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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5337 produtos de "GPCR/Proteína-G"

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  • TSHR antagonist S37

    CAS:
    <p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>
    Fórmula:C25H20N2O3S2
    Pureza:98.35%
    Cor e Forma:Solid
    Peso molecular:460.57
  • Astressin acetate


    <p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>
    Fórmula:C163H273N49O44
    Pureza:96.87%
    Cor e Forma:Solid
    Peso molecular:3623.21
  • Clopidogrel hydrogen sulfate

    CAS:
    <p>Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.</p>
    Fórmula:C16H16ClNO2S·H2SO4
    Pureza:99.57% - 99.79%
    Cor e Forma:Solid
    Peso molecular:419.9
  • MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Fórmula:C27H25N3O4S2
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:519.64
  • YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74
  • BP 897 hydrochloride

    CAS:
    <p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>
    Fórmula:C26H32ClN3O2
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:454
  • Urocortin (rat) acetate


    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Pureza:97.76%
    Cor e Forma:Soild
  • Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Fórmula:C19H24N2O·HCl
    Pureza:99.84% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:332.87
  • Sonepcizumab

    CAS:
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Pureza:SDS-PAGE:95% SEC-HPLC:98.90%
    Cor e Forma:Liquid
    Peso molecular:146.43 kDa
  • Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Fórmula:C9H15ClNO5P
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:283.65
  • Metaraminol tartrate

    CAS:
    <p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Fórmula:C13H19NO8
    Pureza:99.68%
    Cor e Forma:White Powder
    Peso molecular:317.29
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51
  • Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49
  • Thioridazine hydrochloride

    CAS:
    <p>Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4</p>
    Fórmula:C21H27ClN2S2
    Pureza:99.55% - 99.957%
    Cor e Forma:White To Off-White Solid
    Peso molecular:407.04
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Fórmula:C21H25NO·CH4SO3
    Pureza:98.41% - 99.96%
    Cor e Forma:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecular:403.53
  • KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Fórmula:C26H40N4O8
    Pureza:98.46%
    Cor e Forma:Solid
    Peso molecular:536.62
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:348.87
  • Cloperastine hydrochloride

    CAS:
    <p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>
    Fórmula:C20H25Cl2NO
    Pureza:97.74% - 99.42%
    Cor e Forma:Solid
    Peso molecular:366.33
  • Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39
  • Cinnarizine

    CAS:
    <p>Cinnarizine is a piperazine, blocks H1-receptor &amp; Ca-channels, has vasodilating &amp; antiemetic effects, may cause Parkinson-like symptoms.</p>
    Fórmula:C26H28N2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:368.51
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Cor e Forma:Solid
    Peso molecular:508.56
  • Acetophenazine dimaleate

    CAS:
    <p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>
    Fórmula:C31H37N3O10S
    Pureza:99.39% - 99.48%
    Cor e Forma:Solid
    Peso molecular:643.71
  • Agomelatine

    CAS:
    <p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>
    Fórmula:C15H17NO2
    Pureza:99.92%
    Cor e Forma:White Solid
    Peso molecular:243.3
  • LCKLSL hydrochloride


    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Fórmula:C30H58ClN7O8S
    Pureza:98.02% - 99.31%
    Cor e Forma:Solid
    Peso molecular:712.34
  • Nylidrin hydrochloride

    CAS:
    <p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells &amp; human basophils.</p>
    Fórmula:C19H26ClNO2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:335.87
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Fórmula:C19H26ClN5O4
    Pureza:99.69% - 99.91%
    Cor e Forma:Solid
    Peso molecular:423.89
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Fórmula:C22H34Cl2N2O2
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:429.42
  • Clomipramine hydrochloride

    CAS:
    <p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>
    Fórmula:C19H23ClN2·HCl
    Pureza:99.04% - 99.47%
    Cor e Forma:White To Slightly Yellow Crystalline Powder
    Peso molecular:351.31
  • Ifenprodil

    CAS:
    <p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 &amp; GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>
    Fórmula:C21H27NO2
    Pureza:99.58%
    Cor e Forma:White Crystalline Powder
    Peso molecular:325.44
  • Aniracetam

