GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.946 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5360 produtos de "GPCR/Proteína-G"
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Tirzepatide TFA
<p>Tirzepatide TFA, a GIP and GLP-1 agonist, targets type 2 diabetes treatment.</p>Fórmula:C227H349F3N48O70Cor e Forma:SolidPeso molecular:4927.47AC 187 TFA
<p>AC 187 TFA, a potent and orally active amylin receptor antagonist, exhibits an IC50 of 0.48 nM and a Ki of 0.275 nM.</p>Fórmula:C129H206F3N37O42Cor e Forma:SolidPeso molecular:3004.27Misoprostol acid
CAS:<p>Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.</p>Fórmula:C21H36O5Pureza:98%Cor e Forma:SolidPeso molecular:368.51Neurokinin B
CAS:<p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>Fórmula:C55H79N13O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1210.42[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Fórmula:C74H112N22O18SPureza:98%Cor e Forma:SolidPeso molecular:1629.88OXA(17-33) TFA
<p>OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).</p>Fórmula:C81H126F3N23O24Cor e Forma:SolidPeso molecular:1863Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:<p>Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent</p>Fórmula:C45H63N15O11S2Cor e Forma:SolidPeso molecular:1054.21CCR6 antagonist 1
CAS:<p>CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.</p>Fórmula:C17H12F3NO2Pureza:99.83%Cor e Forma:SoildPeso molecular:319.28Isoprenaline
CAS:<p>Isoprenaline is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.</p>Fórmula:C11H17NO3Pureza:99.31%Cor e Forma:SolidPeso molecular:211.26MLN-3897 TFA
<p>MLN-3897 TFA is a potent CCR1 antagonist that inhibits the binding of 125I-MIP-1α to THP-1 cell membranes.</p>Fórmula:C32H32ClF3N2O6Pureza:98.62%Cor e Forma:SolidPeso molecular:633.05Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:<p>Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.</p>Fórmula:C161H240N46O41S2Cor e Forma:SolidPeso molecular:3540.09LY-53857 free base
CAS:<p>LY-53857 free base is a bioactive chemical.</p>Fórmula:C23H32N2O3Cor e Forma:SolidPeso molecular:384.51Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Fórmula:C84H130F3N25O23S2Cor e Forma:SolidPeso molecular:1979.21d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Fórmula:C52H72F3N13O13S2Cor e Forma:SolidPeso molecular:1208.33MGV354
<p>MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].</p>Fórmula:C35H37N5O3Pureza:98%Cor e Forma:SolidPeso molecular:575.7(Pro34)-Peptide YY (human)
CAS:<p>(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .</p>Fórmula:C194H294N54O56Cor e Forma:SolidPeso molecular:4278.73Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Fórmula:C58H73F6N11O14S2Cor e Forma:SolidPeso molecular:1326.39Urocortin III (human)
CAS:<p>Urocortin III, a human peptide, binds CRF-R2, affecting insulin via somatostatin feedback with K i values 13.5-100+ nM.</p>Fórmula:C185H307N53O50S2Cor e Forma:SolidPeso molecular:4137.93HAEGTFTSDVS
CAS:<p>HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.</p>Fórmula:C48H71N13O20Pureza:98%Cor e Forma:SolidPeso molecular:1150.18Endothelin 1 (swine, human), Alexa Fluor 488-labeled
<p>Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.</p>Cor e Forma:SolidPeso molecular:2848.4Amylin (8-37), human
CAS:<p>Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.</p>Fórmula:C138H216N42O45Cor e Forma:SolidPeso molecular:3183.495[Ala1,3,11,15]-Endothelin
CAS:<p>Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).</p>Fórmula:C109H163N25O32SPureza:98%Cor e Forma:SolidPeso molecular:2368Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Fórmula:C184H297N69O43SPureza:98%Cor e Forma:SolidPeso molecular:4195.87Chemerin-9, Mouse
CAS:<p>Chemokine-like receptor 1 (CMKLR1) agonist (EC50 = 42 nM). Corresponds to C-terminal of full length mouse Chemerin, amino acids 148 - 156.</p>Fórmula:C51H68N10O12Cor e Forma:SolidPeso molecular:1013.163Minaprine
