
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.943 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(196 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(69 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(164 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5337 produtos de "GPCR/Proteína-G"
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TSHR antagonist S37
CAS:<p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>Fórmula:C25H20N2O3S2Pureza:98.35%Cor e Forma:SolidPeso molecular:460.57Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Fórmula:C163H273N49O44Pureza:96.87%Cor e Forma:SolidPeso molecular:3623.21Clopidogrel hydrogen sulfate
CAS:<p>Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.</p>Fórmula:C16H16ClNO2S·H2SO4Pureza:99.57% - 99.79%Cor e Forma:SolidPeso molecular:419.9MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Fórmula:C27H25N3O4S2Pureza:97.44%Cor e Forma:SolidPeso molecular:519.64YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Fórmula:C33H37N5O5SPureza:99.67%Cor e Forma:SolidPeso molecular:615.74BP 897 hydrochloride
CAS:<p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>Fórmula:C26H32ClN3O2Pureza:99.42%Cor e Forma:SolidPeso molecular:454Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Pureza:97.76%Cor e Forma:SoildPalonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Cor e Forma:White SolidPeso molecular:332.87Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Pureza:SDS-PAGE:95% SEC-HPLC:98.90%Cor e Forma:LiquidPeso molecular:146.43 kDaFosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Fórmula:C9H15ClNO5PPureza:99.84%Cor e Forma:SolidPeso molecular:283.65Metaraminol tartrate
CAS:<p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Fórmula:C13H19NO8Pureza:99.68%Cor e Forma:White PowderPeso molecular:317.29Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:383.51Naftopidil
CAS:<p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>Fórmula:C24H28N2O3Pureza:99.60% - 99.97%Cor e Forma:White Crystalline PowderPeso molecular:392.49Thioridazine hydrochloride
CAS:<p>Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4</p>Fórmula:C21H27ClN2S2Pureza:99.55% - 99.957%Cor e Forma:White To Off-White SolidPeso molecular:407.04Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53KGA-2727
CAS:<p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>Fórmula:C26H40N4O8Pureza:98.46%Cor e Forma:SolidPeso molecular:536.62Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Fórmula:C18H25ClN4OPureza:99.88% - 99.93%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:348.87Cloperastine hydrochloride
CAS:<p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>Fórmula:C20H25Cl2NOPureza:97.74% - 99.42%Cor e Forma:SolidPeso molecular:366.33Aripiprazole
CAS:<p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Cor e Forma:Colourless Flake Crystalline SolidPeso molecular:448.39Cinnarizine
CAS:<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Fórmula:C26H28N2Pureza:99.94%Cor e Forma:SolidPeso molecular:368.51Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Fórmula:C28H32N2O7Pureza:99.03% - 99.67%Cor e Forma:SolidPeso molecular:508.56Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Cor e Forma:SolidPeso molecular:643.71Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Fórmula:C15H17NO2Pureza:99.92%Cor e Forma:White SolidPeso molecular:243.3LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Fórmula:C30H58ClN7O8SPureza:98.02% - 99.31%Cor e Forma:SolidPeso molecular:712.34Nylidrin hydrochloride
CAS:<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Fórmula:C19H26ClNO2Pureza:99.35%Cor e Forma:SolidPeso molecular:335.87Terazosin hydrochloride
CAS:<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Fórmula:C19H26ClN5O4Pureza:99.69% - 99.91%Cor e Forma:SolidPeso molecular:423.89Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Fórmula:C22H34Cl2N2O2Pureza:98.55%Cor e Forma:SolidPeso molecular:429.42Clomipramine hydrochloride