    CAS:
    <p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>
    Fórmula:C12H13NO3
    Pureza:99.88% - 99.89%
    Cor e Forma:White Crystalline Or Crystalline Powde
    Peso molecular:219.24
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Fórmula:C11H9BrO
    Pureza:98.51%
    Cor e Forma:White To Off-White Powder
    Peso molecular:237.09
  • Ketanserin

    CAS:
    <p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>
    Fórmula:C22H22FN3O3
    Pureza:99.19% - 99.73%
    Cor e Forma:Solid
    Peso molecular:395.43
  • Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Fórmula:C18H26ClN3O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:367.87
  • Doxofylline

    CAS:
    <p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>
    Fórmula:C11H14N4O4
    Pureza:99.958% - >99.99%
    Cor e Forma:Solid
    Peso molecular:266.25
  • Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Fórmula:C17H28ClNO2
    Pureza:97.32% - 99.86%
    Cor e Forma:White Crystalline Powder
    Peso molecular:313.86
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Fórmula:C19H27N5O4·HCl
    Pureza:99.78%
    Cor e Forma:White To Off-White Solid
    Peso molecular:425.91
  • Chlorprothixene hydrochloride

    CAS:
    <p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>
    Fórmula:C18H18ClNS·HCl
    Pureza:99.76%
    Cor e Forma:White Powder
    Peso molecular:352.32
  • Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Fórmula:C19H21N3O
    Pureza:98.50% - 99.44%
    Cor e Forma:Solid
    Peso molecular:307.39
  • CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Fórmula:C15H18Cl2N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:341.24
  • Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53
  • CD80-IN-3

    CAS:
    <p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>
    Fórmula:C17H10FN3O3
    Pureza:98.08%
    Cor e Forma:Solid
    Peso molecular:323.28
  • Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Fórmula:C19H31ClF3NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:413.9
  • Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Fórmula:C26H35NO7
    Pureza:98.53% - 99.43%
    Cor e Forma:Coa
    Peso molecular:473.57
  • Dimenhydrinate

    CAS:
    <p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>
    Fórmula:C24H28ClN5O3
    Pureza:99.57% - 99.77%
    Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Peso molecular:469.96
  • Filorexant

    CAS:
    <p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki &lt;3 nM).</p>
    Fórmula:C24H25FN4O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:420.48
  • Pemirolast potassium

    CAS:
    <p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>
    Fórmula:C10H7KN6O
    Pureza:98.91% - 99.63%
    Cor e Forma:Crystals From Dimethylformamide Crystalline Solid
    Peso molecular:266.31
  • Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Fórmula:C15H20N2O2·HCl
    Pureza:99.64% - 99.92%
    Cor e Forma:Solid
    Peso molecular:296.79
  • Timonacic

    CAS:
    <p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>
    Fórmula:C4H7NO2S
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:133.17
  • Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Fórmula:C9H10O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:182.17
  • Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Cor e Forma:White Crystal Powder
    Peso molecular:365.86
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79
  • Adrenalone hydrochloride

    CAS:
    <p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>
    Fórmula:C9H11NO3·HCl
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:217.65
  • Ro 10-5824 dihydrochloride

    CAS:
    <p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:353.29
  • Fluoxetine hydrochloride

    CAS:
    <p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>
    Fórmula:C17H19ClF3NO
    Pureza:99.6% - 99.98%
    Cor e Forma:White To Off-White Crystalline Solid White To Off-White Powder
    Peso molecular:345.787
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Fórmula:C31H38N2O
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:454.65
  • Sergliflozin A

    CAS:
    <p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>
    Fórmula:C20H24O7
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:376.4
  • Gevotroline

    CAS:
    <p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>
    Fórmula:C19H20FN3
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:309.38
  • Carbetapentane citrate

    CAS:
    <p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>
    Fórmula:C20H31NO3·C6H8O7
    Pureza:99.46%
    Cor e Forma:White To Off-White Solid
    Peso molecular:525.59
  • DPTN dihydrochloride

