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Fórmula:C16H24ClN5Pureza:98%Cor e Forma:SolidPeso molecular:321.85ETAP
CAS:ETAP, a dual inhibitor of both monoamine oxidase A (MAO-A) and monoamine oxidase B (MAO-B), exhibits antidepressant-like effects and is utilized in the researchFórmula:C18H17N3OPureza:98%Cor e Forma:SolidPeso molecular:291.35Amitifadine hydrochloride
CAS:Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Fórmula:C11H12Cl3NPureza:98%Cor e Forma:SolidPeso molecular:264.58Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Fórmula:C17H26N4OPureza:98%Cor e Forma:SolidPeso molecular:302.41OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Fórmula:C11H16N2OPureza:98%Cor e Forma:SolidPeso molecular:192.26Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Fórmula:C15H17Cl2NO2Pureza:99.77%Cor e Forma:SolidPeso molecular:314.21Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Fórmula:C18H19NCor e Forma:SolidPeso molecular:249.35PF-4522654
CAS:PF-4522654 is a potent and selective 5-HT2C receptor agonist.Fórmula:C16H18F2N4Cor e Forma:SolidPeso molecular:304.34Pralidoxime mesylate
CAS:Pralidoxime mesylate is a Cholinesterase ReactivatorFórmula:C8H12N2O4SCor e Forma:SolidPeso molecular:232.25GlyT1 Inhibitor 1
CAS:GlyT1 Inhibitor 1 is a selective and potent GlyT1 inhibitor, inhibiting rGlyT1, used in research on neurological disorders.Fórmula:C22H21N5O2Cor e Forma:SolidPeso molecular:387.43L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Fórmula:C20H21N5O3SPureza:98.36%Cor e Forma:White SolidPeso molecular:411.48HexylHIBO
CAS:HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.Fórmula:C12H20N2O4Pureza:99.55%Cor e Forma:SolidPeso molecular:256.3AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Fórmula:C27H38N6O2Pureza:98.01%Cor e Forma:SolidPeso molecular:478.63ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Fórmula:C13H17ClN2Pureza:98%Cor e Forma:SolidPeso molecular:236.74Ref: TM-T23396
1mg44,00€5mg111,00€1mL*10mM (DMSO)123,00€10mg178,00€25mg316,00€50mg470,00€100mg682,00€200mg954,00€A-794282
CAS:A-794282 is a selective antagonist of mGluR1.Fórmula:C19H18N4OSPureza:99.87%Cor e Forma:SolidPeso molecular:350.44WAY 629
CAS:WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.Fórmula:C15H18N2Cor e Forma:SolidPeso molecular:226.32AVN-101 free base
CAS:AVN-101: potent 5-HT7 antagonist, also targets 5-HT6, 5-HT2A, 5-HT2C. Aims to treat CNS disorders.Fórmula:C21H24N2Cor e Forma:SolidPeso molecular:304.43Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Fórmula:C18H12Cl2N2OCor e Forma:SolidPeso molecular:343.21AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Fórmula:C19H29NO5Pureza:98.19% - 99.55%Cor e Forma:SolidPeso molecular:351.44Octamylamine hydrochloride
CAS:Octamylamine hydrochloride is a P450 inhibitor.Fórmula:C13H30ClNCor e Forma:SolidPeso molecular:235.84TC-1698 dihydrochloride
CAS:TC-1698 dihydrochloride: selective α7 nicotinic agonist, with some β-receptor activity; neuroprotectant.Fórmula:C13H20Cl2N2Cor e Forma:SolidPeso molecular:275.22Octamylamine sulfamate
CAS:Octamylamine sulfamate is a P450 inhibitor.Fórmula:C13H32N2O3SCor e Forma:SolidPeso molecular:296.47Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Fórmula:C16H17BrN2Pureza:98%Cor e Forma:SolidPeso molecular:317.22Hadacidin sodium
CAS:Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.Fórmula:C3H4NNaO4Cor e Forma:SolidPeso molecular:141.06PF-06663195
CAS:PF-06663195 is a potent inhibitor of β-site amyloid precursor protein (APP) Cleaving Enzyme 1 (BACE1, β-Secretase 1).Fórmula:C18H18F3N3O2SCor e Forma:SolidPeso molecular:397.41Neopterin, L-erythro-
CAS:Neopterin, L-erythro- can be used as a cholinergic receptor.Fórmula:C9H11N5O4Cor e Forma:SolidPeso molecular:253.21q-FTAA
CAS:q-FTAA targets Aβ1-42 fibrils (330-630 nM) and ADPBC (300-500 nM), useful in Alzheimer's disease research.Fórmula:C21H14O6S4Cor e Forma:SolidPeso molecular:490.59Atropine Oxide Hydrochloride
CAS:Atropine Oxide, a derivative of anticholinergic Atropine, treats poisonings, slow heart rate, and reduces saliva during surgery.Fórmula:C17H24ClNO4Cor e Forma:SolidPeso molecular:341.83Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Fórmula:C19H21NPureza:99.15% - 99.66%Cor e Forma:SolidPeso molecular:263.38Ethybenztropine HBr
CAS:Ethybenztropine HBr is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.Fórmula:C22H28BrNOCor e Forma:SolidPeso molecular:402.37
