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PKC
Miltefosine
CAS:58066-85-6
Miltefosine is the treatment of visceral and cutaneous leishmaniasis drug , and is proceeding clinical …
Formula:
C21H46NO4P
Purity:
99.51%
Color and Shape:
White To Off-White Powder
Molecular weight:
407.58
Estimated delivery in United States, on Thursday 3 Feb 2022
TAS301
CAS:193620-69-8
TAS-301, an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon …
Formula:
C23H19NO3
Purity:
99.69%
Color and Shape:
solid
Molecular weight:
357.4
Estimated delivery in United States, on Thursday 3 Feb 2022
Ruboxistaurin hydrochloride
CAS:169939-93-9
Isozyme-selective inhibitor of protein kinase C (PKC); competitively and reversibly inhibits PKCI and PKCII (IC50 …
Formula:
C28H28N4O3·HCl
Purity:
95.97%
Molecular weight:
505.01
Estimated delivery in United States, on Thursday 3 Feb 2022
Enzastaurin
CAS:170364-57-5
Enzastaurin (LY317615) is an effective PKC selective inhibitor (IC50: 6 nM), 6- to 20-fold selectivity …
Formula:
C32H29N5O2
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
515.61
Estimated delivery in United States, on Thursday 3 Feb 2022
Go 6983
CAS:133053-19-7
Go 6983 is a pan-PKC inhibitor against for PKC, PKC, PKC, PKC and PKC with …
Formula:
C26H26N4O3
Purity:
99.04%
Color and Shape:
solid
Molecular weight:
442.51
Estimated delivery in United States, on Thursday 3 Feb 2022
Chelerythrine chloride
CAS:3895-92-9
Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the …
Formula:
C21H18ClNO4
Purity:
99.19%
Color and Shape:
Yellow To Orange Solid
Molecular weight:
383.83
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC-iota inhibitor 1
CAS:2328094-11-5
PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC- ; IC50 : 0.34 …
Formula:
C21H22N6O
Color and Shape:
solid
Molecular weight:
374.4
Estimated delivery in United States, on Thursday 3 Feb 2022
6,7,4'-Trihydroxyisoflavone
CAS:17817-31-1
6,7,4'-Trihydroxyisoflavone, is a novel inhibitor of PKC in suppressing solar UV-induced matrix metalloproteinase 1, which …
Formula:
C15H10O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
270.2
Estimated delivery in United States, on Thursday 3 Feb 2022
Chelerythrine
CAS:34316-15-9
1. Chelerythrine may have antimanic effect . 2. Chelerythrine can inhibit telomerase activity. 3. Chelerythrine …
Formula:
C21H18NO4
Purity:
98.86%
Color and Shape:
solid
Molecular weight:
348.37
Estimated delivery in United States, on Thursday 3 Feb 2022
K-252b
CAS:99570-78-2
K-252b is an indolocarbazole isolated from the actinomycete Nocardiopsis and is a PKC inhibitor. K-252b …
Formula:
C26H19N3O5
Purity:
98.00%
Color and Shape:
Ready-To-Use Solution
Molecular weight:
453.45
Estimated delivery in United States, on Thursday 3 Feb 2022
Y-33075
CAS:199433-58-4
Y-33075 is a selective inhibitor of ROCK derived from Y-27632, and is more potent than …
Formula:
C16H16N4O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
280.32
Estimated delivery in United States, on Thursday 3 Feb 2022
Bisindolylmaleimide V
CAS:113963-68-1
Bisindolylmaleimide V (BIM V) is a weak protein kinase C (PKC)inhibitor( IC50 >100 µM)
Formula:
C21H15N3O2
Purity:
98.00%
Color and Shape:
Red Solid
Molecular weight:
341.37
Estimated delivery in United States, on Thursday 3 Feb 2022
LXS196
CAS:1874276-76-2
LXS196 is a potent, selective and orally active protein kinase C (PKC) inhibitor(IC50 values of …
Formula:
C22H23F3N8O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
472.47
Estimated delivery in United States, on Thursday 3 Feb 2022
Midostaurin
CAS:120685-11-2
PKC412(Midostaurin; CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor. Midostaurin inhibits protein kinase C …
Formula:
C35H30N4O4
Purity:
98.86%
Color and Shape:
solid
Molecular weight:
570.64
Estimated delivery in United States, on Thursday 3 Feb 2022
VTX-27
CAS:1321924-70-2
VTX-27 is a selective inhibitor of protein kinase C (PKC ) (Kis: 0.08 nM and …
Formula:
C20H24ClFN6O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
418.9
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC-theta inhibitor 1
CAS:1160501-81-4
PKC-theta inhibitor 1 is an inhibitor of PKC (Ki of 6 nM)
Formula:
C17H15F3N4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
348.32
Estimated delivery in United States, on Thursday 3 Feb 2022
Dequalinium chloride
CAS:522-51-0
Dequalinium Chloride, a topical bacteriostat, is a selective blocker of apamin-sensitive K+ channels. It is …
Formula:
C30H40Cl2N4
Purity:
99.80%
Color and Shape:
solid
Molecular weight:
527.59
Estimated delivery in United States, on Thursday 3 Feb 2022
Phorbol 12,13-dibutyrate
CAS:37558-16-0
Phorbol 12,13-dibutyrate is a PKC activator. It also is a potent skin tumor promoter.