    CAS:
    <p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>
    Fórmula:C22H20Cl2N4OS
    Pureza:99.95%
    Cor e Forma:Soild
    Peso molecular:459.39
  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41
  • Linaclotide

    CAS:
    <p>Linaclotide treats IBS-C &amp; chronic constipation; it's a selective guanylate cyclase C agonist.</p>
    Fórmula:C59H79N15O21S6
    Pureza:97.93% - 98.71%
    Cor e Forma:Solid
    Peso molecular:1526.74
  • Silodosin

    CAS:
    <p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>
    Fórmula:C25H32F3N3O4
    Pureza:99.282% - 99.76%
    Cor e Forma:Colorless To Pink Solid
    Peso molecular:495.53
  • Cericlamine

    CAS:
    <p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>
    Fórmula:C12H17Cl2NO
    Pureza:99.38%
    Cor e Forma:Solid
    Peso molecular:262.18
  • Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Fórmula:C11H17NO3·5H2O4S
    Pureza:98.53% - 99.74%
    Cor e Forma:Solid
    Peso molecular:260.3
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Fórmula:C11H19N5
    Pureza:98.33% - 99.62%
    Cor e Forma:Solid
    Peso molecular:221.3
  • Tetrahydrozoline

    CAS:
    <p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>
    Fórmula:C13H16N2
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:200.28
  • SR59230A

    CAS:
    <p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>
    Fórmula:C23H29NO6
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:415.48
  • Pranazepide

    CAS:
    <p>Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.</p>
    Fórmula:C26H19FN4O2
    Pureza:97.43% - 99.53%
    Cor e Forma:Solid
    Peso molecular:438.45
  • AVN 322 free base

    CAS:
    <p>AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.</p>
    Fórmula:C17H19N5O2S
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:357.43
  • Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Fórmula:C22H23ClN2O2
    Pureza:99.71% - 99.98%
    Cor e Forma:White Powder
    Peso molecular:382.88
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Fórmula:C21H23N3OS
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:365.49
  • Rebamipide

    CAS:
    <p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>
    Fórmula:C19H15ClN2O4
    Pureza:99.48% - 99.61%
    Cor e Forma:White Powder
    Peso molecular:370.79
  • Midodrine hydrochloride

    CAS:
    <p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>
    Fórmula:C12H19ClN2O4
    Pureza:99.79% - >99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:290.74
  • ML-109

    CAS:
    <p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>
    Fórmula:C31H29N3O5
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:523.58
  • Azelastine hydrochloride

    CAS:
    <p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>
    Fórmula:C22H24ClN3O·HCl
    Pureza:98% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:418.36
  • Iobenguane sulfate

    CAS:
    <p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>
    Fórmula:C8H10IN3H2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:324.12
  • Terbutaline

    CAS:
    <p>Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol</p>
    Fórmula:C12H19NO3
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:225.3
  • Nelivaptan

    CAS:
    <p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>
    Fórmula:C30H32ClN3O8S
    Pureza:98.46% - 99.89%
    Cor e Forma:Solid
    Peso molecular:630.11
  • Sarizotan 2HCl

    CAS:
    <p>Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.</p>
    Fórmula:C22H23Cl2FN2O
    Pureza:98.83%
    Cor e Forma:Soild
    Peso molecular:421.34
  • Delequamine

    CAS:
    <p>Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.</p>
    Fórmula:C18H26N2O3S
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:350.48
  • Iloperidone

    CAS:
    <p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>
    Fórmula:C24H27FN2O4
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:426.48
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Fórmula:C21H24N4O2S
    Pureza:99.64%
    Cor e Forma:Light Yellow To Yellow Solid
    Peso molecular:396.51
  • Sertraline hydrochloride

    CAS:
    <p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>
    Fórmula:C17H18Cl3N
    Pureza:99.12% - 99.89%
    Cor e Forma:Solid Powder
    Peso molecular:342.691
  • Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Fórmula:C36H51Cl2N3O4
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:660.71
  • RS 15385-198

    CAS:
    <p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Pureza:>99.99%
    Cor e Forma:Soild
    Peso molecular:350.48
  • Olopatadine hydrochloride

