
Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(230 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(126 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(34 products)
- Vasopressin Receptor(48 products)
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Found 3427 products of "Endocrinology/Hormones"
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[Leu5]-Enkephalin acetate(58822-25-6 free base)
Endogenous [Leu5]-Enkephalin acetate is a δ- and μ-opioid receptor agonist involved in pain; Ki: δ=4.0 nM, μ=3.4 nM.Formula:C30H41N5O9Purity:99.28%Color and Shape:SolidMolecular weight:615.68Sulindac sulfone
CAS:Sulindac sulfone is a metabolite of the nonsteroidal anti-inflammatory drug sulindac. Sulindac sulfone is an inhibitor of aldose reductase (IC50 =367 nM).Formula:C20H17FO4SPurity:98.2% - 98.83%Color and Shape:SolidMolecular weight:372.41Ref: TM-T23403
5mg52.00€1mL*10mM (DMSO)52.00€10mg78.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€GSK5182
CAS:GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)Formula:C27H31NO3Purity:97.63% - 99.42%Color and Shape:SolidMolecular weight:417.54Ref: TM-T8370
1mg50.00€2mg71.00€5mg90.00€1mL*10mM (DMSO)108.00€10mg144.00€25mg260.00€50mg394.00€100mg582.00€Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Formula:C19H19ClN6O2Purity:97.36% - >99.99%Color and Shape:SolidMolecular weight:398.85Ref: TM-T6915
1mg50.00€2mg66.00€5mg100.00€1mL*10mM (DMSO)101.00€10mg158.00€25mg250.00€50mg358.00€100mg512.00€200mg732.00€Obafistat
CAS:Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.Formula:C15H16FN5O3SPurity:99.71%Color and Shape:SolidMolecular weight:365.38Ref: TM-T39635
1mL*10mM (DMSO)33.00€1mg37.00€2mg49.00€5mg80.00€10mg111.00€25mg178.00€50mg290.00€100mg469.00€200mg647.00€WAY-200070
CAS:WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).Formula:C13H8BrNO3Purity:99.45% - 99.75%Color and Shape:SolidMolecular weight:306.11Ref: TM-T3958
2mg39.00€5mg58.00€1mL*10mM (DMSO)64.00€10mg90.00€25mg178.00€50mg295.00€100mg477.00€200mg677.00€EBPC
CAS:EBPC is an inhibitor of aldose reductase.Formula:C14H15NO4Purity:99.55%Color and Shape:SolidMolecular weight:261.27Ref: TM-T22757
1mg40.00€5mg77.00€1mL*10mM (DMSO)86.00€10mg105.00€25mg182.00€50mg261.00€100mg371.00€200mg502.00€Naloxegol (NKTR-118)
CAS:Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].Formula:C34H53NO11Color and Shape:SolidMolecular weight:651.78LY404039
CAS:LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).Formula:C7H9NO6SPurity:99% - 99.92%Color and Shape:SolidMolecular weight:235.22Temocapril hydrochloride
CAS:Temocapril hydrochloride (CS-622 HCl), the hydrochloride of Temocapril, is a long-acting ACE inhibitor used for the therapy of hypertension.Formula:C23H28N2O5S2·HClPurity:99.26% - 99.48%Color and Shape:White Solid PowderMolecular weight:513.07L-Thyroxine sodium
CAS:L-Thyroxine sodium (LT4 sodium), the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.Formula:C15H10I4NO4·NaPurity:98.74%Color and Shape:Yellowish To Buff-Colored Amorphous Powder SolidMolecular weight:798.85AL 082D06
CAS:AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.Formula:C23H24ClN3O2Purity:99.05% - 99.06%Color and Shape:SolidMolecular weight:409.91Estradiol dipropionate
CAS:Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.Formula:C24H32O4Purity:99.68%Color and Shape:SolidMolecular weight:384.51TRV-120027 TFA
TRV-120027 TFA is an angiotensin II–mediated vasoconstriction inhibitor and increases cardiomyocyte contractility.Formula:C45H68F3N13O12Purity:97.45%Color and Shape:SolidMolecular weight:1040.1Ref: TM-TP2158