CAS:<p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>Fórmula:C17H22N4OPureza:98%Cor e Forma:SolidPeso molecular:298.38Cyclosomatostatin TFA
<p>Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.</p>Fórmula:C46H58F3N7O8Cor e Forma:SolidPeso molecular:893.99(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:<p>(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .</p>Fórmula:C41H57N9O10SCor e Forma:SolidPeso molecular:868.01Sauvagine TFA
<p>Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.</p>Fórmula:C204H347F3N56O65S1Cor e Forma:SolidPeso molecular:4713.33Prepro-ANF (56-92), human
CAS:<p>Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.</p>Fórmula:C173H270N44O57Cor e Forma:SolidPeso molecular:3878.26Kisspeptin-10, human TFA
<p>"Kisspeptin-10, human TFA: vasoconstrictor, angiogenesis inhibitor, metastasis suppressor via GPR54, key in kidney development & osteoblast differentiation."</p>Fórmula:C63H83N17O14·C2HF3O2Cor e Forma:SolidPeso molecular:1416.46Protease-Activated Receptor-1, PAR-1 Agonist TFA
<p>PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.</p>Cor e Forma:Liquid[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Fórmula:C67H84N16O13Cor e Forma:SolidPeso molecular:1321.48Bay 55-9837 TFA
<p>Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.</p>Fórmula:C150H240F3ClN44O44Cor e Forma:SolidPeso molecular:3456.22Neuropeptide Y (2-36) (porcine)
CAS:<p>Porcine Neuropeptide Y (2-36) is 97.14% similar to rat/human, an agonist for Y5, Y2, Y1 receptors, used in obesity research.</p>Fórmula:C181H278N54O55Cor e Forma:SolidPeso molecular:4090.47Orexin B, rat, mouse TFA
<p>Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.</p>Fórmula:C128H216F3N45O36SCor e Forma:SolidPeso molecular:3050.42PF-9184
CAS:<p>PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.</p>Fórmula:C21H14Cl2N2O4SPureza:97.43%Cor e Forma:SolidPeso molecular:461.321,8-Cineole
CAS:<p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>Fórmula:C10H18OPureza:97.44% - 97.44%Cor e Forma:SolidPeso molecular:154.25ELA-11(human)
CAS:<p>Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.</p>Fórmula:C58H90N16O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1283.57Retrobradykinin
CAS:<p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>Fórmula:C50H73N15O11Cor e Forma:SolidPeso molecular:1060.228Cenderitide
CAS:<p>Cenderitide fuses CNP with DNP, stimulates pGC-A/B, ups cGMP, curbs aldosterone, and aids GFR, not affecting BP—used in heart failure studies.</p>Fórmula:C158H263N49O50S3Cor e Forma:SolidPeso molecular:3745.27Triamterene
CAS:<p>Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.</p>Fórmula:C12H11N7Pureza:99.77%Cor e Forma:Yellow Yellow SolidPeso molecular:253.26α-CGRP(human) TFA
<p>α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a</p>Fórmula:C165H268F3N51O51S2Cor e Forma:SolidPeso molecular:3903.33Neuropeptide Y (3-36) (human, rat)
CAS:<p>Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.</p>Fórmula:C175H269N53O54SCor e Forma:SolidPeso molecular:4011.5CCR2 antagonist 1
CAS:<p>CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).</p>Fórmula:C28H32BrF3N2OCor e Forma:SolidPeso molecular:549.47Fluphenazine free base
CAS:<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Fórmula:C22H26F3N3OSCor e Forma:SolidPeso molecular:437.52Atilmotin
CAS:<p>Atilmotin is a gastrointestinal agent for treating motility disorders.</p>Fórmula:C86H135N20O19Cor e Forma:SolidPeso molecular:1753.146QWF
CAS:<p>Tripeptide SP antagonist (IC50: 90 μM); blocks SP-MRGPR X2 binding and mast cell degranulation; reduces 48/80-induced scratching in mice.</p>Fórmula:C38H43N5O8Pureza:98%Cor e Forma:SolidPeso molecular:697.78(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Fórmula:C14H22N2O3Pureza:98.72%Cor e Forma:SolidPeso molecular:266.34MM 419447
