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Cell Cycle/Checkpoint

Cell Cycle/Checkpoint

Cell cycle/checkpoint inhibitors are compounds that disrupt the normal progression of the cell cycle, particularly at key regulatory checkpoints. These inhibitors are crucial for studying cell division, understanding cancer cell proliferation, and developing anti-cancer therapies. By targeting specific phases of the cell cycle, these inhibitors can induce cell cycle arrest, leading to apoptosis or senescence in rapidly dividing cells. At CymitQuimica, we offer a diverse range of high-quality cell cycle/checkpoint inhibitors to support your research in cancer biology, cell biology, and drug development.

Subcategories of "Cell Cycle/Checkpoint"

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Found 3675 products of "Cell Cycle/Checkpoint"

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  • USP7-IN-10
    Targetmol
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    USP7-IN-10

    CAS:
    <p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>
    Formula:C26H29ClN4O3S
    Color and Shape:Solid
    Molecular weight:513.05

    Ref: TM-T73136

  • L-2'-Fd4C
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    L-2'-Fd4C

    CAS:
    L-2'-Fd4C is an L-nucleoside analogue with both anti-human immunodeficiency virus (HIV) and anti-hepatitis B virus (HBV) activity [1].
    Formula:C9H10FN3O3
    Color and Shape:Solid
    Molecular weight:227.19

    Ref: TM-T60285

  • 12(S)-HETE
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    12(S)-HETE

    CAS:
    <p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47

    Ref: TM-T37047

  • 2′-O-MOE-CMP
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    2′-O-MOE-CMP

    CAS:
    <p>2′-O-MOE-CMP is a nucleotide analogue utilized in the synthesis of oligonucleotides.</p>
    Formula:C12H20N3O9P
    Color and Shape:Solid
    Molecular weight:381.28

    Ref: TM-TSW-00960

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    Pol I-IN-1

    Pol I-IN-1 is a powerful inhibitor of RNA polymerase I (Pol I), specifically targeting the large catalytic subunit RPA194, demonstrating an inhibition
    Formula:C23H22N4O2
    Color and Shape:Solid
    Molecular weight:386.45

    Ref: TM-T61720

  • YKL-1-116
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    YKL-1-116

    CAS:
    YKL-1-116 is an effective, selective, and covalent CDK7 inhibitor.
    Formula:C34H38N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:606.72

    Ref: TM-T24643

  • Antifolate agent 1
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    Antifolate agent 1

    CAS:
    Antifolateagent 1 (Compound 1) is an antifolate agent featuring a single-carbon bridge. It lacks RFC transport, shows no affinity for FRα and FRβ, and exhibits no GARFTase inhibition activity. Antifolateagent 1 serves as a negative control in the development of folate receptor-targeted antifolate agents.
    Formula:C19H19N5O6
    Color and Shape:Solid
    Molecular weight:413.38

    Ref: TM-T212452

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    IRE1α kinase-IN-5

    <p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>
    Formula:C28H30N6O3S
    Color and Shape:Solid
    Molecular weight:530.64

    Ref: TM-T63734

  • 3'-NH-Tr-2',3'-ddG(iBu)-5'-CE-Phosphoramidite
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    3'-NH-Tr-2',3'-ddG(iBu)-5'-CE-Phosphoramidite

    CAS:
    3'-NH-Tr-2',3'-ddG(iBu)-5'-CE-Phosphoramidite is a nucleoside phosphoramidite monomer featuring protective group modifications, suitable for RNA oligonucleotide synthesis.
    Formula:C42H51N8O5P
    Color and Shape:Solid
    Molecular weight:778.88

    Ref: TM-TSW-01143

  • Deoxythymidine-5'-triphosphate-d15
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    Deoxythymidine-5'-triphosphate-d15

    CAS:
    Deoxythymidine-5'-triphosphate-d15 (dTTP-d15) dilithium is a deuterium-labeled form of deoxythymidine-5'-triphosphate. Deoxythymidine-5'-triphosphate (dTTP) is a triphosphate nucleotide utilized in DNA synthesis.
    Formula:C10H15Li2N2O14P3
    Color and Shape:Solid
    Molecular weight:509.13

    Ref: TM-T211806

  • SCH-1473759
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    SCH-1473759

    CAS:
    SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).
    Formula:C20H26N8OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.54