CAS:<p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>Fórmula:C19H23ClN2·HClPureza:99.04% - 99.47%Cor e Forma:White To Slightly Yellow Crystalline PowderPeso molecular:351.31Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Fórmula:C21H27NO2Pureza:99.58%Cor e Forma:White Crystalline PowderPeso molecular:325.44Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Fórmula:C12H13NO3Pureza:99.88% - 99.89%Cor e Forma:White Crystalline Or Crystalline PowdePeso molecular:219.242-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Fórmula:C11H9BrOPureza:98.51%Cor e Forma:White To Off-White PowderPeso molecular:237.09Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Cor e Forma:SolidPeso molecular:395.43Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Fórmula:C18H26ClN3O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:367.87Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Fórmula:C11H14N4O4Pureza:99.958% - >99.99%Cor e Forma:SolidPeso molecular:266.25Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Cor e Forma:White Crystalline PowderPeso molecular:313.86Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Fórmula:C19H27N5O4·HClPureza:99.78%Cor e Forma:White To Off-White SolidPeso molecular:425.91Chlorprothixene hydrochloride
CAS:<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Fórmula:C18H18ClNS·HClPureza:99.76%Cor e Forma:White PowderPeso molecular:352.32Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White Crystalline PowderPeso molecular:341.43Talastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Fórmula:C19H21N3OPureza:98.50% - 99.44%Cor e Forma:SolidPeso molecular:307.39CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Fórmula:C15H18Cl2N4OPureza:99.5%Cor e Forma:SolidPeso molecular:341.24Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Fórmula:C10H13NO4Pureza:98.95% - 99.86%Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21hGPR91 antagonist 1
CAS:<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Fórmula:C31H23F4N3OPureza:98.89%Cor e Forma:SolidPeso molecular:529.53CD80-IN-3
CAS:<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Fórmula:C17H10FN3O3Pureza:98.08%Cor e Forma:SolidPeso molecular:323.28Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Fórmula:C19H31ClF3NO3Pureza:99.55%Cor e Forma:SolidPeso molecular:413.9Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Fórmula:C26H35NO7Pureza:98.53% - 99.43%Cor e Forma:CoaPeso molecular:473.57Dimenhydrinate
CAS:<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Filorexant
CAS:<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Fórmula:C24H25FN4O2Pureza:98.88%Cor e Forma:SolidPeso molecular:420.48Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Fórmula:C10H7KN6OPureza:98.91% - 99.63%Cor e Forma:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Cor e Forma:SolidPeso molecular:266.55Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Cor e Forma:SolidPeso molecular:296.79Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Fórmula:C4H7NO2SPureza:99.99%Cor e Forma:SolidPeso molecular:133.17Flopropione
CAS:<p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>Fórmula:C9H10O4Pureza:99.93%Cor e Forma:SolidPeso molecular:182.17Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Fórmula:C18H19N3O·HCl·2H2OPureza:99.92%Cor e Forma:White Crystal PowderPeso molecular:365.86Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:463.79Adrenalone hydrochloride
CAS:<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Fórmula:C9H11NO3·HClPureza:99.94%Cor e Forma:SolidPeso molecular:217.65Ro 10-5824 dihydrochloride
CAS:<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Fórmula:C17H22Cl2N4Pureza:99.79%Cor e Forma:SolidPeso molecular:353.29Fluoxetine hydrochloride
CAS:<p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Cor e Forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Fórmula:C31H38N2OPureza:97.49%Cor e Forma:SolidPeso molecular:454.65Sergliflozin A
CAS:<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Fórmula:C20H24O7Pureza:99.43%Cor e Forma:SolidPeso molecular:376.4Gevotroline