CAS:<p>MM 419447, a linaclotide metabolite, is a guanylate cyclase-C agonist showing potential in IBS-C research.</p>Fórmula:C50H70N14O19S6Cor e Forma:SolidPeso molecular:1363.55(+)-Cloprostenol sodium
CAS:<p>Cloprostenol sodium is a water-soluble PGF2α analog and FP receptor agonist, promoting luteolysis in rats and hamsters.</p>Fórmula:C22H28ClNaO6Cor e Forma:SolidPeso molecular:446.9Teprotumumab
CAS:<p>Teprotumumab: human antibody, inhibits IGF-1R, used for thyroid eye diseases.</p>Pureza:SDS-PAGE:95.2%;SEC-HPLC:99.6%Cor e Forma:LiquidPeso molecular:145.62 kDaPG-931 TFA
<p>PG-931 TFA, a potent MC4 receptor agonist (IC50 0.58 nM), excels in selectivity and helps reverse hemorrhagic shock in vivo.</p>Fórmula:C61H86F3N15O13Cor e Forma:SolidPeso molecular:1294.42Fenoldopam
CAS:<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Fórmula:C16H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:305.76A6770
CAS:<p>A6770 inhibits S1P lyase, causing [3H]dhS1P build-up in IT-79MTNC3 cells (EC50 <0.01 μM); less effective with vitamin B6 (EC50 <100 μM).</p>Fórmula:C6H8N2O2Cor e Forma:SolidPeso molecular:140.142(2R,2R)-PF-07258669
CAS:<p>(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.</p>Fórmula:C25H27FN6O2Cor e Forma:SolidPeso molecular:462.52(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
CAS:<p>(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1a</p>Fórmula:C159H267N49O43Cor e Forma:SolidPeso molecular:3553.12RFRP-1(human)
CAS:<p>Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.</p>Fórmula:C67H101N19O14SPureza:98%Cor e Forma:SolidPeso molecular:1428.72Melanostatin, frog
CAS:<p>Melanostatin, frog, is an inhibitor of α-melanocyte-stimulating hormone (α-MSH) release, with an IC50 of 60 nM [1] [2].</p>Fórmula:C189H285N53O57SCor e Forma:SolidPeso molecular:4243.67Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Fórmula:C25H31F3N6O8Pureza:98.08%Cor e Forma:SoildPeso molecular:600.55Calcitonin (8-32), salmon
CAS:<p>Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.</p>Fórmula:C119H198N36O37Pureza:98%Cor e Forma:SolidPeso molecular:2725.06D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Fórmula:C49H68F3N11O13S2Cor e Forma:SolidPeso molecular:1140.25Pancreatic Polypeptide, human
CAS:<p>Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.</p>Fórmula:C185H287N53O54S2Pureza:98%Cor e Forma:SolidPeso molecular:4181.71[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS:<p>'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.</p>Fórmula:C39H64N8O10Cor e Forma:SolidPeso molecular:804.97G-Protein antagonist peptide
CAS:<p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>Fórmula:C57H64N12O9SPureza:98%Cor e Forma:SolidPeso molecular:1093.27Pramlintide TFA
Pramlintide TFA, a polypeptide analogue of human amylin and an antidiabetic agent, exhibits antineoplastic properties in colorectal cancer [1].Fórmula:C173H268N51F3O55S2Cor e Forma:SolidPeso molecular:4063.4(±)5(6)-EET
CAS:<p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>Fórmula:C20H32O3Cor e Forma:SolidPeso molecular:320.473GB-6
CAS:<p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>Fórmula:C32H45N11O8Pureza:98%Cor e Forma:SolidPeso molecular:711.77β2AR/M-receptor agonist-1
CAS:<p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>Fórmula:C43H56BrN3O7Cor e Forma:SolidPeso molecular:806.82AGN 191976
CAS:<p>AGN 191976 is a novel thromboxane A2-mimetic.</p>Fórmula:C21H32O6Cor e Forma:SolidPeso molecular:380.481Zoliprofen
CAS:<p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.295-OMe-UDP trisodium salt
CAS:<p>Potent P2Y6 agonist</p>Fórmula:C10H16N2O13P2Pureza:98%Cor e Forma:SolidPeso molecular:434.19Osanetant
CAS:Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Fórmula:C35H41Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:606.62Peptide YY (PYY), human