Formula:
C28H40O8
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
504.61
Estimated delivery in United States, on Thursday 3 Feb 2022
Hypocrellin A
CAS:77029-83-5
Hypocrellin A is PKC inhibitor, has light-induced antitumor,antifungal and antiviral activities, it also exerts immunomodulatory …
Formula:
C30H26O10
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
546.52
Estimated delivery in United States, on Thursday 3 Feb 2022
Sotrastaurin
CAS:425637-18-9
Sotrastaurin is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKC/I////).
Formula:
C25H22N6O2
Purity:
99.41%
Color and Shape:
solid
Molecular weight:
438.48
Estimated delivery in United States, on Thursday 3 Feb 2022
Cercosporin
CAS:35082-49-6
Cercosporin is produced by a plant pathogen, Cercosporakikuchii, and the elsinochromes. Cercosporin is a potent …
Formula:
C29H26O10
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
534.51
Estimated delivery in United States, on Thursday 3 Feb 2022
PS315
CAS:1221964-50-6
PS315 inhibits the full-length and catalytic domain constructs of PKC (IC50=10 μM) and PKC (IC50=30 …
Formula:
C23H19ClO2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
362.85
Estimated delivery in United States, on Thursday 3 Feb 2022
(-)-Indolactam V
CAS:90365-57-4
(-)-Indolactam V is a PKC activator (Kis: 3.36 nM, 1.03 μM for -CRD2 , -CRD2). …
Formula:
C17H23N3O2
Purity:
98.00%
Color and Shape:
White To Off-White Solid
Molecular weight:
301.38
Estimated delivery in United States, on Thursday 3 Feb 2022
K-252c
CAS:85753-43-1
K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor …
Formula:
C20H13N3O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
311.34
Estimated delivery in United States, on Thursday 3 Feb 2022
Decursin
CAS:5928-25-6
1. Decursin is able to attenuate kainic acid-induced seizures and could have potential as an …
Formula:
C19H20O5
Purity:
97.22%
Color and Shape:
solid
Molecular weight:
328.36
Estimated delivery in United States, on Thursday 3 Feb 2022
Ro 31-8220 Mesylate
CAS:138489-18-6
Ro 31-8220 is a pan-PKC inhibitor for PKC-/I/II// (IC50: 5/24/14/27/24 nM), and also shows potent …
Formula:
C25H23N5O2S·CH4O3S
Purity:
99.02%
Color and Shape:
solid
Molecular weight:
553.65
Estimated delivery in United States, on Thursday 3 Feb 2022
Sodium aurothiomalate
CAS:12244-57-4
Sodium aurothiomalate is a gold compound that is used for its immunosuppressive anti-rheumatic effects. Aurothiomalate …
Formula:
C4H3AuNa2O4S
Molecular weight:
390.07
Estimated delivery in United States, on Thursday 3 Feb 2022
Valrubicin
CAS:56124-62-0
Valrubicin (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and …
Formula:
C34H32F3NO13
Purity:
97.41%
Color and Shape:
solid
Molecular weight:
723.64
Estimated delivery in United States, on Thursday 3 Feb 2022
BJE6-106
CAS:1564249-38-2
BJE6-106 (B106) is a potent, selective PKC inhibitor (IC50: 0.05 μM) and targets selectivity over …
Formula:
C26H23NO2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
381.47
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC-IN-1
CAS:1046787-18-1
PKC-IN-1 is a ATP-competitive and reversible conventional PKC enzymes inhibitor (PKC, PKCI, PKCII, PKC, PKC, …
Formula:
C25H37FN8O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
500.61
Estimated delivery in United States, on Thursday 3 Feb 2022
DCPLA-ME
CAS:56687-67-3
DCPLA-ME is the methyl ester form of DCPLA and can be used to treat neurodegenerative …
Formula:
C21H38O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
322.53
Estimated delivery in United States, on Thursday 3 Feb 2022