1mg43.00€5mg111.00€10mg170.00€1mL*10mM (DMSO)193.00€25mg293.00€50mg423.00€100mg577.00€200mg778.00€Iprodione
CAS:Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.Formula:C13H13Cl2N3O3Purity:98.82%Color and Shape:Colorless Crystals Cream To Colorless Odorless PowderMolecular weight:330.17AZD9496
CAS:AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.Formula:C25H25F3N2O2Purity:97.28% - 98.47%Color and Shape:SolidMolecular weight:442.47Ref: TM-T3975
1mg52.00€2mg73.00€1mL*10mM (DMSO)105.00€5mg110.00€10mg178.00€25mg334.00€50mg494.00€100mg712.00€Beclometasone dipropionate monohydrate
CAS:Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.Formula:C28H39ClO8Color and Shape:SolidMolecular weight:539.06VTP-27999 TFA
CAS:VTP-27999 TFA is an inhibitor of Renin (IC50 : 0.47 nM).Formula:C28H42ClF3N4O7Purity:98.84%Color and Shape:SolidMolecular weight:639.13-chloro-5-hydroxybenzoic Acid
CAS:3-chloro-5-hydroxy Benzoic Acid (3-chloro-5-hydroxy BA) is an agonist of GPR81 (EC50 : 16 μM)Formula:C7H5ClO3Purity:98%Color and Shape:SolidMolecular weight:172.572-Chloro-1-(4-fluorobenzyl)benzimidazole
CAS:2-Chloro-1-(4-fluorobenzyl)benzimidazole is an inhibitor of aldose reductase (ALR2).Formula:C14H10ClFN2Purity:99.64%Color and Shape:SolidMolecular weight:260.69Abaloparatide TFA
Abaloparatide TFA (BIM 44058 TFA) is a parathyroid hormone-related protein (PTHrP) analog drug used to treat osteoporosis like the related drug teriparatide.Formula:C176H301N56F3O51Purity:99.76%Color and Shape:SolidMolecular weight:4074.611-methoxycyclopropanecarboxylic acid
CAS:1-methoxycyclopropanecarboxylic acid is an agonist of free fatty acid receptor 3 (FFAR3, human).
Formula:C5H8O3Purity:99.44%Color and Shape:Light-Yellow To Yellow Solid Or LiquidMolecular weight:116.12Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFormula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Formula:C18H13ClF4N2O3Purity:99.55%Color and Shape:SolidMolecular weight:416.75SNG-1153
CAS:SNG-1153 is a estrogen receptor ER-alpha36 modulator.Formula:C21H17F3O5Purity:99.74%Color and Shape:SolidMolecular weight:406.35Galeterone
CAS:Galeterone (VN 124) is an oral androgen receptor modulator/CYP17 inhibitor with antiandrogen properties, targeting prostate cancer growth.Formula:C26H32N2OPurity:99.47% - 99.773%Color and Shape:SolidMolecular weight:388.55Eprotirome
CAS:Eprotirome (KB2115), a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.Formula:C18H17Br2NO5Purity:98.42% - 98.56%Color and Shape:SolidMolecular weight:487.14Ref: TM-T5360
2mg34.00€5mg50.00€1mL*10mM (DMSO)52.00€10mg80.00€25mg145.00€50mg222.00€100mg356.00€200mg522.00€CLP-3094
CAS:CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.Formula:C15H13ClN2OSPurity:99.84%Color and Shape:SolidMolecular weight:304.79G15
CAS:G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)Formula:C19H16BrNO2Purity:98.46% - 98.59%Color and Shape:SolidMolecular weight:370.24Angiotensin I/II (1-5)
CAS:Angiotensin I/II (1-5) is a peptide (ASP-ARG-VAL-TYR-ILE) that contains the amino acids 1-5 and is converted from Angiotensin I/II.Formula:C30H48N8O9Purity:>99.99%Color and Shape:SolidMolecular weight:664.75Canrenoate potassium
CAS:Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.Formula:C22H29KO4Purity:99.04% - 99.18%Color and Shape:Light Yellow To Tan PowderMolecular weight:396.56Angiotensin II 5-valine TFA
Angiotensin II 5-valine TFA is an agonist of angiotensin receptor.Formula:C51H70F3N13O14Purity:99.69%Color and Shape:SolidMolecular weight:1146.18Sobetirome