    Ref: TM-T16862

  • Morpholino U subunit
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    Morpholino U subunit

    CAS:
    Morpholino U subunit is one of the fundamental components of morpholino oligonucleotides, capable of pairing with adenine in target RNA.
    Formula:C30H32ClN4O5P
    Color and Shape:Solid
    Molecular weight:595.03

    Ref: TM-TSW-01102

  • CDK4/6-IN-3
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    CDK4/6-IN-3

    CAS:
    <p>CDK4/6-IN-3 is a brain-penetrant CDK4/CDK6 inhibitor (Kis: &lt;0.3 nM and 2.2 nM) used for the treatment of glioblastoma. It inhibits CDK1 with a Ki of 110 nM.</p>
    Formula:C25H31FN8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.57

    Ref: TM-T10737

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    Hesperadin hydrochloride

    <p>Hesperadin hydrochloride is an ATP-competitive indolone inhibitor of Aurora A and B, with an IC50 value of 250 nM for Aurora B.</p>
    Formula:C29H33ClN4O3S
    Color and Shape:Solid
    Molecular weight:553.12

    Ref: TM-T63905

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    MtTMPK-IN-8

    <p>MtTMPK-IN-8 inhibits MtbTMPK, has low cytotoxicity, shows 0.78-9.4 μM activity against Mycobacterium, useful for tuberculosis research.</p>
    Formula:C24H24N6O7
    Color and Shape:Solid
    Molecular weight:508.48

    Ref: TM-T63491

  • N-Isobutyryl-2', 3'-acetyl-guanosine
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    N-Isobutyryl-2', 3'-acetyl-guanosine

    CAS:
    <p>N-Isobutyryl-2', 3'-acetyl-guanosine is a derivative of guanosine.</p>
    Formula:C18H23N5O8
    Color and Shape:Solid
    Molecular weight:437.404

    Ref: TM-T206416

  • LIMK1 inhibitor 1
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    LIMK1 inhibitor 1

    CAS:
    <p>LIMK1 inhibitor1 (compound 24) is a LIMK1 inhibitor, potentially useful for cancer research.</p>
    Formula:C12H15N3S2
    Color and Shape:Solid
    Molecular weight:265.398

    Ref: TM-T204784

  • CDK1-IN-7
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    CDK1-IN-7

    CAS:
    <p>CDK1-IN-7 (compound M7) is a potent CDK1 inhibitor. It effectively suppresses the proliferation and migration of HCT116 and Lovo cells, making it a valuable tool for colorectal cancer research.</p>
    Formula:C23H19ClN4O3
    Color and Shape:Solid
    Molecular weight:434.88

    Ref: TM-T207488

  • RNAP-σ interaction inhibitor-2
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    RNAP-σ interaction inhibitor-2

    CAS:
    RNAP-σ interaction inhibitor-2 (compound 7d) is an inhibitor targeting the interaction between RNA polymerase and the sigma factor. It demonstrates inhibitory activity against S. aureus with a minimum inhibitory concentration (MIC) of 2 µg/mL.
    Formula:C27H19Cl3N2O6S2
    Color and Shape:Solid
    Molecular weight:637.939

    Ref: TM-T206884

  • NVP-BQS481
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    NVP-BQS481

    CAS:
    NVP-BQS481 (Compound 1) is a selective inhibitor of spindle motor protein 5 (Eg5), with an IC50 of less than 0.5 nM. It demonstrates significant anti-mitotic and anti-tumor activities, exhibiting an IC50 of 0.09 nM against SK-OV-3ip cells. NVP-BQS481 is suitable for use as a cytotoxic payload in the synthesis of antibody-drug conjugates (ADCs).
    Formula:C27H33F3N4O2
    Color and Shape:Solid
    Molecular weight:502.57

    Ref: TM-T212559

  • DHICA
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    DHICA

    CAS:
    DHICA (5,6-Dihydroxyindole-2-carboxylic acid) is an intermediate in melanin synthesis and a component of eumelanin, as well as acting as a moderate potency agonist of GPR35. In the U2OS cell line, DHICA demonstrates the ability to induce β-arrestin translocation signaling with an EC50 value of 23.2 μM. Additionally, it plays a significant role in promoting and protecting against DNA damage.
    Formula:C9H7NO4
    Color and Shape:Solid
    Molecular weight:193.16