Cholesterol 3-Sulfate Sodium Salt
CAS:2864-50-8
Cholesterol sulfate is a sterol sulfate in human plasma. It is a component of cell …
Formula:
C27H45NaO4S
Purity:
99.82%
Color and Shape:
White To Off-White Solid/Powder
Molecular weight:
488.7
Estimated delivery in United States, on Thursday 3 Feb 2022
Hispidin
CAS:555-55-5
Hispidin is a polyphenol originally, including antioxidant, anti-inflammatory, and cytoprotective properties
Formula:
C13H10O5
Purity:
99.55%
Color and Shape:
White Crystalline Powder
Molecular weight:
246.22
Estimated delivery in United States, on Thursday 3 Feb 2022
Plantainoside D
CAS:147331-98-4
Plantainoside D shows potent antioxidative effects as those of ascorbic acid, it shows angiotensin-converting enzyme …
Formula:
C29H36O16
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
640.6
Estimated delivery in United States, on Thursday 3 Feb 2022
Bisindolylmaleimide X hydrochloride
CAS:145317-11-9
Bisindolylmaleimide X hydrochloride (BIM-X hydrochloride) is a potent and selective PKC inhibitor. It is also …
Formula:
C26H25ClN4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
460.96
Estimated delivery in United States, on Thursday 3 Feb 2022
ZIP acetate(863987-12-6 free base)
ZIP acetate is a novel, cell-permeable inhibitor of protein kinase M (PKM), a constitutively active, …
Formula:
C92H158N30O19
Molecular weight:
1988.43
Estimated delivery in United States, on Thursday 3 Feb 2022
Ingenol
CAS:30220-46-3
1. Ingenol mebutate is an effective treatment for actinic keratosis. 2. Formulating novel derivatives from …
Formula:
C20H28O5
Purity:
99.87%
Color and Shape:
solid
Molecular weight:
348.43
Estimated delivery in United States, on Thursday 3 Feb 2022
Y06137
CAS:2226534-49-0
Y06137 is a potent and selective inhibitor of BET, and used for treatment of castration-resistant …
Formula:
C27H32N4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
444.57
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC inhibitor 1
CAS:257879-35-9
PKC inhibitor 1(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 …
Formula:
C24H21N5O2
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
411.5
Estimated delivery in United States, on Thursday 3 Feb 2022
Protein Kinase C 19-31 acetate
Protein Kinase C 19-31 acetate, a peptide inhibitor of protein kinase C (PKC), derived from …
Formula:
C69H122N26O18
Purity:
100.00%
Molecular weight:
1603.9
Estimated delivery in United States, on Thursday 3 Feb 2022
Myricetrin
CAS:17912-87-7
Myricitrin, a flavonoid compound isolated from the root bark of Myrica cerifera, exerts antinociceptive effects.
Formula:
C21H20O12
Purity:
97.16%
Color and Shape:
Light Yellow To Off-White Crystalline Powder
Molecular weight:
464.38
Estimated delivery in United States, on Thursday 3 Feb 2022
Phorbol
CAS:17673-25-5
Phorbol, a plant-derived diterpene, is a tumor promoter through the activation of protein kinase C.
Formula:
C20H28O6
Purity:
99.10%
Color and Shape:
solid
Molecular weight:
364.43
Estimated delivery in United States, on Thursday 3 Feb 2022
DCP-LA
CAS:28399-31-7
DCP-LA (FR236924), linoleic acid derivatives, selective and direct activation of PKC.
Formula:
C20H36O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
308.5
Estimated delivery in United States, on Thursday 3 Feb 2022
TPPB
CAS:497259-23-1
TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
Formula:
C27H30F3N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
501.54
Estimated delivery in United States, on Thursday 3 Feb 2022
AS2521780
CAS:1214726-89-2
AS2521780 is an inhibitor of PKC (IC50: 0.48 nM).