CAS:Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).Formula:C20H24O4Purity:98.08% - 98.25%Color and Shape:SolidMolecular weight:328.4Ulipristal
CAS:Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.Formula:C28H35NO3Purity:99.82%Color and Shape:SolidMolecular weight:433.58GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purity:99.75%Color and Shape:SolidMolecular weight:530.4Ref: TM-T9459
1mg93.00€2mg136.00€5mg178.00€1mL*10mM (DMSO)236.00€10mg268.00€25mg482.00€50mg688.00€100mg964.00€RU 58841
CAS:RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.Formula:C17H18F3N3O3Purity:99.31% - 99.70%Color and Shape:SolidMolecular weight:369.34Ref: TM-T2236
5mg40.00€1mL*10mM (DMSO)48.00€10mg63.00€25mg99.00€50mg130.00€100mg177.00€200mg245.00€500mg371.00€Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purity:99.45% - 99.78%Color and Shape:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMolecular weight:361.39Tasosartan
CAS:Tasosartan (WAY-ANA 756) is an antagonist of angiotensin II type 2 (AT2) receptor (IC50 = 1.2 nM).Formula:C23H21N7OPurity:98.2% - 98.9%Color and Shape:SolidMolecular weight:411.46Ref: TM-T7797
1mg52.00€2mg77.00€5mg113.00€1mL*10mM (DMSO)124.00€10mg177.00€25mg299.00€50mg447.00€100mg623.00€WAY-169916
CAS:WAY-169916 inhibits ER by blocking NF-kB activity, lacks estrogenic effects.Formula:C17H13F3N2O2Purity:98.63% - 98.64%Color and Shape:SolidMolecular weight:334.29Ref: TM-T8981
2mg39.00€5mg60.00€1mL*10mM (DMSO)89.00€10mg92.00€25mg187.00€50mg313.00€100mg450.00€200mg620.00€Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Formula:C36H55NO15Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:741.83Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS:Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.Formula:C18H18O3Purity:99.85% - 99.96%Color and Shape:SolidMolecular weight:282.33Ref: TM-T9800
1mg93.00€1mL*10mM (DMSO)172.00€5mg182.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,099.00€Chlorotrianisene
CAS:Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.Formula:C23H21ClO3Purity:98.88% - 99.03%Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)Molecular weight:380.86Ref: TM-T2569
1mg54.00€5mg114.00€1mL*10mM (DMSO)126.00€10mg178.00€25mg313.00€50mg464.00€100mg660.00€200mg888.00€Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04Spinorphin
CAS:Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.Formula:C45H64N8O10Purity:99.68%Color and Shape:SolidMolecular weight:877ARV-471
CAS:ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
Formula:C45H49N5O4Purity:97.15% - >99.99%Color and Shape:SolidMolecular weight:723.9Apararenone
CAS:Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.Formula:C17H17FN2O4SPurity:99.79%Color and Shape:SolidMolecular weight:364.39BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purity:>99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-TP1905
2mg39.00€5mg58.00€1mL*10mM (DMSO)73.00€10mg93.00€25mg145.00€50mg260.00€100mg462.00€200mg655.00€Propyl pyrazole triol
CAS:PPT is a selective ERα agonist with 410x higher affinity than for ERβ.Formula:C24H22N2O3Purity:97.86%Color and Shape:SolidMolecular weight:386.44Ref: TM-T16566
1mg43.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg133.00€25mg250.00€50mg378.00€100mg570.00€200mg800.00€[Leu5]-Enkephalin TFA(58822-25-6(free bas))
CAS:[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor agoFormula:C30H38F3N5O9Purity:97.03% - 99.78%Color and Shape:SolidMolecular weight:669.644-Hydroxytamoxifen
CAS:4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.Formula:C26H29NO2Purity:99.37% - 99.93%Color and Shape:SolidMolecular weight:387.51