CAS:<p>PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.</p>Fórmula:C194H295N55O57Pureza:98%Cor e Forma:SolidPeso molecular:4309.75Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Fórmula:C22H37NO4Cor e Forma:SolidPeso molecular:379.541Minesapride
CAS:<p>Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.</p>Fórmula:C21H31ClN4O5Pureza:99.85% - 99.88%Cor e Forma:SolidPeso molecular:454.95PAMP-12 (unmodified) (TFA)
<p>PAMP-12 (unmodified) TFA, an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine secretion</p>Fórmula:C79H119F3N24O17Cor e Forma:SolidPeso molecular:1733.94CH 275
CAS:<p>Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.</p>Fórmula:C74H96N14O15S2Pureza:98%Cor e Forma:SolidPeso molecular:1485.8Amylin (IAPP), feline TFA
<p>Amylin (IAPP), feline TFA: 37-amino acid peptide; inhibits insulin/glucagon; secreted by pancreatic β-cells.</p>Fórmula:C167H271F3N52O56S2Cor e Forma:SolidPeso molecular:4024.47Anthramycin
CAS:<p>Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.</p>Fórmula:C16H17N3O4Cor e Forma:SolidPeso molecular:315.32Dipentylone hydrochloride
CAS:<p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>Fórmula:C14H20ClNO3Pureza:99.94%Cor e Forma:SolidPeso molecular:285.77Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Fórmula:C26H47N7O9SPureza:98%Cor e Forma:SolidPeso molecular:633.76Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Fórmula:C215H358N72O66SPureza:98%Cor e Forma:SolidPeso molecular:5039.65AC-263093
CAS:<p>AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the paraventricular nucleus of the hypothalamus.</p>Fórmula:C8H8Br2N4Pureza:99.78%Cor e Forma:SoildPeso molecular:319.98Kisspeptin 234
CAS:<p>Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.</p>Fórmula:C63H78N18O13Pureza:98%Cor e Forma:SolidPeso molecular:1295.42Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29Neuropeptide Y (human)
CAS:<p>Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.</p>Fórmula:C189H285N55O57SPureza:98%Cor e Forma:SolidPeso molecular:4271.68Glucagon-like peptide 1 (1-37), human
CAS:<p>Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.</p>Fórmula:C186H275N51O59Pureza:98%Cor e Forma:SolidPeso molecular:4169.48Amylin (8-37) (human)
CAS:Amylin (8-37) (human) is a fragment of human IAPP with a hairpin structure.Fórmula:C138H215N41O46Cor e Forma:SolidPeso molecular:3184.43Alsactide
CAS:<p>Alsactide, an adrenocorticotropic hormone (ACTH) agonist and a heptadecapeptide analogue, is utilized in the study of the central nervous system [1].</p>Fórmula:C99H155N29O21SCor e Forma:SolidPeso molecular:2119.53Proglumide hemicalcium
CAS:<p>Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.</p>Fórmula:C18H28CaN2O4Pureza:98%Cor e Forma:SolidPeso molecular:376.51Obestatin(rat)
CAS:<p>Endogenous peptide that suppresses food intake and body weight-gain</p>Fórmula:C114H174N34O31Pureza:98%Cor e Forma:SolidPeso molecular:2516.81Lys-Bradykinin
CAS:<p>Endogenous bradykinin receptor agonist</p>Fórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Latanoprost lactone diol
CAS:<p>Latanoprost lactone diol, a key intermediate for synthesizing Latanoprost (a prostaglandin F2α analogue), lowers IOP by activating FP receptors.</p>Fórmula:C18H24O4Pureza:98%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:304.38Adenosine 2',5'-diphosphate sodium
CAS:<p>Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.</p>Fórmula:C10H15N5NaO10P2Cor e Forma:SolidPeso molecular:450.19217-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:<p>Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.</p>Fórmula:C27H39NO4Cor e Forma:SolidPeso molecular:441.612Glucagon receptor antagonists-1
CAS:<p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>Fórmula:C29H34FNO2Pureza:98%Cor e Forma:SolidPeso molecular:447.58Somatostatin-28 (1-14)