Formula:
C30H41N7OS
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
547.76
Estimated delivery in United States, on Thursday 3 Feb 2022
Procyanidin A1
CAS:103883-03-0
Procyanidin A1 has antiallergic effects, it inhibits degranulation downstream of protein kinase C activation or …
Formula:
C30H24O12
Purity:
99.23%
Color and Shape:
solid
Molecular weight:
576.5
Estimated delivery in United States, on Thursday 3 Feb 2022
Bryostatin 1
CAS:83314-01-6
Bryostatin 1 is a natural macrolide isolated from the bryozoan Bugula neritina and is a …
Formula:
C47H68O17
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
905.03
Estimated delivery in United States, on Thursday 3 Feb 2022
1,2-Dipalmitoyl-sn-glycerol
CAS:30334-71-5
1,2-Dipalmitoyl-sn-glycerol is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC.
Formula:
C35H68O5
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
568.91
Estimated delivery in United States, on Thursday 3 Feb 2022
Staurosporine
CAS:62996-74-1
Staurosporine is a potent PKC inhibitor for PKC// (IC50: 2/5/4 nM), less potent to PKC …
Formula:
C28H26N4O3
Purity:
99.30%
Color and Shape:
Off-White Powder
Molecular weight:
466.53
Estimated delivery in United States, on Thursday 3 Feb 2022
CRT0066854 hydrochloride
CAS:2250019-91-9
CRT0066854 hydrochloride is an effective selective atypical PKCs inhibitor. CRT0066854 is against full-length (FL) PKC, …
Formula:
C24H26ClN5S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
452.01
Estimated delivery in United States, on Thursday 3 Feb 2022
Bisindolylmaleimide IV
CAS:119139-23-0
Bisindolylmaleimide IV is a protein kinase C (PKC) cell permeable inhibitor( IC50 : 0.10 - …
Formula:
C20H13N3O2
Purity:
98.20%
Color and Shape:
Dark Red Solid
Molecular weight:
327.34
Estimated delivery in United States, on Thursday 3 Feb 2022
Leucosceptoside A
CAS:83529-62-8
Leucosceptoside A shows inhibitory activity against PKCalpha with the IC50 value of 19.0 microM; it …
Formula:
C30H38O15
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
638.61
Estimated delivery in United States, on Thursday 3 Feb 2022
[Ala107]-MBP (104-118) acetate
[Ala107]-MBP (104-118) acetate is synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor …
Formula:
C59H108N20O21
Purity:
99.23%
Molecular weight:
1553.72
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC pseudosubstrate acetate
PKC pseudosubstrate acetate is an inhibitor of protein kinase C (PKC) ; attached to cell …
Molecular weight:
N/A
Estimated delivery in United States, on Thursday 3 Feb 2022
Iso-H7 dihydrochloride
CAS:140663-38-3
Iso-H7 dihydrochloride is a less potent inhibitor of phosphokinase C than H-7.
Formula:
C14H19Cl2N3O2S
Color and Shape:
White Crystalline Solid
Molecular weight:
364.29
Estimated delivery in United States, on Thursday 3 Feb 2022
Delcasertib
CAS:949100-39-4
Delcasertib is a potent and selective inhibitor of -protein kinase C (PKC).
Formula:
C120H199N45O34S2
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
2880.28
Estimated delivery in United States, on Thursday 3 Feb 2022
20-Deoxyingenol 3-angelate
CAS:75567-38-3
20-Deoxyingenol 3-angelate and ingenol 20-acetate 3-angelate are known as promoters of tumors of mouse skin. …
Formula:
C25H34O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
414.6
Estimated delivery in United States, on Thursday 3 Feb 2022
Pep2m, myristoylated acetate
Pep2m, myristoylated acetate is a Cell-permeable, myristoylated form of pep2m. Peptide inhibitor of the interaction …
Formula:
C65H122N18O16S
Purity:
99.62%
Molecular weight:
1443.96
Estimated delivery in United States, on Thursday 3 Feb 2022
Clitorin
CAS:55804-74-5
Clitorin has free radical scavenging property. It shows significant interactions with CD38, it may have …
Formula:
C33H40O19
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
740.66
Estimated delivery in United States, on Thursday 3 Feb 2022
PKC-theta inhibitor hcl
CAS:2253640-49-0
PKC-theta inhibitor is a selective PKC-inhibitor(IC50:12 nM).
Formula:
C20H25F3N6O3
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
454.4
Estimated delivery in United States, on Thursday 3 Feb 2022
(Z)-Butylidenephthalide
CAS:72917-31-8
(Z)-Butylidenephthalide has antitumor effect, can effectively inhibit the tumor growth in the glioma.
Formula:
C12H12O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
188.2
Estimated delivery in United States, on Thursday 3 Feb 2022