CAS:<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Fórmula:C19H20FN3Pureza:98.65%Cor e Forma:SolidPeso molecular:309.38Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Cor e Forma:White To Off-White SolidPeso molecular:525.59DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Fórmula:C22H20Cl2N4OSPureza:99.95%Cor e Forma:SoildPeso molecular:459.39Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Fórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:434.41Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Fórmula:C59H79N15O21S6Pureza:97.93% - 98.71%Cor e Forma:SolidPeso molecular:1526.74Silodosin
CAS:<p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Cor e Forma:Colorless To Pink SolidPeso molecular:495.53Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Fórmula:C12H17Cl2NOPureza:99.38%Cor e Forma:SolidPeso molecular:262.18Metaproterenol hemisulfate
CAS:<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Cor e Forma:SolidPeso molecular:260.3JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Fórmula:C11H19N5Pureza:98.33% - 99.62%Cor e Forma:SolidPeso molecular:221.3Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Fórmula:C13H16N2Pureza:97.85% - 99.77%Cor e Forma:SolidPeso molecular:200.28SR59230A
CAS:<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Fórmula:C23H29NO6Pureza:98.84%Cor e Forma:SolidPeso molecular:415.48Pranazepide
CAS:<p>Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.</p>Fórmula:C26H19FN4O2Pureza:97.43% - 99.53%Cor e Forma:SolidPeso molecular:438.45AVN 322 free base
CAS:<p>AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.</p>Fórmula:C17H19N5O2SPureza:99.24%Cor e Forma:SolidPeso molecular:357.43Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Fórmula:C22H23ClN2O2Pureza:99.71% - 99.98%Cor e Forma:White PowderPeso molecular:382.88Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Fórmula:C21H23N3OSPureza:99.61%Cor e Forma:SolidPeso molecular:365.49Rebamipide
CAS:<p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>Fórmula:C19H15ClN2O4Pureza:99.48% - 99.61%Cor e Forma:White PowderPeso molecular:370.79Midodrine hydrochloride
CAS:<p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>Fórmula:C12H19ClN2O4Pureza:99.79% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:290.74ML-109
CAS:<p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>Fórmula:C31H29N3O5Pureza:98.63%Cor e Forma:SolidPeso molecular:523.58Azelastine hydrochloride
CAS:<p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>Fórmula:C22H24ClN3O·HClPureza:98% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:418.36Iobenguane sulfate
CAS:<p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>Fórmula:C8H10IN3H2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:324.12Terbutaline
CAS:<p>Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol</p>Fórmula:C12H19NO3Pureza:99.12%Cor e Forma:SolidPeso molecular:225.3Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Fórmula:C30H32ClN3O8SPureza:98.46% - 99.89%Cor e Forma:SolidPeso molecular:630.11Sarizotan 2HCl
CAS:<p>Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.</p>Fórmula:C22H23Cl2FN2OPureza:98.83%Cor e Forma:SoildPeso molecular:421.34Delequamine
CAS:<p>Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.</p>Fórmula:C18H26N2O3SPureza:99.39%Cor e Forma:SolidPeso molecular:350.48Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Fórmula:C24H27FN2O4Pureza:99.42%Cor e Forma:SolidPeso molecular:426.48Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Fórmula:C21H24N4O2SPureza:99.64%Cor e Forma:Light Yellow To Yellow SolidPeso molecular:396.51Sertraline hydrochloride
CAS:<p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>Fórmula:C17H18Cl3NPureza:99.12% - 99.89%Cor e Forma:Solid PowderPeso molecular:342.691Aripiprazole Lauroxil
CAS:<p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>Fórmula:C36H51Cl2N3O4Pureza:99.64%Cor e Forma:SolidPeso molecular:660.71RS 15385-198
CAS:<p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>Fórmula:C18H26N2O3SPureza:>99.99%Cor e Forma:SoildPeso molecular:350.48Olopatadine hydrochloride
CAS:<p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>Fórmula:C21H23NO3·HClPureza:99.62% - 99.64%Cor e Forma:White SolidPeso molecular:373.87Balovaptan
CAS:<p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>Fórmula:C22H24ClN5OPureza:99.88%Cor e Forma:SolidPeso molecular:409.91Tolnaftate