    CAS:
    <p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>
    Fórmula:C21H23NO3·HCl
    Pureza:99.62% - 99.64%
    Cor e Forma:White Solid
    Peso molecular:373.87
  • Balovaptan

    CAS:
    <p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>
    Fórmula:C22H24ClN5O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Tolnaftate

    CAS:
    <p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>
    Fórmula:C19H17NOS
    Pureza:98.85%
    Cor e Forma:White Powder
    Peso molecular:307.41
  • 2',5'-Dideoxyadenosine

    CAS:
    <p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>
    Fórmula:C10H13N5O2
    Pureza:99.55%
    Cor e Forma:White Solid
    Peso molecular:235.24
  • INCB-9471

    CAS:
    <p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>
    Fórmula:C30H40F3N5O2
    Pureza:98.80%
    Cor e Forma:Solid
    Peso molecular:559.666
  • Mirtazapine

    CAS:
    <p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>
    Fórmula:C17H19N3
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Pheniramine maleate

    CAS:
    <p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>
    Fórmula:C16H20N2·C4H4O4
    Pureza:99.85%
    Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
    Peso molecular:356.42
  • Bromperidol

    CAS:
    <p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>
    Fórmula:C21H23BrFNO2
    Pureza:99.89%
    Cor e Forma:Tan Solid
    Peso molecular:420.32
  • (R)-Terazosin

    CAS:
    <p>R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).</p>
    Fórmula:C19H25N5O4
    Pureza:98.87% - 98.96%
    Cor e Forma:Solid
    Peso molecular:387.43
  • Paroxetine hydrochloride

    CAS:
    <p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>
    Fórmula:C19H21ClFNO3
    Pureza:98% - 99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:365.826
  • Tegaserod maleate

    CAS:
    <p>Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.</p>
    Fórmula:C20H27N5O5
    Pureza:98% - 99.06%
    Cor e Forma:White Powder
    Peso molecular:417.46
  • Moxonidine

    CAS:
    <p>Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.</p>
    Fórmula:C9H12ClN5O
    Pureza:99.81% - 99.94%
    Cor e Forma:Crystal
    Peso molecular:241.68
  • Risperidone

    CAS:
    <p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>
    Fórmula:C23H27FN4O2
    Pureza:99.73%
    Cor e Forma:Crystalline Solid
    Peso molecular:410.48
  • Doxepin hydrochloride

    CAS:
    <p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>
    Fórmula:C19H22ClNO
    Pureza:99.65% - 99.91%
    Cor e Forma:White To Off-White Powder
    Peso molecular:315.84
  • AB928

    CAS:
    <p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>
    Fórmula:C23H22N8O
    Pureza:98.09% - >99.99%
    Cor e Forma:Solid
    Peso molecular:426.47
  • Evocalcet

    CAS:
    <p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>
    Fórmula:C24H26N2O2
    Pureza:98.88% - 99.68%
    Cor e Forma:Solid
    Peso molecular:374.48
  • Ketotifen fumarate

    CAS:
    <p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>
    Fórmula:C23H23NO5S
    Pureza:99.25% - 99.73%
    Cor e Forma:Solid
    Peso molecular:425.50
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Fórmula:C15H24N2O4S·HCl
    Pureza:99.4% - 99.77%
    Cor e Forma:Solid
    Peso molecular:364.89
  • Ranitidine Hydrochloride

    CAS:
    <p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>
    Fórmula:C13H23ClN4O3S
    Pureza:99.30% - 99.49%
    Cor e Forma:Solid
    Peso molecular:350.86
  • JHU 75528

    CAS:
    <p>JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.</p>
    Fórmula:C23H21Cl2N5O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:470.35
  • Tabernanthalog fumarate

    CAS:
    <p>Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.</p>
    Fórmula:C18H22N2O5
    Pureza:99.83%
    Cor e Forma:Soild
    Peso molecular:346.38
  • Lesopitron HCl