CAS:<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Fórmula:C61H105N23O21SPureza:98%Cor e Forma:SolidPeso molecular:1528.71T-10430
<p>T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.</p>Fórmula:C17H22N6OCor e Forma:SolidPeso molecular:326.396(+)-OSU 6162
CAS:<p>(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.</p>Fórmula:C15H23NO2SPureza:98.19%Cor e Forma:SoildPeso molecular:281.41Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Fórmula:C14H20ClN3SCor e Forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85Ilatreotide
CAS:<p>Ilatreotide is a Amadori compound of octreotide.</p>Fórmula:C61H86N10O20S2Pureza:98%Cor e Forma:SolidPeso molecular:1343.53Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Fórmula:C23H27N5O3Cor e Forma:SolidPeso molecular:421.501Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Fórmula:C258H401N79O78·C2HF3O2Cor e Forma:SolidPeso molecular:5971.45α-CGRP, rat
CAS:<p>Endogenous neuropeptide, potent vasodilator</p>Fórmula:C162H262N50O52S2Pureza:98%Cor e Forma:SolidPeso molecular:3806.25Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Fórmula:C21H26Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:433.4Lobeline sulfate
CAS:<p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>Fórmula:C22H29NO6SPureza:98%Cor e Forma:White PowderPeso molecular:435.54CRF(6-33)(human)
CAS:<p>CRFBP inhibitor peptide; blocks CRF, reduces weight gain, boosts activity in obese rats.</p>Fórmula:C141H231N41O43SPureza:98%Cor e Forma:SolidPeso molecular:3220.68Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:<p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Fórmula:C162H267N51O48S3Pureza:98%Cor e Forma:SolidPeso molecular:3793.41Hemokinin 1 (mouse)
CAS:<p>Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.</p>Fórmula:C61H100N22O15SPureza:98%Cor e Forma:White PowderPeso molecular:1413.65Etelcalcetide
CAS:<p>Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.</p>Fórmula:C38H73N21O10S2Pureza:98%Cor e Forma:SolidPeso molecular:1048.26BMS-604992 dihydrochloride
CAS:<p>BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.</p>Fórmula:C24H33Cl2N7O5Cor e Forma:SolidPeso molecular:570.47Cinnamtannin A2
CAS:<p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>Fórmula:C60H50O24Cor e Forma:SolidPeso molecular:1155.02PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44PAMP-12 (unmodified)
CAS:<p>PAMP-12 (unmodified), an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine release from</p>Fórmula:C77H118N24O15Cor e Forma:SolidPeso molecular:1619.91Adrenotensin (human)
CAS:<p>Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.</p>Fórmula:C143H224N42O43Cor e Forma:SolidPeso molecular:3219.56(S, R)-LSN 3318839
CAS:<p>(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.</p>Fórmula:C26H23Cl2N3O2Pureza:99.57%Cor e Forma:SoildPeso molecular:480.39ELA-21 (human)
CAS:<p>Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.</p>Fórmula:C112H184N40O25S3Pureza:98%Cor e Forma:SolidPeso molecular:2587.12Angiopeptin
CAS:<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Fórmula:C54H71N11O10S2Cor e Forma:SolidPeso molecular:1098.34ZL-1101
<p>ZL-1101 is a human monoclonal antibody (mAb) targeting TNFRSF4/OX40/CD134.</p>Cor e Forma:Odour LiquidLys-[Hyp3]-Bradykinin
CAS:<p>Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.</p>Fórmula:C56H85N17O13Cor e Forma:SolidPeso molecular:1204.38Amylin (8-37), rat
CAS:<p>Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.</p>Fórmula:C140H227N43O43Pureza:98%Cor e Forma:SolidPeso molecular:3200.61Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide
<p>Biotin-labeled GLP-1-(7-36) amide; a gut peptide that enhances insulin release.</p>Fórmula:C165H252N44O48SCor e Forma:SolidPeso molecular:3652.1LU AA33810
CAS:<p>LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Fórmula:C19H25N3O2S3Pureza:98%Cor e Forma:SolidPeso molecular:423.62Cyclic SSTR agonist octreotide