CAS:<p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>Fórmula:C19H17NOSPureza:98.85%Cor e Forma:White PowderPeso molecular:307.412',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Fórmula:C10H13N5O2Pureza:99.55%Cor e Forma:White SolidPeso molecular:235.24INCB-9471
CAS:<p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>Fórmula:C30H40F3N5O2Pureza:98.80%Cor e Forma:SolidPeso molecular:559.666Mirtazapine
CAS:<p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>Fórmula:C17H19N3Pureza:99.98%Cor e Forma:SolidPeso molecular:265.35Pheniramine maleate
CAS:<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Fórmula:C16H20N2·C4H4O4Pureza:99.85%Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Bromperidol
CAS:<p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>Fórmula:C21H23BrFNO2Pureza:99.89%Cor e Forma:Tan SolidPeso molecular:420.32(R)-Terazosin
CAS:<p>R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).</p>Fórmula:C19H25N5O4Pureza:98.87% - 98.96%Cor e Forma:SolidPeso molecular:387.43Paroxetine hydrochloride
CAS:<p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>Fórmula:C19H21ClFNO3Pureza:98% - 99.99%Cor e Forma:White Crystalline PowderPeso molecular:365.826Tegaserod maleate
CAS:<p>Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.</p>Fórmula:C20H27N5O5Pureza:98% - 99.06%Cor e Forma:White PowderPeso molecular:417.46Moxonidine
CAS:<p>Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.</p>Fórmula:C9H12ClN5OPureza:99.81% - 99.94%Cor e Forma:CrystalPeso molecular:241.68Risperidone
CAS:<p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>Fórmula:C23H27FN4O2Pureza:99.73%Cor e Forma:Crystalline SolidPeso molecular:410.48Doxepin hydrochloride
CAS:<p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>Fórmula:C19H22ClNOPureza:99.65% - 99.91%Cor e Forma:White To Off-White PowderPeso molecular:315.84AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Fórmula:C23H22N8OPureza:98.09% - >99.99%Cor e Forma:SolidPeso molecular:426.47Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Fórmula:C24H26N2O2Pureza:98.88% - 99.68%Cor e Forma:SolidPeso molecular:374.48Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Fórmula:C23H23NO5SPureza:99.25% - 99.73%Cor e Forma:SolidPeso molecular:425.50Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Fórmula:C15H24N2O4S·HClPureza:99.4% - 99.77%Cor e Forma:SolidPeso molecular:364.89Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86JHU 75528
CAS:<p>JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.</p>Fórmula:C23H21Cl2N5O2Pureza:99.79%Cor e Forma:SolidPeso molecular:470.35Tabernanthalog fumarate
CAS:<p>Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.</p>Fórmula:C18H22N2O5Pureza:99.83%Cor e Forma:SoildPeso molecular:346.38Lesopitron HCl
CAS:<p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>Fórmula:C15H22Cl2N6Pureza:97.05% - 99.89%Cor e Forma:SoildPeso molecular:357.28Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Fórmula:C10H16N6SPureza:99.82%Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecular:252.34Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Fórmula:C21H26NO10PPureza:95.63%Cor e Forma:SoildPeso molecular:483.41Maprotiline hydrochloride
CAS:<p>Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.</p>Fórmula:C20H24ClNPureza:99.68% - 99.84%Cor e Forma:White PowderPeso molecular:313.864Quipazine dimaleate
CAS:<p>Quipazine dimaleate is a selective 5-HT3 agonist.</p>Fórmula:C21H23N3O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:445.42p-MPPI hydrochloride
CAS:<p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>Fórmula:C25H28ClIN4O2Pureza:99.95%Cor e Forma:SolidPeso molecular:578.87Amylin, amide, human
CAS:<p>Amylin, amide, human(DAP Amide) is a 37-amino acid peptide hormone co-secreted with insulin to regulate postprandial glucose levels.</p>Fórmula:C165H261N51O55S2Pureza:98%Cor e Forma:SolidPeso molecular:3903.28EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Fórmula:C23H26N4O4SPureza:99.11%Cor e Forma:SolidPeso molecular:454.54Bucumolol
CAS:<p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>Fórmula:C17H23NO4Pureza:99.66%Cor e Forma:SoildPeso molecular:305.37Ozagrel
CAS:<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Fórmula:C13H12N2O2Pureza:97.90% - 99.38%Cor e Forma:White PowderPeso molecular:228.25CI 169369