    CAS:
    <p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>
    Fórmula:C15H22Cl2N6
    Pureza:97.05% - 99.89%
    Cor e Forma:Soild
    Peso molecular:357.28
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Fórmula:C10H16N6S
    Pureza:99.82%
    Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Peso molecular:252.34
  • Quercetin-3'-o-phosphate TEA


    <p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>
    Fórmula:C21H26NO10P
    Pureza:95.63%
    Cor e Forma:Soild
    Peso molecular:483.41
  • Maprotiline hydrochloride

    CAS:
    <p>Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.</p>
    Fórmula:C20H24ClN
    Pureza:99.68% - 99.84%
    Cor e Forma:White Powder
    Peso molecular:313.864
  • Quipazine dimaleate

    CAS:
    <p>Quipazine dimaleate is a selective 5-HT3 agonist.</p>
    Fórmula:C21H23N3O8
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:445.42
  • p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Fórmula:C25H28ClIN4O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:578.87
  • Amylin, amide, human

    CAS:
    <p>Amylin, amide, human(DAP Amide) is a 37-amino acid peptide hormone co-secreted with insulin to regulate postprandial glucose levels.</p>
    Fórmula:C165H261N51O55S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3903.28
  • EMPA

    CAS:
    <p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>
    Fórmula:C23H26N4O4S
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:454.54
  • Bucumolol

    CAS:
    <p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>
    Fórmula:C17H23NO4
    Pureza:99.66%
    Cor e Forma:Soild
    Peso molecular:305.37
  • Ozagrel

    CAS:
    <p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>
    Fórmula:C13H12N2O2
    Pureza:97.90% - 99.38%
    Cor e Forma:White Powder
    Peso molecular:228.25
  • CI 169369

    CAS:
    <p>CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.</p>
    Fórmula:C19H21ClN2S
    Pureza:98.97%
    Cor e Forma:Soild
    Peso molecular:344.9
  • MRGPRX1 agonist 1

    CAS:
    <p>MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).</p>
    Fórmula:C23H21N3O4S
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:435.5
  • Cloroperone

    CAS:
    <p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>
    Fórmula:C22H23ClFNO2
    Pureza:98.40%
    Cor e Forma:Soild
    Peso molecular:387.88
  • Roluperidone

    CAS:
    <p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>
    Fórmula:C22H23FN2O2
    Pureza:96.46% - 97.77%
    Cor e Forma:Solid
    Peso molecular:366.43
  • Promethazine

    CAS:
    <p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>
    Fórmula:C17H20N2S
    Pureza:99.76%
    Cor e Forma:Crystals
    Peso molecular:284.42
  • Labetalol

    CAS:
    <p>Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.</p>
    Fórmula:C19H24N2O3
    Pureza:99.87% - 99.89%
    Cor e Forma:Solid
    Peso molecular:328.41
  • Nepafenac

    CAS:
    <p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>
    Fórmula:C15H14N2O2
    Pureza:98.94% - 99.43%
    Cor e Forma:Solid
    Peso molecular:254.28
  • PIT

    CAS:
    <p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>
    Fórmula:C20H16N2O5S
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:396.42
  • REV 5901A

    CAS:
    <p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>
    Fórmula:C22H26ClNO2
    Pureza:98.04%
    Cor e Forma:Soild
    Peso molecular:371.90
  • Glycerol phenylbutyrate

    CAS:
    <p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>
    Fórmula:C33H38O6
    Pureza:98.54% - 99.74%
    Cor e Forma:Solid
    Peso molecular:530.65
  • RS102895 hydrochloride

    CAS:
    <p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>
    Fórmula:C21H22ClF3N2O2
    Pureza:98.95%
    Cor e Forma:Solid
    Peso molecular:426.86
  • CCR2-RA-[R]

    CAS:
    <p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>
    Fórmula:C18H19ClFNO3
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:351.8
  • N6-Ethyladenosine

    CAS:
    <p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>
    Fórmula:C12H17N5O4
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:295.29
  • SEP-363856 hydrochloride

    CAS:
    <p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>
    Fórmula:C9H14ClNOS
    Pureza:99.86% - 99.99%
    Cor e Forma:Solid
    Peso molecular:219.73
  • NS-2028