    Ref: TM-T201499

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    CDK1-IN-3

    CDK1-IN-3 is a selective inhibitor targeting CDK1 (36.8 nM), CDK2 (305.17 nM), CDK5 (369.37 nM); used in cancer research.
    Formula:C28H25ClF3N5O2
    Color and Shape:Solid
    Molecular weight:555.98

    Ref: TM-T63933

  • HNC-1664
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    HNC-1664

    CAS:
    <p>HNC-1664 is an orally active inhibitor of RNA-dependent RNA polymerase (RdRP). It exhibits broad-spectrum antiviral activity against coronaviruses, including SARS-CoV-2 wild type and its variants (XBB.1.18, HK.3.1, BF.7.14, BA.1, HCoV-229E, HCoV-OC43), as well as arenaviruses. HNC-1664 also demonstrates anti-infective efficacy in a mouse model infected with the SARS-CoV-2 Delta variant.</p>
    Formula:C12H13FIN3O3
    Color and Shape:Solid
    Molecular weight:393.153

    Ref: TM-T205157

  • DIDS
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    DIDS

    CAS:
    <p>DIDS inhibits anion exchangers reversibly then irreversibly and blocks RAD51.</p>
    Formula:C16H10N2O6S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.52

    Ref: TM-T20694

  • 2'-O-MOE-GMP
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    2'-O-MOE-GMP

    CAS:
    <p>2'-O-MOE-GMP is a nucleotide analogue that can be utilized in the synthesis of oligonucleotides.</p>
    Formula:C13H20N5O9P
    Color and Shape:Solid
    Molecular weight:421.30

    Ref: TM-TSW-00967

  • BET/Aurora kinase-IN-1
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    BET/Aurora kinase-IN-1

    CAS:
    <p>BET/Aurora kinase-IN-1 (Compound 38) is a dual inhibitor of BET and Aurora kinases. It exhibits antiproliferative activity against various tumor cell lines and demonstrates significant antitumor efficacy in xenograft models of renal cell carcinoma and colon cancer, with tumor growth inhibition (TGI) rates of 45.99% and 53.06%, respectively.</p>
    Formula:C25H30FN7O
    Color and Shape:Solid
    Molecular weight:463.55

    Ref: TM-T205073

  • VPC-80051
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    VPC-80051

    CAS:
    <p>VPC-80051 is an hnRNP A1 splicing activity inhibitor that directly interacts with the hnRNP A1 RBD and reduces AR-V7 messenger levels in the 22Rv1 CRPC cell line. VPC-80051 is applicable in prostate cancer research.</p>
    Formula:C16H13F2N3O
    Color and Shape:Solid
    Molecular weight:301.291

    Ref: TM-T204737

  • CLK1/2-IN-1
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    CLK1/2-IN-1

    CAS:
    CLK1/2-IN-1 is a CLK1 and CLK2 inhibitor and it also inhibits SRPK1 and SRPK2.
    Formula:C21H20F3N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.42

    Ref: TM-T23896

  • 2′-OMe-ADP
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    2′-OMe-ADP

    CAS:
    <p>2′-OMe-ADP is a nucleotide analogue used in oligonucleotide synthesis.</p>
    Formula:C11H17N5O10P2
    Color and Shape:Solid
    Molecular weight:441.23

    Ref: TM-TSW-00949

  • DENV-IN-6
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    DENV-IN-6

    CAS:
    <p>DENV-IN-6, a potent anti-DENV (I-IV) and HIV-1 IIIB inhibitor with EC50 ranging 6.8-17.5 μM for DENV and EC50 0.0181 μM for HIV-1.</p>
    Formula:C23H26ClFN4OS
    Color and Shape:Solid
    Molecular weight:461

    Ref: TM-T62908

  • CDK7-IN-26
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    CDK7-IN-26

    CAS:
    CDK7-IN-26 (compound 36) is an orally active CDK7 inhibitor with an IC50 of 7.4 nM. The compound effectively suppresses the growth of xenograft tumors derived from triple-negative breast cancer (TNBC) cell lines in vivo and has an IC50 of 0.15 μM for inhibiting MDA-MB-453 cells in vitro.
    Formula:C22H22FN6OPS
    Molecular weight:468.49