CAS:<p>CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.</p>Fórmula:C19H21ClN2SPureza:98.97%Cor e Forma:SoildPeso molecular:344.9MRGPRX1 agonist 1
CAS:<p>MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).</p>Fórmula:C23H21N3O4SPureza:99.95%Cor e Forma:SolidPeso molecular:435.5Cloroperone
CAS:<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Fórmula:C22H23ClFNO2Pureza:98.40%Cor e Forma:SoildPeso molecular:387.88Roluperidone
CAS:<p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>Fórmula:C22H23FN2O2Pureza:96.46% - 97.77%Cor e Forma:SolidPeso molecular:366.43Promethazine
CAS:<p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>Fórmula:C17H20N2SPureza:99.76%Cor e Forma:CrystalsPeso molecular:284.42Labetalol
CAS:<p>Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.</p>Fórmula:C19H24N2O3Pureza:99.87% - 99.89%Cor e Forma:SolidPeso molecular:328.41Nepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Fórmula:C15H14N2O2Pureza:98.94% - 99.43%Cor e Forma:SolidPeso molecular:254.28PIT
CAS:<p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>Fórmula:C20H16N2O5SPureza:98.63%Cor e Forma:SolidPeso molecular:396.42REV 5901A
CAS:<p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>Fórmula:C22H26ClNO2Pureza:98.04%Cor e Forma:SoildPeso molecular:371.90Glycerol phenylbutyrate
CAS:<p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>Fórmula:C33H38O6Pureza:98.54% - 99.74%Cor e Forma:SolidPeso molecular:530.65RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Fórmula:C21H22ClF3N2O2Pureza:98.95%Cor e Forma:SolidPeso molecular:426.86CCR2-RA-[R]
CAS:<p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>Fórmula:C18H19ClFNO3Pureza:99.7%Cor e Forma:SolidPeso molecular:351.8N6-Ethyladenosine
CAS:<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Fórmula:C12H17N5O4Pureza:99.96%Cor e Forma:SolidPeso molecular:295.29SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Fórmula:C9H14ClNOSPureza:99.86% - 99.99%Cor e Forma:SolidPeso molecular:219.73NS-2028
CAS:<p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>Fórmula:C9H5BrN2O3Pureza:99.44%Cor e Forma:A Crystalline SolidPeso molecular:269.05Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Fórmula:C17H21NO3·HClPureza:99% - 99.52%Cor e Forma:SolidPeso molecular:323.82Dazmegrel HCl
<p>Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.</p>Fórmula:C16H18ClN3O2Pureza:98.30%Cor e Forma:SolidPeso molecular:319.79(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Fórmula:C20H29N3O8Pureza:99.72%Cor e Forma:SoildPeso molecular:439.46Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Fórmula:C22H24ClN5O2Pureza:98% - 99.82%Cor e Forma:SolidPeso molecular:425.91GTS-21 dihydrochloride
CAS:<p>GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.</p>Fórmula:C19H20N2O2·2HClPureza:98.54% - >99.99%Cor e Forma:SolidPeso molecular:381.3Methoxamine hydrochloride
CAS:<p>Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.</p>Fórmula:C11H18ClNO3Pureza:99.84% - >99.99%Cor e Forma:Colorless Or White Plate-Like Crystals Or White Crystalline Powder SolidPeso molecular:247.719Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Fórmula:C16H15FN6OSPureza:98.62% - 99.7%Cor e Forma:SolidPeso molecular:358.39PF-04995274
CAS:<p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>Fórmula:C23H32N2O6Pureza:99.52%Cor e Forma:SolidPeso molecular:432.51Somatostatin acetate
<p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>Pureza:99.11%Cor e Forma:Odour SolidLamotrigine
CAS:<p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>Fórmula:C9H7Cl2N5Pureza:99.76% - 99.95%Cor e Forma:White To Pale Cream-Colored Powder Crystals From Isopropanol SolidPeso molecular:256.09Itopride hydrochloride
CAS:<p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>Fórmula:C20H27ClN2O4Pureza:99.59%Cor e Forma:White Or Pale Brownish CrystalPeso molecular:394.9Sulpiride
CAS:<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Fórmula:C15H23N3O4SPureza:99.94%Cor e Forma:White Crystalline PowderPeso molecular:341.43Triprolidine hydrochloride monohydrate