    CAS:
    <p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>
    Fórmula:C9H5BrN2O3
    Pureza:99.44%
    Cor e Forma:A Crystalline Solid
    Peso molecular:269.05
  • Ritodrine hydrochloride

    CAS:
    <p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>
    Fórmula:C17H21NO3·HCl
    Pureza:99% - 99.52%
    Cor e Forma:Solid
    Peso molecular:323.82
  • Dazmegrel HCl


    <p>Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.</p>
    Fórmula:C16H18ClN3O2
    Pureza:98.30%
    Cor e Forma:Solid
    Peso molecular:319.79
  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    <p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>
    Fórmula:C20H29N3O8
    Pureza:99.72%
    Cor e Forma:Soild
    Peso molecular:439.46
  • Domperidone

    CAS:
    <p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>
    Fórmula:C22H24ClN5O2
    Pureza:98% - 99.82%
    Cor e Forma:Solid
    Peso molecular:425.91
  • GTS-21 dihydrochloride

    CAS:
    <p>GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.</p>
    Fórmula:C19H20N2O2·2HCl
    Pureza:98.54% - >99.99%
    Cor e Forma:Solid
    Peso molecular:381.3
  • Methoxamine hydrochloride

    CAS:
    <p>Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.</p>
    Fórmula:C11H18ClNO3
    Pureza:99.84% - >99.99%
    Cor e Forma:Colorless Or White Plate-Like Crystals Or White Crystalline Powder Solid
    Peso molecular:247.719
  • Fezolinetant

    CAS:
    <p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>
    Fórmula:C16H15FN6OS
    Pureza:98.62% - 99.7%
    Cor e Forma:Solid
    Peso molecular:358.39
  • PF-04995274

    CAS:
    <p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>
    Fórmula:C23H32N2O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:432.51
  • Somatostatin acetate


    <p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>
    Pureza:99.11%
    Cor e Forma:Odour Solid
  • Lamotrigine

    CAS:
    <p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>
    Fórmula:C9H7Cl2N5
    Pureza:99.76% - 99.95%
    Cor e Forma:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Peso molecular:256.09
  • Itopride hydrochloride

    CAS:
    <p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>
    Fórmula:C20H27ClN2O4
    Pureza:99.59%
    Cor e Forma:White Or Pale Brownish Crystal
    Peso molecular:394.9
  • Sulpiride

    CAS:
    <p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>
    Fórmula:C15H23N3O4S
    Pureza:99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • Triprolidine hydrochloride monohydrate

    CAS:
    <p>Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.</p>
    Fórmula:C19H25ClN2O
    Pureza:99.68% - 99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:332.87
  • Loxapine succinate

    CAS:
    <p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>
    Fórmula:C22H24ClN3O5
    Pureza:99.69%
    Cor e Forma:White To Of-White Solid
    Peso molecular:445.9
  • Degarelix acetate(214766-78-6 free base)

    CAS:
    <p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>
    Fórmula:C84H107ClN18O18
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:1692.34
  • BIBO3304 TFA

    CAS:
    <p>BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).</p>
    Fórmula:C31H36F3N7O5
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:643.66
  • Fluphenazine dihydrochloride

    CAS:
    <p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>
    Fórmula:C22H28Cl2F3N3OS
    Pureza:99.23%
    Cor e Forma:Off-White Solid
    Peso molecular:510.44
  • MK-0249 FA


    <p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>
    Fórmula:C24H26F3N3O4
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:477.48
  • Retatrutide sodium salt


    <p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>
    Pureza:99.97%
    Cor e Forma:Soild
  • CE3F4

    CAS:
    <p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>
    Fórmula:C11H10Br2FNO
    Pureza:97.15% - 98.06%
    Cor e Forma:Solid
    Peso molecular:351.01
  • CCX140

    CAS:
    <p>CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.</p>
    Fórmula:C20H13ClF3N5O3S
    Pureza:99.66% - 99.95%
    Cor e Forma:Solid
    Peso molecular:495.86
  • Tipepidine hydrochloride

    CAS:
    <p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>
    Fórmula:C15H18ClNS2
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:311.89
  • Flunarizine dihydrochloride