    Ref: TM-T208352

  • Antimalarial agent 44
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    Antimalarial agent 44

    Antimalarial agent 44 (Compound 3) is an antiparasitic agent effective against malaria. It exhibits good permeability in MDCK-MDR1 cell monolayers and has a high clearance rate in mouse liver microsomes.
    Formula:C37H37N5O7
    Color and Shape:Solid
    Molecular weight:663.72

    Ref: TM-T201453

  • PARG-IN-6
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    PARG-IN-6

    CAS:
    PARG-IN-6 (Compound 2) is an orally bioavailable PARG inhibitor with an IC50 of 0.3 nM. It exhibits significant anticancer activity against cancer cells, with an IC50 of 0.0368 μM for HCC1395 cells. PARG-IN-6 shows potential for research in colon cancer, appendiceal cancer, and pancreatic cancer.
    Formula:C24H25F4N7O4S3
    Color and Shape:Solid
    Molecular weight:647.69

    Ref: TM-T210766

  • FR-145715
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    FR-145715

    CAS:
    FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This compound is utilized in the study of gastric lesions.
    Formula:C16H21N5O2S
    Color and Shape:Solid
    Molecular weight:347.44

    Ref: TM-T201582

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    Antiangiogenic agent 2

    <p>Antiangiogenic agent 2 (compound 3b) is a potent inhibitor of thymidine phosphorylase (IC50: 39.71 μM) and exhibits anti-angiogenic effects.</p>
    Formula:C26H26FN3O4
    Color and Shape:Solid
    Molecular weight:463.5

    Ref: TM-T62931

  • PPA-037
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    PPA-037

    CAS:
    <p>PPA-037 is an orally active and highly selective inhibitor of cyclin-dependent kinase 12 (CDK12). It induces the degradation of Cyclin K, thereby enhancing antiproliferative effects on tumor cells. PPA-037 holds potential for use in cancer research.</p>
    Formula:C25H27N7
    Color and Shape:Solid
    Molecular weight:425.53

    Ref: TM-T207610

  • IIP0943
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    IIP0943

    CAS:
    <p>IIP0943 is a selective PLK1 (polo-like kinase 1) inhibitor with an IC50 of 5.1 nM for PLK1. It also exhibits inhibitory activity on the proliferation of HCT116 cells, with an IC50 of 0.22 µM. IIP0943 shows potential for research in the field of oncology.</p>
    Formula:C26H28N6O3S
    Color and Shape:Solid
    Molecular weight:504.604

    Ref: TM-T206115

  • FT709
    Targetmol
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    FT709

    CAS:
    <p>FT709 is a selective USP9X deubiquitinating enzyme inhibitor (IC50=82 nM) that reduces Makorin and ZNF598 levels, impairing ribosomal quality control pathways.</p>
    Formula:C23H22N4O7S
    Color and Shape:Solid
    Molecular weight:498.51

    Ref: TM-T63375

  • PNR-3-80
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    PNR-3-80

    CAS:
    PNR-3-80 is a selective inhibitor of apoptotic endonuclease G (EndoG), with an IC50 of 0.67 μM, showing greater inhibition than against DNase I. It exhibits no inhibitory activity against DNase II, RNase A, proteases, lactate dehydrogenase, and superoxide dismutase 1. PNR-3-80 effectively protects human prostate cancer cells from cell death induced by Cisplatin and Docetaxel and inhibits DNA damage and autophagy (autophagy) prompted by Etoposide. This compound is applicable in studies of cellular damage.
    Formula:C24H14ClN3O3S
    Color and Shape:Solid
    Molecular weight:459.90

    Ref: TM-T212403

  • DNA polymerase-IN-6
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    DNA polymerase-IN-6

    CAS:
    DNA polymerase-IN-6 (Compound 27) exhibits inhibitory activity against DNA polymerase, with EC50 values of 0.33 µM for HCMV, 1.9 µM for HSV-1, 0.76 µM for HSV-2, and 0.066 µM for EBV.
    Formula:C26H28ClFN8O4
    Color and Shape:Solid
    Molecular weight:571.003

    Ref: TM-T204284

  • OPN expression inhibitor 1
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    OPN expression inhibitor 1