<p>Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .</p>Fórmula:C53H71N11O14S2Cor e Forma:SolidPeso molecular:1150.33{Val1}-Exendin-3/4
<p>{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.</p>Fórmula:NAPureza:98%Cor e Forma:SolidPeso molecular:3241.7(R)-CJ 11974
CAS:<p>(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.</p>Fórmula:C31H38N2OPureza:97.15%Cor e Forma:SoildPeso molecular:454.65A71378
CAS:<p>A71378 is a high potency, selectivity CCK-A receptors agonist.</p>Fórmula:C48H62N8O13SPureza:98%Cor e Forma:SolidPeso molecular:991.12TAK-683 acetate
<p>TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.</p>Fórmula:C66H87N17O15Cor e Forma:SolidPeso molecular:1358.5IRL-3630
CAS:<p>IRL 3460 is an enantiomer.</p>Fórmula:C31H40N4O6SPureza:98%Cor e Forma:SolidPeso molecular:596.74OXA(17-33)
CAS:<p>Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.</p>Fórmula:C79H125N23O22Pureza:98%Cor e Forma:SolidPeso molecular:1749Chemerin-9 (149-157) TFA
<p>Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.</p>Fórmula:C56H67F3N10O15Pureza:99.77%Cor e Forma:SolidPeso molecular:1177.18Galanin (1-30), human
CAS:Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Fórmula:C139H210N42O43Pureza:98%Cor e Forma:SolidPeso molecular:3157.46Enuvaptan
CAS:<p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>Fórmula:C21H15ClF6N8O3Cor e Forma:SolidPeso molecular:576.84I-BOP
CAS:<p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>Fórmula:C23H29IO5Cor e Forma:SolidPeso molecular:512.384CAP-100
<p>CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).</p>Cor e Forma:Odour Liquid16-phenoxy tetranor Prostaglandin F2α methyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Fórmula:C23H32O6Cor e Forma:SolidPeso molecular:404.503NF157
CAS:<p>NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.</p>Fórmula:C49H28F2N6Na6O23S6Pureza:98%Cor e Forma:SolidPeso molecular:1437.1Baloncibart
CAS:<p>Baloncibart is a human IgG4K monoclonal antibody that targets NPR1.</p>Cor e Forma:LiquidIRAK inhibitor 4 trans
<p>IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.</p>Fórmula:C33H35F3N6O3Pureza:98%Cor e Forma:SolidPeso molecular:620.66Biotin-NeurokininA
<p>Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.</p>Fórmula:C60H94N16O16S2Cor e Forma:SolidPeso molecular:1359.61Tirzepatide hydrochloride
<p>Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.</p>Fórmula:C225H349N48O68ClPureza:98%Cor e Forma:SolidPeso molecular:4849.91(Iso)-RJW100
CAS:<p>Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).</p>Fórmula:C28H34OPureza:99.79%Cor e Forma:SoildPeso molecular:386.57Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Cor e Forma:SolidPeso molecular:926.09Parstatin(mouse)
CAS:<p>Peptide inhibits endothelial migration/proliferation (IC50 ~20μM), induces cell cycle arrest, triggers apoptosis, and has cardioprotective effects.</p>Fórmula:C189H326N58O57S3Pureza:98%Cor e Forma:SolidPeso molecular:4419.19[Arg-15,20,21,Leu17]-PACAP-Gly-Lys-Arg-NH2
CAS:<p>[Arg-15,-20,-21, Leu17]-PACAP-Gly-Lys-Arg-NH2 (BM-PACAP) is a synthetic analogue of PACAP 1-27 that exhibits a relaxant effect [1].</p>Fórmula:C157H253N53O42Cor e Forma:SolidPeso molecular:3555.02Zalospirone
CAS:<p>Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.</p>Fórmula:C24H29N5O2Pureza:98.41% - 99.82%Cor e Forma:SolidPeso molecular:419.52Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:<p>LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.</p>Fórmula:C60H73N15O13Pureza:98%Cor e Forma:SolidPeso molecular:1212.31Bombinakinin M
CAS:<p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>Fórmula:C100H159N31O24Pureza:98%Cor e Forma:SolidPeso molecular:2179.55GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Fórmula:C165H254N44O55SPureza:98%Cor e Forma:SolidPeso molecular:3766.19Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Cor e Forma:Odour SolidLAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Fórmula:C39H43ClN4O9S2Cor e Forma:SolidPeso molecular:811.36ELA-11(human) TFA