    CAS:
    <p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>
    Fórmula:C26H28Cl2F2N2
    Pureza:99.53% - 99.89%
    Cor e Forma:White Crystalline Powder Odorless And Tasteless
    Peso molecular:477.42
  • JP1302 dihydrochloride

    CAS:
    <p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>
    Fórmula:C24H26Cl2N4
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:441.4
  • Pizotifen Malate

    CAS:
    <p>Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.</p>
    Fórmula:C19H21NS·C4H6O5
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:429.53
  • Buflomedil hydrochloride

    CAS:
    <p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>
    Fórmula:C17H26ClNO4
    Pureza:99.7% - 99.91%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:343.85
  • Molindone hydrochloride

    CAS:
    <p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>
    Fórmula:C16H24N2O2·HCl
    Pureza:99% - 99.99%
    Cor e Forma:Solid
    Peso molecular:312.84
  • Azasetron hydrochloride

    CAS:
    <p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>
    Fórmula:C17H20ClN3O3·HCl
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:386.27
  • Vibozilimod

    CAS:
    <p>Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .</p>
    Fórmula:C29H36ClN3O5
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:542.07
  • Dexchlorpheniramine Maleate

    CAS:
    <p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.58%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:390.86
  • Clozapine

    CAS:
    <p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>
    Fórmula:C18H19ClN4
    Pureza:99.91% - 99.93%
    Cor e Forma:Yellow Crystals From Acetone-Petroleum Ether Solid
    Peso molecular:326.82
  • Sumatriptan succinate

    CAS:
    <p>Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.</p>
    Fórmula:C18H27N3O6S
    Pureza:97.53% - 99.51%
    Cor e Forma:White Powder
    Peso molecular:413.49
  • Ebalzotan

    CAS:
    <p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>
    Fórmula:C19H30N2O2
    Pureza:98.09% - 99.41%
    Cor e Forma:Solid
    Peso molecular:318.45
  • BMY 25368 HCl

    CAS:
    <p>BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.</p>
    Fórmula:C19H26ClN3O3
    Pureza:98.73% - 99.81%
    Cor e Forma:Soild
    Peso molecular:379.88
  • Amp579 TFA


    <p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>
    Fórmula:C24H29ClF3N5O5S
    Pureza:96.56%
    Cor e Forma:Soild
    Peso molecular:592.03
  • Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Fórmula:C46H54N6O8S2
    Pureza:99.32% - >99.99%
    Cor e Forma:White Crystalline Solid
    Peso molecular:883.09
  • CB1 antagonist 2

    CAS:
    <p>CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.</p>
    Fórmula:C17H12Cl3N3O
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:380.66
  • DF-1012 FA


    <p>DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.</p>
    Fórmula:C17H22N4O3
    Pureza:99.15% - 99.97%
    Cor e Forma:Solid
    Peso molecular:330.382
  • CYM50308

    CAS:
    <p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>
    Fórmula:C20H21F2N3O2S
    Pureza:99.43% - 99.77%
    Cor e Forma:Solid
    Peso molecular:405.46
  • Strontium ranelate

    CAS:
    <p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>
    Fórmula:C12H6N2O8S·2Sr
    Pureza:98.97%
    Cor e Forma:Crystalline Solid
    Peso molecular:513.49
  • Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.64% - 99.98%
    Cor e Forma:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Peso molecular:390.87
  • Duloxetine hydrochloride

    CAS:
    <p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>
    Fórmula:C18H20ClNOS
    Pureza:99.93% - >99.99%
    Cor e Forma:White Or White Crystalline Powder
    Peso molecular:333.88
  • Phenoxybenzamine hydrochloride

    CAS:
    <p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>
    Fórmula:C18H23Cl2NO
    Pureza:98.04% - >99.99%
    Cor e Forma:Antihypertensive Drug
    Peso molecular:340.3
  • J-113863

    CAS:
    <p>J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).</p>
    Fórmula:C30H37Cl2IN2O2
    Pureza:95.11%
    Cor e Forma:Solid
    Peso molecular:655.44
  • Latozinemab