    CAS:
    OPN expression inhibitor 1 is an osteopontin expression inhibitor used in the study of breast cancer metastasis.
    Formula:C25H33N3O5
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:455.55

    Ref: TM-T62820

  • CDK9/PARP-IN-1
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    CDK9/PARP-IN-1

    CAS:
    CDK9/PARP-IN-1 (compound 37) is an inhibitor of CDK9 and PARP. It demonstrates IC50 values of 118 nM for CDK9 and 107 nM for PARP1. This compound exhibits a broad-spectrum anti-proliferative effect across various cancer cell lines.
    Formula:C38H34F2N8O3
    Color and Shape:Solid
    Molecular weight:688.725

    Ref: TM-T205731

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    α5β1 integrin agonist-1

    CAS:
    α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.
    Formula:C24H26FN5O9
    Color and Shape:Solid
    Molecular weight:547.49

    Ref: TM-T63868

  • Chk1-IN-5
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    Chk1-IN-5

    CAS:
    Chk1-IN-5 inhibits Chk1, blocking phosphorylation and suppressing colon cancer growth.
    Formula:C18H18FN7O2
    Color and Shape:Solid
    Molecular weight:383.38

    Ref: TM-T37098

  • Mitotic kinesin-IN-1 hydrochloride
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    Mitotic kinesin-IN-1 hydrochloride

    CAS:
    Mitotic kinesin-IN-1 hydrochloride (Example 80) is an inhibitor of mitotic kinesin, which suppresses cell proliferation by hindering mitosis. This compound is applicable in research related to cancer, cardiac hypertrophy, immune and inflammatory diseases, and fungal infections.
    Formula:C22H26ClF2N3OS
    Color and Shape:Solid
    Molecular weight:453.98

    Ref: TM-T212561

  • WRN inhibitor 13
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    WRN inhibitor 13

    CAS:
    WRN inhibitor 13 is an inhibitor of the WRN helicase with a pIC50 value ranging from 6 to 7.
    Formula:C16H20N2O5S
    Color and Shape:Solid
    Molecular weight:352.405

    Ref: TM-T204389

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    CDK/HDAC-IN-1

    <p>CDK/HDAC-IN-1 inhibits CDK2/4/6 &amp; HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.</p>
    Formula:C20H18N4O4
    Color and Shape:Solid
    Molecular weight:378.38

    Ref: TM-T61583

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    c-Myc inhibitor 4

    <p>Potent oral c-Myc inhibitor 4 reduces the proto-oncogene linked to tumor development.</p>
    Formula:C26H33FN6O3
    Color and Shape:Solid
    Molecular weight:496.58

    Ref: TM-T63359

  • GFB-12811
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    GFB-12811

    CAS:
    <p>GFB-12811 is an orally active, selective, and potent CDK5 inhibitor, used in the study of autosomal dominant polycystic kidney disease.</p>
    Formula:C22H23F4N5O
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:449.44

    Ref: TM-T62695

  • CTPS1-IN-1
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    CTPS1-IN-1

    CAS:
    CTPS1-IN-1 is a cytidine-5′ triphosphate synthase 1 (CTPS1) inhibitor with potential antitumor activity and can be used to study autoimmune diseases.
    Formula:C21H22N6O4S2
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:486.57

    Ref: TM-T86105

  • HRO761
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    HRO761

    CAS:
    HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.
    Formula:C31H31ClF3N9O5
    Purity:98.74% - 99.62%
    Color and Shape:Solid
    Molecular weight:702.08

    Ref: TM-T72107

  • Elacytarabine
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    Elacytarabine

    CAS:
    <p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>
    Formula:C27H45N3O6
    Purity:97.69%
    Color and Shape:Solid
    Molecular weight:507.66

    Ref: TM-T15009

  • SR 11302
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    SR 11302

    CAS:
    SR 11302 is an inhibitor of activator protein-1 (AP-1).
    Formula:C26H32O2
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:376.53

    Ref: TM-T23384

  • LY3143921 hydrate
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    LY3143921 hydrate

    CAS:
    <p>LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].</p>
    Formula:C16H14FN5O2
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:327.31

    Ref: TM-T9064

  • INCB086550
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    INCB086550

    CAS:
    <p>INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 &lt;= 10 nM.</p>
    Formula:C41H39N7O4
    Purity:98.49%
    Color and Shape:Solid
    Molecular weight:693.79