<p>ELA-11(human) TFA: apelin receptor agonist, K i =14 nM, inhibits cAMP, stimulates β-arrestin, from ELA-32 fragment.</p>Fórmula:C60H91F3N16O15S2Cor e Forma:SolidPeso molecular:1397.58ANXA3 degrader 1
<p>ANXA3 degrader 1 (Compound 18a5) is a highly selective ANXA3 degrader with activity against cancer cells. It demonstrates significant inhibitory effects in a triple-negative breast cancer (TNBC) tumor xenograft model, with a tumor growth inhibition (TGI) rate of 96%.</p>Fórmula:C30H32N6O2S2Cor e Forma:SolidPeso molecular:572.74Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Fórmula:C16H28N6O4Pureza:98%Cor e Forma:SolidPeso molecular:368.43Galcanezumab
CAS:<p>Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:144.08 kDaCYN 154806
CAS:<p>CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).</p>Fórmula:C56H68N12O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1197.34Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Fórmula:C24H21N5O5SCor e Forma:SolidPeso molecular:491.52Cianopramine hydrochloride
CAS:<p>Cianopramine hydrochloride is a bio-active chemical.</p>Fórmula:C20H24ClN3Cor e Forma:SolidPeso molecular:341.88Bombinakinin M acetate
<p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>Fórmula:C102H163N31O26Pureza:99.80%Cor e Forma:SolidPeso molecular:2239.58HPP-9
<p>HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET</p>Fórmula:C49H52N6O11Cor e Forma:SolidPeso molecular:900.9712-epi Leukotriene B4
CAS:<p>LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.472Tetrahydro-β-carboline
CAS:<p>Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C11H12N2Pureza:96.31%Cor e Forma:Tan SolidPeso molecular:172.2264Guanylin(human)
CAS:<p>Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.</p>Fórmula:C58H87N15O21S4Pureza:98%Cor e Forma:SolidPeso molecular:1458.65HAEGTFTSD
CAS:<p>HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.</p>Fórmula:C40H57N11O17Pureza:98%Cor e Forma:SolidPeso molecular:963.94Prostaglandin H1
CAS:<p>Prostaglandin H1 is the cyclooxygenase metabolite of DGLA, a CRTh2 agonist and a precursor of a family of 1 anti-inflammatory prostaglandins.</p>Fórmula:C20H34O5Cor e Forma:SolidPeso molecular:354.487Exendin-4 (3-39)
CAS:<p>Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.</p>Fórmula:C176H272N46O58SCor e Forma:SolidPeso molecular:3992.44CKLF1-C27 TFA
<p>CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.</p>Fórmula:C153H244F3N39O39Cor e Forma:SolidPeso molecular:3310.8[Asu1,6-Arg8]Vasopressin
CAS:<p>[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.</p>Fórmula:C48H68N14O12Cor e Forma:SolidPeso molecular:1033.14M40
CAS:<p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>Fórmula:C94H145N23O24Pureza:98%Cor e Forma:SolidPeso molecular:1981.33Sarafotoxin S6c
CAS:<p>Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).</p>Fórmula:C103H147N27O37S5Pureza:98%Cor e Forma:SolidPeso molecular:2516Adrenomedullin (AM) (22-52), human TFA
<p>Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.</p>Fórmula:C161H253N46F3O50Pureza:98%Cor e Forma:SolidPeso molecular:3690.06HAEGTFT
CAS:<p>HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C33H47N9O12Pureza:98%Cor e Forma:SolidPeso molecular:761.78Orexin A (human, rat, mouse)
CAS:<p>Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.</p>Fórmula:C152H243N47O44S4Pureza:98%Cor e Forma:SolidPeso molecular:3561.1SB-408124
CAS:<p>SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x more selective than OX2.</p>Fórmula:C19H18F2N4OPureza:99.81%Cor e Forma:SolidPeso molecular:356.37d[Leu4,Lys8]-VP acetate
<p>d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.</p>Fórmula:C49H71N11O13S2Pureza:98.86%Cor e Forma:SolidPeso molecular:1086.2817-phenyl trinor Prostaglandin E2 ethyl amide