CAS:<p>Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.</p>Fórmula:C19H25ClN2OPureza:99.68% - 99.81%Cor e Forma:White Crystalline PowderPeso molecular:332.87Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Fórmula:C22H24ClN3O5Pureza:99.69%Cor e Forma:White To Of-White SolidPeso molecular:445.9Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Fórmula:C84H107ClN18O18Pureza:98.66%Cor e Forma:SolidPeso molecular:1692.34BIBO3304 TFA
CAS:<p>BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).</p>Fórmula:C31H36F3N7O5Pureza:99.5%Cor e Forma:SolidPeso molecular:643.66Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Fórmula:C22H28Cl2F3N3OSPureza:99.23%Cor e Forma:Off-White SolidPeso molecular:510.44MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Fórmula:C24H26F3N3O4Pureza:99.98%Cor e Forma:SolidPeso molecular:477.48Retatrutide sodium salt
<p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>Pureza:99.97%Cor e Forma:SoildCE3F4
CAS:<p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>Fórmula:C11H10Br2FNOPureza:97.15% - 98.06%Cor e Forma:SolidPeso molecular:351.01CCX140
CAS:<p>CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.</p>Fórmula:C20H13ClF3N5O3SPureza:99.66% - 99.95%Cor e Forma:SolidPeso molecular:495.86Tipepidine hydrochloride
CAS:<p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>Fórmula:C15H18ClNS2Pureza:99.97%Cor e Forma:SolidPeso molecular:311.89Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Fórmula:C26H28Cl2F2N2Pureza:99.53% - 99.89%Cor e Forma:White Crystalline Powder Odorless And TastelessPeso molecular:477.42JP1302 dihydrochloride
CAS:<p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>Fórmula:C24H26Cl2N4Pureza:99.61%Cor e Forma:SolidPeso molecular:441.4Pizotifen Malate
CAS:<p>Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.</p>Fórmula:C19H21NS·C4H6O5Pureza:>99.99%Cor e Forma:SolidPeso molecular:429.53Buflomedil hydrochloride
CAS:<p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>Fórmula:C17H26ClNO4Pureza:99.7% - 99.91%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:343.85Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Fórmula:C16H24N2O2·HClPureza:99% - 99.99%Cor e Forma:SolidPeso molecular:312.84Azasetron hydrochloride
CAS:<p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>Fórmula:C17H20ClN3O3·HClPureza:99.50%Cor e Forma:SolidPeso molecular:386.27Vibozilimod
CAS:<p>Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .</p>Fórmula:C29H36ClN3O5Pureza:99.97%Cor e Forma:SolidPeso molecular:542.07Dexchlorpheniramine Maleate
CAS:<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Fórmula:C20H23ClN2O4Pureza:99.58%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:390.86Clozapine
CAS:<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Fórmula:C18H19ClN4Pureza:99.91% - 99.93%Cor e Forma:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecular:326.82Sumatriptan succinate
CAS:<p>Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.</p>Fórmula:C18H27N3O6SPureza:97.53% - 99.51%Cor e Forma:White PowderPeso molecular:413.49Ebalzotan
CAS:<p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>Fórmula:C19H30N2O2Pureza:98.09% - 99.41%Cor e Forma:SolidPeso molecular:318.45BMY 25368 HCl
CAS:<p>BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.</p>Fórmula:C19H26ClN3O3Pureza:98.73% - 99.81%Cor e Forma:SoildPeso molecular:379.88Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Fórmula:C24H29ClF3N5O5SPureza:96.56%Cor e Forma:SoildPeso molecular:592.03Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:99.32% - >99.99%Cor e Forma:White Crystalline SolidPeso molecular:883.09CB1 antagonist 2
CAS:<p>CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.</p>Fórmula:C17H12Cl3N3OPureza:99.75%Cor e Forma:SolidPeso molecular:380.66DF-1012 FA
<p>DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.</p>Fórmula:C17H22N4O3Pureza:99.15% - 99.97%Cor e Forma:SolidPeso molecular:330.382CYM50308
CAS:<p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>Fórmula:C20H21F2N3O2SPureza:99.43% - 99.77%Cor e Forma:SolidPeso molecular:405.46Strontium ranelate
CAS:<p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>Fórmula:C12H6N2O8S·2SrPureza:98.97%Cor e Forma:Crystalline SolidPeso molecular:513.49Chlorpheniramine maleate