    Ref: TM-T36899

  • Troxacitabine
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    Troxacitabine

    CAS:
    Troxacitabine, a DNA polymerase inhibitor, is potentially used for the treatment of acute myeloid leukemia (AML). In comparison with gemcitabine, troxacitabine was equally active against MiaPaCa and was more efficacious against Panc-01.
    Formula:C8H11N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:213.19

    Ref: TM-T17175

    1mg
    Discontinued
    Discontinued product
  • Bicyclomycin benzoate
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    Bicyclomycin benzoate

    CAS:
    Bicyclomycin benzoate (BCM benzoate, FR2054) is a broad-spectrum antibiotic and selective Rho protein inhibitor active against Gram-negative bacteria.
    Formula:C19H22N2O8
    Color and Shape:Solid
    Molecular weight:406.39

    Ref: TM-T10541

    1mg
    Discontinued
    Discontinued product
  • PLK1-IN-6
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    PLK1-IN-6

    <p>PLK1-IN-6: potent, selective PLK1 inhibitor, IC50 = 0.45 nM, hinders cancer cell growth.</p>
    Formula:C28H37N9O3
    Color and Shape:Solid
    Molecular weight:547.65

    Ref: TM-T74777

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • 5'-DMT-3'-TBDMS-ibu-rG
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    5'-DMT-3'-TBDMS-ibu-rG

    CAS:
    <p>5'-DMT-3'-TBDMS-ibu-rG is a modified nucleoside employed in deoxyribonucleic acid (DNA) synthesis.</p>
    Formula:C41H51N5O8Si
    Color and Shape:Solid
    Molecular weight:769.96

    Ref: TM-T40919

    ne
    Discontinued
    Discontinued product
  • NSC639828
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    NSC639828

    CAS:
    NSC639828 is an efficient inhibitor of DNA polymerase α, exhibiting a remarkable IC50 value of 70 μM. Additionally, NSC639828 demonstrates substantial antitumor activity, making it a promising candidate for cancer research.
    Formula:C18H13BrClN5O3
    Color and Shape:Solid
    Molecular weight:462.69

    Ref: TM-T38742

    ne
    Discontinued
    Discontinued product
  • Ethynylcytidine
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    Ethynylcytidine

    CAS:
    <p>Ethynylcytidine is a nucleoside antimetabolite.</p>
    Formula:C11H13N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.24

    Ref: TM-TQ0006

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Tanuxiciclib
    Targetmol
    + Info

    Tanuxiciclib

    CAS:
    Tanuxiciclib is a cyclin dependent kinase (CDK) inhibitor, specifically designed to interfere with cell cycle progression by inhibiting the activity of CDKs, which are crucial regulators of cell division.
    Formula:C15H13FN6O
    Color and Shape:Solid
    Molecular weight:312.308

    Ref: TM-T39404

    ne
    Discontinued
    Discontinued product
  • N6-Benzoyl-5′-O-(4,4′-dimethoxytrityl)-2′-deoxyadenosine
    Targetmol
    + Info

    N6-Benzoyl-5′-O-(4,4′-dimethoxytrityl)-2′-deoxyadenosine

    CAS:
    N6-Benzoyl-5′-O-(4,4′-dimethoxytrityl)-2′-deoxyadenosine, catalog number T66118 and CAS number 64325-78-6, is a valuable organic compound for life sciences research.
    Formula:C38H35N5O6
    Color and Shape:Solid
    Molecular weight:657.727

    Ref: TM-T66118

    ne
    Discontinued
    Discontinued product
  • Formycin A
    Targetmol
    + Info

    Formycin A

    CAS:
    Formycin A shows antitumor and antiviral activities. Formycin A , a purine nucleoside antibiotic, is a potent human immunodeficiency virus type 1 (HIV-1) inhibitor with an EC50 of 10 μM.
    Formula:C10H13N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.24

    Ref: TM-T11312

    5mg
    Discontinued
    Discontinued product
  • GSK-3/CDK5/CDK2-IN-1
    Targetmol
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    GSK-3/CDK5/CDK2-IN-1

    CAS:
    GSK-3/CDK5/CDK2-IN-1 is an imidazole derivative compound that inhibits cdk5, cdk2, and GSK-3.it has demonstrated applications in cancer research and the study of neurodegenerative diseases [1].
    Formula:C21H22N4O2
    Color and Shape:Solid
    Molecular weight:362.433