CAS:<p>17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.</p>Fórmula:C25H35NO4Cor e Forma:SolidPeso molecular:413.55(Ala13)-Apelin-13
CAS:<p>(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.</p>Fórmula:C63H107N23O16SPureza:98%Cor e Forma:SolidPeso molecular:1474.75Vapitadine
CAS:<p>Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.</p>Fórmula:C17H20N4OPureza:99.77% - 99.86%Cor e Forma:SoildPeso molecular:296.37Apraglutide
CAS:<p>Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.</p>Fórmula:C172H263N43O52Pureza:98%Cor e Forma:SolidPeso molecular:3765.25Picumeterol FA
<p>picumeterol FA is a potent and selective β2-adrenergic receptor agonist.</p>Fórmula:C22H31Cl2N3O4Pureza:99.8%Cor e Forma:SoildPeso molecular:472.4Imipramine N-oxide
CAS:<p>Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.</p>Fórmula:C19H24N2OPureza:99.80%Cor e Forma:SolidPeso molecular:296.41Dexbrompheniramine maleate
CAS:<p>Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.</p>Fórmula:C20H23BrN2O4Cor e Forma:SolidPeso molecular:435.318SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Fórmula:C54H71N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1074.258Peptide YY (PYY) (3-36), porcine TFA
<p>Peptide YY (PYY) (3-36), porcine TFA, functions as a gut hormone that serves as a Y2 receptor agonist, effectively reducing appetite [1].</p>Fórmula:C176H272N52O54·C2HF3O2Cor e Forma:SolidPeso molecular:4094.44Acetyl-Amylin (8-37) (human)
CAS:<p>Acetyl-Amylin (8-37) (human) is a specific amylin antagonist [1] .</p>Fórmula:C140H218N42O46Cor e Forma:SolidPeso molecular:3225.48GLP-1(9-36)amide TFA
<p>GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.</p>Fórmula:C142H215F3N36O45Cor e Forma:SolidPeso molecular:3203.43Cortistatin-8
CAS:<p>ghrelin receptor antagonist</p>Fórmula:C47H68N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1009.25TGR5 agonist 1
<p>Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].</p>Fórmula:C28H48NNaO6SCor e Forma:SolidPeso molecular:549.74AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211Naratriptan D3 Hydrochloride
CAS:<p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>Fórmula:C17H26ClN3O2SPureza:98%Cor e Forma:SolidPeso molecular:374.94LTB4-IN-2
<p>LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with an</p>Fórmula:C24H17N5S2Pureza:98%Cor e Forma:SolidPeso molecular:439.56Amylin (IAPP), feline
<p>Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.</p>Fórmula:C165H270N52O54S2Pureza:98%Cor e Forma:SolidPeso molecular:3910.45Setmelanotide Acetate(920014-72-8 free base)
CAS:<p>Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM</p>Fórmula:C51H72N18O11S2Pureza:99.71%Cor e Forma:SolidPeso molecular:1177.35Elabela(19-32)
CAS:<p>APJ receptor agonist with Ki of 0.93 nM, derived from ELA-32, activates Gαi1, β-arrestin-2, lowers rat heart arterial pressure, effective in vivo.</p>Fórmula:C75H119N25O17S2Pureza:98%Cor e Forma:SolidPeso molecular:1707.03HAEGTFTSDVS acetate
<p>HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.</p>Fórmula:C50H75N13O22Pureza:97.47%Cor e Forma:SolidPeso molecular:1210.2Brexpiprazole S-oxide
CAS:<p>Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).</p>Fórmula:C25H27N3O3SPureza:98%Cor e Forma:SolidPeso molecular:449.57Vanicoside E
CAS:<p>Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .</p>Fórmula:C53H52O22Cor e Forma:SolidPeso molecular:1040.97PACAP (1-38) free acid TFA
<p>PACAP (1-38) free acid TFA, an endogenous neuropeptide, effectively enhances antral motility and somatostatin secretion, while concurrently suppressing gastrin</p>Cor e Forma:Odour Solid15(R)-17-phenyl trinor Prostaglandin F2α
CAS:<p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>Fórmula:C23H32O5Cor e Forma:SolidPeso molecular:388.5
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