CAS:<p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>Fórmula:C20H23ClN2O4Pureza:99.64% - 99.98%Cor e Forma:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecular:390.87Duloxetine hydrochloride
CAS:<p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>Fórmula:C18H20ClNOSPureza:99.93% - >99.99%Cor e Forma:White Or White Crystalline PowderPeso molecular:333.88Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Fórmula:C18H23Cl2NOPureza:98.04% - >99.99%Cor e Forma:Antihypertensive DrugPeso molecular:340.3J-113863
CAS:<p>J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).</p>Fórmula:C30H37Cl2IN2O2Pureza:95.11%Cor e Forma:SolidPeso molecular:655.44Latozinemab
<p>Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:146.28 kDaNaftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Fórmula:C21H22ClNPureza:98.75% - 99.84%Cor e Forma:SolidPeso molecular:323.86Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Fórmula:C20H24ClNPureza:97% - 99.94%Cor e Forma:Crystals White To Off-White PowderPeso molecular:313.86SBI-477
CAS:<p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>Fórmula:C24H25N3O6SPureza:99.3%Cor e Forma:SolidPeso molecular:483.54Avexitide acetate
CAS:<p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>Fórmula:C155H246N40O53SPureza:96.64% - 98.65%Cor e Forma:SolidPeso molecular:3549.91Trimipramine maleate
CAS:<p>Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.</p>Fórmula:C24H30N2O4Pureza:99.47%Cor e Forma:SolidPeso molecular:410.516-Iodopravadoline
CAS:<p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>Fórmula:C23H25IN2O3Pureza:99.29%Cor e Forma:Off-White SolidPeso molecular:504.36Tryptamine hydrochloride
CAS:<p>Tryptamine hydrochloride is a monoamine alkaloid, metabolite of tryptophan and CNS active substance, agonist of 5-HT4 receptor, TAAR1, AHR.</p>Fórmula:C10H13ClN2Pureza:99.89%Cor e Forma:SolidPeso molecular:196.68Apelin-12 acetate
<p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>Fórmula:C66H107N21O16SPureza:98.82%Cor e Forma:SolidPeso molecular:1482.75Gulgafafusp alfa
CAS:<p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>Cor e Forma:LiquidPSB-22269
<p>PSB-22269 is identified as a GPR17 antagonist with a Ki value of 8.91 nM. It exhibits significant inhibitory effects in cAMP and G protein activation assays. Molecular docking studies indicate that the binding site of PSB-22269 includes positively charged arginine residues and a hydrophobic pocket. PSB-22269 promotes myelin regeneration strategies, offering potential for multiple sclerosis research.</p>Fórmula:C26H21NO6Cor e Forma:SolidPeso molecular:443.45PACAP-related Peptide (human) (trifluoroacetate salt)
<p>Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some VIP tumors; secreted by CHO-K1 cells.</p>Cor e Forma:LiquidBAM(8-22)
CAS:<p>Potent MRGPRX1 agonist peptide; first found in bovine adrenal glands. Non-opioid, lacking met-enkephalin motif. EC50: 8-150 nM.</p>Fórmula:C91H127N25O23SPureza:98%Cor e Forma:SolidPeso molecular:1971.22Mitemcinal fumarate
CAS:<p>Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.</p>Fórmula:C84H142N2O28Cor e Forma:SolidPeso molecular:1628.02PACAP (1-38) free acid
CAS:<p>PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.</p>Cor e Forma:SolidParstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Fórmula:C191H330N64O53S3Pureza:98%Cor e Forma:SolidPeso molecular:4467.29Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Fórmula:C49H68N18O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1117.31HPP-9
<p>HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET</p>Fórmula:C49H52N6O11Cor e Forma:SolidPeso molecular:900.97Oxaprotiline hydrochloride
CAS:<p>Oxaprotiline hydrochloride is an antidepressant.</p>Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86Mosliciguat
CAS:<p>Mosliciguat is a guanylate cyclase activator.</p>Fórmula:C41H36ClF3N2O5Cor e Forma:SolidPeso molecular:729.19Substance P (4-11)
CAS:<p>Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.</p>Fórmula:C46H67N11O10SCor e Forma:SolidPeso molecular:966.16Stressin I
<p>Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.</p>Fórmula:C203H337N57O56Pureza:98%Cor e Forma:SolidPeso molecular:4472.24