    Ref: TM-T35555

    ne
    Discontinued
    Discontinued product
  • 5'-O-DMT-N6-ibu-dA
    Targetmol
    + Info

    5'-O-DMT-N6-ibu-dA

    CAS:
    5'-O-DMT-N6-ibu-dA can be utilized in the synthesis of oligodeoxyribonucleotides.
    Formula:C35H37N5O6
    Color and Shape:Solid
    Molecular weight:623.71

    Ref: TM-T39332

    ne
    Discontinued
    Discontinued product
  • 2'-Deoxy-2'-fluoro-5-iodouridine
    Targetmol
    + Info

    2'-Deoxy-2'-fluoro-5-iodouridine

    CAS:
    2'-Deoxy-2'-fluoro-5-iodouridine is a nucleoside, specifically a fluoro-modified and halo-nucleoside.
    Formula:C9H10FIN2O5
    Color and Shape:Solid
    Molecular weight:372.09

    Ref: TM-TNU0622

    ne
    Discontinued
    Discontinued product
  • 3BrB-PP1
    Targetmol
    + Info

    3BrB-PP1

    CAS:
    3BrB-PP1 is an ATP-competitive analog that exhibits specific inhibitory activity towards protein kinase, particularly effective against protein kinases with mutations in the ATP-binding pocket, such as the Thr97 mutation within Sty1's ATP-binding pocket.
    Formula:C16H18BrN5
    Color and Shape:Solid
    Molecular weight:360.259

    Ref: TM-T41113

    ne
    Discontinued
    Discontinued product
  • PF-03814735
    Targetmol
    + Info

    PF-03814735

    CAS:
    PF-03814735 is a novel, potent and reversible inhibitor of Aurora A/B with IC50of 0.8 nM/5 nM, is less potent to Flt3, FAK, TrkA, and minimally active to Met and FGFR1. Phase 1.
    Formula:C23H25F3N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.48

    Ref: TM-T6936

    1mg
    Discontinued
    Discontinued product
  • MitoE10
    Targetmol
    + Info

    MitoE10

    CAS:
    <p>MitoE10 is an effective mitochondrial targeting antioxidant.</p>
    Formula:C42H55O5PS
    Color and Shape:Solid
    Molecular weight:702.92

    Ref: TM-T33406

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Ribocil-C
    Targetmol
    + Info

    Ribocil-C

    CAS:
    Ribocil-C is a selective inhibitor of the bacterial riboflavin riboswitch, a synthetic analogue of flavin mononucleotide (FMN), inhibits bacterial cell growth.
    Formula:C21H21N7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.5

    Ref: TM-T12722L

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • 6-Amino-5-nitropyridin-2-one
    Targetmol
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    6-Amino-5-nitropyridin-2-one

    CAS:
    <p>6-Amino-5-nitropyridin-2-one, a pyridine derivative, serves as a nucleobase within hachimoji DNA, where it is specifically paired with 5-aza-7-deazaguanine.</p>
    Formula:C5H5N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:155.11

    Ref: TM-T19157

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Tibremciclib
    Targetmol
    + Info

    Tibremciclib

    CAS:
    <p>Tibremciclib is a cyclin-dependent kinase 4 (CDK4) inhibitor that exhibits antineoplastic properties [1].</p>
    Formula:C28H32F2N8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.6

    Ref: TM-T79863

    ne
    Discontinued
    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • PHI-101
    Targetmol
    + Info

    PHI-101

    CAS:
    <p>PHI-101 is a checkpoint kinase 2 (Chk2) inhibitor that can be used for the study of refractory acute myeloid leukemia (AML) and ovarian cancer.</p>
    Formula:C19H19FN4O2S
    Purity:99.4%
    Color and Shape:Solid
    Molecular weight:386.44

    Ref: TM-T81490

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    200mg
    Discontinued
    Discontinued product
  • YK-2168
    Targetmol
    + Info

    YK-2168

    CAS:
    <p>YK-2168 is a differentiated selective inhibitor of CDK9.</p>
    Formula:C16H18ClN5
    Color and Shape:Solid
    Molecular weight:315.80

    Ref: TM-T200769

    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product