    <p>Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.</p>
    Pureza:> 95%
    Cor e Forma:Liquid
    Peso molecular:146.28 kDa
  • Naftifine hydrochloride

    CAS:
    <p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>
    Fórmula:C21H22ClN
    Pureza:98.75% - 99.84%
    Cor e Forma:Solid
    Peso molecular:323.86
  • Amitriptyline hydrochloride

    CAS:
    <p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>
    Fórmula:C20H24ClN
    Pureza:97% - 99.94%
    Cor e Forma:Crystals White To Off-White Powder
    Peso molecular:313.86
  • SBI-477

    CAS:
    <p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>
    Fórmula:C24H25N3O6S
    Pureza:99.3%
    Cor e Forma:Solid
    Peso molecular:483.54
  • Avexitide acetate

    CAS:
    <p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>
    Fórmula:C155H246N40O53S
    Pureza:96.64% - 98.65%
    Cor e Forma:Solid
    Peso molecular:3549.91
  • Trimipramine maleate

    CAS:
    <p>Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.</p>
    Fórmula:C24H30N2O4
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:410.51
  • 6-Iodopravadoline

    CAS:
    <p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>
    Fórmula:C23H25IN2O3
    Pureza:99.29%
    Cor e Forma:Off-White Solid
    Peso molecular:504.36
  • Tryptamine hydrochloride

    CAS:
    <p>Tryptamine hydrochloride is a monoamine alkaloid, metabolite of tryptophan and CNS active substance, agonist of 5-HT4 receptor, TAAR1, AHR.</p>
    Fórmula:C10H13ClN2
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:196.68
  • Apelin-12 acetate


    <p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>
    Fórmula:C66H107N21O16S
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:1482.75
  • Gulgafafusp alfa

    CAS:
    <p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>
    Cor e Forma:Liquid
  • PSB-22269


    <p>PSB-22269 is identified as a GPR17 antagonist with a Ki value of 8.91 nM. It exhibits significant inhibitory effects in cAMP and G protein activation assays. Molecular docking studies indicate that the binding site of PSB-22269 includes positively charged arginine residues and a hydrophobic pocket. PSB-22269 promotes myelin regeneration strategies, offering potential for multiple sclerosis research.</p>
    Fórmula:C26H21NO6
    Cor e Forma:Solid
    Peso molecular:443.45
  • PACAP-related Peptide (human) (trifluoroacetate salt)


    <p>Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some VIP tumors; secreted by CHO-K1 cells.</p>
    Cor e Forma:Liquid
  • BAM(8-22)

    CAS:
    <p>Potent MRGPRX1 agonist peptide; first found in bovine adrenal glands. Non-opioid, lacking met-enkephalin motif. EC50: 8-150 nM.</p>
    Fórmula:C91H127N25O23S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1971.22
  • Mitemcinal fumarate

    CAS:
    <p>Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.</p>
    Fórmula:C84H142N2O28
    Cor e Forma:Solid
    Peso molecular:1628.02
  • PACAP (1-38) free acid

    CAS:
    <p>PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.</p>
    Cor e Forma:Solid
  • Parstatin(human)

    CAS:
    Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.
    Fórmula:C191H330N64O53S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4467.29
  • Setmelanotide

    CAS:
    <p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>
    Fórmula:C49H68N18O9S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1117.31
  • HPP-9


    <p>HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET</p>
    Fórmula:C49H52N6O11
    Cor e Forma:Solid
    Peso molecular:900.97
  • Oxaprotiline hydrochloride

    CAS:
    <p>Oxaprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.86
  • Mosliciguat

    CAS:
    <p>Mosliciguat is a guanylate cyclase activator.</p>
    Fórmula:C41H36ClF3N2O5
    Cor e Forma:Solid
    Peso molecular:729.19
  • Substance P (4-11)

    CAS:
    <p>Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.</p>
    Fórmula:C46H67N11O10S
    Cor e Forma:Solid
    Peso molecular:966.16
  • Stressin I


    <p>Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.</p>
    Fórmula:C203H337N57O56
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4472.24